General Information of the Cell Line
Cell Line ID
CL000194
Cell Line Name
RBL-1
Synonyms
RBL 1
RBL-I
RBL
Rat Basophilic Leukemia-1
Category
Cancer cell line
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_0496
Tissue Information
Peripheral blood
Disease
Rat leukemia (NCIt: C60428)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT03816, C-C chemokine receptor type 8
Compound ID Compound Name Compound Formula
CP0215421
(5R)-3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C27H28N4O3
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0922180
3-(1-((1H-indol-2-yl)methyl)piperidin-4-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C27H28N4O3
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0495739
3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-(6-methoxy-1,5-naphthyridin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C26H27N5O3
 1
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
CP0112269
3-[1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C27H31N3O3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0510945
3-[1-[(4-bromophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H26BrN3O3
 1
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
CP0510944
3-[1-[(3,4-dichlorophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H25Cl2N3O3
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0551871
5-(6-methoxyquinolin-4-yl)-3-[1-(3-phenylpropyl)piperidin-4-yl]-1,3-oxazolidin-2-one
   Show/Hide
C27H31N3O3
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0428072
3-(1-hexylpiperidin-4-yl)-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C24H33N3O3
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0449767
3-[1-[(4-chlorophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H26ClN3O3
 1
1
IC50 = 630.96 nM
   TI
   LI
   LO
   TS
CP0409484
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C27H27N3O3S
 1
1
IC50 = 794.33 nM
   TI
   LI
   LO
   TS
CP0464301
3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-quinolin-4-yl-1,3-oxazolidin-2-one
   Show/Hide
C26H26N4O2
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0434488
3-[1-[(4-methoxyphenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C26H29N3O4
 1
1
IC50 = 1258.93 nM
   TI
   LI
   LO
   TS
CP0510947
5-(6-methoxyquinolin-4-yl)-3-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-1,3-oxazolidin-2-one
   Show/Hide
C29H29N3O3
 1
1
IC50 = 1258.93 nM
   TI
   LI
   LO
   TS
CP0551872
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C27H27N3O4
 1
1
IC50 = 1258.93 nM
   TI
   LI
   LO
   TS
CP0551870
3-[3-(1H-indol-2-ylmethylamino)propyl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H26N4O3
 1
1
IC50 = 1584.89 nM
   TI
   LI
   LO
   TS
CP0464300
5-(6-methoxyquinolin-4-yl)-3-[1-[(1-methylindol-2-yl)methyl]piperidin-4-yl]-1,3-oxazolidin-2-one
   Show/Hide
C28H30N4O3
 1
1
IC50 = 3162.28 nM
   TI
   LI
   LO
   TS
CP0526481
5-(6-methoxyquinolin-4-yl)-3-[1-(quinolin-2-ylmethyl)piperidin-4-yl]-1,3-oxazolidin-2-one
   Show/Hide
C28H28N4O3
 1
1
IC50 = 3162.28 nM
   TI
   LI
   LO
   TS
CP0526480
3-[1-(3,4-dichlorobenzoyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H23Cl2N3O4
 1
1
IC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0542191
3-[1-[(3-chlorophenyl)methyl]piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H26ClN3O3
 1
1
IC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0551873
3-[3-[1H-indol-2-ylmethyl(methyl)amino]propyl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C26H28N4O3
 1
1
IC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0510946
3-[1-(cyclohexylmethyl)piperidin-4-yl]-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H33N3O3
 1
1
IC50 = 7943.28 nM
   TI
   LI
   LO
   TS
CP0408027
4-[[4-[5-(6-methoxyquinolin-4-yl)-2-oxo-1,3-oxazolidin-3-yl]piperidin-1-yl]methyl]benzonitrile
   Show/Hide
C26H26N4O3
 1
1
IC50 = 12589.25 nM
   TI
   LI
   LO
   TS
CP0495738
3-(1-benzylpiperidin-4-yl)-5-(6-methoxyquinolin-4-yl)-1,3-oxazolidin-2-one
   Show/Hide
C25H27N3O3
 1
1
IC50 = 12589.25 nM
   TI
   LI
   LO
   TS
CP0876820
3-(1-((1H-indol-3-yl)methyl)piperidin-4-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C27H28N4O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0897623
3-(1-((1H-indol-2-yl)methyl)piperidin-4-yl)-5-(naphthalen-1-yl)oxazolidin-2-one
   Show/Hide
C27H27N3O2
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0897625
3-((1-((1H-indol-2-yl)methyl)piperidin-4-yl)methyl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C28H30N4O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0897811
3-(1-((1H-indol-2-yl)methyl)piperidin-4-yl)-5-(quinolin-3-yl)oxazolidin-2-one
   Show/Hide
C26H26N4O2
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0915883
3-(1-(3,4-dichlorophenylsulfonyl)piperidin-4-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C24H23Cl2N3O5S
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0922178
3-(1-((1H-indol-2-yl)methyl)piperidin-4-yl)-5-(quinolin-2-yl)oxazolidin-2-one
   Show/Hide
C26H26N4O2
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0922179
3-(1-((1H-indol-2-yl)methyl)pyrrolidin-3-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C26H26N4O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0933849
3-(1-((1H-indol-2-yl)methyl)azepan-3-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C28H30N4O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0939746
3-(1-biphenyl-4-ylmethyl-piperidin-4-yl)-5-(6-methoxy-quinolin-4-yl)-oxazolidin-2-one
   Show/Hide
C31H31N3O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0939791
3-(1-(2-chlorobenzyl)piperidin-4-yl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C25H26ClN3O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0955403
5-(6-methoxyquinolin-4-yl)-3-(1-methylpiperidin-4-yl)oxazolidin-2-one
   Show/Hide
C19H23N3O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0955404
3-(1-((1H-indol-2-yl)methyl)piperidin-4-yl)-5-(pyridin-4-yl)oxazolidin-2-one
   Show/Hide
C22H24N4O2
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
CP0955405
3-((1-((1H-indol-2-yl)methyl)piperidin-3-yl)methyl)-5-(6-methoxyquinolin-4-yl)oxazolidin-2-one
   Show/Hide
C28H30N4O3
 1
1
IC50 < 50118.72 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Peripheral blood)
Cell Line Name Organism Disease
SET-2 Homo sapiens (Human) Adult acute megakaryoblastic leukemia
Mono-Mac-6 Homo sapiens (Human) Adult acute monocytic leukemia
HL-60 Homo sapiens (Human) Adult acute myeloid leukemia
MOLM-13 Homo sapiens (Human) Adult acute myeloid leukemia
OCI-AML-2 Homo sapiens (Human) Adult acute myeloid leukemia
HL-60/ADR Homo sapiens (Human) Adult acute myeloid leukemia
MOLM-14 Homo sapiens (Human) Adult acute myeloid leukemia
HL60/MDR Homo sapiens (Human) Adult acute myeloid leukemia
HL60/MRP Homo sapiens (Human) Adult acute myeloid leukemia
NALM-6 Homo sapiens (Human) Adult B acute lymphoblastic leukemia
MOLT-4 Homo sapiens (Human) Adult T acute lymphoblastic leukemia
MOLT-4/CCR5 Homo sapiens (Human) Adult T acute lymphoblastic leukemia
Karpas-299 Homo sapiens (Human) Anaplastic large cell lymphoma, ALK-positive
M-07e Homo sapiens (Human) Childhood acute megakaryoblastic leukemia
THP-1 Homo sapiens (Human) Childhood acute monocytic leukemia
MV4-11 Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Dual Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Dual KO-STING Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Blue ISG Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-ASC-GFP Homo sapiens (Human) Childhood acute monocytic leukemia
PMNL Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Xblue Homo sapiens (Human) Childhood acute monocytic leukemia
SEM Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
SEMK2 Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
Reh Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
Jurkat Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
Jurkat E6.1 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF-CEM Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF/VCR1000 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM/VLB100 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM/VLB500 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM-SS Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
HPB-ALL Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF-SB Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM-T4 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
J-Lat 10.6 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
12D7-MDR1 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
MDR CCRF vcr1000 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
FGS7 Jurkat Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
EoL-1 Homo sapiens (Human) Chronic eosinophilic leukemia, not otherwise specified
CII Homo sapiens (Human) Chronic lymphocytic leukemia
Ku812 Homo sapiens (Human) Chronic myelogenous leukemia, BCR-ABL1 positive
Ri-1 Homo sapiens (Human) Diffuse large B-cell lymphoma activated B-cell type
Daudi Homo sapiens (Human) EBV-related Burkitt lymphoma
HEL Homo sapiens (Human) Erythroleukemia
UKE-1 Homo sapiens (Human) Essential thrombocythemia
L-1236 Homo sapiens (Human) Hodgkin lymphoma
Granta-519 Homo sapiens (Human) Mantle cell lymphoma
JeKo-1 Homo sapiens (Human) Mantle cell lymphoma
Mino Homo sapiens (Human) Mantle cell lymphoma
HMC-1 Homo sapiens (Human) Mast cell leukemia
NK-92 Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
NK Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
KHYG-1 Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
RPMI-8226 Homo sapiens (Human) Plasma cell myeloma
OPM-2 Homo sapiens (Human) Plasma cell myeloma
U266B1 Homo sapiens (Human) Plasma cell myeloma
KMS-18 Homo sapiens (Human) Plasma cell myeloma
MM1.S Homo sapiens (Human) Plasma cell myeloma
MM1.R Homo sapiens (Human) Plasma cell myeloma
OPM-1 Homo sapiens (Human) Plasma cell myeloma
RPMI-8226/Dox40 Homo sapiens (Human) Plasma cell myeloma
HuT 78 Homo sapiens (Human) Sezary syndrome
H9 Homo sapiens (Human) Sezary syndrome
CREM010i-SS9-1 Homo sapiens (Human) Sickle cell disease
RBL-2H3 Rattus norvegicus (Rat) Rat leukemia
LCL Orang Asli K28 Homo sapiens (Human) -
JY Homo sapiens (Human) -
C.M.L. Homo sapiens (Human) -
BON Homo sapiens (Human) -
PBMC iPSC #1 Homo sapiens (Human) -
LCL 721 Homo sapiens (Human) -