Compound ID |
Compound Name |
Compound Formula |
CP0518102
|
1-[2-[3-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-hydroxypropoxy]phenyl]-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O3
|
1
|
1 |
EC50 = 6 nM
|
|
|
CP0425009
|
3-[4-(dimethylamino)phenyl]-1-[2-[2-hydroxy-3-[4-(2-methylphenyl)piperazin-1-yl]propoxy]phenyl]propan-1-one
Show/Hide
|
C31H39N3O3
|
1
|
1 |
EC50 = 13 nM
|
|
|
CP0520452
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-(4-methoxyphenyl)propan-1-one
Show/Hide
|
C30H36N2O4
|
1
|
1 |
EC50 = 14 nM
|
|
|
CP0505681
|
1-(4,5-dichloro-2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H32Cl2N2O3
|
1
|
1 |
EC50 = 17 nM
|
|
|
CP0467026
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-p-tolylpropan-1-one
Show/Hide
|
C30H36N2O3
|
1
|
1 |
EC50 = 18 nM
|
|
|
CP0503964
|
3-(4-chlorophenyl)-1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)propan-1-one
Show/Hide
|
C29H33ClN2O3
|
1
|
1 |
EC50 = 19 nM
|
|
|
CP0444392
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-5-methylphenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O3
|
1
|
1 |
EC50 = 26 nM
|
|
|
CP0444382
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O3
|
1
|
1 |
EC50 = 27 nM
|
|
|
CP0525509
|
3-(4-(dimethylamino)phenyl)-1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-4-methoxyphenyl)propan-1-one
Show/Hide
|
C32H41N3O4
|
1
|
1 |
EC50 = 40 nM
|
|
|
CP0428342
|
1-(2-(2-hydroxy-3-(4-hydroxy-4-phenylpiperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H33NO4
|
1
|
1 |
EC50 = 58 nM
|
|
|
CP0444501
|
1-(5-chloro-2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H33ClN2O3
|
1
|
1 |
EC50 = 59 nM
|
|
|
CP0654265
|
Dexniguldipine
Show/Hide
|
C36H39N3O6
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0383404
|
1-(2-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C28H31FN2O3
|
1
|
1 |
EC50 = 70 nM
|
|
|
CP0502511
|
1-(3-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O3
|
1
|
1 |
EC50 = 74 nM
|
|
|
CP0461690
|
1-(2-(2-hydroxy-3-(4-hydroxy-4-phenylpiperidin-1-yl)propoxy)phenyl)-3-(naphthalen-1-yl)propan-1-one
Show/Hide
|
C33H35NO4
|
1
|
1 |
EC50 = 75 nM
|
|
|
CP0380591
|
N-[2-[(3-acetyl-2,4,6-trimethylphenyl)methylsulfanyl]-1,3-benzothiazol-6-yl]-4-butoxybenzamide
Show/Hide
|
C30H32N2O3S2
|
1
|
1 |
EC50 = 97 nM
|
|
|
CP0502506
|
1-(5-(benzyloxy)-2-(2-hydroxy-3-(propylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C28H33NO4
|
1
|
1 |
EC50 = 110 nM
|
|
|
CP0510219
|
N-[2-[(3-acetyl-2,4,6-trimethylphenyl)methylsulfanyl]-1,3-benzothiazol-6-yl]naphthalene-1-carboxamide
Show/Hide
|
C30H26N2O2S2
|
1
|
1 |
EC50 = 110 nM
|
|
|
CP0520463
|
1-(5-(benzyloxy)-2-(3-(4-benzylpiperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C36H40N2O4
|
1
|
1 |
EC50 = 116 nM
|
|
|
CP0036382
|
CAS_52-53-9
Show/Hide
|
C27H38N2O4
|
1
|
1 |
EC50 = 120 nM
|
|
|
CP0461683
|
1-(4,5-dichloro-2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)ethanone
Show/Hide
|
C22H26Cl2N2O3
|
1
|
1 |
EC50 = 125 nM
|
|
|
CP0377384
|
1-(2-(3-(4-benzoylpiperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H32N2O4
|
1
|
1 |
EC50 = 130 nM
|
|
|
CP0377383
|
3-phenyl-1-(2-(8-(piperidin-1-yl)octyloxy)phenyl)propan-1-one
Show/Hide
|
C28H39NO2
|
1
|
1 |
EC50 = 137 nM
|
|
|
CP0475207
|
1-(3-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O3
|
1
|
1 |
EC50 = 137 nM
|
|
|
CP0405733
|
2-benzyl-4-(2-hydroxy-3-(piperidin-1-yl)propoxy)-2,3-dihydroinden-1-one
Show/Hide
|
C24H29NO3
|
1
|
1 |
EC50 = 142 nM
|
|
|
CP0502513
|
1-(2-(3-(cyclohexyl(phenyl)methylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C31H37NO3
|
1
|
1 |
EC50 = 145 nM
|
|
|
CP0520462
|
(2-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)(phenyl)methanone
Show/Hide
|
C26H27FN2O3
|
1
|
1 |
EC50 = 147 nM
|
|
|
CP0525510
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-4-methylphenyl)ethanone
Show/Hide
|
C23H30N2O3
|
1
|
1 |
EC50 = 162 nM
|
|
|
CP0475196
|
2-benzyl-7-(3-(4-(2,4-dimethylphenyl)piperazin-1-yl)-2-hydroxypropoxy)-2,3-dihydroinden-1-one
Show/Hide
|
C31H36N2O3
|
1
|
1 |
EC50 = 167 nM
|
|
|
CP0503967
|
1-[2-(2-Hydroxy-3-piperidin-1-yl-propoxy)-phenyl]-3-naphthalen-1-yl-propan-1-one
Show/Hide
|
C27H31NO3
|
1
|
1 |
EC50 = 172 nM
|
|
|
CP0521900
|
1-(5-(benzyloxy)-2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H35NO4
|
1
|
1 |
EC50 = 172 nM
|
|
|
CP0496046
|
1-(2-(1-methoxy-3-phenylpropyl)phenoxy)-3-(piperidin-1-yl)propan-2-ol
Show/Hide
|
C24H33NO3
|
1
|
1 |
EC50 = 173 nM
|
|
|
CP0552268
|
2-(4-(2-methoxyphenyl)piperazin-1-yl)-1-(3-phenethylbenzofuran-2-yl)ethanol
Show/Hide
|
C29H32N2O3
|
1
|
1 |
EC50 = 177 nM
|
|
|
CP0520470
|
1-(4-(3-(3,3-diphenylpropylamino)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
|
C26H29NO3
|
1
|
1 |
EC50 = 178 nM
|
|
|
CP0489792
|
3-phenyl-1-(2-(7-(piperidin-1-yl)heptyloxy)phenyl)propan-1-one
Show/Hide
|
C27H37NO2
|
1
|
1 |
EC50 = 179 nM
|
|
|
CP0502515
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-5-methoxyphenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O4
|
1
|
1 |
EC50 = 179 nM
|
|
|
CP0502510
|
1-(3-(3-(3,3-diphenylpropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C33H35NO3
|
1
|
1 |
EC50 = 190 nM
|
|
|
CP0444390
|
1-(2-(4-(4-(4-fluorophenyl)piperazin-1-yl)butoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H33FN2O2
|
1
|
1 |
EC50 = 192 nM
|
|
|
CP0461689
|
1-(2-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
|
C23H30N2O3
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0503966
|
3-phenyl-1-(2-(6-(piperidin-1-yl)hexyloxy)phenyl)propan-1-one
Show/Hide
|
C26H35NO2
|
1
|
1 |
EC50 = 203 nM
|
|
|
CP0501908
|
1-[2-Hydroxy-3-(4-o-tolyl-piperazin-1-yl)-propyl]-5-methyl-2-phenyl-4-(3-phenyl-propionyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
|
C33H38N4O3
|
1
|
1 |
EC50 = 210 nM
|
|
|
CP0505682
|
1-(2-(2-hydroxy-3-(2-methyl-1-phenylpropylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C28H33NO3
|
1
|
1 |
EC50 = 210 nM
|
|
|
CP0461685
|
1-{5-acetyl-2-[2-hydroxy-3-(4-o-tolyl-piperazin-1-yl)-propoxy]-4-methyl-phenyl}-ethanone
Show/Hide
|
C25H32N2O4
|
1
|
1 |
EC50 = 211 nM
|
|
|
CP0496048
|
2-benzyl-7-(2-hydroxy-3-(piperidin-1-yl)propoxy)-2,3-dihydroinden-1-one
Show/Hide
|
C24H29NO3
|
1
|
1 |
EC50 = 212 nM
|
|
|
CP0505678
|
1-(4-(4-fluorophenyl)piperazin-1-yl)-3-(2-(1-methoxy-3-phenylpropyl)phenoxy)propan-2-ol
Show/Hide
|
C29H35FN2O3
|
1
|
1 |
EC50 = 226 nM
|
|
|
CP0461688
|
1-(4-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O3
|
1
|
1 |
EC50 = 227 nM
|
|
|
CP0383406
|
1-(2-(2-hydroxy-3-(4-(2-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O4
|
1
|
1 |
EC50 = 230 nM
|
|
|
CP0522690
|
3-phenyl-1-(2-(5-(piperidin-1-yl)pentyloxy)phenyl)propan-1-one
Show/Hide
|
C25H33NO2
|
1
|
1 |
EC50 = 242 nM
|
|
|
CP0521901
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)ethanone
Show/Hide
|
C22H28N2O3
|
1
|
1 |
EC50 = 249 nM
|
|
|
CP0464357
|
1-(2-(2-hydroxy-3-(4-(4-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O4
|
1
|
1 |
EC50 = 256 nM
|
|
|
CP0444386
|
1-(2-(3-(4-benzylpiperidin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H35NO3
|
1
|
1 |
EC50 = 259 nM
|
|
|
CP0425013
|
N-[2-[(3-acetyl-2,4,6-trimethylphenyl)methylsulfanyl]-1,3-benzothiazol-6-yl]-4-tert-butylbenzamide
Show/Hide
|
C30H32N2O2S2
|
1
|
1 |
EC50 = 280 nM
|
|
|
CP0379039
|
3-(4-butan-2-ylphenyl)-2-(4-propan-2-ylphenyl)-1,2-dihydroquinazolin-4-one
Show/Hide
|
C27H30N2O
|
1
|
1 |
EC50 = 290 nM
|
|
|
CP0522692
|
1-(2-(3-(2,2-dimethyl-1-phenylpropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-ol
Show/Hide
|
C29H35NO3
|
1
|
1 |
EC50 = 292 nM
|
|
|
CP0503972
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-4-methoxyphenyl)-3-phenylpropan-1-one
Show/Hide
|
C30H36N2O4
|
1
|
1 |
EC50 = 296 nM
|
|
|
CP0552426
|
1-(2-(2-hydroxy-3-(4-hydroxy-4-phenylpiperidin-1-yl)propoxy)phenyl)propan-1-one
Show/Hide
|
C23H29NO4
|
1
|
1 |
EC50 = 299 nM
|
|
|
CP0425010
|
N-[2-[(3-acetyl-2,4,6-trimethylphenyl)methylsulfanyl]-1,3-benzothiazol-6-yl]-3-phenylpropanamide
Show/Hide
|
C28H28N2O2S2
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0505677
|
(2-(2-hydroxy-3-(4-hydroxy-4-phenylpiperidin-1-yl)propoxy)phenyl)(phenyl)methanone
Show/Hide
|
C27H29NO4
|
1
|
1 |
EC50 = 307 nM
|
|
|
CP0011846
|
1-(2-(2-hydroxy-3-(propylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C21H27NO3
|
2
|
1 |
EC50 = 320 nM
|
|
|
2 |
EC50 = 329 nM
|
|
|
CP0502516
|
1-(2-(3-phenylpropanoyl)phenoxy)-3-(piperidin-1-yl)propan-2-yl acetate
Show/Hide
|
C25H31NO4
|
1
|
1 |
EC50 = 336 nM
|
|
|
CP0522689
|
1-(2-(3-(cyclohexylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C24H31NO3
|
1
|
1 |
EC50 = 341 nM
|
|
|
CP0444384
|
1-(2-(3-(4-benzylpiperidin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
|
C23H29NO3
|
1
|
1 |
EC50 = 357 nM
|
|
|
CP0444383
|
1-(2-(3-(diisopropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C24H33NO3
|
1
|
1 |
EC50 = 377 nM
|
|
|
CP0502512
|
1-(3-acetylphenoxy)-3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propan-2-one
Show/Hide
|
C23H28N2O3
|
1
|
1 |
EC50 = 379 nM
|
|
|
CP0461686
|
1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-5-methylphenyl)ethanone
Show/Hide
|
C23H30N2O3
|
1
|
1 |
EC50 = 396 nM
|
|
|
CP0503963
|
1-(2-(2-hydroxy-3-(methyl(propyl)amino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C22H29NO3
|
1
|
1 |
EC50 = 416 nM
|
|
|
CP0502508
|
1-(3-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C23H29NO3
|
1
|
1 |
EC50 = 424 nM
|
|
|
CP0552265
|
1-(2-(1-isopropoxy-3-phenylpropyl)phenoxy)-3-(piperidin-1-yl)propan-2-ol
Show/Hide
|
C26H37NO3
|
1
|
1 |
EC50 = 460 nM
|
|
|
CP0475197
|
1-(2-(3-(diisopropylamino)-2-hydroxypropoxy)phenyl)-3-(naphthalen-1-yl)propan-1-one
Show/Hide
|
C28H35NO3
|
1
|
1 |
EC50 = 465 nM
|
|
|
CP0520469
|
1-(4-(3-(3,3-diphenylpropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C33H35NO3
|
1
|
1 |
EC50 = 505 nM
|
|
|
CP0483815
|
3-phenyl-1-(2-(4-(piperidin-1-yl)butoxy)phenyl)propan-1-one
Show/Hide
|
C24H31NO2
|
1
|
1 |
EC50 = 533 nM
|
|
|
CP0496047
|
1-(3-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)ethanone
Show/Hide
|
C22H28N2O3
|
1
|
1 |
EC50 = 537 nM
|
|
|
CP0502055
|
1-(2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C23H29NO3
|
1
|
1 |
EC50 = 599 nM
|
|
|
CP0505684
|
1-(2-(2-hydroxy-3-(4-phenylpiperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C28H32N2O3
|
1
|
1 |
EC50 = 610 nM
|
|
|
CP0432626
|
3-phenyl-1-(2-(3-(piperidin-1-yl)propoxy)phenyl)propan-1-one
Show/Hide
|
C23H29NO2
|
1
|
1 |
EC50 = 651 nM
|
|
|
CP0552406
|
1-(diisopropylamino)-3-(2-(1-methoxy-3-phenylpropyl)phenoxy)propan-2-ol
Show/Hide
|
C25H37NO3
|
1
|
1 |
EC50 = 658 nM
|
|
|
CP0498132
|
1-(2-(3-(4-benzylpiperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O3
|
1
|
1 |
EC50 = 659 nM
|
|
|
CP0520467
|
1-(2-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-ol
Show/Hide
|
C28H33FN2O3
|
1
|
1 |
EC50 = 671 nM
|
|
|
CP0502504
|
1-(2-(2-hydroxy-3-(4-(3-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C29H34N2O4
|
1
|
1 |
EC50 = 678 nM
|
|
|
CP0912172
|
(4Z)-5-methyl-4-[[4-(2-methylphenyl)piperazin-1-yl]-phenylmethylidene]-2-phenylpyrazol-3-one
Show/Hide
|
C28H28N4O
|
1
|
1 |
EC50 = 680 nM
|
|
|
CP0552266
|
1-(2-(3-(3,3-diphenylpropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C33H35NO3
|
1
|
1 |
EC50 = 717 nM
|
|
|
CP0464359
|
1-(2-(3-(3,3-diphenylpropylamino)-2-hydroxypropoxy)phenyl)-3-(naphthalen-1-yl)propan-1-one
Show/Hide
|
C37H37NO3
|
1
|
1 |
EC50 = 723 nM
|
|
|
CP0377385
|
1-(2-(2-hydroxy-3-morpholinopropoxy)phenyl)-3-(naphthalen-1-yl)propan-1-one
Show/Hide
|
C26H29NO4
|
1
|
1 |
EC50 = 730 nM
|
|
|
CP0526056
|
2-(1,3-benzodioxol-5-yl)-3-(4-tert-butylphenyl)-1,2-dihydroquinazolin-4-one
Show/Hide
|
C25H24N2O3
|
1
|
1 |
EC50 = 730 nM
|
|
|
CP0503965
|
1-(2-(3-(cyclohexa-1,5-dienyl)-1-methoxypropyl)phenoxy)-3-(3,3-diphenylpropylamino)propan-2-ol
Show/Hide
|
C34H41NO3
|
1
|
1 |
EC50 = 752 nM
|
|
|
CP0379034
|
3-(4-butan-2-ylphenyl)-2-(4-methoxyphenyl)-1,2-dihydroquinazolin-4-one
Show/Hide
|
C25H26N2O2
|
1
|
1 |
EC50 = 760 nM
|
|
|
CP0428325
|
1-(2-(3-(2,2-diphenylethylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
|
C32H33NO3
|
1
|
1 |
EC50 = 797 nM
|
|
|
CP0425011
|
2-(4-butan-2-ylphenyl)-3-(4-chlorophenyl)-1,2-dihydroquinazolin-4-one
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C24H23ClN2O
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1
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1 |
EC50 = 820 nM
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CP0522691
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1-(2-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)-5-methoxyphenyl)ethanone
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C23H30N2O4
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1
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1 |
EC50 = 859 nM
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CP0516038
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4-Benzoyl-1-[2-hydroxy-3-(4-o-tolyl-piperazin-1-yl)-propyl]-5-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one
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C31H34N4O3
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1
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1 |
EC50 = 890 nM
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CP0383408
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1-(2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-ol
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C23H31NO3
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1
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1 |
EC50 = 901 nM
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CP0428344
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1-(2-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
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C22H29NO3
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1
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1 |
EC50 = 907 nM
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CP0444385
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1-(4-(3-(diisopropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
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C24H33NO3
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1
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1 |
EC50 = 915 nM
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CP0505685
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1-(4-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
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C23H29NO3
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1
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1 |
EC50 = 972 nM
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CP0496045
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1-(2-(3-phenethylbenzofuran-2-yl)ethyl)piperidine
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C23H27NO
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1
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1 |
EC50 = 980 nM
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CP0510220
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2-(4-methoxyphenyl)-3-(4-phenoxyphenyl)-1,2-dihydroquinazolin-4-one
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C27H22N2O3
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1
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1 |
EC50 = 1000 nM
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CP0380586
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1-(2-(4-morpholinobutoxy)phenyl)-3-phenylpropan-1-one
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C23H29NO3
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1
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1 |
EC50 = 1006 nM
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CP0520464
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1-(2-(3-(diisopropylamino)-2-hydroxypropoxy)-5-hydroxyphenyl)-3-phenylpropan-1-one
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C24H33NO4
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1
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1 |
EC50 = 1036 nM
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CP0444387
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(S)-1-(3-phenethylbenzofuran-2-yl)-2-(propylamino)ethanol
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C21H25NO2
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1
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1 |
EC50 = 1059 nM
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CP0480446
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[5-[3-[di(propan-2-yl)amino]-2-hydroxypropoxy]-3-methyl-1-phenylpyrazol-4-yl]-phenylmethanone
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C26H33N3O3
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1
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1 |
EC50 = 1060 nM
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CP0483814
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(R)-1-(3-phenethylbenzofuran-2-yl)-2-(propylamino)ethanol
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C21H25NO2
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1
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1 |
EC50 = 1103 nM
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CP0475191
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1-(3-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
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C28H31FN2O3
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1
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1 |
EC50 = 1120 nM
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CP0380481
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[5-[3-[di(propan-2-yl)amino]-2-hydroxypropoxy]-1,3-dimethylpyrazol-4-yl]-phenylmethanone
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C21H31N3O3
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1
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1 |
EC50 = 1210 nM
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CP0378989
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3-(4-ethylphenyl)-2-[4-(2-methylpropoxy)phenyl]-1,2-dihydroquinazolin-4-one
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C26H28N2O2
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1
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1 |
EC50 = 1210 nM
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CP0552421
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1-(4-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
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C23H30N2O3
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1
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1 |
EC50 = 1349 nM
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CP0464358
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3-phenyl-1-(2-(2-(piperidin-1-yl)ethoxy)phenyl)propan-1-one
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C22H27NO2
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1
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1 |
EC50 = 1452 nM
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CP0541676
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4-{2-Hydroxy-3-[2-(3-phenyl-propionyl)-phenoxy]-propylamino}-benzoic acid methyl ester
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C26H27NO5
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1
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1 |
EC50 = 1536 nM
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CP0541675
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1-(4-(2-hydroxy-3-(4-o-tolylpiperazin-1-yl)propoxy)phenyl)ethanone
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C22H28N2O3
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1
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1 |
EC50 = 1550 nM
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CP0520472
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1-((3-phenethyl-2,3-dihydrobenzofuran-2-yl)methyl)piperidine
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C22H27NO
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1
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1 |
EC50 = 1619 nM
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CP0377386
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N-benzyl-N-[2-hydroxy-3-[2-(3-phenylpropanoyl)phenoxy]propyl]propanamide
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C28H31NO4
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1
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1 |
EC50 = 1649 nM
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CP0520489
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N-[2-hydroxy-3-[2-(3-phenylpropanoyl)phenoxy]propyl]-N-propylbenzamide
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C28H31NO4
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1
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1 |
EC50 = 1686 nM
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CP0502505
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1-(5-hydroxy-2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)-3-phenylpropan-1-one
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C23H29NO4
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1
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1 |
EC50 = 1727 nM
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CP0502507
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1-(2-(3-(diisopropylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-ol
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C24H35NO3
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1
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1 |
EC50 = 1741 nM
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CP0552405
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1-(2-(1-methoxy-3-phenylpropyl)phenoxy)-3-morpholinopropan-2-ol
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C23H31NO4
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1
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1 |
EC50 = 1807 nM
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CP0395443
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1-(2-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
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C21H25FN2O3
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1
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1 |
EC50 = 2087 nM
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CP0475190
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(2-(3-(diethylamino)-2-hydroxypropoxy)phenyl)(phenyl)methanone
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C20H25NO3
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1
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1 |
EC50 = 2322 nM
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CP0496050
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1-(2-(3-(dimethylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
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C20H25NO3
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1
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1 |
EC50 = 2479 nM
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CP0502509
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1-(4-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C28H31FN2O3
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1
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1 |
EC50 = 2535 nM
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CP0377387
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1-(2-(2-hydroxy-3-(4-nitrophenylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C24H24N2O5
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1
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1 |
EC50 = 2568 nM
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CP0447914
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1-(3-Butylamino-2-hydroxy-propyl)-5-methyl-2-phenyl-4-(3-phenyl-propionyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C26H33N3O3
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1
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1 |
EC50 = 2690 nM
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CP0333258
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1-(5-hydroxy-2-(2-hydroxy-3-(propylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C21H27NO4
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1
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1 |
EC50 = 3021 nM
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CP0871109
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6-amino-4-(4-(dimethylamino)phenyl)-3-p-tolyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
Show/Hide
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C22H21N5O
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1
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1 |
EC50 = 3080 nM
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CP0428324
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1-(2-(2-hydroxy-3-(4-hydroxy-4-phenylpiperidin-1-yl)propoxy)phenyl)ethanone
Show/Hide
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C22H27NO4
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1
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1 |
EC50 = 3197 nM
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CP0383409
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1-(3-(2-hydroxy-3-morpholinopropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C22H27NO4
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1
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1 |
EC50 = 3475 nM
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CP0510224
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2-butylsulfanyl-3-prop-2-enylspiro[6H-benzo[h]quinazoline-5,1'-cyclopentane]-4-one
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C23H28N2OS
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1
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1 |
EC50 = 3500 nM
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CP0552403
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1-(2-(2-hydroxy-3-morpholinopropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C22H27NO4
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1
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1 |
EC50 = 3645 nM
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CP0860235
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5-Methyl-2-phenyl-4-[3-phenyl-1-propylamino-prop-(Z)-ylidene]-2,4-dihydro-pyrazol-3-one
Show/Hide
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C22H25N3O
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1
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1 |
EC50 = 3790 nM
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CP0444388
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1-(2-(2-hydroxy-3-(piperidin-1-yl)propoxy)-5-methylphenyl)ethanone
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C17H25NO3
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1
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1 |
EC50 = 5470 nM
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CP0883234
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2-(2-chlorophenyl)-4-pyrrolidin-1-ylquinazoline
Show/Hide
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C18H16ClN3
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1
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1 |
EC50 = 5940 nM
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CP0536633
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1-(2-Hydroxy-3-propylamino-propyl)-5-methyl-2-phenyl-4-(3-phenyl-propionyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C25H31N3O3
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1
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1 |
EC50 = 6310 nM
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CP0552404
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1-(2-(2-hydroxy-3-(phenylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C24H25NO3
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1
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1 |
EC50 = 6467 nM
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CP0520473
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(3-phenethyl-2,3-dihydrobenzofuran-2-yl)(piperidin-1-yl)methanone
Show/Hide
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C22H25NO2
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1
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1 |
EC50 = 6658 nM
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CP0475192
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1-(4-(2-hydroxy-3-morpholinopropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C22H27NO4
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1
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1 |
EC50 = 6875 nM
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CP0392857
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1-(3-tert-Butylamino-2-hydroxy-propyl)-5-methyl-2-phenyl-4-(3-phenyl-propionyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C26H33N3O3
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1
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1 |
EC50 = 7760 nM
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CP0537793
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1-(3-Methyl-1-phenyl-5-propylamino-1H-pyrazol-4-yl)-3-phenyl-propan-1-one
Show/Hide
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C22H25N3O
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1
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1 |
EC50 = 8380 nM
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CP0444391
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1-(2-(2-hydroxy-3-(4-(trifluoromethyl)phenylamino)propoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C25H24F3NO3
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1
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1 |
EC50 = 8490 nM
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CP0674318
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N-(2-ethoxyphenyl)-6-methyl-4-(thiophen-2-yl)-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
Show/Hide
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C18H19N3O2S2
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1
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1 |
EC50 = 8770 nM
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CP0502514
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1-(3-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)ethanone
Show/Hide
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C16H23NO3
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1
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1 |
EC50 = 9073 nM
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CP0377382
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1-(2-(2-hydroxy-3-morpholinopropoxy)phenyl)-3-phenylpropan-1-ol
Show/Hide
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C22H29NO4
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1
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1 |
EC50 = 9540 nM
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CP0552424
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7-(2-hydroxy-3-(piperidin-1-yl)propoxy)-2-methyl-2,3-dihydroinden-1-one
Show/Hide
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C18H25NO3
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1
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1 |
EC50 = 9684 nM
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CP0405734
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1-(3-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
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C21H25FN2O3
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1
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1 |
EC50 = 10070 nM
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CP0552267
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1-(2-(3-(dibenzhydrylamino)-2-hydroxypropoxy)phenyl)-3-phenylpropan-1-one
Show/Hide
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C44H41NO3
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1
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1 |
EC50 = 10400 nM
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CP0406058
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(3-Methyl-1-phenyl-5-propylamino-1H-pyrazol-4-yl)-phenyl-methanone
Show/Hide
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C20H21N3O
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1
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1 |
EC50 = 11030 nM
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CP0552423
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4-(2-hydroxy-3-(piperidin-1-yl)propoxy)-2,3-dihydroinden-1-one
Show/Hide
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C17H23NO3
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1
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1 |
EC50 = 11190 nM
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CP0542996
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1-(3-Ethyl-benzofuran-2-yl)-2-propylamino-ethanol
Show/Hide
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C15H21NO2
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1
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1 |
EC50 = 11520 nM
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CP0519405
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1-(2-Hydroxy-3-isopropylamino-propyl)-5-methyl-2-phenyl-4-(3-phenyl-propionyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C25H31N3O3
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1
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1 |
EC50 = 11750 nM
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CP0552425
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1-(4-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-hydroxypropoxy)phenyl)ethanone
Show/Hide
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C21H25FN2O3
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1
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1 |
EC50 = 11890 nM
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CP0538354
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4-Benzoyl-1-(3-diisopropylamino-2-hydroxy-propyl)-5-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one
Show/Hide
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C26H33N3O3
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1
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1 |
EC50 = 12590 nM
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CP0525507
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1-(2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)propan-1-one
Show/Hide
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C17H25NO3
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1
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1 |
EC50 = 14310 nM
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CP0378990
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diethyl 2-[(2,4,6-trichlorophenyl)hydrazinylidene]propanedioate
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C13H13Cl3N2O4
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1
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1 |
EC50 = 17700 nM
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CP0379038
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4-tert-butyl-N-[2-(naphthalen-1-ylmethylsulfanyl)-1,3-benzothiazol-6-yl]benzamide
Show/Hide
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C29H26N2OS2
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1
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1 |
EC50 > 20000 nM
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CP0436007
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N-[4-[2-(4-methoxyphenyl)-4-oxo-1,2-dihydroquinazolin-3-yl]phenyl]acetamide
Show/Hide
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C23H21N3O3
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1
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1 |
EC50 = 20930 nM
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CP0475195
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ethyl 2-[2-(3-phenylpropanoyl)phenoxy]acetate
Show/Hide
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C19H20O4
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1
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1 |
EC50 = 23180 nM
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CP0457323
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4-Benzoyl-1-(3-diisopropylamino-2-hydroxy-propyl)-2,5-dimethyl-1,2-dihydro-pyrazol-3-one
Show/Hide
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C21H31N3O3
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1
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1 |
EC50 = 24120 nM
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CP0543797
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2-[4-(dimethylamino)phenyl]-3-(4-ethoxyphenyl)-1,2-dihydroquinazolin-4-one
Show/Hide
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C24H25N3O2
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1
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1 |
EC50 = 25130 nM
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CP0537243
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4-Benzoyl-1-(2-hydroxy-3-propylamino-propyl)-5-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one
Show/Hide
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C23H27N3O3
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1
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1 |
EC50 = 28210 nM
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CP0496051
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1-(2-(2-hydroxy-3-(piperidin-1-yl)propoxy)phenyl)ethanone
Show/Hide
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C16H23NO3
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1
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1 |
EC50 = 31960 nM
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CP0505679
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1-((3-methyl-2,3-dihydrobenzofuran-2-yl)methyl)piperidine
Show/Hide
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C15H21NO
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1
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1 |
EC50 = 48920 nM
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CP0467804
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1-[4-(2-hydroxy-3-piperidin-1-ylpropoxy)phenyl]ethanone
Show/Hide
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C16H23NO3
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1
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1 |
EC50 = 49000 nM
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CP0428330
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4-tert-butyl-N-[2-[(4-tert-butylphenyl)methylsulfanyl]-1,3-benzothiazol-6-yl]benzamide
Show/Hide
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C29H32N2OS2
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1
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1 |
EC50 > 50000 nM
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CP0379036
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1-[2-(2-hydroxy-3-morpholin-4-ylpropoxy)phenyl]propan-1-one
Show/Hide
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C16H23NO4
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1
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1 |
EC50 = 67000 nM
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CP0501929
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1-(2-Hydroxy-3-propylamino-propyl)-5-methyl-2-phenyl-4-(thiophene-2-carbonyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C21H25N3O3S
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1
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1 |
EC50 = 72440 nM
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CP0511174
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1-(3-tert-Butylamino-2-hydroxy-propyl)-5-methyl-2-phenyl-4-(thiophene-2-carbonyl)-1,2-dihydro-pyrazol-3-one
Show/Hide
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C22H27N3O3S
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1
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1 |
EC50 = 72440 nM
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CP0384923
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4-Benzoyl-1-(3-tert-butylamino-2-hydroxy-propyl)-5-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one
Show/Hide
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C24H29N3O3
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1
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1 |
EC50 = 81280 nM
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CP0544009
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4-Benzoyl-1-(2-hydroxy-3-isopropylamino-propyl)-5-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one
Show/Hide
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C23H27N3O3
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1
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1 |
EC50 = 83180 nM
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CP0425012
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3-(4-ethylphenyl)-2-(4-phenylmethoxyphenyl)-1,2-dihydroquinazolin-4-one
Show/Hide
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C29H26N2O2
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1
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1 |
EC50 > 100000 nM
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CP0435917
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4-[4,6-bis(trifluoromethyl)-1,3,5-triazin-2-yl]-N,N-dimethylaniline
Show/Hide
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C13H10F6N4
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1
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1 |
EC50 > 100000 nM
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