Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01196 , Somatostatin receptor type 5
Gene Name SSTR5
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P35346
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01196
 
Compound ID Compound Name Compound Formula
CP0089773
N-[1-[[3,5-diethoxy-4-[4-(trifluoromethoxy)phenyl]phenyl]methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C30H34F3N3O4
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 2.4 nM
   TI
   LI
   LO
   TS
CP0093165
N-[1-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
   Show/Hide
C29H34FN3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 4.4 nM
   TI
   LI
   LO
   TS
CP0093166
6-chloro-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl)methyl)piperidin-4-yl)nicotinamide
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C28H31ClFN3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 7.9 nM
   TI
   LI
   LO
   TS
CP0093360
N-[1-[(3,5-diethoxy-4-fluorophenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C23H30FN3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 25 nM
   TI
   LI
   LO
   TS
CP0105230
6-amino-N-(1-((2-(benzyloxy)-6-ethoxy-4'-fluorobiphenyl-4-yl)methyl)piperidin-4-yl)nicotinamide
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C33H35FN4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 6.7 nM
   TI
   LI
   LO
   TS
CP0105231
N-[1-[(3,5-diethoxy-4-fluorophenyl)methyl]piperidin-4-yl]-6-(propan-2-ylamino)pyridine-3-carboxamide
   Show/Hide
C25H35FN4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 6.3 nM
   TI
   LI
   LO
   TS
CP0233778
N-[1-[(3,5-diethoxy-4-imidazol-1-ylphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C26H33N5O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 11 nM
   TI
   LI
   LO
   TS
CP0243209
N-[1-[(4-chloro-3,5-diethoxyphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C23H30ClN3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 4.4 nM
   TI
   LI
   LO
   TS
CP0285421
6-amino-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl)methyl)piperidin-4-yl)nicotinamide
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C28H33FN4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 7.1 nM
   TI
   LI
   LO
   TS
CP0285422
N-[1-[[3-ethoxy-4-(4-fluorophenyl)phenyl]methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C27H30FN3O2
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 4.9 nM
   TI
   LI
   LO
   TS
CP0287624
6-amino-N-[1-[(3-ethoxy-4,5-difluorophenyl)methyl]azepan-4-yl]pyridine-3-carboxamide
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C21H26F2N4O2
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 436 nM
   TI
   LI
   LO
   TS
CP0293088
N-[1-[(3,5-diethoxy-4-phenylphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
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C29H35N3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 5.4 nM
   TI
   LI
   LO
   TS
CP0294860
N-[1-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]azepan-4-yl]-5-methylpyridine-3-carboxamide
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C30H36FN3O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 9.3 nM
   TI
   LI
   LO
   TS
CP0294861
N-[1-[(3,5-diethoxy-4-phenylphenyl)methyl]piperidin-4-yl]-6-(methylamino)pyridine-3-carboxamide
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C29H36N4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 6.9 nM
   TI
   LI
   LO
   TS
CP0297376
6-amino-N-(1-(3-ethoxy-4-methylbenzyl)piperidin-4-yl)nicotinamide
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C21H28N4O2
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 19 nM
   TI
   LI
   LO
   TS
CP0357897
N-[1-[(3,5-diethoxy-4-fluorophenyl)methyl]piperidin-4-yl]-6-(methylamino)pyridine-3-carboxamide
   Show/Hide
C23H31FN4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 18 nM
   TI
   LI
   LO
   TS
CP0357900
N-[1-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]piperidin-4-yl]-6-(methylamino)pyridine-3-carboxamide
   Show/Hide
C29H35FN4O3
 2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 2.5 nM
   TI
   LI
   LO
   TS
CP0072332
1-[2-[[5-cyclopropyl-4-(4-fluorophenyl)-2-propan-2-yloxyphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C31H38FN3O4
 1
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
CP0207041
1-[2-[[5-cyclopropyl-2-ethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C30H36FN3O4
 1
1
IC50 = 2.6 nM
   TI
   LI
   LO
   TS
CP0517967
1-[2-[[5-cyclopropyl-4-(4-fluorophenyl)-2-methoxyphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C29H34FN3O4
 1
1
IC50 = 3.9 nM
   TI
   LI
   LO
   TS
CP0411749
1-[2-[[2-cyclopropyl-5-ethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C30H36FN3O4
 1
1
IC50 = 4.6 nM
   TI
   LI
   LO
   TS
CP0408223
1-[2-[[5-cyclopropyl-2-ethyl-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C30H36FN3O3
 1
1
IC50 = 5.1 nM
   TI
   LI
   LO
   TS
CP0116714
1-[2-[[3-cyclopropyl-5-ethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C30H36FN3O4
 1
1
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
CP0085871
1-[2-[[3-ethoxy-4-(4-fluorophenyl)-5-methylphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C28H34FN3O4
 1
1
IC50 = 6.1 nM
   TI
   LI
   LO
   TS
CP0493214
1-[2-[[3-ethoxy-5-ethyl-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C29H36FN3O4
 1
1
IC50 = 6.1 nM
   TI
   LI
   LO
   TS
CP0365008
1-[2-[[3-chloro-5-cyclopropyl-4-(4-fluorophenyl)-2-methoxyphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C29H33ClFN3O4
 1
1
IC50 = 6.2 nM
   TI
   LI
   LO
   TS
CP0079035
1-[2-[[5-cyclopropyl-2-ethoxy-4-(4-fluorophenyl)-3-methylphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C31H38FN3O4
 1
1
IC50 = 6.7 nM
   TI
   LI
   LO
   TS
CP0236074
1-[2-[[3-chloro-5-cyclopropyl-2-ethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C30H35ClFN3O4
 1
1
IC50 = 7.3 nM
   TI
   LI
   LO
   TS
CP0529623
4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C29H29FN2O5
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0274343
1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]piperidine-4-carboxylic acid
   Show/Hide
C28H34FN3O5
 1
1
IC50 = 9.6 nM
   TI
   LI
   LO
   TS
CP0460414
1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-ethylpiperidine-4-carboxylic acid
   Show/Hide
C30H38FN3O5
 1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0520082
1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C29H36FN3O5
 1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0323968
1-[2-[[3-ethoxy-4-(4-fluorophenyl)-5-methoxyphenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-methylpiperidine-4-carboxylic acid
   Show/Hide
C28H34FN3O5
 1
1
IC50 = 18 nM
   TI
   LI
   LO
   TS
CP0546703
CHEMBL4072189
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C29H35FN2O5
 1
1
IC50 = 30 nM
   TI
   LI
   LO
   TS
CP0465677
3-chloro-4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C29H28ClFN2O5
 1
1
IC50 = 46 nM
   TI
   LI
   LO
   TS
CP0472685
1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-4-fluoropiperidine-4-carboxylic acid
   Show/Hide
C28H33F2N3O5
 1
1
IC50 = 58 nM
   TI
   LI
   LO
   TS
CP0561817
6-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]pyridine-3-carboxylic acid
   Show/Hide
C28H28FN3O5
 1
1
IC50 = 61 nM
   TI
   LI
   LO
   TS
CP0073983
2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid
   Show/Hide
C24H28FN3O5
 2
1
IC50 = 72 nM
   TI
   LI
   LO
   TS
2
Ki = 18 nM
   TI
   LI
   LO
   TS
CP0478370
4-[2-[1-[3,5-diethoxy-4-(4-fluorophenyl)phenyl]ethyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C30H31FN2O5
 1
1
IC50 = 95 nM
   TI
   LI
   LO
   TS
CP0106411
2-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid
   Show/Hide
C22H24ClN3O4
 2
1
IC50 = 98 nM
   TI
   LI
   LO
   TS
2
Ki = 23 nM
   TI
   LI
   LO
   TS
CP0390087
4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]cyclohexane-1-carboxylic acid
   Show/Hide
C29H35FN2O5
 1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
CP0389778
4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]-3-methylbenzoic acid
   Show/Hide
C30H31FN2O5
 1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS
CP0410576
4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzamide
   Show/Hide
C29H30FN3O4
 1
1
IC50 = 150 nM
   TI
   LI
   LO
   TS
CP0389777
1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]pyrrolidine-3-carboxylic acid;hydrochloride
   Show/Hide
C27H33ClFN3O5
 1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS
CP0884345
1-(2-((2,6-Diethoxy-4'-fluorobiphenyl-4-yl)methyl)-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl)azetidine-3-carboxylic acid hydrochloride
   Show/Hide
C26H31ClFN3O5
 1
1
IC50 = 200 nM
   TI
   LI
   LO
   TS
CP0864095
(4-(2-((2,6-Diethoxy-4'-fluorobiphenyl-4-yl)methyl)-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl)phenyl)acetic acid hydrochloride
   Show/Hide
C30H32ClFN2O5
 1
1
IC50 = 220 nM
   TI
   LI
   LO
   TS
CP0072718
3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole
   Show/Hide
C27H23FN8O
 1
1
IC50 = 533 nM
   TI
   LI
   LO
   TS
CP0396535
3-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C29H29FN2O5
 1
1
IC50 = 550 nM
   TI
   LI
   LO
   TS
CP0135724
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H27N3O3
 2
1
IC50 = 740 nM
   TI
   LI
   LO
   TS
2
Ki = 121 nM
   TI
   LI
   LO
   TS
CP0483118
[4-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]phenyl]methanol
   Show/Hide
C29H31FN2O4
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0390090
2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-7-phenyl-5-oxa-2,6-diazaspiro[3.4]oct-6-ene
   Show/Hide
C28H29FN2O3
 1
1
IC50 = 2800 nM
   TI
   LI
   LO
   TS
CP0520914
3-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]propanoic acid
   Show/Hide
C25H29FN2O5
 1
1
IC50 = 3200 nM
   TI
   LI
   LO
   TS
CP0651917
5-((1R,3R)-1-(1-ethyl-1H-pyrazol-4-yl)-3-(4-(5-fluoropyridin-2-yl)-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one
   Show/Hide
C27H24FN9O2
 1
1
IC50 = 9240 nM
   TI
   LI
   LO
   TS
CP0237736
2-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridine-4-carboxylic acid
   Show/Hide
C30H24FN7O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0390088
4-[2-[3,5-diethoxy-4-(4-fluorophenyl)benzoyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C29H27FN2O6
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0495640
2-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]benzoic acid
   Show/Hide
C29H29FN2O5
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0076698
(1R,3R)-1-(oxan-4-yl)-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
   Show/Hide
C25H26N4O
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0049566
15-28-Somatostatin-28
   Show/Hide
C76H104N18O19S2
 1
1
Ki = 0.14 nM
   TI
   LI
   LO
   TS
CP0050675
(4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37-{2-[(2S)-2-[(2S)-6-amino-2-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2R)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-hydroxypropanamido]propanamido]-3-carbamoylpropanamido]-3-hydroxypropanamido]-3-carbamoylpropanoyl]pyrrolidin-2-yl]formamido}propanamido]-4-(methylsulfanyl)butanamido]propanoyl]pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamido]-4-carboxybutanamido]-5-carbamimidamidopentanamido]hexanamido]propanamido]a
   Show/Hide
C137H207N41O39S3
 1
1
Ki = 0.4 nM
   TI
   LI
   LO
   TS
CP0470520
(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S,34R,37S)-19,34-bis(4-aminobutyl)-31-(2-amino-2-oxoethyl)-37-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-13,25,28-tribenzyl-16-[(1S)-1-hydroxyethyl]-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacontane-4-carboxylic acid
   Show/Hide
C76H104N18O19S2
 1
1
Ki = 1.4 nM
   TI
   LI
   LO
   TS
CP0063692
2-(1-(4-chloro-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxylic acid
   Show/Hide
C24H28ClN3O5
 1
1
Ki = 3 nM
   TI
   LI
   LO
   TS
CP0142932
N-[1-[(3,5-diethoxy-4-methylphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
   Show/Hide
C24H33N3O3
 1
1
Ki = 4 nM
   TI
   LI
   LO
   TS
CP0858062
Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 5.98 nM
   TI
   LI
   LO
   TS
CP0269624
2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxamide
   Show/Hide
C24H29FN4O4
 1
1
Ki = 8 nM
   TI
   LI
   LO
   TS
CP0293090
N-[1-[[3-ethoxy-4-[4-(trifluoromethyl)phenyl]phenyl]methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
   Show/Hide
C28H30F3N3O2
 1
1
Ki = 11 nM
   TI
   LI
   LO
   TS
CP0073900
2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide
   Show/Hide
C23H31N5O5S
 1
1
Ki = 13 nM
   TI
   LI
   LO
   TS
CP0142929
N-[1-[(4-chloro-3-ethoxyphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
   Show/Hide
C21H26ClN3O2
 1
1
Ki = 15 nM
   TI
   LI
   LO
   TS
CP0553008
2-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide
   Show/Hide
C21H25ClN4O4S
 1
1
Ki = 17 nM
   TI
   LI
   LO
   TS
CP0105229
(R)-N-(1-(4-chloro-3-ethoxybenzyl)azepan-4-yl)-5-methylnicotinamide
   Show/Hide
C22H28ClN3O2
 1
1
Ki = 18 nM
   TI
   LI
   LO
   TS
CP0104467
N-[1-[(3-ethoxy-4-methylphenyl)methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
   Show/Hide
C22H29N3O2
 1
1
Ki = 21 nM
   TI
   LI
   LO
   TS
CP0229715
(R)-N-(1-(3-ethoxy-4-methylbenzyl)azepan-4-yl)-5-methylnicotinamide
   Show/Hide
C23H31N3O2
 1
1
Ki = 22 nM
   TI
   LI
   LO
   TS
CP0287622
(R)-N-(1-(3,5-diethoxy-4-fluorobenzyl)azepan-4-yl)-5-methylnicotinamide
   Show/Hide
C24H32FN3O3
 1
1
Ki = 22 nM
   TI
   LI
   LO
   TS
CP0281598
N-[1-[[4-methoxy-3-(2-methylpropoxy)phenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C24H31N3O3
 1
1
Ki = 23 nM
   TI
   LI
   LO
   TS
CP0136510
N-[1-[[3,5-di(propan-2-yloxy)phenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C25H33N3O3
 1
1
Ki = 31 nM
   TI
   LI
   LO
   TS
CP0063620
N-[1-[(4-amino-3,5-diethoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C23H30N4O3
 1
1
Ki = 33 nM
   TI
   LI
   LO
   TS
CP0063654
N-[1-[(3-ethoxy-4-methylphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H27N3O2
 1
1
Ki = 37 nM
   TI
   LI
   LO
   TS
CP0917823
NMeCpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 40.1 nM
   TI
   LI
   LO
   TS
CP0854677
Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-Nal-NH2
   Show/Hide
C59H69F3N12O9S2
 1
1
Ki = 45.5 nM
   TI
   LI
   LO
   TS
CP0208127
2-(1-(3,5-diethoxy-4-(1H-pyrrol-1-yl)benzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide
   Show/Hide
C29H37N5O5S
 1
1
Ki = 52 nM
   TI
   LI
   LO
   TS
CP0115766
N-[1-[[3-ethoxy-5-(oxan-4-yloxy)phenyl]methyl]piperidin-4-yl]-5-ethylsulfonyl-1,3-benzoxazol-2-amine
   Show/Hide
C28H37N3O6S
 1
1
Ki = 55 nM
   TI
   LI
   LO
   TS
CP0115593
4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenol
   Show/Hide
C21H25N3O3
 1
1
Ki = 66 nM
   TI
   LI
   LO
   TS
CP0136960
(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
   Show/Hide
C58H68ClN11O10S2
 1
1
Ki = 70.7 nM
   TI
   LI
   LO
   TS
CP0045800
N-[1-[(3-cyclopentyloxy-4-methoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C25H31N3O3
 1
1
Ki = 83 nM
   TI
   LI
   LO
   TS
CP0862999
Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 88.5 nM
   TI
   LI
   LO
   TS
CP0847584
Cpa-cyclo(DCys-Pal-NMeDTrp-Lys-Thr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 93 nM
   TI
   LI
   LO
   TS
CP0847417
Cpa-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
   Show/Hide
C56H68ClN13O9S2
 1
1
Ki = 101 nM
   TI
   LI
   LO
   TS
CP0886292
Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
   Show/Hide
C59H72N12O9S2
 1
1
Ki = 106 nM
   TI
   LI
   LO
   TS
CP0912534
Cpa-cyclo(DCys-Pal-NMeDTrp-NMeLys-Thr-Cys)-Nal-NH2
   Show/Hide
C59H71ClN12O9S2
 1
1
Ki = 112 nM
   TI
   LI
   LO
   TS
CP0063576
N-[1-[(4-chloro-3-ethoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C21H24ClN3O2
 1
1
Ki = 113 nM
   TI
   LI
   LO
   TS
CP0847340
Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-Nal-NH2
   Show/Hide
C57H67ClN12O9S2
 1
1
Ki = 140 nM
   TI
   LI
   LO
   TS
CP0489286
4-((4-(benzo[d]thiazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenol
   Show/Hide
C21H25N3O2S
 1
1
Ki = 149 nM
   TI
   LI
   LO
   TS
CP0106410
ethyl 4-[[4-(1,3-benzoxazol-2-ylamino)piperidin-1-yl]methyl]-2,6-diethoxybenzoate
   Show/Hide
C26H33N3O5
 1
1
Ki = 156 nM
   TI
   LI
   LO
   TS
CP0861120
Cpa-cyclo(DCys-Pal-DTrp-Lys-NMeThr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 161 nM
   TI
   LI
   LO
   TS
CP0045806
N-[2-[[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]amino]-1,3-benzoxazol-5-yl]-1-methylimidazole-4-sulfonamide
   Show/Hide
C26H32N6O5S
 1
1
Ki = 175 nM
   TI
   LI
   LO
   TS
CP0902700
Nal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
   Show/Hide
C60H71N13O9S2
 1
1
Ki = 176 nM
   TI
   LI
   LO
   TS
CP0115594
N-[1-[(3,5-diethoxy-4-fluorophenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C23H28FN3O3
 1
1
Ki = 178 nM
   TI
   LI
   LO
   TS
CP0074097
N-[2-[[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]amino]-1,3-benzoxazol-5-yl]cyclobutanecarboxamide
   Show/Hide
C27H34N4O4
 1
1
Ki = 182 nM
   TI
   LI
   LO
   TS
CP0106403
2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide
   Show/Hide
C22H28N4O5S
 2
1
Ki = 185 nM
   TI
   LI
   LO
   TS
2
Ki = 529 nM
   TI
   LI
   LO
   TS
CP0045791
N-[1-[(3-ethoxy-4-fluorophenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C21H24FN3O2
 1
1
Ki = 194 nM
   TI
   LI
   LO
   TS
CP0096309
5-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine
   Show/Hide
C22H26ClN3O3
 1
1
Ki = 194 nM
   TI
   LI
   LO
   TS
CP0063599
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-5-ethylsulfonyl-1,3-benzoxazol-2-amine
   Show/Hide
C24H31N3O5S
 1
1
Ki = 196 nM
   TI
   LI
   LO
   TS
CP0045803
N-[1-[[3-ethoxy-5-(oxan-4-yloxy)phenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C26H33N3O4
 1
1
Ki = 199 nM
   TI
   LI
   LO
   TS
CP0063569
N-[2-[[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]amino]-1,3-benzoxazol-5-yl]benzenesulfonamide
   Show/Hide
C28H32N4O5S
 1
1
Ki = 205 nM
   TI
   LI
   LO
   TS
CP0287134
2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide
   Show/Hide
C24H32N4O5S
 1
1
Ki = 226 nM
   TI
   LI
   LO
   TS
CP0063635
6-chloro-N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine
   Show/Hide
C21H23Cl2N3O2
 1
1
Ki = 239 nM
   TI
   LI
   LO
   TS
CP0045726
5-chloro-2-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide
   Show/Hide
C21H24ClFN4O4S
 1
1
Ki = 252 nM
   TI
   LI
   LO
   TS
CP0063602
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-5-nitro-1,3-benzoxazol-2-amine
   Show/Hide
C22H26N4O5
 1
1
Ki = 252 nM
   TI
   LI
   LO
   TS
CP0063633
5-chloro-2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide
   Show/Hide
C23H28ClFN4O5S
 1
1
Ki = 252 nM
   TI
   LI
   LO
   TS
CP0115657
N-[1-[(4-methoxy-3-propoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C23H29N3O3
 1
1
Ki = 293 nM
   TI
   LI
   LO
   TS
CP0096099
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-[1,3]thiazolo[5,4-b]pyridin-2-amine
   Show/Hide
C21H26N4O2S
 1
1
Ki = 309 nM
   TI
   LI
   LO
   TS
CP0880716
Pal-cyclo(DCys-Pal-DTrp-NMeLys-Thr-Cys)-DTrp-NH2
   Show/Hide
C55H68N14O9S2
 1
1
Ki = 313 nM
   TI
   LI
   LO
   TS
CP0371966
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-1,3-benzothiazol-2-amine
   Show/Hide
C22H27N3O2S
 1
1
Ki = 326 nM
   TI
   LI
   LO
   TS
CP0229734
N-[1-(3-ethoxy-4-methoxyphenyl)piperidin-4-yl]-1,3-benzothiazol-2-amine
   Show/Hide
C21H25N3O2S
 1
1
Ki = 330 nM
   TI
   LI
   LO
   TS
CP0063687
5-chloro-2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide
   Show/Hide
C22H27ClN4O5S
 1
1
Ki = 343 nM
   TI
   LI
   LO
   TS
CP0063685
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-5-(trifluoromethoxy)-1,3-benzoxazol-2-amine
   Show/Hide
C23H26F3N3O4
 1
1
Ki = 354 nM
   TI
   LI
   LO
   TS
CP0106805
N-[2-[[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]amino]-1,3-benzoxazol-5-yl]acetamide
   Show/Hide
C24H30N4O4
 1
1
Ki = 357 nM
   TI
   LI
   LO
   TS
CP0096067
6-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]thiazol-2-amine
   Show/Hide
C22H26ClN3O2S
 1
1
Ki = 361 nM
   TI
   LI
   LO
   TS
CP0063688
N-[1-[[3-(ethylamino)-4-methoxyphenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H28N4O2
 1
1
Ki = 371 nM
   TI
   LI
   LO
   TS
CP0063612
N-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C21H25N3O3
 1
1
Ki = 472 nM
   TI
   LI
   LO
   TS
CP0073981
N-[1-[[3-(2-fluoroethoxy)-4-methoxyphenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H26FN3O3
 1
1
Ki = 487 nM
   TI
   LI
   LO
   TS
CP0530284
N-[1-[[3-ethoxy-4-(trifluoromethoxy)phenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H24F3N3O3
 1
1
Ki = 524 nM
   TI
   LI
   LO
   TS
CP0063618
N-[1-[[3-ethoxy-4-(trifluoromethyl)phenyl]methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C22H24F3N3O2
 1
1
Ki = 524 nM
   TI
   LI
   LO
   TS
CP0115658
N-[1-[(4-cyclopropyloxy-3-ethoxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C24H29N3O3
 1
1
Ki = 537 nM
   TI
   LI
   LO
   TS
CP0096070
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-[1,3]oxazolo[5,4-b]pyridin-2-amine
   Show/Hide
C21H26N4O3
 1
1
Ki = 633 nM
   TI
   LI
   LO
   TS
CP0093361
(S)-N-(1-(4-chloro-3-ethoxybenzyl)azepan-4-yl)-5-methylnicotinamide
   Show/Hide
C22H28ClN3O2
 1
1
Ki = 637 nM
   TI
   LI
   LO
   TS
CP0371967
N-[1-[(1,4-dimethoxynaphthalen-2-yl)methyl]piperidin-4-yl]-1,3-benzothiazol-2-amine
   Show/Hide
C25H27N3O2S
 1
1
Ki = 683 nM
   TI
   LI
   LO
   TS
CP0487505
4-Chloro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
   Show/Hide
C26H22ClN5
 1
1
Ki = 691 nM
   TI
   LI
   LO
   TS
CP0060372
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-[1,3]oxazolo[5,4-c]pyridin-2-amine
   Show/Hide
C21H26N4O3
 1
1
Ki = 720 nM
   TI
   LI
   LO
   TS
CP0880603
Cpa-cyclo(NMeDCys-Pal-DTrp-Lys-Thr-Cys)-Dip-NHMe
   Show/Hide
C61H73ClN12O9S2
 1
1
Ki = 766 nM
   TI
   LI
   LO
   TS
CP0489292
N-[1-[(1,4-dimethoxynaphthalen-2-yl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C25H27N3O3
 1
1
Ki = 794 nM
   TI
   LI
   LO
   TS
CP0845116
Cpa-cyclo(DCys-Pal-DTrp-Dab-Thr-Cys)-Nal-NH2
   Show/Hide
C55H63ClN12O9S2
 1
1
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0847290
Cpa-cyclo(DCys-Pal-DTrp-DDap-Thr-Cys)-Nal-NH2
   Show/Hide
C54H61ClN12O9S2
 1
1
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0859471
Cpa-cyclo(DCys-Pal-DTrp-Lys-Thr-Cys)-NMeNal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0888162
Cpa-cyclo(DCys-NMePal-DTrp-Lys-Thr-Cys)-Nal-NH2
   Show/Hide
C58H69ClN12O9S2
 1
1
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0421312
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethoxy)benzenecarboximidamide
   Show/Hide
C27H22F3N5O
 1
1
Ki = 1130 nM
   TI
   LI
   LO
   TS
CP0415095
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]ethanimidamide
   Show/Hide
C21H21N5
 1
1
Ki = 1190 nM
   TI
   LI
   LO
   TS
CP0510832
1-(4-fluorobenzyl)-N-(1-((1,4-dimethoxynaphthalen-2-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
   Show/Hide
C32H33FN4O2
 1
1
Ki = 1230 nM
   TI
   LI
   LO
   TS
CP0372257
1-(4-fluorobenzyl)-N-(1-((7-methyl-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
   Show/Hide
C29H30FN5
 1
1
Ki = 1440 nM
   TI
   LI
   LO
   TS
CP0421355
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-methoxybenzenecarboximidamide
   Show/Hide
C27H25N5O
 1
1
Ki = 1620 nM
   TI
   LI
   LO
   TS
CP0371968
1-(4-fluorobenzyl)-N-(1-((2,3-dihydrobenzofuran-5-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
   Show/Hide
C28H29FN4O
 1
1
Ki = 1630 nM
   TI
   LI
   LO
   TS
CP0391029
N-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-1,3-benzothiazol-2-amine
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C21H25N3O2S
 1
1
Ki = 1789 nM
   TI
   LI
   LO
   TS
CP0377054
4-tert-Butyl-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
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C30H31N5
 1
1
Ki = 1870 nM
   TI
   LI
   LO
   TS
CP0404417
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-4-(trifluoromethyl)benzenecarboximidamide
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C27H22F3N5
 1
1
Ki = 2120 nM
   TI
   LI
   LO
   TS
CP0495082
2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-benzamidine
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C26H21F2N5
 1
1
Ki = 2250 nM
   TI
   LI
   LO
   TS
CP0392901
N'-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]benzenecarboximidamide
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C26H23N5
 1
1
Ki = 2360 nM
   TI
   LI
   LO
   TS
CP0395005
1-(2,4-Difluoro-phenyl)-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea
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C26H21F2N5O
 1
1
Ki = 3650 nM
   TI
   LI
   LO
   TS
CP0467228
1-(4-fluorobenzyl)-N-(1-(4-methoxybenzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C27H29FN4O
 1
1
Ki = 3950 nM
   TI
   LI
   LO
   TS
CP0504975
1-[(4-fluorophenyl)methyl]-N-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]benzimidazol-2-amine
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C28H28FN5
 1
1
Ki = 3950 nM
   TI
   LI
   LO
   TS
CP0040184
1-[(4-fluorophenyl)methyl]-N-{1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}-1H-1,3-benzodiazol-2-amine
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C28H31FN4O
 1
1
Ki = 4070 nM
   TI
   LI
   LO
   TS
CP0515175
1-(4-fluorobenzyl)-N-(1-phenethylpiperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C27H29FN4
 1
1
Ki = 5000 nM
   TI
   LI
   LO
   TS
CP0391030
4-((4-(benzo[d]thiazol-2-ylamino)piperidin-1-yl)methyl)-2-methoxyphenol
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C20H23N3O2S
 1
1
Ki = 5128 nM
   TI
   LI
   LO
   TS
CP0391032
1-(4-fluorobenzyl)-N-(1-benzylpiperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C26H27FN4
 1
1
Ki = 6120 nM
   TI
   LI
   LO
   TS
CP0376599
1-tert-Butyl-3-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-urea
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C24H27N5O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0382365
tert-butyl N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]carbamate
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C24H26N4O2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0430098
N-[(1R)-2-(1H-indol-3-yl)-1-(5-phenyl-1H-imidazol-2-yl)ethyl]-2-[3-(trifluoromethyl)phenyl]acetamide
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C28H23F3N4O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0427900
1-(4-fluorobenzyl)-N-(1-(3-phenylpropyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C28H31FN4
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0471388
1-(4-fluorobenzyl)-N-(1-((1,2,3,4-tetrahydronaphthalen-2-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C30H33FN4
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0523733
1-[(4-fluorophenyl)methyl]-N-[1-[2-[4-(trifluoromethoxy)phenyl]ethyl]piperidin-4-yl]benzimidazol-2-amine
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C28H28F4N4O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0553069
1-(4-fluorobenzyl)-N-(1-(4-fluorophenethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine
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C27H28F2N4
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0045798
N-(1,3-benzothiazol-2-yl)-4-(3-ethoxy-4-methoxyphenyl)piperazine-1-carboxamide
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C21H24N4O3S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0063595
N-(1,3-benzothiazol-2-yl)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidine-4-carboxamide
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C23H27N3O3S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0063597
4-N-(1,3-benzothiazol-2-yl)-1-N-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine
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C22H27N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0073866
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-1H-benzimidazol-2-amine
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C22H28N4O2
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0096064
1-(benzo[d]thiazol-2-yl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine
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C21H25N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0096098
1-(benzo[d]thiazol-2-ylmethyl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine
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C22H27N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0106405
N-[1-[(5-ethoxy-6-methoxypyridin-3-yl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
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C21H26N4O3
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0115595
2-(4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxy-5-fluorophenoxy)ethanol
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C23H28FN3O4
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0115653
N-[3-[(3-ethoxy-4-methoxyanilino)methyl]phenyl]-1,3-benzothiazol-2-amine
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C23H23N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0136504
1-N-(1,3-benzothiazol-2-ylmethyl)-4-N-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine
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C23H29N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0193949
N-[1-[(3-ethoxy-4-propan-2-yloxyphenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
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C24H31N3O3
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0194006
N-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-[1,3]oxazolo[4,5-b]pyridin-2-amine
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C21H26N4O3
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0225953
N-[1-[(3,5-diethoxy-2-fluorophenyl)methyl]piperidin-4-yl]-1,3-benzoxazol-2-amine
   Show/Hide
C23H28FN3O3
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0277635
N-[1-[(3,5-diethoxy-4-fluorophenyl)methyl]azetidin-3-yl]-5-methylpyridine-3-carboxamide
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C21H26FN3O3
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS