| Compound ID |
Compound Name |
Compound Formula |
|
CP0403274
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-(furan-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acid
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|
C23H20BFN4O4
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0513114
|
[6-[[benzyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]pyridin-3-yl]boronic acid
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|
C24H21BFN5O3
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0470776
|
US8981106, 2 (SX-576)
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|
C20H15BF4N2O4S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0427146
|
[6-[[benzyl-[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C25H22BFN4O3
|
1
|
| 1 |
IC50 = 326 nM
|
|
|
|
CP0513113
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-(furan-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C22H19BFN5O4
|
1
|
| 1 |
IC50 = 444 nM
|
|
|
|
CP0444575
|
[3-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]phenyl]boronic acid
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|
C19H17BFN3O3
|
1
|
| 1 |
IC50 = 611 nM
|
|
|
|
CP0464167
|
[4-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]phenyl]boronic acid
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|
C19H18BFN4O3
|
1
|
| 1 |
IC50 = 681 nM
|
|
|
|
CP0484020
|
[3-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]phenyl]boronic acid
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|
C18H16BFN4O3
|
1
|
| 1 |
IC50 = 1340 nM
|
|
|
|
CP0534769
|
[4-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]phenyl]boronic acid
Show/Hide
|
C20H19BFN3O3
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0403272
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C19H18BFN4O3
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0539316
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C18H17BFN5O3
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0545486
|
[4-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]phenyl]boronic acid
Show/Hide
|
C18H16BFN4O3
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0464244
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-(pyridin-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C23H20BFN6O3
|
1
|
| 1 |
IC50 = 2050 nM
|
|
|
|
CP0413760
|
[3-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]phenyl]boronic acid
Show/Hide
|
C19H18BFN4O3
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0464170
|
[3-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]phenyl]boronic acid
Show/Hide
|
C20H19BFN3O3
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0536889
|
[4-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]phenyl]boronic acid
Show/Hide
|
C19H17BFN3O3
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0403273
|
[2-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]phenyl]boronic acid
Show/Hide
|
C20H19BFN3O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0464169
|
[2-[[[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]phenyl]boronic acid
Show/Hide
|
C19H18BFN4O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0464171
|
2-[(5-boronopyridin-2-yl)methyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]acetic acid
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|
C19H17BFN5O5
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0470380
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-(oxan-4-ylmethyl)amino]methyl]pyridin-3-yl]boronic acid
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|
C24H26BFN4O4
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0513117
|
[6-[[2-aminoethyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C19H20BFN6O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0536890
|
[2-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]phenyl]boronic acid
Show/Hide
|
C19H17BFN3O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0549121
|
[6-[[[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]-(pyridin-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acid
Show/Hide
|
C24H21BFN5O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
