| Compound ID |
Compound Name |
Compound Formula |
|
CP0010057
|
2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetic acid
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|
C19H16ClNO4
|
2
|
| 1 |
IC50 = 18 nM
|
|
|
| 2 |
IC50 = 39 nM
|
|
|
|
CP0511926
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-methoxyphenyl)-5-phenyl-1H-pyrazole
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|
C29H29FN2O4
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0061060
|
5-Bromo-2-(4-fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-thiophene
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|
C17H12BrFO2S2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0448740
|
6-(4-Methylsulfanyl-phenyl)-5-phenyl-imidazo[2,1-b]thiazole
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|
C18H14N2S2
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0460409
|
1-(4,4-Dimethyl-3-methylene-2-phenyl-cyclobut-1-enyl)-4-methanesulfonyl-benzene
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|
C20H20O2S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0049684
|
5-(4-Fluoro-phenyl)-6-(4-methanesulfonyl-phenyl)-spiro[2.4]hept-5-ene
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|
C20H19FO2S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0404461
|
5-(4-Methylsulfanyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole
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|
C18H14N2S2
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0377648
|
2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-4,4-dimethyl-cyclobut-2-enone
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|
C19H17FO3S
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0395145
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-spiro[3.4]oct-2-en-1-one
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|
C21H20O3S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0470554
|
1-Methanesulfonyl-4-(3-methylene-2-phenyl-cyclobut-1-enyl)-benzene
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|
C18H16O2S
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0428132
|
2-Isopropyl-5-(4-methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
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|
C20H19N3O2S2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0449755
|
5-(4-Methanesulfonyl-phenyl)-6-m-tolyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
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|
C19H14F3N3O2S2
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0401298
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
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|
C18H12F3N3O2S2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0405545
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-fluorophenyl)-5-phenyl-1H-pyrazole
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|
C28H26F2N2O3
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0475206
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1-(4-methylphenyl)-5-phenyl-1H-pyrazole
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|
C29H29FN2O3
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
|
CP0405546
|
1-(4-chlorophenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
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|
C28H26ClFN2O3
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0383216
|
2-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-3-phenyl-cyclobut-2-enone
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|
C19H18O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0475726
|
3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enone
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|
C19H18O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0441647
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-thiazolo[2,3-c][1,2,4]triazole
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|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0449758
|
2-Ethyl-5-(4-methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
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|
C19H17N3O2S2
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0489046
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-cyclobut-2-enone
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|
C17H14O3S
|
1
|
| 1 |
IC50 = 4400 nM
|
|
|
|
CP0420498
|
3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-1,5-diphenyl-1H-pyrazole
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|
C28H27FN2O3
|
1
|
| 1 |
IC50 = 7140 nM
|
|
|
|
CP0498180
|
6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
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|
C18H11F4N3O2S2
|
1
|
| 1 |
IC50 = 8500 nM
|
|
|
|
CP0405020
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-2-trifluoromethyl-thiazolo[3,2-b][1,2,4]triazole
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|
C18H12F3N3O2S2
|
1
|
| 1 |
IC50 = 9000 nM
|
|
|
|
CP0430344
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-2-vinyl-thiazolo[3,2-b][1,2,4]triazole
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|
C19H15N3O2S2
|
1
|
| 1 |
IC50 = 9600 nM
|
|
|
|
CP0011191
|
4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzene-1-sulfonamide
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|
C17H14F3N3O2S
|
1
|
| 1 |
IC50 = 13500 nM
|
|
|
|
CP0502197
|
6-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
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|
C17H12FN3O2S2
|
1
|
| 1 |
IC50 = 15000 nM
|
|
|
|
CP0427141
|
1-(4-methanesulfonylphenyl)-3-[(3,4-methylenedioxy)-phenoxymethyl]-5-phenyl-1H-pyrazole
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|
C24H20N2O5S
|
1
|
| 1 |
IC50 = 15810 nM
|
|
|
|
CP0437319
|
1-(4-methanesulfonylphenyl)-3-[(3,4,5-trimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
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|
C26H26N2O6S
|
1
|
| 1 |
IC50 = 17590 nM
|
|
|
|
CP0522693
|
1-(4-methanesulfonylphenyl)-3-[(3,5-dimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
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|
C25H24N2O5S
|
1
|
| 1 |
IC50 = 25050 nM
|
|
|
|
CP0420193
|
1-(4-aminosulfonylphenyl)-3-[3-fluoro-5-(4-methoxytetrahydropyran-4-yl)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C28H28FN3O5S
|
1
|
| 1 |
IC50 = 25700 nM
|
|
|
|
CP0096361
|
3-((3-fluoro-5-(1-methoxycyclohexyl)phenoxy)methyl)-1-(4-(methylsulfonyl)phenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C29H29FN2O5S
|
1
|
| 1 |
IC50 = 26080 nM
|
|
|
|
CP0437782
|
6-(3,4-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H11F2N3O2S2
|
1
|
| 1 |
IC50 = 30000 nM
|
|
|
|
CP0879971
|
3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enone oxime
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|
C19H19NO3S
|
1
|
| 1 |
IC50 = 34000 nM
|
|
|
|
CP0427142
|
1-(4-methanesulfonylphenyl)-3-[3-(4-morpholino)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C27H27N3O4S
|
1
|
| 1 |
IC50 = 38080 nM
|
|
|
|
CP0498156
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 = 43000 nM
|
|
|
|
CP0427145
|
3-[(3-fluoro-5-methoxy)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C24H21FN2O4S
|
1
|
| 1 |
IC50 = 44330 nM
|
|
|
|
CP0535156
|
3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl-cyclobut-2-enol
Show/Hide
|
C19H20O3S
|
1
|
| 1 |
IC50 = 45000 nM
|
|
|
|
CP0376557
|
6-(4-Methanesulfonyl-phenyl)-2,3-dimethyl-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C20H18N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0383382
|
2-Chloro-6-(4-chloro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H12Cl2N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0402232
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole-3-carboxylic acid
Show/Hide
|
C19H14N2O4S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0402569
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-3,5-dihydro-1lambda*4*-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0404472
|
5-(4-Methanesulfonyl-phenyl)-3-methyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0406295
|
5-(4-Methanesulfonyl-phenyl)-6-phenyl-imidazo[2,1-b]thiazole-3-carboxylic acid ethyl ester
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|
C21H18N2O4S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0409180
|
6-(4-Methanesulfonyl-phenyl)-2-methyl-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0410010
|
6-(4-Methanesulfonyl-phenyl)-3-methyl-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0437670
|
5-(4-Methanesulfonyl-phenyl)-2,3-dimethyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C20H18N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0467337
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C18H14N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0483637
|
2,3-Dichloro-6-(4-chloro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H11Cl3N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0492730
|
6-(3,4-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H12F2N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0494744
|
2-(4-Methanesulfonyl-phenyl)-3-phenyl-benzo[d]imidazo[2,1-b]thiazole
Show/Hide
|
C22H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0502348
|
6-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-imidazo[2,1-b]thiazole
Show/Hide
|
C18H13FN2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0524161
|
3-(4-Methanesulfonyl-phenyl)-2-phenyl-benzo[d]imidazo[2,1-b]thiazole
Show/Hide
|
C22H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0527628
|
5-(4-Methanesulfonyl-phenyl)-2-methyl-6-phenyl-imidazo[2,1-b]thiazole
Show/Hide
|
C19H16N2O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0376342
|
5-(4-Methanesulfonyl-phenyl)-6-(3-methoxy-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H15N3O3S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0419384
|
5-(4-Methanesulfonyl-phenyl)-2-methyl-6-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H15N3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0449756
|
6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2-methyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C18H14FN3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0449757
|
6-(3-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H12FN3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0459216
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0497173
|
6-(4-Methanesulfonyl-phenyl)-5-phenyl-thiazolo[2,3-c][1,2,4]triazole
Show/Hide
|
C17H13N3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0505496
|
6-(3,5-Difluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-thiazolo[3,2-b][1,2,4]triazole
Show/Hide
|
C17H11F2N3O2S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0379346
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-phenylsulfanyl-5H-furan-2-one
Show/Hide
|
C19H18O4S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0465037
|
4-(4-Methanesulfonyl-phenyl)-5,5-dimethyl-3-phenoxy-5H-furan-2-one
Show/Hide
|
C19H18O5S
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0505182
|
3-Benzoyl-4-(4-methanesulfonyl-phenyl)-5,5-dimethyl-5H-furan-2-one
Show/Hide
|
C20H18O5S
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0427144
|
3-[(5-cyano-3-fluoro)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C24H18FN3O3S
|
1
|
| 1 |
IC50 = 99560 nM
|
|
|
|
CP0341579
|
6-((3-fluoro-5-(4-methoxytetrahydro-2H-pyran-4-yl)phenoxy)methyl)-1-methylquinolin-2(1H)-one
Show/Hide
|
C23H24FNO4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0428151
|
1-(4-methanesulfonylphenyl)-3-[(3-nitro)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C23H19N3O5S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0437318
|
1-(4-methanesulfonylphenyl)-3-[(3,4-dimethoxy)phenoxymethyl]-5-phenyl-1H-pyrazole
Show/Hide
|
C25H24N2O5S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0511927
|
3-[(3-ethoxy)phenoxymethyl]-1-(4-methanesulfonylphenyl)-5-phenyl-1H-pyrazole
Show/Hide
|
C25H24N2O4S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
