Protein Information

General Information of the Protein

Protein ID	PT01838
Protein Name	Sphingosine 1-phosphate receptor 3
Secondarily Protein Name	Endothelial differentiation G-protein coupled receptor 3 Sphingosine 1-phosphate receptor Edg-3
Gene Name	S1PR3
Secondarily Gene Name	C9orf108 C9orf47 EDG3
Sequence	MATALPPRLQPVRGNETLREHYQYVGKLAGRLKEASEGSTLTTVLFLVICSFIVLENLMVLIAIWKNNKFHNRMYFFIGNLALCDLLAGIAYKVNILMSGKKTFSLSPTVWFLREGSMFVALGASTCSLLAIAIERHLTMIKMRPYDANKRHRVFLLIGMCWLIAFTLGALPILGWNCLHNLPDCSTILPLYSKKYIAFCISIFTAILVTIVILYARIYFLVKSSSRKVANHNNSERSMALLRTVVIVVSVFIACWSPLFILFLIDVACRVQACPILFKAQWFIVLAVLNSAMNPVIYTLASKEMRRAFFRLVCNCLVRGRGARASPIQPALDPSRSKSSSSNNSSHSPKVKEDLPHTAPSSCIMDKNAALQNGIFCN Show/Hide
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor > Family A G protein-coupled receptor > Small molecule receptor (family A GPCR) > Lipid-like ligand receptor (family A GPCR) > EDG receptor
Function	Receptor for the lysosphingolipid sphingosine 1-phosphate (S1P). S1P is a bioactive lysophospholipid that elicits diverse physiological effect on most types of cells and tissues. When expressed in rat HTC4 hepatoma cells, is capable of mediating S1P-induced cell proliferation and suppression of apoptosis. Show/Hide
Uniprot ID	Primary ID: Q99500 Secondarily ID: Q5SQD8 Q7Z5I2 Show/Hide
HGNC ID	HGNC:3167
Subcellular Location	Cell membrane

Map of Molecular Bioactivity Related to the Protein

Map of Molecular Bioactivity Related to the Protein Protein Cell Line Compound Bioactivity Value: <= 0.1 μM > 0.1 μM and <= 10 μM > 10 μM Imprecise Activity

Table of Molecular Bioactivities Related to the Protein

Cell Line ID: CL000011 , CHO

Cell Line Info

Compound ID	Compound Name	Compound Formula
CP0386360 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(3,5,5-triethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C30H41N3O5S	1
1	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0414585 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-[[methyl(2-methylpropyl)amino]methyl]-5-propan-2-ylphenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C31H44N4O5	1
1	EC50 = 1.4 nM Bioactivity Info	TI LI LO TS
CP0014534 Compound Info	(2S,3R,4E)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate Show/Hide	C18H38NO5P	3
1	EC50 = 1.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.04 nM Bioactivity Info	TI LI LO TS
3	IC50 = 0.26 nM Bioactivity Info	TI LI LO TS
CP0372160 Compound Info	[(2R)-2-amino-2-(hydroxymethyl)-4-(4-octylphenyl)butyl] dihydrogen phosphate Show/Hide	C19H34NO5P	2
1	EC50 = 1.7 nM Bioactivity Info	TI LI LO TS
2	EC50 = 2.5 nM Bioactivity Info	TI LI LO TS
CP0440020 Compound Info	N-[(2S)-3-[4-[5-(2-cyclopentyl-6-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O5	1
1	EC50 = 2.4 nM Bioactivity Info	TI LI LO TS
CP0420270 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-[[methyl(2-methylpropyl)amino]methyl]-5-propylphenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C31H44N4O5	1
1	EC50 = 3.5 nM Bioactivity Info	TI LI LO TS
CP0392887 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(2-ethyl-6-pentan-3-ylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 3.6 nM Bioactivity Info	TI LI LO TS
CP0899061 Compound Info	2-amino-4-(4-(3-(4-ethylphenyl)propyl)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C22H32NO5P	1
1	EC50 = 3.72 nM Bioactivity Info	TI LI LO TS
CP0490818 Compound Info	2-Amino-4-(4'-benzyloxy-2'-fluorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C24H27FNO6P	1
1	EC50 = 4.1 nM Bioactivity Info	TI LI LO TS
CP0452125 Compound Info	2-Amino-4-(2'-fluoro-4'-phenylthiobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C23H25FNO5PS	1
1	EC50 = 4.9 nM Bioactivity Info	TI LI LO TS
CP0505145 Compound Info	N-[(2S)-3-[4-[5-(2-cyclobutyl-6-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 5 nM Bioactivity Info	TI LI LO TS
CP0430641 Compound Info	(S)-2-amino-4-(4-(heptyloxy)phenyl)-2-methylbutyl dihydrogen phosphate Show/Hide	C18H32NO5P	1
1	EC50 = 5.4 nM Bioactivity Info	TI LI LO TS
CP0393043 Compound Info	3-[2-[2-ethyl-4-[5-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]ethylamino]propanoic acid Show/Hide	C28H37N3O4S	1
1	EC50 = 5.8 nM Bioactivity Info	TI LI LO TS
CP0395616 Compound Info	N-[3-[2,6-dimethyl-4-[5-[(2S,4R)-3,3,9-trimethyl-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-dien-7-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H31N3O5S	2
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
2	EC50 = 66 nM Bioactivity Info	TI LI LO TS
CP0554783 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[3-ethyl-5-[[methyl(2-methylpropyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C30H42N4O5	1
1	EC50 = 8 nM Bioactivity Info	TI LI LO TS
CP0435144 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H37N3O5S	1
1	EC50 = 8.9 nM Bioactivity Info	TI LI LO TS
CP0379596 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(3-ethylspiro[6,7-dihydro-4H-2-benzothiophene-5,1'-cyclopentane]-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C30H39N3O5S	1
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0379603 Compound Info	N-[(2S)-3-[4-[5-(5,5-dimethyl-3-propyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H39N3O5S	1
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0047332 Compound Info	[2-azaniumyl-2-(hydroxymethyl)-4-(4-octylphenyl)butyl] hydrogen phosphate Show/Hide	C19H34NO5P	4
1	EC50 = 12 nM Bioactivity Info	TI LI LO TS
2	EC50 = 35.1 nM Bioactivity Info	TI LI LO TS
3	EC50 = 44 nM Bioactivity Info	TI LI LO TS
4	IC50 = 6.3 nM Bioactivity Info	TI LI LO TS
CP0477265 Compound Info	2-Amino-4-(4'-benzyloxy-3-chlorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C24H27ClNO6P	1
1	EC50 = 13 nM Bioactivity Info	TI LI LO TS
CP0379610 Compound Info	N-[3-[2,6-dimethyl-4-[5-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H33N3O5S	1
1	EC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0443215 Compound Info	(2S)-3-[2-ethyl-4-[5-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-methylpropan-1-ol Show/Hide	C27H36N2O3S	1
1	EC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0419852 Compound Info	1-(4-(5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C24H18F3N3O3S	2
1	EC50 = 17 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0380075 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyl-6-methoxypyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 17 nM Bioactivity Info	TI LI LO TS
CP0472429 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-cyclohexyl-2-isopropyliminothiazolidin-4-one Show/Hide	C19H23ClN2O2S	1
1	EC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0876518 Compound Info	(S)-3-(2,6-Dimethyl-4-(3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)-1,2,4-oxadiazol-5-yl)phenoxy)-propane-1,2-diol Show/Hide	C24H28N2O4S	1
1	EC50 = 19.9 nM Bioactivity Info	TI LI LO TS
CP0568784 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[4-ethyl-5-[[methyl(propyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H38N4O5S	1
1	EC50 = 20 nM Bioactivity Info	TI LI LO TS
CP0909868 Compound Info	2-amino-2-(hydroxymethyl)-4-(4-(4-propylphenethyl)phenyl)butyl dihydrogen phosphate Show/Hide	C22H32NO5P	1
1	EC50 = 21 nM Bioactivity Info	TI LI LO TS
CP0469652 Compound Info	N-[(2S)-3-[4-[5-(2-cyclobutyl-6-methoxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H32N4O6	1
1	EC50 = 22 nM Bioactivity Info	TI LI LO TS
CP0386357 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(3-ethylspiro[6,7-dihydro-4H-2-benzothiophene-5,1'-cyclopropane]-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H35N3O5S	1
1	EC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0440017 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyl-5-ethylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O5	1
1	EC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0446792 Compound Info	N-[(2S)-3-[4-[5-(2-cyclobutyl-6-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H32N4O5	1
1	EC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0379604 Compound Info	N-[(2S)-3-[4-[3-(5,5-dimethyl-3-propyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-3-oxopropyl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C30H43NO5S	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0392959 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3,5,5-triethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C28H40O4S	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0392958 Compound Info	N-[(2S)-3-[4-[5-(2-cyclohexyl-6-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H38N4O5	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0445536 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyl-5-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0493876 Compound Info	3-[2-ethyl-4-[5-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]propanoic acid Show/Hide	C26H32N2O4S	1
1	EC50 = 26 nM Bioactivity Info	TI LI LO TS
CP0531251 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[2-methoxy-6-(2-methylpropyl)pyridin-4-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O6	1
1	EC50 = 27 nM Bioactivity Info	TI LI LO TS
CP0440022 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[5-ethyl-6-(2-methylpropyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 29 nM Bioactivity Info	TI LI LO TS
CP0446799 Compound Info	N-[(2S)-3-[4-[5-[6-(diethylamino)-5-ethylpyridin-3-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H37N5O5	1
1	EC50 = 30 nM Bioactivity Info	TI LI LO TS
CP0446796 Compound Info	US9617250, S-entiomer of Example 22 of D1 Show/Hide	C26H34N4O5	1
1	EC50 = 33 nM Bioactivity Info	TI LI LO TS
CP0372311 Compound Info	(Z,Z)-2-Isopropylimino-5-(3-methoxy-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O2S	1
1	EC50 = 35 nM Bioactivity Info	TI LI LO TS
CP0508754 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyloxy-6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 38 nM Bioactivity Info	TI LI LO TS
CP0895768 Compound Info	(S)-3-(2,6-Dimethyl-4-(5-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]-thiophen-1-yl)-1,2,4-oxadiazol-3-yl)phenoxy)-propane-1,2-diol Show/Hide	C24H28N2O4S	1
1	EC50 = 40.6 nM Bioactivity Info	TI LI LO TS
CP0459613 Compound Info	N-[(2S)-3-[4-[5-[5-[(dimethylamino)methyl]-4-ethylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H34N4O5S	1
1	EC50 = 45 nM Bioactivity Info	TI LI LO TS
CP0392888 Compound Info	BDBM50165434 Show/Hide	C27H36N4O5	1
1	EC50 = 46 nM Bioactivity Info	TI LI LO TS
CP0390242 Compound Info	US9617250, Example 233 of D1 Show/Hide	C27H34N4O5	1
1	EC50 = 47 nM Bioactivity Info	TI LI LO TS
CP0372314 Compound Info	(Z,Z)-5-(4-Hydroxy-3-methyl-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O2S	1
1	EC50 = 50 nM Bioactivity Info	TI LI LO TS
CP0401799 Compound Info	N-[(2S)-3-[4-[5-(2-cyclopentyloxy-6-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O6	1
1	EC50 = 50 nM Bioactivity Info	TI LI LO TS
CP0897100 Compound Info	2-Amino-4-(4'-butoxy-2'-fluorobiphenyl-4-yl)-2-(phosphoryloxymethy)butanol Show/Hide	C21H30F2NO6P	1
1	EC50 = 51 nM Bioactivity Info	TI LI LO TS
CP0372309 Compound Info	(Z,Z)-5-[4-(3-Hydroxy-propyl)-benzylidene]-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C22H24N2O2S	1
1	EC50 = 54 nM Bioactivity Info	TI LI LO TS
CP0420001 Compound Info	N-[(2S)-3-[4-[5-(2-cyclobutyloxy-6-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 55 nM Bioactivity Info	TI LI LO TS
CP0490776 Compound Info	(5Z)-2-butan-2-ylimino-5-[(3-chloro-4-hydroxyphenyl)methylidene]-3-phenyl-1,3-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0495817 Compound Info	(Z,Z)-5-[4-(2-Hydroxy-ethyl)-benzylidene]-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H22N2O2S	1
1	EC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0469848 Compound Info	3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimidine-4-carboxamido)-3-methylphenylsulfonamido)propanoic acid Show/Hide	C25H33N5O5S	1
1	EC50 = 62 nM Bioactivity Info	TI LI LO TS
CP0443219 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3-ethylspiro[6,7-dihydro-4H-2-benzothiophene-5,1'-cyclopentane]-1-yl)propan-1-one Show/Hide	C28H38O4S	1
1	EC50 = 62 nM Bioactivity Info	TI LI LO TS
CP0869582 Compound Info	(2RS)-3-(2,6-Dimethyl-4-(5-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)-1,3,4-oxadiazol-2-yl)phenoxy)propane-1,2-diol Show/Hide	C24H28N2O4S	1
1	EC50 = 65.3 nM Bioactivity Info	TI LI LO TS
CP0495815 Compound Info	(Z,Z)-5-[4-(3-Hydroxy-propoxy)-benzylidene]-2-isopropylimino-3-phenylthiazolidin-4-one Show/Hide	C22H24N2O3S	1
1	EC50 = 68 nM Bioactivity Info	TI LI LO TS
CP0508753 Compound Info	N-[(2S)-3-[4-[5-(2-cyclopentyl-6-methoxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 71 nM Bioactivity Info	TI LI LO TS
CP0570889 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyl-5-methoxypyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 71 nM Bioactivity Info	TI LI LO TS
CP0379595 Compound Info	N-[3-[4-[5-[3,5-dimethyl-4-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2,6-dimethylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H33N3O5S	1
1	EC50 = 74 nM Bioactivity Info	TI LI LO TS
CP0472432 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-propylimino-3-o-tolyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 81 nM Bioactivity Info	TI LI LO TS
CP0495852 Compound Info	2-Amino-4-[2'-fluoro-4'-(4-methylphenoxy)biphenyl-4-yl]-2-(phosphoryloxymethyl)butanol Show/Hide	C24H28NO6P	1
1	EC50 = 83 nM Bioactivity Info	TI LI LO TS
CP0379602 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(3-methoxy-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H35N3O6S	1
1	EC50 = 83 nM Bioactivity Info	TI LI LO TS
CP0401704 Compound Info	(Z,Z)-5-(4-Hydroxymethyl-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O2S	1
1	EC50 = 86 nM Bioactivity Info	TI LI LO TS
CP0407075 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-p-tolyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 88 nM Bioactivity Info	TI LI LO TS
CP0454281 Compound Info	(Z,Z)-5-(4-Hydroxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H18N2O2S	1
1	EC50 = 95 nM Bioactivity Info	TI LI LO TS
CP0390335 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-methyl-6-propan-2-yloxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O6	1
1	EC50 = 95 nM Bioactivity Info	TI LI LO TS
CP0495814 Compound Info	(Z,Z)-2-tert-Butylimino-5-(3-chloro-4-hydroxy-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0531252 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(2-methoxy-6-pentan-3-ylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O6	1
1	EC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0373469 Compound Info	(Z,Z)-5-(3-Fluoro-4-hydroxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H17FN2O2S	1
1	EC50 = 99 nM Bioactivity Info	TI LI LO TS
CP0420267 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[3-ethyl-4-[[ethyl(methyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0434662 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-5-[[methyl(2-methylpropyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0374262 Compound Info	(Z,Z)-5-(3-Hydroxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H18N2O2S	1
1	EC50 = 103 nM Bioactivity Info	TI LI LO TS
CP0253199 Compound Info	N,N-dicyclohexyl-5-phenyl-1,2-oxazole-3-carboxamide Show/Hide	C22H28N2O2	1
1	EC50 = 103 nM Bioactivity Info	TI LI LO TS
CP0106181 Compound Info	N,N-dicyclohexyl-5-cyclopropyl-1,2-oxazole-3-carboxamide Show/Hide	C19H28N2O2	1
1	EC50 = 105 nM Bioactivity Info	TI LI LO TS
CP0495820 Compound Info	(Z,Z)-2-Isopropylimino-5-(4-methoxy-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O2S	1
1	EC50 = 106 nM Bioactivity Info	TI LI LO TS
CP0466516 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyl-4-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 106 nM Bioactivity Info	TI LI LO TS
CP0438157 Compound Info	(Z,Z)-5-[3-Chloro-4-((2S)-2,3-dihydroxy-propoxy)-benzylidene]-2-propylimino-3-otolyl-thiazolidin-4-one Show/Hide	C23H25ClN2O4S	1
1	EC50 = 109 nM Bioactivity Info	TI LI LO TS
CP0372367 Compound Info	3-(3-methyl-4-{5-[4-(propan-2-yloxy)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl}phenyl)propanoic acid Show/Hide	C22H21F3N2O4	1
1	EC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0880198 Compound Info	(2RS)-3-(2,6-Dimethyl-4-(2-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)oxazol-5-yl)phenoxy)propane-1,2-diol Show/Hide	C25H29NO4S	1
1	EC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0534605 Compound Info	N-[(2S)-3-[4-[5-(2-cyclobutyloxy-6-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H32N4O6	1
1	EC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0854263 Compound Info	2-amino-4-(4-(4-(2-ethyl-1H-imidazol-4-yl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C22H28N3O6P	1
1	EC50 = 113 nM Bioactivity Info	TI LI LO TS
CP0372305 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-cyclopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H15ClN2O2S	1
1	EC50 = 114 nM Bioactivity Info	TI LI LO TS
CP0372307 Compound Info	(Z,Z)-5-[4-(3-Dimethylamino-propoxy)-benzylidene]-2-isopropylimino-3-phenylthiazolidin-4-one Show/Hide	C24H29N3O2S	1
1	EC50 = 114 nM Bioactivity Info	TI LI LO TS
CP0495813 Compound Info	(Z,Z)-5-[4-(2-Hydroxy-ethoxy)-benzylidene]-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H22N2O3S	1
1	EC50 = 114 nM Bioactivity Info	TI LI LO TS
CP0372316 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-hexyl-2-isopropylimino-thiazolidin-4-one Show/Hide	C19H25ClN2O2S	1
1	EC50 = 118 nM Bioactivity Info	TI LI LO TS
CP0454283 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H17ClN2O2S	1
1	EC50 = 120 nM Bioactivity Info	TI LI LO TS
CP0414582 Compound Info	N-[(2S)-3-[4-[5-[5-[[butyl(methyl)amino]methyl]-4-methylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H38N4O5S	1
1	EC50 = 120 nM Bioactivity Info	TI LI LO TS
CP0559242 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-5-[[methyl(propyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H36N4O5S	1
1	EC50 = 120 nM Bioactivity Info	TI LI LO TS
CP0392960 Compound Info	N-[3-[2-ethyl-6-methyl-4-[5-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H35N3O5S	1
1	EC50 = 122 nM Bioactivity Info	TI LI LO TS
CP0906035 Compound Info	(1R,2R)-2-(4-(5-(4-isopropoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)cyclopropanecarboxylic acid Show/Hide	C23H21F3N2O4	1
1	EC50 = 123 nM Bioactivity Info	TI LI LO TS
CP0372514 Compound Info	(Z,Z)-5-[3-Chloro-4-((2R)-2,3-dihydroxy-propoxy)-benzylidene]-2-propylimino-3-o-tolyl-thiazolidin-4-one Show/Hide	C23H25ClN2O4S	1
1	EC50 = 123 nM Bioactivity Info	TI LI LO TS
CP0490773 Compound Info	(Z,Z)-5-[3-Chloro-4-(2-hydroxy-ethoxy)-benzylidene]-2-propylimino-3-o-tolylthiazolidin-4-one Show/Hide	C22H23ClN2O3S	1
1	EC50 = 124 nM Bioactivity Info	TI LI LO TS
CP0514180 Compound Info	(Z,Z)-3-[5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-4-oxo-thiazolidin-3-yl]-propionicacidethylester Show/Hide	C18H21ClN2O4S	1
1	EC50 = 125 nM Bioactivity Info	TI LI LO TS
CP0446797 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-6-(2-methylpropyl)pyridin-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 125 nM Bioactivity Info	TI LI LO TS
CP0379600 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C26H36O4S	1
1	EC50 = 126 nM Bioactivity Info	TI LI LO TS
CP0373470 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-(4-methoxy-phenyl)-thiazolidin-4-one Show/Hide	C20H19ClN2O3S	1
1	EC50 = 127 nM Bioactivity Info	TI LI LO TS
CP0372155 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-cyclobutylimino-3-phenyl-thiazolidin-4-one Show/Hide	C20H17ClN2O2S	1
1	EC50 = 128 nM Bioactivity Info	TI LI LO TS
CP0407073 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(3-chloro-phenyl)-2-isopropyliminothiazolidin-4-one Show/Hide	C19H16Cl2N2O2S	1
1	EC50 = 129 nM Bioactivity Info	TI LI LO TS
CP0851079 Compound Info	2-amino-4-(4-(4-ethylphenethyl)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H30NO5P	1
1	EC50 = 130 nM Bioactivity Info	TI LI LO TS
CP0514580 Compound Info	(Z,Z)-5-(4-Bromo-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H17BrN2OS	1
1	EC50 = 136 nM Bioactivity Info	TI LI LO TS
CP0372294 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-o-tolyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 139 nM Bioactivity Info	TI LI LO TS
CP0541599 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[6-methyl-4-(2-methylpropyl)pyridin-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 139 nM Bioactivity Info	TI LI LO TS
CP0372306 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-(dimethyl-hydrazono)-3-phenylthiazolidin-4-one Show/Hide	C18H16ClN3O2S	1
1	EC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0474138 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyloxy-5-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0403889 Compound Info	N-[3-[2-ethyl-4-[3-(3-ethyl-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-3-oxopropyl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H41NO5S	1
1	EC50 = 141 nM Bioactivity Info	TI LI LO TS
CP0504085 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(3-chloro-4-methyl-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C20H18Cl2N2O2S	1
1	EC50 = 144 nM Bioactivity Info	TI LI LO TS
CP0177664 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-5-[[methyl(2-methylpropyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H38N4O5S	1
1	EC50 = 145 nM Bioactivity Info	TI LI LO TS
CP0446791 Compound Info	N-[(2S)-3-[4-[5-(2-cyclohexyl-6-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O5	1
1	EC50 = 149 nM Bioactivity Info	TI LI LO TS
CP0420274 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[5-[[ethyl(methyl)amino]methyl]-4-methylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H34N4O5S	1
1	EC50 = 150 nM Bioactivity Info	TI LI LO TS
CP0390201 Compound Info	(S)-3-amino-5-(4-(heptyloxy)phenyl)-3-methylpentylphosphonic acid Show/Hide	C19H34NO4P	1
1	EC50 = 151 nM Bioactivity Info	TI LI LO TS
CP0445535 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-5-(2-methylpropyl)pyridin-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 154 nM Bioactivity Info	TI LI LO TS
CP0390634 Compound Info	3-(4-(5-(5-chloro-6-(1,1,1-trifluoropropan-2-yloxy)pyridin-3-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C20H17ClF3N3O4	1
1	EC50 = 160 nM Bioactivity Info	TI LI LO TS
CP0394082 Compound Info	3-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C24H26N2O3	1
1	EC50 = 160 nM Bioactivity Info	TI LI LO TS
CP0388697 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-isopropyl-2-isopropylimino-thiazolidin-4-one Show/Hide	C16H19ClN2O2S	1
1	EC50 = 162 nM Bioactivity Info	TI LI LO TS
CP0372312 Compound Info	(Z,Z)-5-(4-Dimethylamino-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H23N3OS	1
1	EC50 = 165 nM Bioactivity Info	TI LI LO TS
CP0379598 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(3-ethyl-4,5,6,7-tetrahydro-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H33N3O5S	1
1	EC50 = 172 nM Bioactivity Info	TI LI LO TS
CP0403890 Compound Info	N-[3-[4-[5-[3-ethyl-5-methyl-4-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2,6-dimethylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N3O5S	1
1	EC50 = 172 nM Bioactivity Info	TI LI LO TS
CP0915931 Compound Info	rac-(Z,Z)-5-[3-Chloro-4-(2,3-dihydroxy-propoxy)-benzylidene]-2-propylimino-3-otolyl-thiazolidin-4-one Show/Hide	C23H25ClN2O4S	1
1	EC50 = 174 nM Bioactivity Info	TI LI LO TS
CP0440021 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(5-ethyl-6-pyrrolidin-1-ylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H35N5O5	1
1	EC50 = 176 nM Bioactivity Info	TI LI LO TS
CP0474136 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(6-methoxy-4-pentan-3-ylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O6	1
1	EC50 = 180 nM Bioactivity Info	TI LI LO TS
CP0372150 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-phenethylthiazolidin-4-one Show/Hide	C21H21ClN2O2S	1
1	EC50 = 183 nM Bioactivity Info	TI LI LO TS
CP0409183 Compound Info	3-(3-methyl-4-{5-[4-(propan-2-yloxy)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl}phenyl)butanoic acid Show/Hide	C23H23F3N2O4	1
1	EC50 = 184 nM Bioactivity Info	TI LI LO TS
CP0909865 Compound Info	2-amino-2-(hydroxymethyl)-4-(4-(4-(4-isopropylphenyl)butyl)phenyl)butyl dihydrogen phosphate Show/Hide	C24H36NO5P	1
1	EC50 = 184 nM Bioactivity Info	TI LI LO TS
CP0372157 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-phenyl-2-propylimino-thiazolidin-4-one Show/Hide	C19H17ClN2O2S	1
1	EC50 = 189 nM Bioactivity Info	TI LI LO TS
CP0508775 Compound Info	N-[(2S)-3-[4-[5-(2-cyclopentyloxy-6-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 190 nM Bioactivity Info	TI LI LO TS
CP0372130 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-m-tolyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 200 nM Bioactivity Info	TI LI LO TS
CP0875386 Compound Info	2-((3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)propyl)amino)-acetic acid Show/Hide	C27H35NO4S	1
1	EC50 = 201 nM Bioactivity Info	TI LI LO TS
CP0210525 Compound Info	5-cyclopropyl-N,N-bis(2-methylcyclohexyl)-1,2-oxazole-3-carboxamide Show/Hide	C21H32N2O2	1
1	EC50 = 202 nM Bioactivity Info	TI LI LO TS
CP0906687 Compound Info	2-amino-4-(4-(4-butylphenoxy)-2-fluorophenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H29FNO6P	1
1	EC50 = 204 nM Bioactivity Info	TI LI LO TS
CP0414583 Compound Info	N-[(2S)-3-[4-[5-[4-(diethylaminomethyl)-3-ethylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 210 nM Bioactivity Info	TI LI LO TS
CP0534606 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyl-4-methoxypyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 210 nM Bioactivity Info	TI LI LO TS
CP0373472 Compound Info	(Z,Z)-5-(3-Hydroxy-4-methoxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O3S	1
1	EC50 = 212 nM Bioactivity Info	TI LI LO TS
CP0522088 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-(4-phenyl-butyl)-thiazolidin-4-one Show/Hide	C23H25ClN2O2S	1
1	EC50 = 212 nM Bioactivity Info	TI LI LO TS
CP0848818 Compound Info	2-amino-2-(hydroxymethyl)-4-(4-(4-(4-methylbenzyl)phenoxy)phenyl)butyl dihydrogen phosphate Show/Hide	C25H30NO6P	1
1	EC50 = 225 nM Bioactivity Info	TI LI LO TS
CP0372129 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-pyridin-3-ylthiazolidin-4-one Show/Hide	C18H16ClN3O2S	1
1	EC50 = 228 nM Bioactivity Info	TI LI LO TS
CP0467328 Compound Info	3-(4-(5-(3-bromo-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H21BrN2O4	1
1	EC50 = 230 nM Bioactivity Info	TI LI LO TS
CP0496093 Compound Info	1-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimidine-4-carboxamido)-3-methylbenzyl)azetidine-3-carboxylic acid Show/Hide	C27H35N5O3	1
1	EC50 = 236 nM Bioactivity Info	TI LI LO TS
CP0379609 Compound Info	N-[3-[2,6-dimethyl-4-[5-[5-methyl-4-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H31N3O5S	1
1	EC50 = 236 nM Bioactivity Info	TI LI LO TS
CP0456032 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-(4-propan-2-ylphenyl)-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C23H29N2O6P	1
1	EC50 = 237 nM Bioactivity Info	TI LI LO TS
CP0411203 Compound Info	(5Z)-5-[[4-(2,3-dihydroxypropoxy)phenyl]methylidene]-3-phenyl-2-propan-2-ylimino-1,3-thiazolidin-4-one Show/Hide	C22H24N2O4S	1
1	EC50 = 240 nM Bioactivity Info	TI LI LO TS
CP0404698 Compound Info	N-[3-[4-[3-[5,5-dimethyl-3-(trifluoromethyl)-6,7-dihydro-4H-2-benzothiophen-1-yl]-3-oxopropyl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36F3NO5S	1
1	EC50 = 242 nM Bioactivity Info	TI LI LO TS
CP0414338 Compound Info	[2-amino-4-[4-[2-(4-fluorophenyl)-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C20H22FN2O6P	1
1	EC50 = 245 nM Bioactivity Info	TI LI LO TS
CP0514181 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(3-chloro-2-methyl-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C20H18Cl2N2O2S	1
1	EC50 = 246 nM Bioactivity Info	TI LI LO TS
CP0481261 Compound Info	N-[3-[2,6-dimethyl-4-[5-[5-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H29N3O5S	1
1	EC50 = 247 nM Bioactivity Info	TI LI LO TS
CP0433972 Compound Info	N-[(2S)-3-[4-[5-(4-cyclopentyl-6-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 258 nM Bioactivity Info	TI LI LO TS
CP0374261 Compound Info	(Z,Z)-2-Butylimino-5-(3-chloro-4-hydroxy-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 264 nM Bioactivity Info	TI LI LO TS
CP0375772 Compound Info	(S)-3-amino-5-(4-(heptyloxy)phenyl)-3-methylpentanoic acid Show/Hide	C19H31NO3	1
1	EC50 = 300 nM Bioactivity Info	TI LI LO TS
CP0372153 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-cyclopentylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H19ClN2O2S	1
1	EC50 = 302 nM Bioactivity Info	TI LI LO TS
CP0869940 Compound Info	2-amino-4-(4-(4-butylphenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H30NO6P	1
1	EC50 = 302 nM Bioactivity Info	TI LI LO TS
CP0411204 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2,6-dimethyl-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C21H21ClN2O2S	1
1	EC50 = 307 nM Bioactivity Info	TI LI LO TS
CP0392956 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-methyl-6-pyrrolidin-1-ylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H33N5O5	1
1	EC50 = 307 nM Bioactivity Info	TI LI LO TS
CP0372145 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-cyclohexylimino-3-phenyl-thiazolidin-4-one Show/Hide	C22H21ClN2O2S	1
1	EC50 = 310 nM Bioactivity Info	TI LI LO TS
CP0392961 Compound Info	US9617250, Example 101 of D1 Show/Hide	C25H32N4O5	1
1	EC50 = 310 nM Bioactivity Info	TI LI LO TS
CP0379607 Compound Info	N-[3-[4-[5-(5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H33N3O5S	1
1	EC50 = 314 nM Bioactivity Info	TI LI LO TS
CP0374263 Compound Info	(Z,Z)-5-Benzylidene-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H18N2OS	1
1	EC50 = 317 nM Bioactivity Info	TI LI LO TS
CP0390240 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[5-methyl-6-(2-methylpropyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 318 nM Bioactivity Info	TI LI LO TS
CP0440024 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[5-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H31N3O5S	1
1	EC50 = 320 nM Bioactivity Info	TI LI LO TS
CP0262673 Compound Info	N,N-dicyclohexyl-5-(4-methoxyphenyl)-1,2-oxazole-3-carboxamide Show/Hide	C23H30N2O3	1
1	EC50 = 323 nM Bioactivity Info	TI LI LO TS
CP0374219 Compound Info	(Z,Z)-5-(4-Hydroxy-3-methoxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O3S	1
1	EC50 = 335 nM Bioactivity Info	TI LI LO TS
CP0407074 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2-ethyl-phenyl)-2-isopropyliminothiazolidin-4-one Show/Hide	C21H21ClN2O2S	1
1	EC50 = 335 nM Bioactivity Info	TI LI LO TS
CP0110354 Compound Info	N-cyclohexyl-5-cyclopropyl-N-(2-methylcyclohexyl)-1,2-oxazole-3-carboxamide Show/Hide	C20H30N2O2	1
1	EC50 = 337 nM Bioactivity Info	TI LI LO TS
CP0334414 Compound Info	N,N-dicyclohexyl-5-cyclopentyl-1,2-oxazole-3-carboxamide Show/Hide	C21H32N2O2	1
1	EC50 = 339 nM Bioactivity Info	TI LI LO TS
CP0421315 Compound Info	3-(4-(5-(3-cyano-4-(1,1,1,3,3,3-hexafluoropropan-2-yloxy)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C22H15F6N3O4	1
1	EC50 = 340 nM Bioactivity Info	TI LI LO TS
CP0874453 Compound Info	(2R/S)-2-((3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)propyl)amino)-succinic acid Show/Hide	C29H37NO6S	1
1	EC50 = 348 nM Bioactivity Info	TI LI LO TS
CP0854261 Compound Info	2-amino-4-(2-chloro-4-(4-(2-ethyloxazol-4-yl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C22H26ClN2O7P	1
1	EC50 = 349 nM Bioactivity Info	TI LI LO TS
CP0374220 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2,3-dimethyl-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C21H21ClN2O2S	1
1	EC50 = 350 nM Bioactivity Info	TI LI LO TS
CP0420042 Compound Info	N-[(2S)-3-[4-[5-[4-[[butyl(methyl)amino]methyl]-3-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 350 nM Bioactivity Info	TI LI LO TS
CP0399288 Compound Info	N-[(2S)-3-[4-[5-[2-(diethylamino)-6-methylpyridin-4-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	2
1	EC50 = 350 nM Bioactivity Info	TI LI LO TS
2	EC50 = 352 nM Bioactivity Info	TI LI LO TS
CP0396855 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H22F3N2O6P	1
1	EC50 = 356 nM Bioactivity Info	TI LI LO TS
CP0474123 Compound Info	N-[(2S)-3-[4-[5-[3,4-dimethyl-5-[[methyl(propyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H38N4O5S	1
1	EC50 = 370 nM Bioactivity Info	TI LI LO TS
CP0474142 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-5-[[methyl(propyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 380 nM Bioactivity Info	TI LI LO TS
CP0848817 Compound Info	4-(4-([1,1'-biphenyl]-4-yloxy)phenyl)-2-amino-2-(hydroxymethyl)butyldihydrogen phosphate Show/Hide	C23H26NO6P	1
1	EC50 = 383 nM Bioactivity Info	TI LI LO TS
CP0851078 Compound Info	2-amino-4-(4-(4-benzylphenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C24H28NO6P	1
1	EC50 = 391 nM Bioactivity Info	TI LI LO TS
CP0415715 Compound Info	N-[3-[2,6-dimethyl-4-[3-oxo-3-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propyl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H37NO5S	1
1	EC50 = 392 nM Bioactivity Info	TI LI LO TS
CP0463957 Compound Info	2-methyl-3-(3-methyl-4-{5-[4-(propan-2-yloxy)-3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-3-yl}phenyl)propanoic acid Show/Hide	C23H23F3N2O4	1
1	EC50 = 400 nM Bioactivity Info	TI LI LO TS
CP0869520 Compound Info	3-(4-(2-Aminoethoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C24H31NO2S	1
1	EC50 = 407 nM Bioactivity Info	TI LI LO TS
CP0415286 Compound Info	6-((cyclopropylmethyl)(propyl)amino)-N-(1H-indazol-5-yl)pyrimidine-4-carboxamide Show/Hide	C19H22N6O	1
1	EC50 = 416 nM Bioactivity Info	TI LI LO TS
CP0456028 Compound Info	[2-amino-4-[4-[2-(4-ethylphenyl)-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C22H27N2O6P	1
1	EC50 = 416 nM Bioactivity Info	TI LI LO TS
CP0504086 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2-chloro-phenyl)-2-isopropyliminothiazolidin-4-one Show/Hide	C19H16Cl2N2O2S	1
1	EC50 = 425 nM Bioactivity Info	TI LI LO TS
CP0414586 Compound Info	N-[(2S)-3-[4-[5-[3-[[butyl(methyl)amino]methyl]-5-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 425 nM Bioactivity Info	TI LI LO TS
CP0407072 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-(2-methoxy-phenyl)-thiazolidin-4-one Show/Hide	C20H19ClN2O3S	1
1	EC50 = 428 nM Bioactivity Info	TI LI LO TS
CP0446801 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(5-methyl-6-propan-2-ylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 = 429 nM Bioactivity Info	TI LI LO TS
CP0466509 Compound Info	N-[(2S)-3-[4-[5-[6-(diethylamino)-4-methylpyridin-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	1
1	EC50 = 429 nM Bioactivity Info	TI LI LO TS
CP0393042 Compound Info	N-[3-[2,6-dimethyl-4-[3-oxo-3-[(2S,4R)-3,3,9-trimethyl-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-dien-7-yl]propyl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H35NO5S	2
1	EC50 = 430 nM Bioactivity Info	TI LI LO TS
2	EC50 = 437 nM Bioactivity Info	TI LI LO TS
CP0106190 Compound Info	MLS000116372 Show/Hide	C19H30N2O2	1
1	EC50 = 434 nM Bioactivity Info	TI LI LO TS
CP0490775 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2,4-dimethyl-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C21H21ClN2O2S	1
1	EC50 = 458 nM Bioactivity Info	TI LI LO TS
CP0381848 Compound Info	3-(4-(5-(4-ethoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H19F3N2O4	1
1	EC50 = 460 nM Bioactivity Info	TI LI LO TS
CP0390653 Compound Info	3-(4-(5-(4-isopropoxy-3-methylphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C22H24N2O4	1
1	EC50 = 460 nM Bioactivity Info	TI LI LO TS
CP0394075 Compound Info	3-(4-(5-(4-(S)-sec-butoxy-3-cyanophenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C23H23N3O4	1
1	EC50 = 470 nM Bioactivity Info	TI LI LO TS
CP0408502 Compound Info	3-(4-(5-(5-(1,1-difluoro-2-methylpropyl)pyridin-2-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H21F2N3O3	1
1	EC50 = 470 nM Bioactivity Info	TI LI LO TS
CP0427573 Compound Info	1-(4-(5-benzylthiazolo[5,4-b]pyridin-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 = 478 nM Bioactivity Info	TI LI LO TS
CP0414584 Compound Info	N-[(2S)-3-[4-[5-[4-[(dimethylamino)methyl]-3-ethylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 480 nM Bioactivity Info	TI LI LO TS
CP0409138 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[4-(2-propyl-1,3-oxazol-4-yl)phenyl]phenyl]butyl] dihydrogen phosphate;hydrochloride Show/Hide	C23H30ClN2O6P	1
1	EC50 = 484 nM Bioactivity Info	TI LI LO TS
CP0880199 Compound Info	3-(4-((R)-2,3-Dihydroxypropoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H32O4S	1
1	EC50 = 489 nM Bioactivity Info	TI LI LO TS
CP0545730 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-(4-propan-2-ylphenyl)triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C22H29N4O5P	1
1	EC50 = 496 nM Bioactivity Info	TI LI LO TS
CP0381832 Compound Info	3-(4-(5-(3-cyano-4-(1,1,1-trifluoropropan-2-yloxy)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C22H18F3N3O4	1
1	EC50 = 500 nM Bioactivity Info	TI LI LO TS
CP0869942 Compound Info	2-amino-4-(2-hexylchroman-6-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C20H34NO6P	1
1	EC50 = 508 nM Bioactivity Info	TI LI LO TS
CP0472428 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-3-(3-methoxy-phenyl)-thiazolidin-4-one Show/Hide	C20H19ClN2O3S	1
1	EC50 = 514 nM Bioactivity Info	TI LI LO TS
CP0549747 Compound Info	N-[(2R)-3-[2-ethyl-6-methyl-4-[5-[5-methyl-6-(2-methylpropyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 519 nM Bioactivity Info	TI LI LO TS
CP0469651 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(4-methoxy-6-pentan-3-ylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O6	1
1	EC50 = 520 nM Bioactivity Info	TI LI LO TS
CP0454282 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-3-(2,4-dimethoxy-phenyl)-2-isopropylimino-thiazolidin-4-one Show/Hide	C21H21ClN2O4S	1
1	EC50 = 525 nM Bioactivity Info	TI LI LO TS
CP0390197 Compound Info	N-[3-[2,6-dimethyl-4-[5-[3-methyl-4-(2-methylpropyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H31N3O5S	1
1	EC50 = 528 nM Bioactivity Info	TI LI LO TS
CP0372308 Compound Info	(Z,Z)-5-[3-(2-Hydroxy-ethoxy)-benzylidene]-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H22N2O3S	1
1	EC50 = 531 nM Bioactivity Info	TI LI LO TS
CP0270537 Compound Info	N-cycloheptyl-5-cyclopropyl-N-(2-methylcyclohexyl)-1,2-oxazole-3-carboxamide Show/Hide	C21H32N2O2	1
1	EC50 = 535 nM Bioactivity Info	TI LI LO TS
CP0876019 Compound Info	N-(3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)propyl)-2-hydroxyacetamide Show/Hide	C27H35NO4S	1
1	EC50 = 555 nM Bioactivity Info	TI LI LO TS
CP0286386 Compound Info	N,N,5-tricyclohexyl-1,2-oxazole-3-carboxamide Show/Hide	C22H34N2O2	1
1	EC50 = 559 nM Bioactivity Info	TI LI LO TS
CP0420271 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-methyl-6-[[methyl(2-methylpropyl)amino]methyl]pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H39N5O5	1
1	EC50 = 560 nM Bioactivity Info	TI LI LO TS
CP0483485 Compound Info	N-[(2S)-3-[4-[5-[4-(diethylaminomethyl)-3-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 560 nM Bioactivity Info	TI LI LO TS
CP0876016 Compound Info	N-(2-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)ethyl)methane-sulfonamide Show/Hide	C25H33NO4S2	1
1	EC50 = 566 nM Bioactivity Info	TI LI LO TS
CP0403893 Compound Info	3-[[3-[2,6-dimethyl-4-[3-oxo-3-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propyl]phenoxy]-2-hydroxypropyl]amino]propanoic acid Show/Hide	C28H39NO5S	1
1	EC50 = 569 nM Bioactivity Info	TI LI LO TS
CP0473849 Compound Info	[2-amino-4-[4-[2-(4-chlorophenyl)-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C20H22ClN2O6P	1
1	EC50 = 569 nM Bioactivity Info	TI LI LO TS
CP0483484 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-4-[[methyl(2-methylpropyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 570 nM Bioactivity Info	TI LI LO TS
CP0379605 Compound Info	N-[3-[2,6-dimethyl-4-[3-[5-(2-methylpropyl)thiophen-2-yl]-3-oxopropyl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H33NO5S	1
1	EC50 = 590 nM Bioactivity Info	TI LI LO TS
CP0875385 Compound Info	(2R/S)-2-((3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)-2-hydroxy-propyl)amino)acetic acid Show/Hide	C27H35NO5S	1
1	EC50 = 597 nM Bioactivity Info	TI LI LO TS
CP0381995 Compound Info	3-[4-(2,3-dihydroxypropoxy)-3,5-dimethylphenyl]-1-(3-ethyl-5-methyl-4,5,6,7-tetrahydro-2-benzothiophen-1-yl)propan-1-one Show/Hide	C25H34O4S	1
1	EC50 = 599 nM Bioactivity Info	TI LI LO TS
CP0440035 Compound Info	N-[(2S)-3-[4-[5-[6-(diethylamino)-5-methylpyridin-3-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	1
1	EC50 = 616 nM Bioactivity Info	TI LI LO TS
CP0414361 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-[4-(trifluoromethyl)phenyl]triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C20H22F3N4O5P	1
1	EC50 = 616 nM Bioactivity Info	TI LI LO TS
CP0392892 Compound Info	N-[(2S)-3-[4-[5-[5-(diethylamino)-4-methylpyridin-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	1
1	EC50 = 617 nM Bioactivity Info	TI LI LO TS
CP0394080 Compound Info	3-(4-(5-(4-isopropoxy-3-methoxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C22H24N2O5	1
1	EC50 = 620 nM Bioactivity Info	TI LI LO TS
CP0876020 Compound Info	3-(4-((S)-2,3-Dihydroxypropoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H32O4S	1
1	EC50 = 623 nM Bioactivity Info	TI LI LO TS
CP0572693 Compound Info	N-[(2S)-3-[4-[5-[5-[(dimethylamino)methyl]-4-methylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H32N4O5S	1
1	EC50 = 660 nM Bioactivity Info	TI LI LO TS
CP0454269 Compound Info	(Z,Z)-3-Benzyl-5-(3-chloro-4-hydroxy-benzylidene)-2-isopropylimino-thiazolidin-4-one Show/Hide	C20H19ClN2O2S	1
1	EC50 = 674 nM Bioactivity Info	TI LI LO TS
CP0898303 Compound Info	2-amino-4-(4-(4-butylphenethyl)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C23H34NO5P	1
1	EC50 = 674 nM Bioactivity Info	TI LI LO TS
CP0499809 Compound Info	N-[(2S)-3-[4-[5-(2-cyclohexyl-6-methoxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O6	1
1	EC50 = 690 nM Bioactivity Info	TI LI LO TS
CP0445537 Compound Info	N-[(2S)-3-[4-[5-(2-butylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 = 700 nM Bioactivity Info	TI LI LO TS
CP0445533 Compound Info	N-[(2S)-3-[4-[5-(2-cyclopentylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H32N4O5	1
1	EC50 = 736 nM Bioactivity Info	TI LI LO TS
CP0428791 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-(2-methylpropyl)pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 = 757 nM Bioactivity Info	TI LI LO TS
CP0865102 Compound Info	3-(3,5-Dimethyl-4-(2-(methylamino)ethoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H33NO2S	1
1	EC50 = 780 nM Bioactivity Info	TI LI LO TS
CP0469650 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyl-4-methoxypyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 800 nM Bioactivity Info	TI LI LO TS
CP0403891 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3-ethylspiro[6,7-dihydro-4H-2-benzothiophene-5,1'-cyclopropane]-1-yl)propan-1-one Show/Hide	C26H34O4S	1
1	EC50 = 819 nM Bioactivity Info	TI LI LO TS
CP0454270 Compound Info	(Z,Z)-3-Allyl-5-(3-chloro-4-hydroxy-benzylidene)-2-isopropylimino-thiazolidin-4-one Show/Hide	C16H17ClN2O2S	1
1	EC50 = 821 nM Bioactivity Info	TI LI LO TS
CP0397029 Compound Info	[2-amino-4-[4-[2-[(4-fluorophenyl)methyl]-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C21H24FN2O6P	1
1	EC50 = 828 nM Bioactivity Info	TI LI LO TS
CP0456275 Compound Info	(3R)-3-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]-4-oxobutanoic acid Show/Hide	C25H21FN4O3S	1
1	EC50 = 834 nM Bioactivity Info	TI LI LO TS
CP0385931 Compound Info	1-((3-fluoro-4-(5-(1-phenylcyclohexyl)thiazolo[5,4-b]pyridin-2-yl)phenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C29H28FN3O2S	1
1	EC50 = 836 nM Bioactivity Info	TI LI LO TS
CP0542201 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-(4-propylphenyl)-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C23H29N2O6P	1
1	EC50 = 844 nM Bioactivity Info	TI LI LO TS
CP0390246 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyl-6-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 860 nM Bioactivity Info	TI LI LO TS
CP0445534 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyl-4-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O5	1
1	EC50 = 866 nM Bioactivity Info	TI LI LO TS
CP0440019 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[2-(ethylamino)-6-methylpyridin-4-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H31N5O5	1
1	EC50 = 868 nM Bioactivity Info	TI LI LO TS
CP0554584 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-(2-thiophen-2-yl-1,3-oxazol-4-yl)phenyl]butyl] dihydrogen phosphate Show/Hide	C18H21N2O6PS	1
1	EC50 = 869 nM Bioactivity Info	TI LI LO TS
CP0878803 Compound Info	2-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)-N-methyl-acetamide Show/Hide	C25H31NO3S	1
1	EC50 = 870 nM Bioactivity Info	TI LI LO TS
CP0444984 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-methyl-6-[[methyl(propyl)amino]methyl]pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H37N5O5	1
1	EC50 = 870 nM Bioactivity Info	TI LI LO TS
CP0875990 Compound Info	2-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)acetamide Show/Hide	C24H29NO3S	1
1	EC50 = 875 nM Bioactivity Info	TI LI LO TS
CP0514883 Compound Info	1-((3-fluoro-4-(5-((S)-1-phenylethyl)thiazolo[5,4-b]pyridin-2-yl)phenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C25H22FN3O2S	1
1	EC50 = 877 nM Bioactivity Info	TI LI LO TS
CP0865106 Compound Info	3-(4-(2-Hydroxyethoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C24H30O3S	1
1	EC50 = 879 nM Bioactivity Info	TI LI LO TS
CP0072186 Compound Info	1-((3-fluoro-4-(5-(1-phenylcyclopropyl)thiazolo[5,4-b]pyridin-2-yl)phenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C26H22FN3O2S	1
1	EC50 = 888 nM Bioactivity Info	TI LI LO TS
CP0480178 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[(4-methoxyphenyl)methyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C22H27N2O7P	1
1	EC50 = 899.2 nM Bioactivity Info	TI LI LO TS
CP0390593 Compound Info	1-[[3-fluoro-4-[6-(2-propan-2-yl-1,3-thiazolidine-3-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C25H26FN3O3S2	1
1	EC50 = 900 nM Bioactivity Info	TI LI LO TS
CP0501218 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[4-[[ethyl(methyl)amino]methyl]-3-methylphenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 910 nM Bioactivity Info	TI LI LO TS
CP0568660 Compound Info	N-[(2S)-3-[4-[5-(5-cyclopentyl-6-methoxypyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 920 nM Bioactivity Info	TI LI LO TS
CP0456029 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[(4-propan-2-ylphenyl)methyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C24H31N2O6P	1
1	EC50 = 925 nM Bioactivity Info	TI LI LO TS
CP0534607 Compound Info	N-[(2S)-3-[4-[5-(6-cyclopentyloxy-4-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 930 nM Bioactivity Info	TI LI LO TS
CP0436469 Compound Info	3-[1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinolin-7-yl]propanoic acid Show/Hide	C27H21F3N2O4	1
1	EC50 = 940 nM Bioactivity Info	TI LI LO TS
CP0403320 Compound Info	3-(4-(5-(5-chloro-6-isopropoxypyridin-3-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C20H20ClN3O4	1
1	EC50 = 950 nM Bioactivity Info	TI LI LO TS
CP0233337 Compound Info	N,N-dicyclohexyl-5-propan-2-yl-1,2-oxazole-3-carboxamide Show/Hide	C19H30N2O2	1
1	EC50 = 959 nM Bioactivity Info	TI LI LO TS
CP0508745 Compound Info	[2-amino-4-[4-[2-[(4-chlorophenyl)methyl]-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C21H24ClN2O6P	1
1	EC50 = 970 nM Bioactivity Info	TI LI LO TS
CP0385945 Compound Info	1-((3-fluoro-4-(5-((R)-1-phenylethyl)thiazolo[5,4-b]pyridin-2-yl)phenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C25H22FN3O2S	1
1	EC50 = 996 nM Bioactivity Info	TI LI LO TS
CP0454284 Compound Info	(2Z,5Z)-2-(2,2-dimethylhydrazono)-5-(4-hydroxy-3-methoxybenzylidene)-3-phenylthiazolidin-4-one Show/Hide	C19H19N3O3S	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0876613 Compound Info	1-((2R/S)-3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)-2-hydroxy-propyl)azetidine-3-carboxylic acid Show/Hide	C29H37NO5S	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0851048 Compound Info	2-amino-2-(hydroxymethyl)-4-(4'-(2-methyloxazol-4-yl)-[1,1'-biphenyl]-4-yl)butyl dihydrogen phosphate Show/Hide	C21H25N2O6P	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0869939 Compound Info	2-amino-2-(hydroxymethyl)-4-(4'-(2-propyloxazol-4-yl)-[1,1'-biphenyl]-4-yl)butyl dihydrogen phosphate Show/Hide	C23H29N2O6P	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0898301 Compound Info	2-amino-4-(4-(4-(2-ethyloxazol-4-yl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C22H27N2O7P	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0909869 Compound Info	2-amino-4-(6-hexylnaphthalen-1-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H32NO5P	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0863963 Compound Info	3-(6-(2,5-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl3NO4	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0380863 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-(4-methylphenyl)-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H25N2O6P	1
1	EC50 = 1020 nM Bioactivity Info	TI LI LO TS
CP0895803 Compound Info	3-(4-(2-((2-Hydroxyethyl)amino)ethoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C26H35NO3S	1
1	EC50 = 1040 nM Bioactivity Info	TI LI LO TS
CP0403242 Compound Info	[2-amino-4-[4-[4-(2-ethyl-1,3-oxazol-4-yl)phenyl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate;hydrochloride Show/Hide	C22H28ClN2O6P	1
1	EC50 = 1058 nM Bioactivity Info	TI LI LO TS
CP0908208 Compound Info	1-(3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)propyl)azetidine-3-carboxylic acid Show/Hide	C29H37NO4S	1
1	EC50 = 1070 nM Bioactivity Info	TI LI LO TS
CP0442591 Compound Info	3-[4-[(2R)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C25H34O4S	1
1	EC50 = 1098 nM Bioactivity Info	TI LI LO TS
CP0394078 Compound Info	3-(4-{5-[3-cyano-4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazol-3-yl}-3-methylphenyl)propanoic acid Show/Hide	C22H21N3O4	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0408513 Compound Info	4-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)butanoic acid Show/Hide	C25H28N2O3	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0489829 Compound Info	1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinoline-8-carboxylic acid Show/Hide	C25H17F3N2O4	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0427262 Compound Info	3-[[2-bromo-4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C26H30BrF3N2O3	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0508073 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-(4-methoxyphenyl)-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H25N2O7P	1
1	EC50 = 1113 nM Bioactivity Info	TI LI LO TS
CP0390243 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-propylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 = 1120 nM Bioactivity Info	TI LI LO TS
CP0392507 Compound Info	(3S)-3-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]-4-oxobutanoic acid Show/Hide	C25H21FN4O3S	1
1	EC50 = 1130 nM Bioactivity Info	TI LI LO TS
CP0851080 Compound Info	2-amino-4-(4-(4-(2-cyclopropyloxazol-4-yl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C23H27N2O7P	1
1	EC50 = 1130 nM Bioactivity Info	TI LI LO TS
CP0869941 Compound Info	2-amino-4-(4-(4-(4-fluorobenzyl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C24H27FNO6P	1
1	EC50 = 1141 nM Bioactivity Info	TI LI LO TS
CP0434024 Compound Info	N-[3-[2,6-dimethyl-4-[5-(5-propylthiophen-2-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C22H27N3O5S	1
1	EC50 = 1150 nM Bioactivity Info	TI LI LO TS
CP0394070 Compound Info	3-(4-(5-(5-isobutylpyridin-2-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H23N3O3	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0501361 Compound Info	3-(4-(4-(3-phenylpropoxy)phenyl)-5,6-dihydropyridin-1(2H)-yl)propanoic acid Show/Hide	C23H27NO3	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0483482 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-3-[[methyl(2-methylpropyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0389002 Compound Info	1-(4-(5-benzylbenzo[d]thiazol-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C25H21FN2O2S	1
1	EC50 = 1210 nM Bioactivity Info	TI LI LO TS
CP0379838 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-[4-(trifluoromethoxy)phenyl]triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C20H22F3N4O6P	1
1	EC50 = 1219 nM Bioactivity Info	TI LI LO TS
CP0421194 Compound Info	6-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)hexanoic acid Show/Hide	C27H32N2O3	1
1	EC50 = 1220 nM Bioactivity Info	TI LI LO TS
CP0372159 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-ethylimino-3-phenyl-thiazolidin-4-one Show/Hide	C18H15ClN2O2S	1
1	EC50 = 1229 nM Bioactivity Info	TI LI LO TS
CP0404704 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(5-methyl-6-pyrrolidin-1-ylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H33N5O5	1
1	EC50 = 1230 nM Bioactivity Info	TI LI LO TS
CP0568786 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[3-[[ethyl(methyl)amino]methyl]-5-methylphenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 1250 nM Bioactivity Info	TI LI LO TS
CP0445563 Compound Info	N-[3-[4-[5-(5-butylthiophen-2-yl)-1,2,4-oxadiazol-3-yl]-2,6-dimethylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H29N3O5S	1
1	EC50 = 1253 nM Bioactivity Info	TI LI LO TS
CP0559385 Compound Info	US10179791, Compound 128 Show/Hide	C23H25Cl2NO4	1
1	EC50 = 1258.93 nM Bioactivity Info	TI LI LO TS
CP0851014 Compound Info	2-amino-2-(hydroxymethyl)-4-(4-(4-(2-methyloxazol-4-yl)phenoxy)phenyl)butyl dihydrogen phosphate Show/Hide	C21H25N2O7P	1
1	EC50 = 1273 nM Bioactivity Info	TI LI LO TS
CP0385338 Compound Info	3-[1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]-1,6-naphthyridin-7-yl]propanoic acid Show/Hide	C26H20F3N3O4	1
1	EC50 = 1300 nM Bioactivity Info	TI LI LO TS
CP0410679 Compound Info	3-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-cyclopropylphenyl]methylamino]propanoic acid Show/Hide	C29H35F3N2O3	1
1	EC50 = 1300 nM Bioactivity Info	TI LI LO TS
CP0385932 Compound Info	1-(3-fluoro-4-(5-(1-phenylcyclobutyl)thiazolo[5,4-b]pyridin-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C27H24FN3O2S	1
1	EC50 = 1310 nM Bioactivity Info	TI LI LO TS
CP0431227 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-pentan-3-ylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 1340 nM Bioactivity Info	TI LI LO TS
CP0865103 Compound Info	3-(3-Chloro-4-(2-hydroxyethoxy)-5-methylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C23H27ClO3S	1
1	EC50 = 1350 nM Bioactivity Info	TI LI LO TS
CP0106185 Compound Info	N,N-dicyclohexyl-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide Show/Hide	C20H32N2O2	1
1	EC50 = 1375 nM Bioactivity Info	TI LI LO TS
CP0495819 Compound Info	(Z,Z)-5-(3,4-Dimethoxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C21H22N2O3S	1
1	EC50 = 1385 nM Bioactivity Info	TI LI LO TS
CP0397028 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-(4-methylphenyl)triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C20H25N4O5P	1
1	EC50 = 1388 nM Bioactivity Info	TI LI LO TS
CP0419837 Compound Info	[2-amino-4-[4-[1-(4-cyanophenyl)triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C20H22N5O5P	1
1	EC50 = 1390 nM Bioactivity Info	TI LI LO TS
CP0463484 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[[4-(trifluoromethyl)phenyl]methyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C22H24F3N2O6P	1
1	EC50 = 1391 nM Bioactivity Info	TI LI LO TS
CP0415391 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C25H34O4S	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0414581 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-5-[(2-methylpropylamino)methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H36N4O5S	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0380074 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[4-methoxy-6-(2-methylpropyl)pyridin-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O6	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0511185 Compound Info	N-[(2S)-3-[4-[5-(4-cyclopentyloxy-6-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0407071 Compound Info	(Z,Z)-5-[4-(2-Hydroxy-1-hydroxymethyl-ethoxy)-benzylidene]-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C22H24N2O4S	1
1	EC50 = 1430 nM Bioactivity Info	TI LI LO TS
CP0380310 Compound Info	1-(4-(5-(piperidin-1-yl)benzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C24H26N2O3	1
1	EC50 = 1440 nM Bioactivity Info	TI LI LO TS
CP0392503 Compound Info	2-[2-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]ethylamino]acetic acid Show/Hide	C25H22FN3O2S	1
1	EC50 = 1440 nM Bioactivity Info	TI LI LO TS
CP0408509 Compound Info	3-(4-(5-(3-chloro-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H21ClN2O4	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0405884 Compound Info	1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C24H17F3N2O2	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0385153 Compound Info	3-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C26H31F3N2O3	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0469682 Compound Info	N-[(2S)-3-[4-[5-[2-[[butyl(methyl)amino]methyl]-6-methylpyridin-4-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H39N5O5	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0399285 Compound Info	N-[(2S)-3-[4-[5-(4-cyclopentyl-6-methoxypyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H34N4O6	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0392889 Compound Info	US9617250, Example 57 of D1 Show/Hide	C24H30N4O5	1
1	EC50 = 1532 nM Bioactivity Info	TI LI LO TS
CP0379843 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-(2-pentyl-1,3-oxazol-4-yl)phenyl]butyl] dihydrogen phosphate Show/Hide	C19H29N2O6P	1
1	EC50 = 1544 nM Bioactivity Info	TI LI LO TS
CP0488280 Compound Info	2-[[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]methylamino]acetic acid Show/Hide	C24H20FN3O2S	1
1	EC50 = 1560 nM Bioactivity Info	TI LI LO TS
CP0444335 Compound Info	US10179791, Compound 258 Show/Hide	C26H33NO4	1
1	EC50 = 1584.89 nM Bioactivity Info	TI LI LO TS
CP0862081 Compound Info	3-(6-(3-phenylpropoxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C24H30ClNO4	1
1	EC50 = 1584.89 nM Bioactivity Info	TI LI LO TS
CP0381831 Compound Info	3-(4-(5-(3-cyano-4-(2,2,2-trifluoroethoxy)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H16F3N3O4	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0450699 Compound Info	2-[1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinolin-7-yl]acetic acid Show/Hide	C26H19F3N2O4	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0505506 Compound Info	3-[[4-[(E)-N-[[4-cyclopentyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C25H29F3N2O3	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0474137 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(2-methoxy-6-phenylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H30N4O6	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0876018 Compound Info	3-(4-(2-Hydroxyethoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]-thiophen-1-yl)propan-1-one Show/Hide	C22H26O3S	1
1	EC50 = 1610 nM Bioactivity Info	TI LI LO TS
CP0459673 Compound Info	N-cyclohexyl-N-cyclopentyl-5-cyclopropyl-1,2-oxazole-3-carboxamide Show/Hide	C18H26N2O2	1
1	EC50 = 1683 nM Bioactivity Info	TI LI LO TS
CP0566502 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[5-[[2-hydroxyethyl(methyl)amino]methyl]-4-methylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H34N4O6S	1
1	EC50 = 1700 nM Bioactivity Info	TI LI LO TS
CP0541600 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[6-(2-methylpropyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 = 1710 nM Bioactivity Info	TI LI LO TS
CP0851077 Compound Info	2-amino-4-(4-(4-(4-chlorobenzyl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C24H27ClNO6P	1
1	EC50 = 1711 nM Bioactivity Info	TI LI LO TS
CP0882274 Compound Info	2-amino-4-(4-(4-(4-ethylbenzyl)phenoxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C26H32NO6P	1
1	EC50 = 1739 nM Bioactivity Info	TI LI LO TS
CP0334412 Compound Info	N-cyclopentyl-5-cyclopropyl-N-(2-methylcyclohexyl)-1,2-oxazole-3-carboxamide Show/Hide	C19H28N2O2	1
1	EC50 = 1740 nM Bioactivity Info	TI LI LO TS
CP0395614 Compound Info	1-[3-[2,6-dimethyl-4-[3-oxo-3-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propyl]phenoxy]-2-hydroxypropyl]azetidine-3-carboxylic acid Show/Hide	C29H39NO5S	1
1	EC50 = 1755 nM Bioactivity Info	TI LI LO TS
CP0392893 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(6-propylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 = 1770 nM Bioactivity Info	TI LI LO TS
CP0898296 Compound Info	2-amino-4-(4-(4-butylphenoxy)-3-fluorophenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H29FNO6P	1
1	EC50 = 1790 nM Bioactivity Info	TI LI LO TS
CP0876614 Compound Info	3-(4-(3-Hydroxypropoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H32O3S	1
1	EC50 = 1800 nM Bioactivity Info	TI LI LO TS
CP0386358 Compound Info	N-[3-[4-[5-(5-ethylthiophen-2-yl)-1,2,4-oxadiazol-3-yl]-2,6-dimethylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C21H25N3O5S	1
1	EC50 = 1860 nM Bioactivity Info	TI LI LO TS
CP0398773 Compound Info	1-(4-(5-isobutylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H25NO3	1
1	EC50 = 1900 nM Bioactivity Info	TI LI LO TS
CP0492133 Compound Info	3-[[(E)-2-methyl-3-[4-(3-phenylpropoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C22H27NO3	1
1	EC50 = 1900 nM Bioactivity Info	TI LI LO TS
CP0481056 Compound Info	3-[[2-chloro-4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C26H30ClF3N2O3	1
1	EC50 = 1900 nM Bioactivity Info	TI LI LO TS
CP0550854 Compound Info	[2-amino-4-[4-[1-(4-ethylphenyl)triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C21H27N4O5P	1
1	EC50 = 1910 nM Bioactivity Info	TI LI LO TS
CP0556777 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-(1-pentyltriazol-4-yl)phenyl]butyl] dihydrogen phosphate Show/Hide	C18H29N4O5P	1
1	EC50 = 1945 nM Bioactivity Info	TI LI LO TS
CP0863962 Compound Info	3-(6-(2-chloro-6-propylbenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C25H31Cl2NO4	1
1	EC50 = 1995.26 nM Bioactivity Info	TI LI LO TS
CP0480177 Compound Info	[2-amino-4-[4-[1-(4-chlorophenyl)triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C19H22ClN4O5P	1
1	EC50 = 1997 nM Bioactivity Info	TI LI LO TS
CP0554782 Compound Info	N-[(2S)-3-[4-[5-[3-[(dimethylamino)methyl]-5-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 2000 nM Bioactivity Info	TI LI LO TS
CP0403666 Compound Info	1-[[3-fluoro-4-[6-(2-methyl-1,3-thiazolidine-3-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C23H22FN3O3S2	1
1	EC50 = 2040 nM Bioactivity Info	TI LI LO TS
CP0909864 Compound Info	2-amino-4-(6-hexylnaphthalen-2-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H32NO5P	1
1	EC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0420269 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-5-[(2-methylpropylamino)methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0508074 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[4-(trifluoromethoxy)phenyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H22F3N2O7P	1
1	EC50 = 2110 nM Bioactivity Info	TI LI LO TS
CP0909867 Compound Info	2-amino-2-(hydroxymethyl)-4-(4-((3'-methoxy-[1,1'-biphenyl]-4-yl)oxy)phenyl)butyl dihydrogen phosphate Show/Hide	C24H28NO7P	1
1	EC50 = 2197 nM Bioactivity Info	TI LI LO TS
CP0465580 Compound Info	3-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-fluorophenyl]methylamino]propanoic acid Show/Hide	C26H30F4N2O3	1
1	EC50 = 2200 nM Bioactivity Info	TI LI LO TS
CP0853015 Compound Info	3-(4-(3-Hydroxy-2-(hydroxymethyl)propoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C26H34O4S	1
1	EC50 = 2200 nM Bioactivity Info	TI LI LO TS
CP0407397 Compound Info	N-[(2S)-3-[4-[5-[3,4-dimethyl-5-[[methyl(2-methylpropyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H40N4O5S	1
1	EC50 = 2300 nM Bioactivity Info	TI LI LO TS
CP0430361 Compound Info	6-(dipropylamino)-N-(4-hydroxyphenyl)pyrimidine-4-carboxamide Show/Hide	C17H22N4O2	1
1	EC50 = 2320 nM Bioactivity Info	TI LI LO TS
CP0447433 Compound Info	5-[(S)-3-Amino-5-(4-heptyloxy-phenyl)-3-methyl-pentyl]-1,1-dioxo-1lambda6-[1,2,5]thiadiazolidin-3-one Show/Hide	C21H35N3O4S	1
1	EC50 = 2400 nM Bioactivity Info	TI LI LO TS
CP0463725 Compound Info	3-[[5-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]furan-2-yl]methylamino]propanoic acid Show/Hide	C24H29F3N2O4	1
1	EC50 = 2500 nM Bioactivity Info	TI LI LO TS
CP0389006 Compound Info	1-(3-fluoro-4-(5-(2-phenylpropan-2-yl)thiazolo[5,4-b]pyridin-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C26H24FN3O2S	1
1	EC50 = 2510 nM Bioactivity Info	TI LI LO TS
CP0084726 Compound Info	2-(4-octylphenethyl)-2-aminopropane-1,3-diol Show/Hide	C19H33NO2	2
1	EC50 = 2511.89 nM Bioactivity Info	TI LI LO TS
2	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0372310 Compound Info	(Z,Z)-5-(2-Chloro-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H17ClN2OS	1
1	EC50 = 2583 nM Bioactivity Info	TI LI LO TS
CP0878807 Compound Info	3-(4-(2-Hydroxyethoxy)-3-methylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C23H28O3S	1
1	EC50 = 2590 nM Bioactivity Info	TI LI LO TS
CP0507797 Compound Info	3-[[6-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]pyridin-3-yl]methylamino]propanoic acid Show/Hide	C25H30F3N3O3	1
1	EC50 = 2600 nM Bioactivity Info	TI LI LO TS
CP0389626 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-(3-methylbutyl)pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 2600 nM Bioactivity Info	TI LI LO TS
CP0446794 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(5-methyl-6-pentan-3-ylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 2630 nM Bioactivity Info	TI LI LO TS
CP0401204 Compound Info	1-[[4-[6-(2,2-dimethyl-1,3-thiazolidine-3-carbonyl)-1,3-benzothiazol-2-yl]-3-fluorophenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C24H24FN3O3S2	1
1	EC50 = 2680 nM Bioactivity Info	TI LI LO TS
CP0258904 Compound Info	N-cycloheptyl-N-cyclopentyl-5-cyclopropyl-1,2-oxazole-3-carboxamide Show/Hide	C19H28N2O2	1
1	EC50 = 2753 nM Bioactivity Info	TI LI LO TS
CP0434248 Compound Info	3-(5-{5-[3-cyano-4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridin-2-yl)propanoic acid Show/Hide	C21H20N4O4	1
1	EC50 = 2760 nM Bioactivity Info	TI LI LO TS
CP0865104 Compound Info	3-(4-(2-Hydroxyethoxy)-2-methoxyphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C23H28O4S	1
1	EC50 = 2780 nM Bioactivity Info	TI LI LO TS
CP0350596 Compound Info	5-cyclopropyl-N-(2-methylcyclohexyl)-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide Show/Hide	C19H28N2O3	1
1	EC50 = 2820 nM Bioactivity Info	TI LI LO TS
CP0876017 Compound Info	3-(4-(2-(Dimethylamino)ethoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C26H35NO2S	1
1	EC50 = 2840 nM Bioactivity Info	TI LI LO TS
CP0387947 Compound Info	3-[2-ethyl-6-methyl-4-[5-[(2S,4R)-3,3,9-trimethyl-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-dien-7-yl]-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid Show/Hide	C25H28N2O3S	1
1	EC50 = 2880 nM Bioactivity Info	TI LI LO TS
CP0389001 Compound Info	1-((4-(6-benzylthiazolo[5,4-b]pyridin-2-yl)-3-fluorophenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 = 2890 nM Bioactivity Info	TI LI LO TS
CP0906431 Compound Info	1-((6-(3-(2-fluorophenyl)propoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C25H29ClFNO3	1
1	EC50 = 2900 nM Bioactivity Info	TI LI LO TS
CP0440023 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(6-propan-2-ylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 = 2900 nM Bioactivity Info	TI LI LO TS
CP0509642 Compound Info	N-[(2S)-3-[4-[5-[3-[[butyl(methyl)amino]methyl]-4-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 = 2900 nM Bioactivity Info	TI LI LO TS
CP0380878 Compound Info	[2-amino-4-[4-[2-(4-cyanophenyl)-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C21H22N3O6P	1
1	EC50 = 2973 nM Bioactivity Info	TI LI LO TS
CP0436615 Compound Info	3-[[(E)-2-methyl-3-[4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C23H29NO3	1
1	EC50 = 3000 nM Bioactivity Info	TI LI LO TS
CP0511321 Compound Info	3-[[4-[(E)-N-[[4-(furan-2-yl)-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C24H23F3N2O4	1
1	EC50 = 3000 nM Bioactivity Info	TI LI LO TS
CP0456030 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-(4-methoxyphenyl)triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C20H25N4O6P	1
1	EC50 = 3008 nM Bioactivity Info	TI LI LO TS
CP0386332 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[6-methyl-5-(2-methylpropyl)pyridin-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 3080 nM Bioactivity Info	TI LI LO TS
CP0381221 Compound Info	(S)-4-amino-6-(4-(heptyloxy)phenyl)-4-methylhexanoic acid Show/Hide	C20H33NO3	1
1	EC50 = 3100 nM Bioactivity Info	TI LI LO TS
CP0420273 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-4-(pyrrolidin-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H36N4O5	1
1	EC50 = 3100 nM Bioactivity Info	TI LI LO TS
CP0915964 Compound Info	1-((6-(3-(4-fluorophenyl)propoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C25H29ClFNO3	1
1	EC50 = 3200 nM Bioactivity Info	TI LI LO TS
CP0417590 Compound Info	1-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-methylphenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C28H33F3N2O3	1
1	EC50 = 3200 nM Bioactivity Info	TI LI LO TS
CP0469680 Compound Info	N-[(2S)-3-[4-[5-[4-[(dimethylamino)methyl]-3-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 3200 nM Bioactivity Info	TI LI LO TS
CP0383844 Compound Info	6-(cyclohexyl(cyclopropylmethyl)amino)-N-(6-methyl-1H-indazol-5-yl)pyrimidine-4-carboxamide Show/Hide	C23H28N6O	1
1	EC50 = 3270 nM Bioactivity Info	TI LI LO TS
CP0422247 Compound Info	(E/Z)-3-(3-(4-(3-phenylpropoxy)phenyl)allylamino)propanoic acid Show/Hide	C21H25NO3	1
1	EC50 = 3300 nM Bioactivity Info	TI LI LO TS
CP0480441 Compound Info	1-[(E)-3-[4-(3-phenylpropoxy)phenyl]prop-2-enyl]azetidine-3-carboxylic acid Show/Hide	C22H25NO3	1
1	EC50 = 3300 nM Bioactivity Info	TI LI LO TS
CP0874455 Compound Info	2-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)-N-(2-hydroxy-ethyl)acetamide Show/Hide	C26H33NO4S	1
1	EC50 = 3410 nM Bioactivity Info	TI LI LO TS
CP0393734 Compound Info	1-(4-(5-benzylbenzofuran-2-yl)-2-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C26H22FNO3	1
1	EC50 = 3430 nM Bioactivity Info	TI LI LO TS
CP0262672 Compound Info	N-cyclohexyl-N-(cyclohexylmethyl)-5-cyclopropyl-1,2-oxazole-3-carboxamide Show/Hide	C20H30N2O2	1
1	EC50 = 3430 nM Bioactivity Info	TI LI LO TS
CP0389000 Compound Info	1-(4-(6-benzylbenzo[d]thiazol-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C25H21FN2O2S	1
1	EC50 = 3470 nM Bioactivity Info	TI LI LO TS
CP0210527 Compound Info	N-cyclohexyl-5-cyclopropyl-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide Show/Hide	C18H26N2O3	1
1	EC50 = 3536 nM Bioactivity Info	TI LI LO TS
CP0541601 Compound Info	N-[3-[2-ethyl-6-methyl-4-[5-[2-(3-methylbutyl)pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 = 3730 nM Bioactivity Info	TI LI LO TS
CP0379606 Compound Info	3-[4-[(2S)-2,3-dihydroxypropoxy]-3,5-dimethylphenyl]-1-(3-ethyl-4,5,6,7-tetrahydro-2-benzothiophen-1-yl)propan-1-one Show/Hide	C24H32O4S	1
1	EC50 = 3830 nM Bioactivity Info	TI LI LO TS
CP0854743 Compound Info	1-((6-(3-(3-fluorophenyl)propoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C25H29ClFNO3	1
1	EC50 = 3900 nM Bioactivity Info	TI LI LO TS
CP0442590 Compound Info	N-[3-[2-ethyl-4-[3-(3-methoxy-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-3-oxopropyl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H39NO6S	1
1	EC50 = 3910 nM Bioactivity Info	TI LI LO TS
CP0392890 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-propan-2-ylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 = 3940 nM Bioactivity Info	TI LI LO TS
CP0863958 Compound Info	3-(6-(2,6-dichlorobenzylthio)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl3NO3S	1
1	EC50 = 3981.07 nM Bioactivity Info	TI LI LO TS
CP0478376 Compound Info	3-[[5-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]thiophen-2-yl]methylamino]propanoic acid Show/Hide	C24H29F3N2O3S	1
1	EC50 = 4000 nM Bioactivity Info	TI LI LO TS
CP0390654 Compound Info	3-(4-(5-(3-fluoro-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H21FN2O4	1
1	EC50 = 4070 nM Bioactivity Info	TI LI LO TS
CP0377161 Compound Info	3-(3-(4-(5-phenylpentyloxy)phenyl)propylamino)propanoic acid Show/Hide	C23H31NO3	1
1	EC50 = 4200 nM Bioactivity Info	TI LI LO TS
CP0851941 Compound Info	3-(4-(3-Aminopropoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H33NO2S	1
1	EC50 = 4200 nM Bioactivity Info	TI LI LO TS
CP0851940 Compound Info	3-(3,5-Dichloro-4-(2-hydroxyethoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C22H24Cl2O3S	1
1	EC50 = 4250 nM Bioactivity Info	TI LI LO TS
CP0487810 Compound Info	3-[[5-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]pyridin-2-yl]methylamino]propanoic acid Show/Hide	C25H30F3N3O3	1
1	EC50 = 4300 nM Bioactivity Info	TI LI LO TS
CP0420266 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[3-ethyl-4-(pyrrolidin-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H38N4O5	1
1	EC50 = 4300 nM Bioactivity Info	TI LI LO TS
CP0474129 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-3-[[methyl(propyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 = 4300 nM Bioactivity Info	TI LI LO TS
CP0414532 Compound Info	N-[(2S)-3-[4-[5-[5-[(dimethylamino)methyl]-3,4-dimethylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H34N4O5S	1
1	EC50 = 4400 nM Bioactivity Info	TI LI LO TS
CP0393039 Compound Info	N-[3-[2-ethyl-6-methyl-4-[3-oxo-3-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propyl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H39NO5S	1
1	EC50 = 4418 nM Bioactivity Info	TI LI LO TS
CP0395618 Compound Info	3-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C24H32O3S	1
1	EC50 = 4447 nM Bioactivity Info	TI LI LO TS
CP0403894 Compound Info	3-[4-(3-hydroxypropoxy)-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C25H34O3S	1
1	EC50 = 4450 nM Bioactivity Info	TI LI LO TS
CP0420265 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[5-[[ethyl(methyl)amino]methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H32N4O5S	1
1	EC50 = 4600 nM Bioactivity Info	TI LI LO TS
CP0876610 Compound Info	3-(3-Chloro-4-(2-hydroxyethoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C22H25ClO3S	1
1	EC50 = 4630 nM Bioactivity Info	TI LI LO TS
CP0407755 Compound Info	1-((3-fluoro-4-(6-(1-phenylcyclopropyl)benzo[d]thiazol-2-yl)phenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C27H23FN2O2S	1
1	EC50 = 4670 nM Bioactivity Info	TI LI LO TS
CP0379846 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-(4-propylphenyl)triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C22H29N4O5P	1
1	EC50 = 4689 nM Bioactivity Info	TI LI LO TS
CP0380314 Compound Info	1-(4-(5-(cyclopropylmethoxy)benzofuran-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C23H22FNO4	1
1	EC50 = 4800 nM Bioactivity Info	TI LI LO TS
CP0856515 Compound Info	1-((1-methyl-6-(3-phenylpropoxy)-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C25H30ClNO3	1
1	EC50 = 5000 nM Bioactivity Info	TI LI LO TS
CP0214241 Compound Info	1-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-ethylphenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C29H35F3N2O3	1
1	EC50 = 5000 nM Bioactivity Info	TI LI LO TS
CP0899669 Compound Info	3-(3,5-Dimethyl-4-(3-(methylamino)propoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C26H35NO2S	1
1	EC50 = 5030 nM Bioactivity Info	TI LI LO TS
CP0899670 Compound Info	3-(2-Chloro-4-(2-hydroxyethoxy)phenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C22H25ClO3S	1
1	EC50 = 5200 nM Bioactivity Info	TI LI LO TS
CP0869583 Compound Info	3-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenyl)propanoic acid Show/Hide	C25H30O3S	1
1	EC50 = 5210 nM Bioactivity Info	TI LI LO TS
CP0541598 Compound Info	N-[(2S)-3-[4-[5-[4-(diethylamino)-6-methylpyridin-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	1
1	EC50 = 5240 nM Bioactivity Info	TI LI LO TS
CP0395617 Compound Info	N-[(2S)-3-[4-[3-(5,5-dimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)-3-oxopropyl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H37NO5S	1
1	EC50 = 5270 nM Bioactivity Info	TI LI LO TS
CP0443773 Compound Info	N-[3-[4-[3-[3,5-dimethyl-4-(2-methylpropyl)thiophen-2-yl]-3-oxopropyl]-2,6-dimethylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H37NO5S	1
1	EC50 = 5270 nM Bioactivity Info	TI LI LO TS
CP0389005 Compound Info	1-(4-(6-benzylthiazolo[4,5-c]pyridin-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 = 5460 nM Bioactivity Info	TI LI LO TS
CP0420268 Compound Info	N-[(2S)-3-[4-[5-[4-[(dimethylamino)methyl]-3,5-dimethylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 5500 nM Bioactivity Info	TI LI LO TS
CP0392504 Compound Info	4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]-4-oxobutanoic acid Show/Hide	C25H20FN3O3S	1
1	EC50 = 5560 nM Bioactivity Info	TI LI LO TS
CP0450697 Compound Info	8-(aminomethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C25H20F3N3O2	1
1	EC50 = 5600 nM Bioactivity Info	TI LI LO TS
CP0457393 Compound Info	N-[(2R)-3-[2-ethyl-6-methyl-4-[5-[6-(2-methylpropyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 = 5740 nM Bioactivity Info	TI LI LO TS
CP0372148 Compound Info	(Z,Z)-2-Isopropylimino-5-(2-methyl-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2OS	1
1	EC50 = 5791 nM Bioactivity Info	TI LI LO TS
CP0410678 Compound Info	3-[[4-[(E)-C-methyl-N-[[4-thiophen-2-yl-3-(trifluoromethyl)phenyl]methoxy]carbonimidoyl]phenyl]methylamino]propanoic acid Show/Hide	C24H23F3N2O3S	1
1	EC50 = 5900 nM Bioactivity Info	TI LI LO TS
CP0481055 Compound Info	3-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-methylphenyl]methylamino]propanoic acid Show/Hide	C27H33F3N2O3	1
1	EC50 = 5900 nM Bioactivity Info	TI LI LO TS
CP0539722 Compound Info	N-[(2S)-3-[4-[5-[5-(diethylamino)-6-methylpyridin-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H35N5O5	1
1	EC50 = 5960 nM Bioactivity Info	TI LI LO TS
CP0390203 Compound Info	(S)-1-(4-(heptyloxy)phenyl)-3-methyl-5-(1H-tetrazol-5-yl)pentan-3-amine Show/Hide	C20H33N5O	1
1	EC50 = 6400 nM Bioactivity Info	TI LI LO TS
CP0224930 Compound Info	N-benzyl-5-cyclopropyl-N-pyridin-2-yl-1,2-oxazole-3-carboxamide Show/Hide	C19H17N3O2	1
1	EC50 = 6563 nM Bioactivity Info	TI LI LO TS
CP0437510 Compound Info	MLS000087301 Show/Hide	C17H26N2O2	1
1	EC50 = 6595 nM Bioactivity Info	TI LI LO TS
CP0407077 Compound Info	(Z,Z)-2-Isopropylimino-5-(2-methoxy-benzylidene)-3-phenyl-thiazolidin-4-one Show/Hide	C20H20N2O2S	1
1	EC50 = 6689 nM Bioactivity Info	TI LI LO TS
CP0501178 Compound Info	3-[[(E)-3-[4-(5-phenylpentoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C23H29NO3	1
1	EC50 = 6700 nM Bioactivity Info	TI LI LO TS
CP0232742 Compound Info	N-benzyl-5-cyclopropyl-N-phenyl-1,2-oxazole-3-carboxamide Show/Hide	C20H18N2O2	1
1	EC50 = 7000 nM Bioactivity Info	TI LI LO TS
CP0391882 Compound Info	4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]butanoic acid Show/Hide	C25H22FN3O2S	1
1	EC50 = 7120 nM Bioactivity Info	TI LI LO TS
CP0503489 Compound Info	3-[[(E)-3-[2-chloro-4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C22H26ClNO3	1
1	EC50 = 7200 nM Bioactivity Info	TI LI LO TS
CP0385152 Compound Info	3-[[4-[(E)-N-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-C-methylcarbonimidoyl]-2-ethylphenyl]methylamino]propanoic acid Show/Hide	C28H35F3N2O3	1
1	EC50 = 7200 nM Bioactivity Info	TI LI LO TS
CP0391835 Compound Info	1-[[3-fluoro-4-[6-(1,3-thiazolidine-3-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C22H20FN3O3S2	1
1	EC50 = 7420 nM Bioactivity Info	TI LI LO TS
CP0869584 Compound Info	(2R/S)-3-(4-(2-Hydroxy-3-((2-hydroxyethyl)amino)propoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)-propan-1-one Show/Hide	C27H37NO4S	1
1	EC50 = 7470 nM Bioactivity Info	TI LI LO TS
CP0511453 Compound Info	3-[[6-(4-phenylbutoxy)-3,4-dihydronaphthalen-2-yl]methylamino]propanoic acid Show/Hide	C24H29NO3	1
1	EC50 = 7800 nM Bioactivity Info	TI LI LO TS
CP0341701 Compound Info	N-cyclohexyl-N-cyclopentyl-5-propyl-1,2-oxazole-3-carboxamide Show/Hide	C18H28N2O2	1
1	EC50 = 7985 nM Bioactivity Info	TI LI LO TS
CP0232744 Compound Info	N,N-dicyclohexyl-5-(3,4-diethoxyphenyl)-1,2-oxazole-3-carboxamide Show/Hide	C26H36N2O4	1
1	EC50 = 8070 nM Bioactivity Info	TI LI LO TS
CP0469683 Compound Info	N-[(2S)-3-[4-[5-[2-(diethylaminomethyl)-6-methylpyridin-4-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H37N5O5	1
1	EC50 = 8100 nM Bioactivity Info	TI LI LO TS
CP0876004 Compound Info	(S)-1-((6-(3-(4-chlorophenyl)-2-methylpropoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H31Cl2NO3	1
1	EC50 = 8200 nM Bioactivity Info	TI LI LO TS
CP0893675 Compound Info	3-(4-(3-((2-Hydroxyethyl)amino)propoxy)-3,5-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C27H37NO3S	1
1	EC50 = 8420 nM Bioactivity Info	TI LI LO TS
CP0395615 Compound Info	3-[4-(2-aminoethoxy)-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C24H33NO2S	1
1	EC50 = 8558 nM Bioactivity Info	TI LI LO TS
CP0374264 Compound Info	(Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-methylimino-3-phenyl-thiazolidin-4-one Show/Hide	C17H13ClN2O2S	1
1	EC50 = 8810 nM Bioactivity Info	TI LI LO TS
CP0478097 Compound Info	3-(3-(4-(3-phenylpropoxy)phenyl)propylamino)propanoic acid Show/Hide	C21H27NO3	1
1	EC50 = 9000 nM Bioactivity Info	TI LI LO TS
CP0542112 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[3-[[ethyl(methyl)amino]methyl]-4-methylphenyl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 = 9000 nM Bioactivity Info	TI LI LO TS
CP0856516 Compound Info	(S)-1-((6-(3-(4-fluorophenyl)-2-methylpropoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H31ClFNO3	1
1	EC50 = 9450 nM Bioactivity Info	TI LI LO TS
CP0442126 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(2-ethylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H28N4O5	1
1	EC50 = 9950 nM Bioactivity Info	TI LI LO TS
CP0381566 Compound Info	4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)-3-methylbenzoic acid Show/Hide	C22H22N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0381847 Compound Info	3-(4-(5-(4-methoxy-3-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C20H17F3N2O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0394068 Compound Info	3-(4-(5-(6-isopropoxypyridin-3-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C20H21N3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0394073 Compound Info	3-(4-(5-(5-butylpyridin-2-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H23N3O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0408158 Compound Info	5-(4-cyclohexylphenyl)-3-o-tolyl-1,2,4-oxadiazole Show/Hide	C21H22N2O	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0372152 Compound Info	(Z,Z)-3-[5-(3-Chloro-4-hydroxy-benzylidene)-2-isopropylimino-4-oxo-thiazolidin-3-yl]-propionicacid Show/Hide	C16H17ClN2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0454271 Compound Info	(Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-imino-3-phenyl-thiazolidin-4-one Show/Hide	C16H11ClN2O2S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0495818 Compound Info	(Z,Z)-5-(3,4-Dihydroxy-benzylidene)-2-isopropylimino-3-phenyl-thiazolidin-4-one Show/Hide	C19H18N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0447149 Compound Info	3-(4-(4-(3-phenylpropoxy)phenyl)piperidin-1-yl)propanoic acid Show/Hide	C23H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0447150 Compound Info	3-(3-(4-(6-phenylhexyloxy)phenyl)propylamino)propanoic acid Show/Hide	C24H33NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0487579 Compound Info	3-[(3E)-3-[[4-(3-phenylpropoxy)phenyl]methylidene]piperidin-1-yl]propanoic acid Show/Hide	C24H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0494650 Compound Info	3-(3-(4-(4-phenylbutoxy)phenyl)propylamino)propanoic acid Show/Hide	C22H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0501458 Compound Info	3-[[(E)-3-[4-(3-phenylpropoxy)phenyl]but-2-enyl]amino]propanoic acid Show/Hide	C22H27NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0503563 Compound Info	3-[[(Z)-3-[4-(3-phenylpropoxy)phenyl]but-2-enyl]amino]propanoic acid Show/Hide	C22H27NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0436609 Compound Info	1-[(E)-3-[4-(3-phenylpropoxy)phenyl]prop-2-enyl]piperidine-4-carboxylic acid Show/Hide	C24H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0436614 Compound Info	3-[[(E)-3-[4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C22H27NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0455131 Compound Info	1-[[5-methyl-2-(4-phenylbutoxy)-8,9-dihydro-7H-benzo[7]annulen-6-yl]methyl]azetidine-3-carboxylic acid Show/Hide	C27H33NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0475006 Compound Info	3-[[(E)-3-[2-methoxy-4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C23H29NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0478314 Compound Info	3-[[(E)-3-[2-methyl-4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C23H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0494106 Compound Info	3-[[(E)-3-[3-methyl-4-(4-phenylbutoxy)phenyl]prop-2-enyl]amino]propanoic acid Show/Hide	C23H29NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0501179 Compound Info	3-[[1-methyl-6-(4-phenylbutoxy)-3,4-dihydronaphthalen-2-yl]methylamino]propanoic acid Show/Hide	C25H31NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0501185 Compound Info	1-[[1-methyl-6-(4-phenylbutoxy)-3,4-dihydronaphthalen-2-yl]methyl]azetidine-3-carboxylic acid Show/Hide	C26H31NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0389617 Compound Info	(2S)-2-[[4-[3-[(4-chloro-2,5-dimethylphenyl)sulfonylamino]phenyl]-2,6-dimethylbenzoyl]-methylamino]-4-(dimethylamino)butanoic acid Show/Hide	C30H36ClN3O5S	2
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
2	IC50 = 802 nM Bioactivity Info	TI LI LO TS
CP0851931 Compound Info	(2RS)-3-(2,6-Dimethyl-4-(2-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)thiazol-5-yl)phenoxy)propane-1,2-diol Show/Hide	C25H29NO3S2	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0853014 Compound Info	(3bS,4aR)-N-(2-(2-Hydroxyethoxy)benzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0865105 Compound Info	(3bS,4aR)-N-(2,5-Dimethoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0869521 Compound Info	(3bS,4aR)-N-(3-(2-Hydroxyethoxy)benzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]-thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0869522 Compound Info	(3bS,4aR)-N-(2,4-Dimethoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0875387 Compound Info	3-(3-Ethyl-4-(2-hydroxyethoxy)-5-methylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H32O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0875389 Compound Info	3-(4-(2-Hydroxyethoxy)-3,5-dimethoxyphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C24H30O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0875390 Compound Info	(3bS,4aR)-N-(4-(2-Hydroxyethoxy)-2-methoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C22H27NO4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0875391 Compound Info	(3bS,4aR)-N-(4-(2-Hydroxyethoxy)benzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0875985 Compound Info	(2RS)-3-(2,6-Dimethyl-4-(5-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)-1,3,4-thiadiazol-2-yl)phenoxy)propane-1,2-diol Show/Hide	C24H28N2O3S2	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0876021 Compound Info	2-(3-Methoxy-4-(((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydro-cyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamido)methyl)phenoxy)acetic acid Show/Hide	C22H25NO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0876612 Compound Info	(3bS,4aR)-N-(2,6-Dimethoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0878804 Compound Info	3-(4-(2-Hydroxyethoxy)-2,6-dimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C24H30O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0878805 Compound Info	3-(4-(2-Hydroxyethoxy)-2,6-dimethoxyphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C24H30O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0878806 Compound Info	2-(2,6-Dimethyl-4-(3-oxo-3-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propyl)phenoxy)acetic acid Show/Hide	C24H28O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0880200 Compound Info	(3bS,4aR)-N-(2-Methoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C20H23NO2S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0895696 Compound Info	(3bS,4aR)-N-(2,3-Dimethoxybenzyl)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophene-1-carboxamide Show/Hide	C21H25NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0895771 Compound Info	3-(4-(2-Hydroxyethoxy)-3-methoxyphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C23H28O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0901837 Compound Info	3-(4-(2-Hydroxyethoxy)-2,3,5-trimethylphenyl)-1-((3bS,4aR)-3,4,4-trimethyl-3b,4,4a,5-tetrahydrocyclopropa[3,4]cyclopenta[1,2-c]thiophen-1-yl)propan-1-one Show/Hide	C25H32O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0379608 Compound Info	3-[4-(3-amino-2-hydroxypropoxy)-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C25H35NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0390199 Compound Info	3-(4-hydroxy-3,5-dimethylphenyl)-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C22H28O2S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0393041 Compound Info	3-[4-[3-(2-hydroxyethylamino)propoxy]-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C27H39NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0395619 Compound Info	3-[4-[2-(2-hydroxyethylamino)ethoxy]-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C26H37NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0403887 Compound Info	3-[4-(2,3-dihydroxypropoxy)-3,5-dimethylphenyl]-1-[(5S)-5-(dimethylamino)-3-ethyl-4,5,6,7-tetrahydro-2-benzothiophen-1-yl]propan-1-one Show/Hide	C26H37NO4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0403888 Compound Info	3-[4-(2,3-dihydroxypropoxy)-3,5-dimethylphenyl]-1-[(5S)-3-ethyl-5-hydroxy-5-methyl-6,7-dihydro-4H-2-benzothiophen-1-yl]propan-1-one Show/Hide	C25H34O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0434450 Compound Info	3-[4-[2-hydroxy-3-(2-hydroxyethylamino)propoxy]-3,5-dimethylphenyl]-1-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propan-1-one Show/Hide	C27H39NO4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0442592 Compound Info	3-[4-(2,3-dihydroxypropoxy)-3,5-dimethylphenyl]-1-[(5S)-3-ethyl-5-hydroxy-4,5,6,7-tetrahydro-2-benzothiophen-1-yl]propan-1-one Show/Hide	C24H32O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0471597 Compound Info	3-[2,6-dimethyl-4-[3-oxo-3-(3,5,5-trimethyl-6,7-dihydro-4H-2-benzothiophen-1-yl)propyl]phenyl]propanoic acid Show/Hide	C25H32O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0433971 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-(5-pyridin-4-yl-1,2,4-oxadiazol-3-yl)phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C21H24N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0440018 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C22H26N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0445538 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-(2-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C22H26N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0466512 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(6-ethylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H28N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0096517 Compound Info	2-amino-2-[2-[4-[4-(2-ethyl-1,3-oxazol-4-yl)phenyl]phenyl]ethyl]propane-1,3-diol;hydrochloride Show/Hide	C22H27ClN2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0429299 Compound Info	2-amino-2-[2-[4-[4-[2-(1-hydroxyethyl)-1,3-oxazol-4-yl]phenyl]phenyl]ethyl]propane-1,3-diol;hydrochloride Show/Hide	C22H27ClN2O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0444011 Compound Info	2-amino-2-[2-[4-[4-[2-(2-hydroxypropyl)-1,3-oxazol-4-yl]phenyl]phenyl]ethyl]propane-1,3-diol;hydrochloride Show/Hide	C23H29ClN2O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0444012 Compound Info	2-amino-2-[2-[4-[4-(2-propyl-1,3-oxazol-4-yl)phenyl]phenyl]ethyl]propane-1,3-diol;hydrochloride Show/Hide	C23H29ClN2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0407395 Compound Info	N-[(2S)-3-[4-[5-[4-[(dimethylamino)methyl]-2-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0407396 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-5-(methylaminomethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H30N4O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0414527 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-methyl-6-(pyrrolidin-1-ylmethyl)pyridin-4-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H35N5O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0414529 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-[(2-methylpropylamino)methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H36N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0414531 Compound Info	N-[(2S)-3-[4-[5-[4-[(dimethylamino)methyl]phenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H32N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0414580 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-[5-(ethylaminomethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H30N4O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0420272 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-(methylaminomethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0420275 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[5-[(propan-2-ylamino)methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H32N4O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0459612 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-(methylaminomethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C24H30N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0459614 Compound Info	N-[(2S)-3-[2-ethyl-4-[5-(5-formyl-4-methylthiophen-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C22H25N3O6S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0474126 Compound Info	N-[(2S)-3-[4-[5-[2-[(dimethylamino)methyl]-6-methylpyridin-4-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C25H33N5O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0483477 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-methyl-4-[(2-methylpropylamino)methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0483483 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[2-methyl-5-[[methyl(2-methylpropyl)amino]methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C29H40N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0501219 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[5-(methylaminomethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C22H28N4O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0501220 Compound Info	N-[(2S)-3-[4-[5-[5-[(dimethylamino)methyl]thiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C23H30N4O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0542113 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[4-methyl-3-[(2-methylpropylamino)methyl]phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C28H38N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0554784 Compound Info	N-[(2S)-3-[4-[5-[3-[(dimethylamino)methyl]-4-methylphenyl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0554785 Compound Info	N-[(2S)-3-[4-[5-[5-[[2-(dimethylamino)ethyl-methylamino]methyl]-4-methylthiophen-2-yl]-1,2,4-oxadiazol-3-yl]-2-ethyl-6-methylphenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C27H39N5O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0559244 Compound Info	N-[(2S)-3-[2-ethyl-6-methyl-4-[5-[3-(propylaminomethyl)phenyl]-1,2,4-oxadiazol-3-yl]phenoxy]-2-hydroxypropyl]-2-hydroxyacetamide Show/Hide	C26H34N4O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0410304 Compound Info	3-[6-[(2-chloro-6-ethylphenyl)methoxy]spiro[2H-1-benzofuran-3,4'-piperidine]-1'-yl]-2-methylpropanoic acid;hydrochloride Show/Hide	C25H31Cl2NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0475809 Compound Info	3-[6-[(2-chloro-6-ethylphenyl)methoxy]spiro[2H-1-benzofuran-3,3'-piperidine]-1'-yl]propanoic acid;hydrochloride Show/Hide	C24H29Cl2NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0862080 Compound Info	3-(6-((2,6-dichloropyridin-4-yl)methoxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C21H23Cl3N2O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0863955 Compound Info	3-(6-(2,6-dichlorobenzyloxy)-7-fluoro-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H23Cl3FNO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0863957 Compound Info	3-(6-(2,3-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0863960 Compound Info	(E)-3-(6-(2,6-dichlorostyryl)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H24Cl3NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0863961 Compound Info	3-(6-(2,6-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)-2-methylpropanoic acid hydrochloride Show/Hide	C23H26Cl3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0863964 Compound Info	3-(6-(2,6-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0882546 Compound Info	2-(6-(2,6-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)ethyl dihydrogen phosphate hydrochloride Show/Hide	C21H25Cl3NO6P	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0882547 Compound Info	3-(6-(2,6-dichloro-4-methylbenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H26Cl3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0882548 Compound Info	3-(6-((2-chlorophenyl)ethynyl)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H23Cl2NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0882550 Compound Info	3-(6-(2-chloro-6-ethylbenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C24H29Cl2NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0882551 Compound Info	3-(6-(3-chlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H25Cl2NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0931379 Compound Info	3-(6-(2,6-dichlorobenzyloxy)-2H-spiro[benzofuran-3,3'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0948587 Compound Info	3-(6-(2-chloro-6-fluorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H24Cl2FNO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0950442 Compound Info	3-(6-(2-chloro-6-(trifluoromethoxy)benzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H24Cl2F3NO5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0952523 Compound Info	3-(6-(2-chloro-6-(trifluoromethyl)benzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H24Cl2F3NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0952524 Compound Info	3-(6-(benzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C22H26ClNO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0952542 Compound Info	3-(6-(phenylethynyl)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C23H24ClNO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0960370 Compound Info	2-(6-(2,6-dichlorobenzylsulfonyl)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)acetic acid hydrochloride Show/Hide	C21H22Cl3NO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0960909 Compound Info	3-(6-(2-chloro-6-isopropylbenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C25H31Cl2NO4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0385933 Compound Info	1-((4-(5-benzylthiazolo[4,5-b]pyridin-2-yl)-3-fluorophenyl)methyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 = 10100 nM Bioactivity Info	TI LI LO TS
CP0380313 Compound Info	1-(4-(5-butoxybenzofuran-2-yl)-3-chlorobenzyl)azetidine-3-carboxylic acid Show/Hide	C23H24ClNO4	1
1	EC50 = 10300 nM Bioactivity Info	TI LI LO TS
CP0873458 Compound Info	(R)-1-((6-(3-(4-fluorophenyl)-2-methylpropoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H31ClFNO3	1
1	EC50 = 11000 nM Bioactivity Info	TI LI LO TS
CP0854745 Compound Info	1-((1-methyl-6-(4-phenylbutan-2-yloxy)-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H32ClNO3	1
1	EC50 = 14000 nM Bioactivity Info	TI LI LO TS
CP0868470 Compound Info	rac-1-((1-methyl-6-(2-methyl-3-phenylpropoxy)-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H32ClNO3	1
1	EC50 = 20800 nM Bioactivity Info	TI LI LO TS
CP0375771 Compound Info	(S)-2-amino-4-(4-(heptyloxy)phenyl)-2-methylbutanoic acid Show/Hide	C18H29NO3	1
1	EC50 > 22000 nM Bioactivity Info	TI LI LO TS
CP0873010 Compound Info	rac-1-((1-methyl-6-(3-phenylbutoxy)-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C26H32ClNO3	1
1	EC50 = 22000 nM Bioactivity Info	TI LI LO TS
CP0380308 Compound Info	1-(4-(5-butylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H25NO3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0380309 Compound Info	1-(4-(5-cyclohexylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C25H27NO3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0380311 Compound Info	1-((6-(5-cyclohexylbenzofuran-2-yl)pyridin-3-yl)methyl)azetidine-3-carboxylic acid Show/Hide	C24H26N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0393723 Compound Info	1-(4-(5-(pyridin-3-yl)benzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C24H20N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0393727 Compound Info	1-((2-(5-butoxybenzofuran-2-yl)thiazol-5-yl)methyl)azetidine-3-carboxylic acid Show/Hide	C20H22N2O4S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0393732 Compound Info	1-(4-(5-cyclohexylbenzofuran-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C25H26FNO3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0398775 Compound Info	1-(4-(5-phenethylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C27H25NO3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0398778 Compound Info	1-(4-(5-(cyclopentylmethoxy)benzofuran-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C25H26FNO4	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0425181 Compound Info	1-(4-(5-butoxybenzofuran-2-yl)-3-methoxybenzyl)azetidine-3-carboxylic acid Show/Hide	C24H27NO5	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0477215 Compound Info	1-(4-(6-butoxybenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H25NO4	1
1	EC50 = 25000 nM Bioactivity Info	TI LI LO TS
CP0522161 Compound Info	1-(4-(5-phenoxybenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C25H21NO4	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0412287 Compound Info	1-(4-(5-benzylthiazolo[5,4-c]pyridin-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0412289 Compound Info	1-(4-(6-benzylthiazolo[4,5-b]pyridin-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0382585 Compound Info	1-[[3-fluoro-4-[5-(pyridin-2-ylmethyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0390590 Compound Info	1-[[3-fluoro-4-[6-(pyrrolidine-1-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C23H22FN3O3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0392730 Compound Info	1-[[3-fluoro-4-[6-(pyridin-2-ylmethyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C24H20FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0392732 Compound Info	1-[[4-[6-(azepane-1-carbonyl)-1,3-benzothiazol-2-yl]-3-fluorophenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C25H26FN3O3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0403668 Compound Info	1-[[3-fluoro-4-[6-(pyridine-2-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C24H18FN3O3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0441117 Compound Info	1-[[3-fluoro-4-[6-(piperidine-1-carbonyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C24H24FN3O3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0457178 Compound Info	1-[[3-fluoro-4-[5-(1-pyridin-2-ylethyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C25H22FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0460017 Compound Info	1-[[3-fluoro-4-[6-(1-pyridin-2-ylcyclopropyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C26H22FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0500205 Compound Info	1-[[3-fluoro-4-[6-(1-pyridin-2-ylethyl)-1,3-benzothiazol-2-yl]phenyl]methyl]azetidine-3-carboxylic acid Show/Hide	C25H22FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0391739 Compound Info	5-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]pentanoic acid Show/Hide	C26H23FN2O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0391876 Compound Info	2-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]ethanamine Show/Hide	C23H20FN3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0391878 Compound Info	3-[[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]methyl-methylamino]propanoic acid Show/Hide	C26H24FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0391879 Compound Info	4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]butanoic acid Show/Hide	C25H21FN2O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0391880 Compound Info	3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]aniline Show/Hide	C21H16FN3S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0405808 Compound Info	3-[[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]methylamino]propanoic acid Show/Hide	C25H22FN3O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0456273 Compound Info	2-(2-fluorophenyl)-5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridine Show/Hide	C21H15FN2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0457172 Compound Info	3-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]propanoic acid Show/Hide	C24H19FN2O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0457208 Compound Info	3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]benzoic acid Show/Hide	C22H15FN2O2S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0242679 Compound Info	1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]-1,6-naphthyridine-3-carboxamide Show/Hide	C23H16F3N3O2	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0385335 Compound Info	8-(2-hydroxyethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C26H21F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0385337 Compound Info	1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinoline-7-carboxylic acid Show/Hide	C25H17F3N2O4	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0385339 Compound Info	7-(hydroxymethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]-1,6-naphthyridine-3-carboxamide Show/Hide	C24H18F3N3O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0410263 Compound Info	7-(3-hydroxypropyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C27H23F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0416499 Compound Info	6-(hydroxymethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C25H19F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0433036 Compound Info	7-(hydroxymethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C25H19F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0436527 Compound Info	7-(2-hydroxyethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C26H21F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0436528 Compound Info	3-[[1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinolin-7-yl]amino]propanoic acid Show/Hide	C27H22F3N3O4	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0450696 Compound Info	8-(hydroxymethyl)-1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C25H19F3N2O3	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0450698 Compound Info	1-[[1-methyl-4-oxo-3-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]quinolin-7-yl]methyl]azetidine-3-carboxylic acid Show/Hide	C29H24F3N3O4	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0291779 Compound Info	1-(4-(5-benzylbenzofuran-2-yl)-3-fluorobenzyl)azetidine-3-carboxylic acid Show/Hide	C26H22FNO3	1
1	EC50 = 27000 nM Bioactivity Info	TI LI LO TS
CP0873459 Compound Info	(S)-1-((6-(2-(4-fluorobenzyl)butoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C27H33ClFNO3	1
1	EC50 = 29300 nM Bioactivity Info	TI LI LO TS
CP0373573 Compound Info	6-(cyclohexylamino)-N-(4-hydroxyphenyl)pyrimidine-4-carboxamide Show/Hide	C17H20N4O2	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0373788 Compound Info	6-(Cyclohexylamino)-N-(4-hydroxy-2-methylphenyl)pyrimidine-4-carboxamide Show/Hide	C18H22N4O2	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0390430 Compound Info	6-(cyclohexyl(cyclopropylmethyl)amino)-N-(4-hydroxy-2-methylphenyl)pyrimidine-4-carboxamide Show/Hide	C22H28N4O2	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0400300 Compound Info	6-(cyclohexylamino)-N-(2-methyl-4-sulfamoylphenyl)pyrimidine-4-carboxamide Show/Hide	C18H23N5O3S	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0469845 Compound Info	6-(cyclohexyl(cyclopropylmethyl)amino)-N-(2-methyl-4-sulfamoylphenyl)pyrimidine-4-carboxamide Show/Hide	C22H29N5O3S	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0873456 Compound Info	(R)-1-((6-(2-(4-fluorobenzyl)-3-methylbutoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C28H35ClFNO3	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0873457 Compound Info	1-((6-(2,2-dimethyl-3-phenylpropoxy)-1-methyl-3,4-dihydronaphthalen-2-yl)methyl)azetidine-3-carboxylic acid hydrochloride Show/Hide	C27H34ClNO3	1
1	EC50 > 30000 nM Bioactivity Info	TI LI LO TS
CP0882552 Compound Info	2,2,2-trifluoroacetic acid compound with 3-(6-(2-chlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid Show/Hide	C24H25ClF3NO6	1
1	EC50 > 31622.78 nM Bioactivity Info	TI LI LO TS
CP0104446 Compound Info	N-cyclohexyl-5-propyl-1,2-oxazole-3-carboxamide Show/Hide	C13H20N2O2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0210528 Compound Info	N-cyclohexyl-5-cyclopropyl-1,2-oxazole-3-carboxamide Show/Hide	C13H18N2O2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0224929 Compound Info	N-cyclohexyl-N-phenyl-5-propyl-1,2-oxazole-3-carboxamide Show/Hide	C19H24N2O2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0334413 Compound Info	N,N-dicyclohexyl-2-cyclopropyl-1,3-oxazole-4-carboxamide Show/Hide	C19H28N2O2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0338186 Compound Info	N,N-dicyclohexyl-1,2-benzoxazole-3-carboxamide Show/Hide	C20H26N2O2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0455035 Compound Info	N,N-dicyclohexyl-5-cyclopropylfuran-2-carboxamide Show/Hide	C20H29NO2	1
1	EC50 > 50000 nM Bioactivity Info	TI LI LO TS
CP0381087 Compound Info	3-[(4-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]propanoic acid Show/Hide	C22H19NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0388429 Compound Info	4-[[(4-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]methyl]benzoic acid Show/Hide	C27H21NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0388439 Compound Info	5-[(4-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]pentanoic acid Show/Hide	C24H23NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0388447 Compound Info	4-[(7-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]butanoic acid Show/Hide	C23H21NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0414869 Compound Info	1-[(5-naphthalen-2-yl-1-benzothiophen-2-yl)methyl]azetidine-3-carboxylic acid Show/Hide	C23H19NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0464445 Compound Info	4-[(4-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]butanoic acid Show/Hide	C23H21NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0464446 Compound Info	2-[(4-naphthalen-2-yl-1-benzothiophen-2-yl)methylamino]acetic acid Show/Hide	C21H17NO2S	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0372154 Compound Info	(2R,3S,5S)-2-[(hydrogen phosphonatooxy)methyl]-5-(hydroxymethyl)-3-(4-octylphenyl)pyrrolidin-1-ium Show/Hide	C20H34NO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0372156 Compound Info	(2R,3S,5S)-5-[(hydrogen phosphonatooxy)methyl]-2-(hydroxymethyl)-3-(4-octylphenyl)pyrrolidin-1-ium Show/Hide	C20H34NO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0372158 Compound Info	(2S,3R,5R)-2-[(hydrogen phosphonatooxy)methyl]-5-(hydroxymethyl)-3-(4-octylphenyl)pyrrolidin-1-ium Show/Hide	C20H34NO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0496074 Compound Info	(2S,3R,5R)-5-[(hydrogen phosphonatooxy)methyl]-2-(hydroxymethyl)-3-(4-octylphenyl)pyrrolidin-1-ium Show/Hide	C20H34NO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0876631 Compound Info	(1R,2S)-2-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)cyclopropanecarboxylic acid Show/Hide	C23H21N3O4	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0421165 Compound Info	3-(4-(5-(6-isobutylpyridin-3-yl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid Show/Hide	C21H23N3O3	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0400334 Compound Info	2-Amino-4-(4'-butoxy-3-chlorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C21H29ClNO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0428867 Compound Info	2-Amino-4-(4'-butoxy-3'-fluorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C21H29FNO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0430689 Compound Info	2-amino-4-(4'-butoxybiphenyl-4-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H30NO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0430690 Compound Info	2-amino-4-(4'-butoxy-2',5'-difluorobiphenyl-4-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H28F2NO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0430691 Compound Info	2-Amino-4-[3-chloro-2'-fluoro-4'-(4-methylphenylthio)biphenyl-4-yl]-2-(phosphoryloxymethyl)butanol Show/Hide	C24H26ClFNO5PS	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0433658 Compound Info	2-Amino-4-(3-chloro-4'-phenoxybiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C23H25ClNO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0463736 Compound Info	2-Amino-4-(4'-phenoxybiphenyl-4-yl)-2-(phosphoryloxymethyl)-butanol Show/Hide	C23H26NO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0495853 Compound Info	2-amino-4-(2-fluoro-4-pentylphenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C16H27FNO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0502881 Compound Info	2-Amino-4-(4'-butoxy-3'-chlorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C21H29ClNO6P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0506447 Compound Info	2-Amino-4-[2'-fluoro-4'-(4-methylphenylthio)biphenyl-4-yl]-2-(phosphoryloxymethyl)butanol Show/Hide	C24H27FNO5PS	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0510033 Compound Info	2-amino-4-(3-chloro-4'-pentylbiphenyl-4-yl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C22H31ClNO5P	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0510858 Compound Info	2-Amino-4-[2'-fluoro-4'-(3-methylphenylthio)biphenyl-4-yl]-2-(phosphoryloxymethyl)butanol Show/Hide	C24H27FNO5PS	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0513279 Compound Info	2-Amino-4-(4'-benzylthio-2'-fluorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C24H27FNO5PS	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0874736 Compound Info	2-Amino-4-(4'-benzylthio-3-chlorobiphenyl-4-yl)-2-(phosphoryloxymethyl)butanol Show/Hide	C25H29ClNO4PS	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0882549 Compound Info	3-(6-(2-chloro-6-ethylbenzylthio)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)propanoic acid hydrochloride Show/Hide	C24H29Cl2NO3S	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0930972 Compound Info	2-(6-(2,6-dichlorobenzyloxy)-2H-spiro[benzofuran-3,4'-piperidine]-1'-yl)acetic acid hydrochloride Show/Hide	C21H22Cl3NO4	1
1	EC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0094968 Compound Info	(2R)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]-2-methylbutanoic acid Show/Hide	C26H24FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0391877 Compound Info	3-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]propan-1-amine Show/Hide	C24H22FN3S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0392476 Compound Info	(2R)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]-4-oxobutanoic acid Show/Hide	C25H21FN4O3S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0392477 Compound Info	(2S)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]-4-oxobutanoic acid Show/Hide	C25H21FN4O3S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0392508 Compound Info	(2S)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]-2-methylbutanoic acid Show/Hide	C26H24FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0401223 Compound Info	(2R)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]butanoic acid Show/Hide	C25H22FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0456274 Compound Info	3-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]anilino]propanoic acid Show/Hide	C24H20FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0456276 Compound Info	(2S)-2-amino-4-[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]butanoic acid Show/Hide	C25H22FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0463062 Compound Info	[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]methanamine Show/Hide	C22H18FN3S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0481868 Compound Info	4-[[3-fluoro-4-[5-(1-phenylcyclopropyl)-[1,3]thiazolo[5,4-b]pyridin-2-yl]phenyl]methylamino]butanoic acid Show/Hide	C26H24FN3O2S	1
1	EC50 > 2500 nM Bioactivity Info	TI LI LO TS
CP0393726 Compound Info	1-(4-(5-benzylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C26H23NO3	1
1	EC50 > 4300 nM Bioactivity Info	TI LI LO TS
CP0848807 Compound Info	2-amino-4-(4-((4'-ethyl-[1,1'-biphenyl]-4-yl)oxy)phenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C25H30NO6P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0854262 Compound Info	2-amino-4-(4-(4-butylphenoxy)-2-chlorophenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C21H29ClNO6P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0906686 Compound Info	2-amino-4-(4-(3-(benzyloxy)phenylthio)-2-chlorophenyl)-2-(hydroxymethyl)butyl dihydrogen phosphate Show/Hide	C24H27ClNO6PS	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0380879 Compound Info	[2-amino-4-[4-[2-(furan-2-yl)-1,3-oxazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C18H21N2O7P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0380883 Compound Info	[2-amino-4-[4-[1-[(4-chlorophenyl)methyl]triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C20H24ClN4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0396852 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-[[4-(trifluoromethyl)phenyl]methyl]triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H24F3N4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0414334 Compound Info	[2-amino-4-[4-[1-(4-fluorophenyl)triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C19H22FN4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0480179 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[1-[(4-methylphenyl)methyl]triazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C21H27N4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0480181 Compound Info	[2-amino-4-[4-[1-[(4-fluorophenyl)methyl]triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C20H24FN4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0542202 Compound Info	[2-amino-2-(hydroxymethyl)-4-[4-[2-[(4-methylphenyl)methyl]-1,3-oxazol-4-yl]phenyl]butyl] dihydrogen phosphate Show/Hide	C22H27N2O6P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0542205 Compound Info	[2-amino-4-[4-[1-[(4-ethylphenyl)methyl]triazol-4-yl]phenyl]-2-(hydroxymethyl)butyl] dihydrogen phosphate Show/Hide	C22H29N4O5P	1
1	EC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0380312 Compound Info	1-(4-(5-butoxybenzofuran-2-yl)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H25NO4	1
1	EC50 > 7200 nM Bioactivity Info	TI LI LO TS
CP0409297 Compound Info	[2-amino-4-(4-octylphenyl)butyl] dihydrogen phosphate Show/Hide	C18H32NO4P	1
1	IC50 = 0.71 nM Bioactivity Info	TI LI LO TS
CP0402395 Compound Info	3-(10-phenyldecylamino)propylphosphonic acid Show/Hide	C19H34NO3P	1
1	IC50 = 0.91 nM Bioactivity Info	TI LI LO TS
CP0506943 Compound Info	3-[(4-nonoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0409210 Compound Info	3-[(3-fluoro-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H31FNO4P	1
1	IC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0414924 Compound Info	(3-Amino-13-phenyl-tridecyl)-phosphonic acid Show/Hide	C19H34NO3P	1
1	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0380620 Compound Info	(3-Pentadecylamino-propyl)-phosphonic acid Show/Hide	C18H40NO3P	1
1	IC50 = 2.7 nM Bioactivity Info	TI LI LO TS
CP0376811 Compound Info	3-[(4-nonylphenyl)methylamino]propylphosphonic acid Show/Hide	C19H34NO3P	2
1	IC50 = 2.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 3.1 nM Bioactivity Info	TI LI LO TS
CP0453571 Compound Info	(3-Tridecylamino-propyl)-phosphonic acid Show/Hide	C16H36NO3P	1
1	IC50 = 2.8 nM Bioactivity Info	TI LI LO TS
CP0406502 Compound Info	(3-Tetradecylamino-propyl)-phosphonic acid Show/Hide	C17H38NO3P	1
1	IC50 = 3.6 nM Bioactivity Info	TI LI LO TS
CP0378040 Compound Info	1,2,4-oxadiazole based compound, 22 Show/Hide	C24H27N3O3	1
1	IC50 = 3.86 nM Bioactivity Info	TI LI LO TS
CP0402450 Compound Info	3-[2-(4-octylphenyl)ethylamino]propylphosphonic acid Show/Hide	C19H34NO3P	1
1	IC50 = 4.3 nM Bioactivity Info	TI LI LO TS
CP0392505 Compound Info	[(1S,3S)-3-[(4-nonylphenyl)methylamino]cyclohexyl]phosphonic acid Show/Hide	C22H38NO3P	1
1	IC50 = 4.7 nM Bioactivity Info	TI LI LO TS
CP0453216 Compound Info	3-[(3-chloro-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H31ClNO4P	1
1	IC50 = 4.9 nM Bioactivity Info	TI LI LO TS
CP0379285 Compound Info	2-[(2R,5S)-5-tetradecylpyrrolidin-2-yl]ethylphosphonic acid Show/Hide	C20H42NO3P	1
1	IC50 = 5.2 nM Bioactivity Info	TI LI LO TS
CP0377169 Compound Info	3-[(3-methyl-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0881026 Compound Info	3-(N-alkylamino) propylphosphonic acid derivative Show/Hide	C19H36NO5P	1
1	IC50 = 6.3 nM Bioactivity Info	TI LI LO TS
CP0398427 Compound Info	[2-amino-1-hydroxy-4-(4-octylphenyl)butan-2-yl] dihydrogen phosphate Show/Hide	C18H32NO5P	1
1	IC50 = 6.3 nM Bioactivity Info	TI LI LO TS
CP0275274 Compound Info	[(2S)-2-amino-2-(hydroxymethyl)-4-(4-octylphenyl)butyl] dihydrogen phosphate Show/Hide	C19H34NO5P	1
1	IC50 = 6.3 nM Bioactivity Info	TI LI LO TS
CP0457473 Compound Info	3-[(4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H32NO4P	1
1	IC50 = 8.5 nM Bioactivity Info	TI LI LO TS
CP0445772 Compound Info	3-[methyl(tetradecyl)amino]propylphosphonic acid Show/Hide	C18H40NO3P	1
1	IC50 = 9.8 nM Bioactivity Info	TI LI LO TS
CP0418882 Compound Info	(3-Amino-hexadecyl)-phosphonic acid Show/Hide	C16H36NO3P	1
1	IC50 = 10 nM Bioactivity Info	TI LI LO TS
CP0374881 Compound Info	1,2,4-oxadiazole based compound, 26 Show/Hide	C23H25N3O3	1
1	IC50 = 12 nM Bioactivity Info	TI LI LO TS
CP0379112 Compound Info	(3-Dodecylamino-propyl)-phosphonic acid Show/Hide	C15H34NO3P	1
1	IC50 = 13 nM Bioactivity Info	TI LI LO TS
CP0453944 Compound Info	3-[(3,5-dichloro-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H30Cl2NO4P	1
1	IC50 = 13 nM Bioactivity Info	TI LI LO TS
CP0373301 Compound Info	3-[3-(4-heptylphenyl)propylamino]propylphosphonic acid Show/Hide	C19H34NO3P	1
1	IC50 = 14 nM Bioactivity Info	TI LI LO TS
CP0374689 Compound Info	(3-Amino-heptadecyl)-phosphonic acid Show/Hide	C17H38NO3P	1
1	IC50 = 14 nM Bioactivity Info	TI LI LO TS
CP0373686 Compound Info	(3-Hexadecylamino-propyl)-phosphonic acid Show/Hide	C19H42NO3P	1
1	IC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0916381 Compound Info	[Hydroxy-(1-tetradecyl-pyrrolidin-3-yl)-methyl]-phosphonic acid Show/Hide	C19H40NO4P	1
1	IC50 = 17 nM Bioactivity Info	TI LI LO TS
CP0403262 Compound Info	1-(4-nonylbenzyl)pyrrolidin-3-ylphosphonic acid Show/Hide	C20H34NO3P	2
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
2	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0863137 Compound Info	[(1S,3R)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0403977 Compound Info	[(1R,3R)-3-amino-1-hydroxy-5-(4-octylphenyl)pentyl]phosphonic acid Show/Hide	C19H34NO4P	2
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
2	IC50 = 85 nM Bioactivity Info	TI LI LO TS
CP0393499 Compound Info	(3-Hydroxy-1-tetradecyl-pyrrolidin-3-yl)-phosphonic acid Show/Hide	C18H38NO4P	1
1	IC50 = 19 nM Bioactivity Info	TI LI LO TS
CP0431648 Compound Info	3-[(4-octylphenyl)methylamino]propylphosphonic acid Show/Hide	C18H32NO3P	1
1	IC50 = 21 nM Bioactivity Info	TI LI LO TS
CP0404437 Compound Info	3-[(3-bromo-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H31BrNO4P	1
1	IC50 = 26 nM Bioactivity Info	TI LI LO TS
CP0393677 Compound Info	(3-Amino-pentadecyl)-phosphonic acid Show/Hide	C15H34NO3P	1
1	IC50 = 40 nM Bioactivity Info	TI LI LO TS
CP0453952 Compound Info	3-[(3,5-dimethyl-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C20H36NO4P	1
1	IC50 = 44 nM Bioactivity Info	TI LI LO TS
CP0498260 Compound Info	3-[[4-(5-heptyl-1,2,4-oxadiazol-3-yl)phenyl]methylamino]propylphosphonic acid Show/Hide	C19H30N3O4P	1
1	IC50 = 46 nM Bioactivity Info	TI LI LO TS
CP0373279 Compound Info	(3-Amino-octadecyl)-phosphonic acid Show/Hide	C18H40NO3P	1
1	IC50 = 47 nM Bioactivity Info	TI LI LO TS
CP0464605 Compound Info	(4-Hydroxy-1-tetradecyl-piperidin-4-yl)-methyl-phosphinic acid Show/Hide	C20H42NO3P	1
1	IC50 = 51 nM Bioactivity Info	TI LI LO TS
CP0448991 Compound Info	3-[[4-(2-heptyltetrazol-5-yl)phenyl]methylamino]propylphosphonic acid Show/Hide	C18H30N5O3P	1
1	IC50 = 55 nM Bioactivity Info	TI LI LO TS
CP0848005 Compound Info	[3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 62 nM Bioactivity Info	TI LI LO TS
CP0868637 Compound Info	[3-Amino-2-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 68 nM Bioactivity Info	TI LI LO TS
CP0463921 Compound Info	3-[(3-ethoxy-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C20H36NO5P	1
1	IC50 = 74 nM Bioactivity Info	TI LI LO TS
CP0434360 Compound Info	3-[(3,5-dibromo-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H30Br2NO4P	1
1	IC50 = 94 nM Bioactivity Info	TI LI LO TS
CP0453956 Compound Info	3-[(3-methoxy-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C19H34NO5P	1
1	IC50 = 99 nM Bioactivity Info	TI LI LO TS
CP0430984 Compound Info	3-[[4-(1-hydroxynonyl)phenyl]methylamino]propylphosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0437625 Compound Info	3-[(3-hydroxy-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H32NO5P	1
1	IC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0403972 Compound Info	(3-Amino-henicosyl)-phosphonic acid Show/Hide	C21H46NO3P	1
1	IC50 = 130 nM Bioactivity Info	TI LI LO TS
CP0413075 Compound Info	3-Hydroxy-4-(4-nonyl-benzylamino)-butyric acid Show/Hide	C20H33NO3	1
1	IC50 = 170 nM Bioactivity Info	TI LI LO TS
CP0419093 Compound Info	methyl-[3-[(4-nonylphenyl)methylamino]propyl]phosphinic acid Show/Hide	C20H36NO2P	1
1	IC50 = 170 nM Bioactivity Info	TI LI LO TS
CP0404436 Compound Info	3-[[4-(4-hexylphenyl)phenyl]methylamino]propylphosphonic acid Show/Hide	C22H32NO3P	1
1	IC50 = 180 nM Bioactivity Info	TI LI LO TS
CP0393495 Compound Info	2-(1-tetradecylpyrrolidin-2-yl)ethylphosphonic acid Show/Hide	C20H42NO3P	1
1	IC50 = 190 nM Bioactivity Info	TI LI LO TS
CP0492236 Compound Info	3-[(3-bromo-4-decoxy-5-methoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C21H37BrNO5P	1
1	IC50 = 200 nM Bioactivity Info	TI LI LO TS
CP0379286 Compound Info	(2-Tetradecylamino-cyclohexylmethyl)-phosphonic acid Show/Hide	C21H44NO3P	1
1	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0433608 Compound Info	(4-Hydroxy-2-tetradecyl-piperidin-4-yl)-methyl-phosphinic acid Show/Hide	C20H42NO3P	1
1	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0382451 Compound Info	3-[(4-nonanoylphenyl)methylamino]propylphosphonic acid Show/Hide	C19H32NO4P	1
1	IC50 = 260 nM Bioactivity Info	TI LI LO TS
CP0393661 Compound Info	[3-amino-5-(4-octylphenyl)pentyl]phosphonic acid Show/Hide	C19H34NO3P	1
1	IC50 = 280 nM Bioactivity Info	TI LI LO TS
CP0409209 Compound Info	4-[(3-Phosphono-propylamino)-methyl]-benzoic acid heptyl ester Show/Hide	C18H30NO5P	1
1	IC50 = 280 nM Bioactivity Info	TI LI LO TS
CP0850212 Compound Info	[(1R,3S)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 320 nM Bioactivity Info	TI LI LO TS
CP0860724 Compound Info	[(1S,3S)-3-Amino-1-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid Show/Hide	C19H34NO4P	1
1	IC50 = 320 nM Bioactivity Info	TI LI LO TS
CP0447807 Compound Info	3-Fluoro-4-(4-nonyl-benzylamino)-butyric acid Show/Hide	C20H32FNO2	1
1	IC50 = 350 nM Bioactivity Info	TI LI LO TS
CP0379287 Compound Info	(3-Tetradecylamino-cyclopentyl)-phosphonic acid Show/Hide	C19H40NO3P	1
1	IC50 = 370 nM Bioactivity Info	TI LI LO TS
CP0384390 Compound Info	2-Hydroxy-4-(4-nonyl-benzylamino)-butyric acid Show/Hide	C20H33NO3	1
1	IC50 = 370 nM Bioactivity Info	TI LI LO TS
CP0404002 Compound Info	2,2-Difluoro-4-(4-nonyl-benzylamino)-butyric acid Show/Hide	C20H31F2NO2	1
1	IC50 = 390 nM Bioactivity Info	TI LI LO TS
CP0485396 Compound Info	3-(2-tridecylpiperidin-1-yl)propylphosphonic acid Show/Hide	C21H44NO3P	1
1	IC50 = 410 nM Bioactivity Info	TI LI LO TS
CP0404466 Compound Info	3-[(3-bromo-5-methoxy-4-undecoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C22H39BrNO5P	1
1	IC50 = 430 nM Bioactivity Info	TI LI LO TS
CP0384392 Compound Info	2-(trans-5-(4-(5-(4-(4,4-difluorocyclohexyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C26H27F2N3O3	1
1	IC50 = 460 nM Bioactivity Info	TI LI LO TS
CP0478347 Compound Info	[3-amino-3-(hydroxymethyl)-5-(4-octylphenyl)pentyl]phosphonic acid Show/Hide	C20H36NO4P	1
1	IC50 = 510 nM Bioactivity Info	TI LI LO TS
CP0384362 Compound Info	1-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H20F3NO3S	1
1	IC50 = 530 nM Bioactivity Info	TI LI LO TS
CP0391327 Compound Info	3-[(3-chloro-5-methoxy-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C19H33ClNO5P	1
1	IC50 = 610 nM Bioactivity Info	TI LI LO TS
CP0860694 Compound Info	[3-Amino-2-hydroxy-5-(4-octyl-phenyl)-pentyl]-phosphonic acid; compound with [(E)-3-amino-5-(4-octyl-phenyl)-pent-1-enyl]-phosphonic acid Show/Hide	C38H66N2O7P2	1
1	IC50 = 720 nM Bioactivity Info	TI LI LO TS
CP0389839 Compound Info	3-[(3-bromo-5-methoxy-4-nonoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C20H35BrNO5P	1
1	IC50 = 830 nM Bioactivity Info	TI LI LO TS
CP0384389 Compound Info	3-[4-(4-heptylphenyl)butylamino]propylphosphonic acid Show/Hide	C20H36NO3P	1
1	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0854351 Compound Info	hydrogen (3-{[(4-nonylphenyl)methyl]amino}propyl)phosphonite Show/Hide	C19H34NO2P	1
1	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0410003 Compound Info	3-[(3-methoxy-5-methyl-4-octoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C20H36NO5P	1
1	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0428538 Compound Info	1-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)pyrrolidine-3-carboxylic acid Show/Hide	C24H22F3NO3S	1
1	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0430889 Compound Info	3-(2-tetradecylpyrrolidin-1-yl)propylphosphonic acid Show/Hide	C21H44NO3P	1
1	IC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0403608 Compound Info	4-(4-Nonyl-benzylamino)-butyric acid Show/Hide	C20H33NO2	1
1	IC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0390461 Compound Info	2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C24H27N3O3	1
1	IC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0378761 Compound Info	(+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C26H29N3O3	1
1	IC50 = 1700 nM Bioactivity Info	TI LI LO TS
CP0419853 Compound Info	1-(3-chloro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H19ClF3NO3S	1
1	IC50 = 2000 nM Bioactivity Info	TI LI LO TS
CP0384401 Compound Info	2-(5-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C24H22F3NO3S	1
1	IC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0428536 Compound Info	3-(3-bromo-5-methoxy-4-(octyloxy)benzylamino)propylphosphonic acid Show/Hide	C19H33BrNO5P	1
1	IC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0405741 Compound Info	1-(4-nonylbenzyl)pyrrolidine-3-carboxylic acid Show/Hide	C21H33NO2	1
1	IC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0419848 Compound Info	1-(3-fluoro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H19F4NO3S	1
1	IC50 = 2100 nM Bioactivity Info	TI LI LO TS
CP0378760 Compound Info	(+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopentyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C25H25F2N3O3	1
1	IC50 = 2200 nM Bioactivity Info	TI LI LO TS
CP0384397 Compound Info	2-(trans-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C26H29N3O3	1
1	IC50 = 3100 nM Bioactivity Info	TI LI LO TS
CP0391846 Compound Info	1,2,4-oxadiazole based compound, 37 Show/Hide	C24H23F2N3O3	1
1	IC50 = 4018 nM Bioactivity Info	TI LI LO TS
CP0391844 Compound Info	1,2,4-oxadiazole based compound, 36 Show/Hide	C24H23F2N3O3	1
1	IC50 = 4282 nM Bioactivity Info	TI LI LO TS
CP0405750 Compound Info	1-(3-ethyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C25H24F3NO3S	1
1	IC50 = 4300 nM Bioactivity Info	TI LI LO TS
CP0446328 Compound Info	5-(4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)phenyl)pyrrolidine-3-carboxylic acid Show/Hide	C23H20F3NO3S	1
1	IC50 = 4800 nM Bioactivity Info	TI LI LO TS
CP0419846 Compound Info	1-(4-nonylbenzyl)azetidine-3-carboxylic acid Show/Hide	C20H31NO2	1
1	IC50 = 4900 nM Bioactivity Info	TI LI LO TS
CP0872791 Compound Info	sodium 4-[(4-butoxyphenyl)thio]-20-[1-hydroxy-4-[(5-hydroxyheptyl)oxy]but-2-yn-1-yl]biphenyl-3-sulfonate Show/Hide	C33H39NaO7S2	1
1	IC50 = 5000 nM Bioactivity Info	TI LI LO TS
CP0454272 Compound Info	4-Amino-6-(4-octyl-phenyl)-hexanoic acid Show/Hide	C20H33NO2	1
1	IC50 = 6600 nM Bioactivity Info	TI LI LO TS
CP0378774 Compound Info	(+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)propanoic acid Show/Hide	C25H29N3O3	1
1	IC50 = 6700 nM Bioactivity Info	TI LI LO TS
CP0419851 Compound Info	1-(3-methyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C24H22F3NO3S	1
1	IC50 = 7500 nM Bioactivity Info	TI LI LO TS
CP0454291 Compound Info	3-Amino-5-(4-octyl-phenyl)-pentane-1-sulfonic acid Show/Hide	C19H33NO3S	1
1	IC50 = 7600 nM Bioactivity Info	TI LI LO TS
CP0378775 Compound Info	(+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C25H26FN3O3	1
1	IC50 = 7600 nM Bioactivity Info	TI LI LO TS
CP0421389 Compound Info	3-[(3-bromo-4-hexoxy-5-methoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C17H29BrNO5P	1
1	IC50 = 8200 nM Bioactivity Info	TI LI LO TS
CP0393963 Compound Info	1,2,4-oxadiazole based compound, 24 Show/Hide	C23H25N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0393967 Compound Info	1,2,4-oxadiazole based compound, 29 Show/Hide	C22H23N3O4	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0393969 Compound Info	1,2,4-oxadiazole based compound, 30 Show/Hide	C22H21N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0431020 Compound Info	1,2,4-oxadiazole based compound, 25 Show/Hide	C25H29N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0431223 Compound Info	1,2,4-oxadiazole based compound, 34 Show/Hide	C25H21N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0446402 Compound Info	1,2,4-oxadiazole based compound, 31 Show/Hide	C23H23N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0487372 Compound Info	3-Amino-5-(4-octyl-phenyl)-pentanoic acid Show/Hide	C19H31NO2	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0453348 Compound Info	3-[(3-bromo-4-heptoxy-5-methoxyphenyl)methylamino]propylphosphonic acid Show/Hide	C18H31BrNO5P	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0378758 Compound Info	(+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidine-2-carboxylic acid Show/Hide	C23H25N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0378772 Compound Info	(+/-)-3-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)propanoic acid Show/Hide	C25H29N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0378773 Compound Info	(+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C24H27N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0424726 Compound Info	(+/-)-2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C24H27N3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0436082 Compound Info	(+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-2-yl)acetic acid Show/Hide	C25H26FN3O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0441771 Compound Info	(+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidine-2-carboxylic acid Show/Hide	C23H25N3O3	1
1	IC50 = 10000 nM Bioactivity Info	TI LI LO TS
CP0405742 Compound Info	3-(2,4-dichlorophenyl)-5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazole Show/Hide	C19H9Cl2F3N2OS	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0419845 Compound Info	3-phenyl-5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-1,2,4-oxadiazole Show/Hide	C19H11F3N2OS	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0419847 Compound Info	1-(3,5-dichloro-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H18Cl2F3NO3S	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0419849 Compound Info	1-(3-bromo-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C23H19BrF3NO3S	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0419850 Compound Info	1-(3-methoxy-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C24H22F3NO4S	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0425423 Compound Info	1-(3,5-dimethyl-4-((4-phenyl-5-(trifluoromethyl)thiophen-2-yl)methoxy)benzyl)azetidine-3-carboxylic acid Show/Hide	C25H24F3NO3S	1
1	IC50 = 10000 nM Bioactivity Info	TI LI LO TS
CP0443173 Compound Info	26-tert-butyl-13-(2,4,4-trimethylpentan-2-yl)-3,6,9,16,19,22-hexaoxatricyclo[22.3.1.0^{10,15}]octacosa-1(28),10(15),11,13,24,26-hexaene-28-carboxylic acid Show/Hide	C24H19F6NO3S	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0393962 Compound Info	1,2,4-oxadiazole based compound, 21 Show/Hide	C23H25N3O3	1
1	IC50 = 12000 nM Bioactivity Info	TI LI LO TS
CP0485409 Compound Info	1,2,4-oxadiazole based compound, 33 Show/Hide	C25H27N3O3	1
1	IC50 = 12000 nM Bioactivity Info	TI LI LO TS
CP0882743 Compound Info	sodium 4-[(4-butoxyphenyl)thio]-20-(1-hydroxytridec-2-yn-1-yl)biphenyl-3-sulfonate Show/Hide	C35H43NaO5S2	1
1	IC50 = 13000 nM Bioactivity Info	TI LI LO TS
CP0431224 Compound Info	1,2,4-oxadiazole based compound, 35 Show/Hide	C22H20F3N3O3	1
1	IC50 = 13000 nM Bioactivity Info	TI LI LO TS
CP0436128 Compound Info	1,2,4-oxadiazole based compound, 32 Show/Hide	C24H25N3O3	1
1	IC50 = 14000 nM Bioactivity Info	TI LI LO TS
CP0387271 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-4-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C29H34FN3O4	1
1	IC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0398647 Compound Info	N-[3,5-bis(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C30H34F2N2O4	1
1	IC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0398735 Compound Info	N-[3-(4-cyanophenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C31H34FN3O4	1
1	IC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0411434 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-2-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C29H34FN3O4	1
1	IC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0477277 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-3-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C29H34FN3O4	1
1	IC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0436191 Compound Info	1,2,4-oxadiazole based compound, 23 Show/Hide	C22H23N3O3	1
1	IC50 = 58000 nM Bioactivity Info	TI LI LO TS
CP0306592 Compound Info	5-(4-phenyl-5-(trifluoromethyl)thiophen-2-yl)-3-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazole Show/Hide	C20H10F6N2OS	1
1	IC50 > 10 nM Bioactivity Info	TI LI LO TS
CP0393959 Compound Info	1,3,4-oxadiazole based compound, 9 Show/Hide	C23H25N3O3	1
1	IC50 > 10 nM Bioactivity Info	TI LI LO TS
CP0456422 Compound Info	1,2,4-oxadiazole based compound, 13 Show/Hide	C23H25N3O3	1
1	IC50 > 10 nM Bioactivity Info	TI LI LO TS
CP0355224 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-[4-(methylcarbamoyl)phenoxy]phenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C32H38FN3O5	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0375037 Compound Info	N-[3-(4-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C31H36FN3O5	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0379497 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-sulfamoylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C30H36FN3O6S	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0387270 Compound Info	N-[3-(3-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C31H36FN3O5	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0388589 Compound Info	N-[3-[4-(dimethylcarbamoyl)phenoxy]-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C33H40FN3O5	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0398734 Compound Info	N-[3-(2-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide Show/Hide	C31H36FN3O5	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0411436 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-methylsulfonylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C31H37FN2O6S	1
1	IC50 > 800 nM Bioactivity Info	TI LI LO TS
CP0384395 Compound Info	2-(trans-5-(4-(5-(4-(3,3,3-trifluoropropyl)phenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C23H22F3N3O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0384399 Compound Info	2-(trans-5-(4-(5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C25H27N3O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0384400 Compound Info	2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)phenyl)pyrrolidin-3-yl)acetic acid Show/Hide	C24H27N3O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0485046 Compound Info	1,2,4-oxadiazole based compound, 28 Show/Hide	C21H21N3O4	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0496784 Compound Info	1,3,4-oxadiazole based compound, 5 Show/Hide	C18H19N3O	1
1	IC50 > 5000 nM Bioactivity Info	TI LI LO TS
CP0431023 Compound Info	1,2,4-oxadiazole based compound, 27 Show/Hide	C24H27N3O3	1
1	IC50 ~ 10000 nM Bioactivity Info	TI LI LO TS

Cell Line ID: CL000064 , Chem-1

Cell Line Info

Cell Line ID: CL000026 , CHO-K1

Cell Line Info

Cell Line ID: CL001050 , EDG3-Ga15-bla HEK293T

Cell Line Info

Cell Line ID: CL000025 , HEK-293T

Cell Line Info

Cell Line ID: CL000006 , HEK293

Cell Line Info

Cell Line ID: CL000436 , PathHunter CHO-K1 EDG1 beta-arrestin

Cell Line Info

Cell Line ID: CL000194 , RBL-1

Cell Line Info

Cell Line ID: CL000043 , U2OS

Cell Line Info

Biochemical Assays

Compound ID	Compound Name	Compound Formula
CP0047332 Compound Info	[2-azaniumyl-2-(hydroxymethyl)-4-(4-octylphenyl)butyl] hydrogen phosphate Show/Hide	C19H34NO5P	3
1	EC50 = 2 nM
2	EC50 = 3.57 nM
3	EC50 = 13.6 nM
CP0084726 Compound Info	2-(4-octylphenethyl)-2-aminopropane-1,3-diol Show/Hide	C19H33NO2	1
1	EC50 = 3 nM
CP0014534 Compound Info	(2S,3R,4E)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate Show/Hide	C18H38NO5P	3
1	EC50 = 8.7 nM
2	IC50 = 0.4 nM
3	IC50 = 0.66 nM
CP0405884 Compound Info	1-methyl-4-oxo-N-[4-phenyl-3-(trifluoromethyl)phenyl]quinoline-3-carboxamide Show/Hide	C24H17F3N2O2	1
1	EC50 = 1500 nM
CP0096517 Compound Info	2-amino-2-[2-[4-[4-(2-ethyl-1,3-oxazol-4-yl)phenyl]phenyl]ethyl]propane-1,3-diol;hydrochloride Show/Hide	C22H27ClN2O3	1
1	EC50 > 10000 nM
CP0362401 Compound Info	1-[[4-ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]thiophen-2-yl]methyl]azetidine-3-carboxylic acid Show/Hide	C25H23N3O4S	1
1	EC50 > 20000 nM
CP0070558 Compound Info	(R)-2-amino-2-(4-(4-(biphenyl-4-ylmethoxy)phenyl)-1H-imidazol-2-yl)propyl dihydrogen phosphate Show/Hide	C25H26N3O5P	1
1	IC50 = 20 nM
CP0163457 Compound Info	(S)-2-amino-3-(4-(2-(biphenyl-4-yl)ethoxy)phenylamino)-2-methyl-3-oxopropyl dihydrogen phosphate Show/Hide	C24H27N2O6P	1
1	IC50 = 200 nM
CP0387271 Compound Info	4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-4-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide Show/Hide	C29H34FN3O4	1
1	Kd > 100 nM
CP0409055 Compound Info	2-[4-[3-(4-fluorophenoxy)-5-[[3-hydroxy-3-(2-methylpropyl)pyrrolidine-1-carbonyl]amino]phenoxy]phenyl]-2-methylpropanoic acid Show/Hide	C31H35FN2O6	1
1	Kd > 100 nM

Clinical Information about the Protein

Target 1 ( Sphingosine-1-phosphate receptor 3 (S1PR3) )

Target Type	Patented-recorded Target

Cite

About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han