General Information of the Cell Line
Cell Line ID
CL000828
Cell Line Name
HL60/MDR
Category
Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0002
Tissue Information
Peripheral blood
Disease
Adult acute myeloid leukemia (NCIt: C9154)
Acute myeloid leukemia (ORDO: Orphanet_519)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT01546, ATP-dependent translocase ABCB1
Compound ID Compound Name Compound Formula
CP0514373
3'',5''-dimethoxy-[1,1';2',1'']-terphenyl-4-ol
   Show/Hide
C20H18O3
 2
1
AC50 = 24000 nM
   TI
   LI
   LO
   TS
2
IC50 = 28000 nM
   TI
   LI
   LO
   TS
CP0436560
3'',5''-dimethoxy-[1,1';4,1'']-terphenyl-4-ol
   Show/Hide
C20H18O3
 2
1
AC50 = 32000 nM
   TI
   LI
   LO
   TS
2
IC50 = 23000 nM
   TI
   LI
   LO
   TS
CP0451875
6-(3,5-dimethoxy-phenyl)-naphthalen-2-ol
   Show/Hide
C18H16O3
 2
1
AC50 = 33000 nM
   TI
   LI
   LO
   TS
2
IC50 = 16000 nM
   TI
   LI
   LO
   TS
CP0514372
5-[2-(4-hydroxyphenyl)phenyl]benzene-1,3-diol
   Show/Hide
C18H14O3
 2
1
AC50 = 40000 nM
   TI
   LI
   LO
   TS
2
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0451790
4,3'',5''-trimethoxy-[1,1';2',1'']-terphenyl
   Show/Hide
C21H20O3
 2
1
AC50 = 48000 nM
   TI
   LI
   LO
   TS
2
IC50 = 16000 nM
   TI
   LI
   LO
   TS
CP0486929
3'',5''-dimethoxy-[1,1';3',1'']-terphenyl-4-ol
   Show/Hide
C20H18O3
 2
1
AC50 = 48000 nM
   TI
   LI
   LO
   TS
2
IC50 = 20000 nM
   TI
   LI
   LO
   TS
CP0274708
1,3-dimethoxy-5-[(E)-2-(4-methoxyphenyl)ethenyl]benzene
   Show/Hide
C17H18O3
 2
1
AC50 = 50000 nM
   TI
   LI
   LO
   TS
2
IC50 = 8000 nM
   TI
   LI
   LO
   TS
CP0436915
5-[4-(4-hydroxyphenyl)phenyl]benzene-1,3-diol
   Show/Hide
C18H14O3
 2
1
AC50 = 60000 nM
   TI
   LI
   LO
   TS
2
IC50 = 23000 nM
   TI
   LI
   LO
   TS
CP0408205
2-[(E)-2-(3,5-dimethoxyphenyl)vinyl]-6-methoxyphenol
   Show/Hide
C17H18O4
 2
1
AC50 = 82000 nM
   TI
   LI
   LO
   TS
2
IC50 = 34000 nM
   TI
   LI
   LO
   TS
CP0124683
(E)-4-(3,5-dimethoxystyryl)phenol
   Show/Hide
C16H16O3
 2
1
AC50 = 85000 nM
   TI
   LI
   LO
   TS
2
IC50 = 42000 nM
   TI
   LI
   LO
   TS
CP0340894
5-(6-Hydroxy-naphthalen-2-yl)-benzene-1,3-diol
   Show/Hide
C16H12O3
 2
1
AC50 = 92000 nM
   TI
   LI
   LO
   TS
2
IC50 = 53000 nM
   TI
   LI
   LO
   TS
CP0376091
5-[(E)-2-(3,5-dimethoxy-phenyl)-vinyl]-2-ethoxy-phenol
   Show/Hide
C18H20O4
 2
1
AC50 = 98000 nM
   TI
   LI
   LO
   TS
2
IC50 = 42000 nM
   TI
   LI
   LO
   TS
CP0041805
(E)-resveratrol
   Show/Hide
C14H12O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 = 60000 nM
   TI
   LI
   LO
   TS
CP0376089
2-(3,5-Dimethoxy-phenyl)-6-methoxy-naphthalene
   Show/Hide
C19H18O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376090
4-[(E)-2-(3,5-dimethoxy-phenyl)-vinyl]-2,6-dimethoxy-phenol
   Show/Hide
C18H20O5
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376092
2-[(E)-2-(3,5-dimethoxy-phenyl)-vinyl]-phenol
   Show/Hide
C16H16O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 = 68000 nM
   TI
   LI
   LO
   TS
CP0419733
4,3'',5''-trimethoxy-[1,1';3',1'']-terphenyl
   Show/Hide
C21H20O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 = 80000 nM
   TI
   LI
   LO
   TS
CP0436561
2,6-di-tert-butyl-4-[(E)-2-(3,5-dimethoxy-phenyl)-vinyl]-phenol
   Show/Hide
C24H32O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0441875
5-[3-(4-hydroxyphenyl)phenyl]benzene-1,3-diol
   Show/Hide
C18H14O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 = 58000 nM
   TI
   LI
   LO
   TS
CP0441876
3-[(E)-2-(3,5-Dimethoxy-phenyl)-vinyl]-phenol
   Show/Hide
C16H16O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0455669
4,3'',5''-trimethoxy-[1,1';4',1'']-terphenyl
   Show/Hide
C21H20O3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0526033
4-chloro-2-[(E)-2-(3,5-dimethoxy-phenyl)-vinyl]-phenol
   Show/Hide
C16H15ClO3
 2
1
AC50 > 100000 nM
   TI
   LI
   LO
   TS
2
IC50 = 73000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Peripheral blood)
Cell Line Name Organism Disease
SET-2 Homo sapiens (Human) Adult acute megakaryoblastic leukemia
Mono-Mac-6 Homo sapiens (Human) Adult acute monocytic leukemia
HL-60 Homo sapiens (Human) Adult acute myeloid leukemia
MOLM-13 Homo sapiens (Human) Adult acute myeloid leukemia
OCI-AML-2 Homo sapiens (Human) Adult acute myeloid leukemia
HL-60/ADR Homo sapiens (Human) Adult acute myeloid leukemia
MOLM-14 Homo sapiens (Human) Adult acute myeloid leukemia
HL60/MRP Homo sapiens (Human) Adult acute myeloid leukemia
NALM-6 Homo sapiens (Human) Adult B acute lymphoblastic leukemia
MOLT-4 Homo sapiens (Human) Adult T acute lymphoblastic leukemia
MOLT-4/CCR5 Homo sapiens (Human) Adult T acute lymphoblastic leukemia
Karpas-299 Homo sapiens (Human) Anaplastic large cell lymphoma, ALK-positive
M-07e Homo sapiens (Human) Childhood acute megakaryoblastic leukemia
THP-1 Homo sapiens (Human) Childhood acute monocytic leukemia
MV4-11 Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Dual Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Dual KO-STING Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Blue ISG Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-ASC-GFP Homo sapiens (Human) Childhood acute monocytic leukemia
PMNL Homo sapiens (Human) Childhood acute monocytic leukemia
THP1-Xblue Homo sapiens (Human) Childhood acute monocytic leukemia
SEM Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
SEMK2 Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
Reh Homo sapiens (Human) Childhood B acute lymphoblastic leukemia
Jurkat Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
Jurkat E6.1 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF-CEM Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF/VCR1000 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM/VLB100 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM/VLB500 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM-SS Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
HPB-ALL Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CCRF-SB Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
CEM-T4 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
J-Lat 10.6 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
12D7-MDR1 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
MDR CCRF vcr1000 Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
FGS7 Jurkat Homo sapiens (Human) Childhood T acute lymphoblastic leukemia
EoL-1 Homo sapiens (Human) Chronic eosinophilic leukemia, not otherwise specified
CII Homo sapiens (Human) Chronic lymphocytic leukemia
Ku812 Homo sapiens (Human) Chronic myelogenous leukemia, BCR-ABL1 positive
Ri-1 Homo sapiens (Human) Diffuse large B-cell lymphoma activated B-cell type
Daudi Homo sapiens (Human) EBV-related Burkitt lymphoma
HEL Homo sapiens (Human) Erythroleukemia
UKE-1 Homo sapiens (Human) Essential thrombocythemia
L-1236 Homo sapiens (Human) Hodgkin lymphoma
Granta-519 Homo sapiens (Human) Mantle cell lymphoma
JeKo-1 Homo sapiens (Human) Mantle cell lymphoma
Mino Homo sapiens (Human) Mantle cell lymphoma
HMC-1 Homo sapiens (Human) Mast cell leukemia
NK-92 Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
NK Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
KHYG-1 Homo sapiens (Human) Natural killer cell lymphoblastic leukemia/lymphoma
RPMI-8226 Homo sapiens (Human) Plasma cell myeloma
OPM-2 Homo sapiens (Human) Plasma cell myeloma
U266B1 Homo sapiens (Human) Plasma cell myeloma
KMS-18 Homo sapiens (Human) Plasma cell myeloma
MM1.S Homo sapiens (Human) Plasma cell myeloma
MM1.R Homo sapiens (Human) Plasma cell myeloma
OPM-1 Homo sapiens (Human) Plasma cell myeloma
RPMI-8226/Dox40 Homo sapiens (Human) Plasma cell myeloma
HuT 78 Homo sapiens (Human) Sezary syndrome
H9 Homo sapiens (Human) Sezary syndrome
CREM010i-SS9-1 Homo sapiens (Human) Sickle cell disease
RBL-1 Rattus norvegicus (Rat) Rat leukemia
RBL-2H3 Rattus norvegicus (Rat) Rat leukemia
LCL Orang Asli K28 Homo sapiens (Human) -
JY Homo sapiens (Human) -
C.M.L. Homo sapiens (Human) -
BON Homo sapiens (Human) -
PBMC iPSC #1 Homo sapiens (Human) -
LCL 721 Homo sapiens (Human) -