Brief Information of the Compound and Protein
Compound Name
N-[1-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]piperidin-4-yl]-5-methylpyridine-3-carboxamide
    Show/Hide
PubChem ID
CID: 46911015
SID: 99371994
Canonical SMILES
CCOc1cc(CN2CCC(CC2)NC(=O)c2cncc(C)c2)cc(OCC)c1-c1ccc(F)cc1
    Show/Hide
Compound Formula C29H34FN3O3
Compound Structure
Protein Name
Somatostatin receptor type 5
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Somatostatin receptor
Uniprot ID
P35346
Gene Name
SSTR5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 4.4 nM
   TI
   LI
   LO
   TS
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  2
1
IC50 = 1.3 nM
   TI
   LI
   LO
   TS
2
IC50 = 3.1 nM
   TI
   LI
   LO
   TS