| Compound ID |
Compound Name |
Compound Formula |
|
CP0198642
|
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C21H25ClO6
|
12
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
EC50 = 2 nM
|
|
|
| 3 |
EC50 = 3 nM
|
|
|
| 4 |
IC50 = 0.49 nM
|
|
|
| 5 |
IC50 = 1.05 nM
|
|
|
| 6 |
IC50 = 1.3 nM
|
|
|
| 7 |
IC50 = 1.35 nM
|
|
|
| 8 |
IC50 = 1.4 nM
|
|
|
| 9 |
IC50 = 1.5 nM
|
|
|
| 10 |
IC50 = 3 nM
|
|
|
| 11 |
IC50 = 4 nM
|
|
|
| 12 |
IC50 = 22 nM
|
|
|
|
CP0042564
|
3-(1-benzofuran-5-yl)-1-(2-hydroxy-4-methyl-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)propan-1-one
Show/Hide
|
C24H26O9
|
2
|
| 1 |
EC50 = 6.6 nM
|
|
|
| 2 |
IC50 = 5.2 nM
|
|
|
|
CP0438225
|
(2R,3S,4S,5R,6S)-2-Hydroxymethyl-6-[2-(4-methyl-benzyl)-phenoxy]-tetrahydro-pyran-3,4,5-triol
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|
C20H24O6
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0165583
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-{2-[(4-methoxyphenyl)methyl]phenoxy}oxane-3,4,5-triol
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|
C20H24O7
|
2
|
| 1 |
EC50 = 9.2 nM
|
|
|
| 2 |
IC50 = 6.25 nM
|
|
|
|
CP0341643
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(4-methylbenzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C20H24O5
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0050531
|
1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one
Show/Hide
|
C21H24O10
|
6
|
| 1 |
EC50 = 35 nM
|
|
|
| 2 |
EC50 = 35.6 nM
|
|
|
| 3 |
EC50 = 79 nM
|
|
|
| 4 |
EC50 = 108 nM
|
|
|
| 5 |
IC50 = 16.4 nM
|
|
|
| 6 |
IC50 = 752 nM
|
|
|
|
CP0468848
|
(2R,3S,4R,5R,6S)-2-[(E)-(benzylhydrazinylidene)methyl]-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
|
C28H31ClN2O5
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0536986
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-hydroxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C21H24ClNO6
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0559037
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(methoxyamino)methyl]oxane-3,4,5-triol
Show/Hide
|
C22H28ClNO6
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0431758
|
4-chloro-N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]benzamide
Show/Hide
|
C28H28Cl2N2O6
|
1
|
| 1 |
EC50 = 65 nM
|
|
|
|
CP0495617
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(p-tolylthio)phenyl)-tetrahydro-2H-pyran-3,4,5-triol
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|
C19H22O5S
|
1
|
| 1 |
EC50 = 69 nM
|
|
|
|
CP0383609
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-(2-hydroxyethylhydrazinylidene)methyl]oxane-3,4,5-triol
Show/Hide
|
C23H29ClN2O6
|
1
|
| 1 |
EC50 = 88 nM
|
|
|
|
CP0548766
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-methoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C22H26ClNO6
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0431757
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(hydroxyamino)methyl]oxane-3,4,5-triol
Show/Hide
|
C21H26ClNO6
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
|
CP0559038
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]benzamide
Show/Hide
|
C28H29ClN2O6
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0559042
|
N'-[[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methyl]furan-2-carbohydrazide
Show/Hide
|
C26H29ClN2O7
|
1
|
| 1 |
EC50 = 151 nM
|
|
|
|
CP0409806
|
4-Chloro-3-(4-cyclopropylbenzyl)-1-(beta-D-xylopyranosyl)-1Hindole
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|
C23H24ClNO4
|
1
|
| 1 |
EC50 = 161 nM
|
|
|
|
CP0477383
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]pyridine-4-carboxamide
Show/Hide
|
C27H28ClN3O6
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0559043
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]thiophene-2-carboxamide
Show/Hide
|
C26H27ClN2O6S
|
1
|
| 1 |
EC50 = 175 nM
|
|
|
|
CP0509805
|
(2S,3R,4R,5S,6R)-2-(3-benzylphenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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|
C19H22O5
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0573606
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-2-hydroxyethoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C23H28ClNO7
|
1
|
| 1 |
EC50 = 194 nM
|
|
|
|
CP0536984
|
(2R,3S,4R,5R,6S)-2-[(E)-(1,3-benzothiazol-2-ylhydrazinylidene)methyl]-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
|
C28H28ClN3O5S
|
1
|
| 1 |
EC50 = 204 nM
|
|
|
|
CP0536983
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]thiophene-3-carboxamide
Show/Hide
|
C26H27ClN2O6S
|
1
|
| 1 |
EC50 = 208 nM
|
|
|
|
CP0536982
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[[2-(4-nitrophenyl)hydrazinyl]methyl]oxane-3,4,5-triol
Show/Hide
|
C27H30ClN3O7
|
1
|
| 1 |
EC50 = 211 nM
|
|
|
|
CP0508789
|
4-Chloro-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(beta-Dxylopyranosyl)-1H-indole
Show/Hide
|
C22H22ClNO6
|
1
|
| 1 |
EC50 = 233 nM
|
|
|
|
CP0379728
|
4-Bromo-3-(4-cyclopropylbenzyl)-1-(beta-D-xylopyranosyl)-1Hindole
Show/Hide
|
C23H24BrNO4
|
1
|
| 1 |
EC50 = 241 nM
|
|
|
|
CP0379730
|
4-Chloro-3-(4-hydroxybenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20ClNO5
|
1
|
| 1 |
EC50 = 255 nM
|
|
|
|
CP0378600
|
4-Chloro-3-(4-methoxybenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H22ClNO5
|
1
|
| 1 |
EC50 = 275 nM
|
|
|
|
CP0511458
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(4'-methyl-biphenyl-3-yl)-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C19H22O5
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0523408
|
4-Chloro-3-[4-(N,N-dimethylamino)benzyl]-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C22H25ClN2O4
|
1
|
| 1 |
EC50 = 297 nM
|
|
|
|
CP0532119
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]furan-2-carboxamide
Show/Hide
|
C26H27ClN2O7
|
1
|
| 1 |
EC50 = 301 nM
|
|
|
|
CP0431755
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-ethoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C23H28ClNO6
|
1
|
| 1 |
EC50 = 335 nM
|
|
|
|
CP0455459
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-[(4-nitrophenyl)hydrazinylidene]methyl]oxane-3,4,5-triol
Show/Hide
|
C27H28ClN3O7
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0559044
|
N-[(E)-[(2R,3S,4R,5R,6S)-6-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-3,4,5-trihydroxyoxan-2-yl]methylideneamino]acetamide
Show/Hide
|
C23H27ClN2O6
|
1
|
| 1 |
EC50 = 395 nM
|
|
|
|
CP0559045
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-pent-2-ynoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C26H30ClNO6
|
1
|
| 1 |
EC50 = 396 nM
|
|
|
|
CP0478522
|
4-Chloro-3-[4-(methylsulfanyl)benzyl]-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H22ClNO4S
|
1
|
| 1 |
EC50 = 426 nM
|
|
|
|
CP0563817
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-(4,5-dihydro-1H-imidazol-2-ylhydrazinylidene)methyl]oxane-3,4,5-triol
Show/Hide
|
C24H29ClN4O5
|
1
|
| 1 |
EC50 = 429 nM
|
|
|
|
CP0511313
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-[3-(2-p-tolyl-ethyl)-phenyl]-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C21H26O5
|
1
|
| 1 |
EC50 = 430 nM
|
|
|
|
CP0477944
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-prop-2-ynoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C24H26ClNO6
|
1
|
| 1 |
EC50 = 431 nM
|
|
|
|
CP0557684
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-[(2-nitrophenyl)hydrazinylidene]methyl]oxane-3,4,5-triol
Show/Hide
|
C27H28ClN3O7
|
1
|
| 1 |
EC50 = 457 nM
|
|
|
|
CP0522169
|
4-Chloro-3-(3-fluoro-4-methoxybenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H21ClFNO5
|
1
|
| 1 |
EC50 = 473 nM
|
|
|
|
CP0494750
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(3-phenylpropyl)phenyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H26O5
|
1
|
| 1 |
EC50 = 480 nM
|
|
|
|
CP0399750
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-[3-(3-methyl-benzyl)-phenyl]-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C20H24O5
|
1
|
| 1 |
EC50 = 510 nM
|
|
|
|
CP0379726
|
4-Chloro-3-[4-(prop-2-yn-1-yloxy)benzyl]-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C23H22ClNO5
|
1
|
| 1 |
EC50 = 530 nM
|
|
|
|
CP0511456
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(p-tolyloxy)phenyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H22O6
|
1
|
| 1 |
EC50 = 540 nM
|
|
|
|
CP0523647
|
4-Chloro-3-{4-[2-(2-ethoxyethoxy)ethoxy]benzyl}-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C26H32ClNO7
|
1
|
| 1 |
EC50 = 577 nM
|
|
|
|
CP0511314
|
(2S,3R,4R,5S,6R)-2-Biphenyl-3-yl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C18H20O5
|
1
|
| 1 |
EC50 = 623 nM
|
|
|
|
CP0399745
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-[3-(3-p-tolyl-propyl)-phenyl]-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C22H28O5
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
|
CP0523405
|
4-Chloro-3-(6-methoxy-2-naphthylmethyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C25H24ClNO5
|
1
|
| 1 |
EC50 = 633 nM
|
|
|
|
CP0549735
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-2-methoxyethoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C24H30ClNO7
|
1
|
| 1 |
EC50 = 678 nM
|
|
|
|
CP0511457
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-phenethylphenyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H24O5
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
|
CP0522163
|
3-(1,3-Benzodioxol-5-ylmethyl)-4-chloro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H20ClNO6
|
1
|
| 1 |
EC50 = 863 nM
|
|
|
|
CP0505692
|
3-Benzyl-4-chloro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20ClNO4
|
1
|
| 1 |
EC50 = 865 nM
|
|
|
|
CP0523416
|
4-Chloro-3-(3-methoxybenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H22ClNO5
|
1
|
| 1 |
EC50 = 893 nM
|
|
|
|
CP0472461
|
3-Benzyl-4-bromo-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20BrNO4
|
1
|
| 1 |
EC50 = 923 nM
|
|
|
|
CP0399748
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-[3-(2-m-tolyl-ethyl)-phenyl]-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C21H26O5
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
|
CP0494851
|
3-Benzyl-4-methyl-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 1094 nM
|
|
|
|
CP0501732
|
4-Chloro-3-(3-fluorobenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H19ClFNO4
|
1
|
| 1 |
EC50 = 1161 nM
|
|
|
|
CP0399746
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-[3-(3-m-tolyl-propyl)-phenyl]-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C22H28O5
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0511459
|
(2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(3'-methyl-biphenyl-3-yl)-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C19H22O5
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0523407
|
4-Chloro-3-(4-isopropylbenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C23H26ClNO4
|
1
|
| 1 |
EC50 = 1288 nM
|
|
|
|
CP0052037
|
C-aryl glucoside, 5
Show/Hide
|
C23H29NO9
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0494622
|
4-Chloro-3-[4-(2-phenoxyethoxy)benzyl]-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C28H28ClNO6
|
1
|
| 1 |
EC50 = 1334 nM
|
|
|
|
CP0518445
|
4-Chloro-3-(4-fluorobenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H19ClFNO4
|
1
|
| 1 |
EC50 = 1376 nM
|
|
|
|
CP0410065
|
4-Chloro-3-(4-n-propylbenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C23H26ClNO4
|
1
|
| 1 |
EC50 = 1410 nM
|
|
|
|
CP0505706
|
4-Chloro-3-(2-thienylmethyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C18H18ClNO4S
|
1
|
| 1 |
EC50 = 1682 nM
|
|
|
|
CP0494857
|
3-Benzyl-4-nitro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20N2O6
|
1
|
| 1 |
EC50 = 1819 nM
|
|
|
|
CP0536985
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-cyclopropylmethoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C25H30ClNO6
|
1
|
| 1 |
EC50 = 1953 nM
|
|
|
|
CP0373411
|
3-Benzyl-4-fluoro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 2237 nM
|
|
|
|
CP0464769
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-phenylmethoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C28H30ClNO6
|
1
|
| 1 |
EC50 = 2251 nM
|
|
|
|
CP0503745
|
3-Benzyl-6-methyl-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 3033 nM
|
|
|
|
CP0517146
|
3-Benzyl-4-methoxy-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H23NO5
|
1
|
| 1 |
EC50 = 5487 nM
|
|
|
|
CP0472390
|
3-Benzyl-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H21NO4
|
1
|
| 1 |
EC50 = 7129 nM
|
|
|
|
CP0561843
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-6-[(E)-3,3-dimethylbutoxyiminomethyl]oxane-3,4,5-triol
Show/Hide
|
C27H36ClNO6
|
1
|
| 1 |
EC50 = 8541 nM
|
|
|
|
CP0517147
|
3-Benzyl-6-chloro-5-fluoro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H19ClFNO4
|
1
|
| 1 |
EC50 = 8600 nM
|
|
|
|
CP0494856
|
3-Benzyl-7-fluoro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 9821 nM
|
|
|
|
CP0508801
|
3-Benzyl-6-chloro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20ClNO4
|
1
|
| 1 |
EC50 = 10279 nM
|
|
|
|
CP0472391
|
3-Benzyl-7-chloro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20ClNO4
|
1
|
| 1 |
EC50 = 10680 nM
|
|
|
|
CP0508795
|
4-Chloro-3-(4-phenylbenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C26H24ClNO4
|
1
|
| 1 |
EC50 = 11137 nM
|
|
|
|
CP0508800
|
3-Benzyl-5-fluoro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 12415 nM
|
|
|
|
CP0378598
|
4-Chloro-3-(2-methoxybenzyl)-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H22ClNO5
|
1
|
| 1 |
EC50 = 12915 nM
|
|
|
|
CP0494855
|
3-Benzyl-7-methyl-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 12956 nM
|
|
|
|
CP0478519
|
3-Benzyl-6-fluoro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 23627 nM
|
|
|
|
CP0502133
|
3-Benzyl-5-chloro-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H20ClNO4
|
1
|
| 1 |
EC50 = 28217 nM
|
|
|
|
CP0522162
|
4-Chloro-3-(2,4-dimethoxybenzyl)-1-(beta-D-xylopyranosyl)-1Hindole
Show/Hide
|
C22H24ClNO6
|
1
|
| 1 |
EC50 = 30931 nM
|
|
|
|
CP0494853
|
3-Benzyl-5-methyl-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
EC50 = 40589 nM
|
|
|
|
CP0378596
|
3-Benzyl-4-hydroxy-1-(beta-D-xylopyranosyl)-1H-indole
Show/Hide
|
C20H21NO5
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0564560
|
US9034921, E171
Show/Hide
|
C23H25ClO6
|
1
|
| 1 |
IC50 = 0.37 nM
|
|
|
|
CP0545470
|
US9034921, E001
Show/Hide
|
C23H27BrO6
|
1
|
| 1 |
IC50 = 0.44 nM
|
|
|
|
CP0578807
|
US9034921, E172
Show/Hide
|
C24H27ClO6
|
1
|
| 1 |
IC50 = 0.46 nM
|
|
|
|
CP0536117
|
(2S,3R,4R,5S,6R)-2-[4-chloro-5-[(4-ethylphenyl)methyl]-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0568442
|
US9034921, E005
Show/Hide
|
C23H27ClO6
|
1
|
| 1 |
IC50 = 0.68 nM
|
|
|
|
CP0425348
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO6S
|
2
|
| 1 |
IC50 = 0.72 nM
|
|
|
| 2 |
IC50 = 1.75 nM
|
|
|
|
CP0564527
|
US9034921, E020
Show/Hide
|
C23H27ClO6
|
1
|
| 1 |
IC50 = 0.72 nM
|
|
|
|
CP0530034
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO5S2
|
1
|
| 1 |
IC50 = 0.772 nM
|
|
|
|
CP0450860
|
(1S,16R,17S,18R,19R)-5-chloro-4-[(4-methylsulfanylphenyl)methyl]-8,14,20-trioxatricyclo[14.3.1.02,7]icosa-2(7),3,5-triene-17,18,19-triol
Show/Hide
|
C25H31ClO6S
|
1
|
| 1 |
IC50 = 0.778 nM
|
|
|
|
CP0564589
|
US9034921, E007
Show/Hide
|
C24H30O6
|
1
|
| 1 |
IC50 = 0.79 nM
|
|
|
|
CP0577050
|
US9034921, E181
Show/Hide
|
C24H29ClO6
|
1
|
| 1 |
IC50 = 0.79 nM
|
|
|
|
CP0498302
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-hydroxyphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO7S
|
1
|
| 1 |
IC50 = 0.797 nM
|
|
|
|
CP0485581
|
(2S,3R,4R,5S,6R)-2-[4-chloro-2-hydroxy-5-[(4-methylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0499382
|
(1S,16R,17S,18R,19R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,14,20-trioxatricyclo[14.3.1.02,7]icosa-2(7),3,5-triene-17,18,19-triol
Show/Hide
|
C26H33ClO7
|
1
|
| 1 |
IC50 = 0.899 nM
|
|
|
|
CP0498301
|
(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C23H24ClNO6S2
|
1
|
| 1 |
IC50 = 0.934 nM
|
|
|
|
CP0397860
|
(1S,10Z,15R,16S,17R,18R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,13,19-trioxatricyclo[13.3.1.02,7]nonadeca-2(7),3,5,10-tetraene-16,17,18-triol
Show/Hide
|
C25H29ClO7
|
1
|
| 1 |
IC50 = 0.974 nM
|
|
|
|
CP0572322
|
US9034921, E016
Show/Hide
|
C23H27ClO7
|
1
|
| 1 |
IC50 = 0.98 nM
|
|
|
|
CP0481747
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-methoxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0573915
|
(1R,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-(difluoromethoxy)-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
|
C22H23ClF2O7
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0536116
|
(2S,3R,4R,5S,6R)-2-[4-chloro-5-[(4-ethoxyphenyl)methyl]-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO7
|
1
|
| 1 |
IC50 = 1.03 nM
|
|
|
|
CP0390165
|
(2S,3R,4R,5S,6R)-2-[4-chloro-2-hydroxy-5-[(4-methoxyphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C20H23ClO7
|
1
|
| 1 |
IC50 = 1.08 nM
|
|
|
|
CP0487788
|
2-[[(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-2,3,4-trihydroxy-6,8-dioxabicyclo[3.2.1]octan-1-yl]oxy]acetonitrile
Show/Hide
|
C23H24ClNO7
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0527637
|
(2S,3R,4R,6R)-2-[4-chloro-2-hydroxy-5-[(4-methoxyphenyl)methyl]phenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
|
C20H21ClF2O6
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0502878
|
((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((2-(thiophen-3-yl)thiazol-5-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO5S2
|
1
|
| 1 |
IC50 = 1.11 nM
|
|
|
|
CP0506109
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO5S2
|
1
|
| 1 |
IC50 = 1.14 nM
|
|
|
|
CP0578329
|
US9034921, E233
Show/Hide
|
C26H31ClO6
|
1
|
| 1 |
IC50 = 1.16 nM
|
|
|
|
CP0567318
|
US9034921, E187
Show/Hide
|
C24H29ClO6
|
1
|
| 1 |
IC50 = 1.17 nM
|
|
|
|
CP0462919
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C22H24ClNO6S2
|
1
|
| 1 |
IC50 = 1.18 nM
|
|
|
|
CP0576780
|
US9034921, E194
Show/Hide
|
C24H29ClO7
|
1
|
| 1 |
IC50 = 1.22 nM
|
|
|
|
CP0484164
|
(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C23H24ClNO7S
|
1
|
| 1 |
IC50 = 1.24 nM
|
|
|
|
CP0470212
|
(2R,3S,4R,5R,6S)-2-(Hydroxymethyl)-6-(4-methyl-3-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H23NO5S2
|
1
|
| 1 |
IC50 = 1.28 nM
|
|
|
|
CP0462916
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-2-methoxy-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C21H22ClNO6S2
|
1
|
| 1 |
IC50 = 1.29 nM
|
|
|
|
CP0404716
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-ethylbenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0394824
|
(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-methoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
|
C22H25ClO7
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0562522
|
(2S,3R,4R,6R)-2-[5-(3,4-dihydro-2H-chromen-6-ylmethyl)-2-hydroxy-4-methoxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
|
C23H26F2O7
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0511523
|
(1S,13R,14S,15R,16R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,11,17-trioxatricyclo[11.3.1.02,7]heptadeca-2(7),3,5-triene-14,15,16-triol
Show/Hide
|
C23H27ClO7
|
1
|
| 1 |
IC50 = 1.34 nM
|
|
|
|
CP0499383
|
(1S,15R,16S,17R,18R)-5-chloro-4-[(4-methylsulfanylphenyl)methyl]-8,13,19-trioxatricyclo[13.3.1.02,7]nonadeca-2(7),3,5-triene-16,17,18-triol
Show/Hide
|
C24H29ClO6S
|
1
|
| 1 |
IC50 = 1.35 nM
|
|
|
|
CP0498831
|
(1S,16R,17S,18R,19R)-5-chloro-4-[(4-ethylphenyl)methyl]-8,14,20-trioxatricyclo[14.3.1.02,7]icosa-2(7),3,5-triene-17,18,19-triol
Show/Hide
|
C26H33ClO6
|
1
|
| 1 |
IC50 = 1.38 nM
|
|
|
|
CP0499384
|
(1S,16R,17S,18R,19R)-5-chloro-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-8,14,20-trioxatricyclo[14.3.1.02,7]icosa-2(7),3,5-triene-17,18,19-triol
Show/Hide
|
C26H31ClO8
|
1
|
| 1 |
IC50 = 1.38 nM
|
|
|
|
CP0389025
|
(1S,17R,18S,19R,20R)-5-chloro-4-[(4-ethylphenyl)methyl]-8,15,21-trioxatricyclo[15.3.1.02,7]henicosa-2(7),3,5-triene-18,19,20-triol
Show/Hide
|
C27H35ClO6
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0472691
|
(1S,15R,16S,17R,18R)-5-chloro-4-[(4-ethylphenyl)methyl]-8,13,19-trioxatricyclo[13.3.1.02,7]nonadeca-2(7),3,5-triene-16,17,18-triol
Show/Hide
|
C25H31ClO6
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0429521
|
(3S,3'R,4'S,5'S,6'R)-5-[(4-ethylphenyl)methyl]-6'-(hydroxymethyl)-6-methylspiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
|
C23H28O6
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0516130
|
(3S,3'R,4'S,5'S,6'R)-5-[(4-ethylphenyl)methyl]-6-ethynyl-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
|
C24H26O6
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0507517
|
(2S,3R,4R,6R)-2-[4-chloro-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-hydroxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
|
C21H21ClF2O7
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0502877
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((2-(furan-2-yl)thiazol-5-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO6S
|
1
|
| 1 |
IC50 = 1.42 nM
|
|
|
|
CP0508237
|
(2S,3R,4R,5S,6R)-2-(3-((5-(Furan-2-yl)thiazol-2-yl)methyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H23NO6S
|
1
|
| 1 |
IC50 = 1.43 nM
|
|
|
|
CP0580220
|
(2S,3R,4R,5S,6R)-2-[7-chloro-6-[(4-methylphenyl)methyl]-2,3-dihydro-1-benzofuran-4-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 1.44 nM
|
|
|
|
CP0490987
|
(2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H28O5
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0073918
|
LP-802034
Show/Hide
|
C21H25ClO5S
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0478538
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-(2-hydroxyethoxy)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H24ClNO8S
|
1
|
| 1 |
IC50 = 1.51 nM
|
|
|
|
CP0564590
|
US9034921, E024
Show/Hide
|
C23H27ClO7
|
1
|
| 1 |
IC50 = 1.52 nM
|
|
|
|
CP0552001
|
US9034921, E019
Show/Hide
|
C22H25ClO7
|
1
|
| 1 |
IC50 = 1.53 nM
|
|
|
|
CP0484165
|
(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C23H24ClNO7S
|
1
|
| 1 |
IC50 = 1.54 nM
|
|
|
|
CP0504578
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClNO6S
|
1
|
| 1 |
IC50 = 1.57 nM
|
|
|
|
CP0524884
|
(2S,3R,4R,5S,6R)-2-(4-chloro-2-methoxy-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H22ClNO6S2
|
1
|
| 1 |
IC50 = 1.59 nM
|
|
|
|
CP0452455
|
(1S,14R,15S,16R,17R)-5-chloro-4-[(4-ethylphenyl)methyl]-8,12,18-trioxatricyclo[12.3.1.02,7]octadeca-2(7),3,5-triene-15,16,17-triol
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C24H29ClO6
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1
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| 1 |
IC50 = 1.59 nM
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CP0487900
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(3S,3'R,4'S,5'S,6'R)-5-[(4-cyclopropylphenyl)methyl]-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C23H26O6
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1
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| 1 |
IC50 = 1.6 nM
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CP0484166
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(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C23H24ClNO6S2
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1
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| 1 |
IC50 = 1.69 nM
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CP0578330
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US9034921, E021
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C22H25ClO7
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1
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| 1 |
IC50 = 1.72 nM
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CP0489166
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(2S,3R,4R,5S,6R)-2-(4-Bromo-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C20H20BrNO6S
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1
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| 1 |
IC50 = 1.89 nM
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CP0484162
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-methoxy-5-((5-phenylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H24ClNO6S
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1
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| 1 |
IC50 = 2.01 nM
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CP0571361
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US9034921, E006
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C23H27FO6
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1
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| 1 |
IC50 = 2.03 nM
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CP0580129
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US9034921, E156
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C23H27ClO7
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1
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| 1 |
IC50 = 2.09 nM
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CP0562524
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(2S,3R,4R,5S,6R)-2-[4-chloro-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-hydroxyphenyl]-5-fluoro-6-(hydroxymethyl)-5-methyloxane-3,4-diol
Show/Hide
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C22H24ClFO7
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1
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| 1 |
IC50 = 2.1 nM
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CP0484168
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5e((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C20H19ClFNO5S2
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1
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| 1 |
IC50 = 2.12 nM
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CP0373293
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-methoxyphenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO7S
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1
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| 1 |
IC50 = 2.15 nM
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CP0488884
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1-(beta-D-Glucopyranosyl)-4-methyl-3-(5-(4-fluorophenyl)-2-thienylmethyl)benzene
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C24H25FO6S
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1
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| 1 |
IC50 = 2.2 nM
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CP0178282
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CANAGLIFLOZIN
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C24H25FO5S
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1
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| 1 |
IC50 = 2.2 nM
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CP0513204
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(2S,3R,4R,5S,6R)-2-(4-chloro-2-(hydroxymethyl)-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H22ClNO6S2
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1
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| 1 |
IC50 = 2.23 nM
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CP0528684
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(2S,3R,4R,5S,6R)-2-(4-Chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-(prop-2-ynyloxy)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H22ClNO7S
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1
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| 1 |
IC50 = 2.23 nM
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CP0529848
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(2S,3R,4R,5S,6R)-2-(2,4-Dichloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H19Cl2NO6S
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1
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| 1 |
IC50 = 2.24 nM
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CP0397861
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(1S,15R,16S,17R,18R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,13,19-trioxatricyclo[13.3.1.02,7]nonadeca-2(7),3,5-triene-16,17,18-triol
Show/Hide
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C25H31ClO7
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1
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| 1 |
IC50 = 2.27 nM
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CP0484169
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(2S,3R,4R,5S,6R)-2-(2,4-Dichloro-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C20H19Cl2NO5S2
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1
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| 1 |
IC50 = 2.31 nM
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CP0390432
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(2S,3R,4S,5S,6R)-2-(4-chloro-3-(4-methoxybenzyl)phenyl)-6-methyltetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H23ClO5
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1
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| 1 |
IC50 = 2.4 nM
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CP0470818
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1-(beta-D-Glucopyranosyl)-4-chloro-3-(5-chloro-2-thienylmethyl)benzene
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C17H18Cl2O6S
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1
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| 1 |
IC50 = 2.4 nM
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CP0149289
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(1S,2S,3S,4R,5S)-5-[4-Chloro-3-(4-ethoxybenzyl)phenyl]-1-(hydroxymethyl)-6,8-dioxa-bicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C22H25ClO7
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1
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| 1 |
IC50 = 2.4 nM
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CP0567743
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US9315438, Compound represented by formula (II)
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C25H29ClO6
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1
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| 1 |
IC50 = 2.5 nM
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CP0394825
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-ethoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C23H27ClO7
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1
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| 1 |
IC50 = 2.5 nM
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CP0578397
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(2S,3R,4R,6R)-2-[4-chloro-2-hydroxy-5-[(3-methoxyphenyl)methyl]phenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
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C20H21ClF2O6
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1
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| 1 |
IC50 = 2.6 nM
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CP0380477
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((2-(thiophen-2-yl)thiazol-5-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H20ClNO5S2
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1
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| 1 |
IC50 = 2.79 nM
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CP0484163
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5-((5-phenylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H26ClNO6S
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1
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| 1 |
IC50 = 2.87 nM
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CP0076249
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TOFOGLIFLOZIN
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C22H26O6
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1
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| 1 |
IC50 = 2.9 nM
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CP0511524
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(1S,14R,15S,16R,17R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,12,18-trioxatricyclo[12.3.1.02,7]octadeca-2(7),3,5-triene-15,16,17-triol
Show/Hide
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C24H29ClO7
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1
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| 1 |
IC50 = 2.95 nM
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CP0447422
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(5S,6R,7R,8S)-5-(3-(4-ethylbenzyl)-4-methylphenyl)-4-oxaspiro[2.5]octane-6,7,8-triol
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C23H28O4
|
1
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| 1 |
IC50 = 3 nM
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CP0465081
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6,8-dichloro-4-((5-(5-chloropyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C19H13Cl3F3N5O2
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1
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| 1 |
IC50 = 3 nM
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CP0534081
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4-((5-(5-chloropyridin-2-yl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-6,8-dimethyl-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C21H22ClN5O2
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1
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| 1 |
IC50 = 3 nM
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CP0530035
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(2S,3R,4R,5S,6R)-2-(3-(2,5'-Bithiazol-2'-ylmethyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H19ClN2O5S2
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1
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| 1 |
IC50 = 3.13 nM
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CP0429520
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-propan-2-ylphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
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C23H28O6
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1
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| 1 |
IC50 = 3.2 nM
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CP0373295
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(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-phenylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H26ClNO6S
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1
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| 1 |
IC50 = 3.38 nM
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CP0501855
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(6S,7R,8R,9S)-6-(3-(4-ethylbenzyl)-4-methylphenyl)-2,5-dioxaspiro[3.5]nonane-7,8,9-triol
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C23H28O5
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1
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| 1 |
IC50 = 3.4 nM
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CP0469922
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(1R,2S,3R,4R,5S)-5-[4-chloro-3-[[4-[(3S)-oxolan-3-yl]oxyphenyl]methyl]phenyl]-1-(difluoromethoxy)-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C24H25ClF2O8
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1
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| 1 |
IC50 = 3.4 nM
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CP0373298
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C20H19ClFNO6S
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1
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| 1 |
IC50 = 3.49 nM
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CP0521419
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H19ClN2O5S2
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1
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| 1 |
IC50 = 3.51 nM
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CP0516131
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-methylsulfanylphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
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C21H24O6S
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1
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| 1 |
IC50 = 3.6 nM
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CP0466558
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(1S,17R,18S,19R,20R)-5-chloro-4-[(4-ethoxyphenyl)methyl]-8,15,21-trioxatricyclo[15.3.1.02,7]henicosa-2(7),3,5-triene-18,19,20-triol
Show/Hide
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C27H35ClO7
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1
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| 1 |
IC50 = 3.63 nM
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CP0511959
|
US9315438, Reference compound 1
Show/Hide
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C25H29ClO6
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1
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| 1 |
IC50 = 3.63 nM
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CP0389026
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(1S,15R,16S,17R,18R)-5-chloro-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-8,13,19-trioxatricyclo[13.3.1.02,7]nonadeca-2(7),3,5-triene-16,17,18-triol
Show/Hide
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C25H29ClO8
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1
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| 1 |
IC50 = 3.65 nM
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CP0508412
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(2S,3R,4R,5S,6R)-2-[3-(1-benzothiophen-2-ylmethyl)-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H21ClO5S
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1
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| 1 |
IC50 = 3.7 nM
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CP0528687
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C20H19ClFNO5S2
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1
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| 1 |
IC50 = 3.88 nM
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CP0373294
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C22H24ClNO7S
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1
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| 1 |
IC50 = 3.98 nM
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CP0494443
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4-((5-(5-chloropyridin-2-yl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-6-methyl-8-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H19ClN6O4
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1
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| 1 |
IC50 = 4 nM
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CP0376549
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2-(2-Chloro-5-((2S,3S,4R,5R,6R)-3,4,5-tris(benzyloxy)-6-(benzyloxymethyl)-tetrahydro-2H-pyran-2-yl)benzyl)-5-(pyrazin-2-yl)-1,3,4-thiadiazole
Show/Hide
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C19H19ClN4O5S
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1
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| 1 |
IC50 = 4.06 nM
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CP0553328
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(2S,3R,4R,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-4-chloro-2-hydroxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C21H19ClF2O5S
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1
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| 1 |
IC50 = 4.2 nM
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CP0373296
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(2S,3R,4R,5S,6R)-2-(2-(Allyloxy)-4-chloro-5-((5-(4-fluorophenyl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H25ClFNO6S
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1
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| 1 |
IC50 = 4.22 nM
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CP0578495
|
US9034921, E166
Show/Hide
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C21H23ClO6
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1
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| 1 |
IC50 = 4.22 nM
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CP0462918
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C22H24ClNO6S2
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1
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| 1 |
IC50 = 4.29 nM
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CP0562523
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(2S,3R,4R,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-4-chloro-2-methoxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C22H21ClF2O5S
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1
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| 1 |
IC50 = 4.3 nM
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CP0573087
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(2S,3R,4R,5S,6R)-2-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-hydroxy-4-methoxyphenyl]-5-fluoro-6-(hydroxymethyl)-5-methyloxane-3,4-diol
Show/Hide
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C23H27FO8
|
1
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| 1 |
IC50 = 4.3 nM
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CP0528683
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C22H24ClNO7S
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1
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| 1 |
IC50 = 4.35 nM
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CP0469918
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-cyclopropyloxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C24H27ClO7
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1
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| 1 |
IC50 = 4.4 nM
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CP0504582
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((2-(furan-3-yl)thiazol-5-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H20ClNO6S
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1
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| 1 |
IC50 = 4.47 nM
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CP0501224
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-ethylphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C19H23ClO5S
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1
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| 1 |
IC50 = 4.47 nM
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CP0504917
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5-((5-phenylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H21ClFNO5S
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1
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| 1 |
IC50 = 4.57 nM
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CP0504576
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(2S,3R,4R,5S,6R,E)-2-(3-((5-(but-2-en-2-yl)thiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H24ClNO5S
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1
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| 1 |
IC50 = 4.69 nM
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CP0373299
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(2S,3R,4R,5S,6R)-2-(2,4-Dichloro-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
Show/Hide
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C20H19Cl2NO5S2
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1
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| 1 |
IC50 = 4.77 nM
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CP0492184
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-methylphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
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C21H24O6
|
1
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| 1 |
IC50 = 4.8 nM
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CP0398864
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-hexylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H30ClNO5S
|
1
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| 1 |
IC50 = 5 nM
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CP0049115
|
4-((5-(2,3-dihydro-1H-inden-2-yl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-6,8-dimethyl-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C25H28N4O2
|
1
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| 1 |
IC50 = 5 nM
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CP0521656
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6-chloro-4-((5-(5-chloropyridin-2-yl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-8-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C19H16Cl2N6O4
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1
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| 1 |
IC50 = 5 nM
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CP0394826
|
(1S,2S,3R,4R,5S)-5-[3-[(4-ethoxyphenyl)methyl]phenyl]-1-methoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C22H26O7
|
1
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| 1 |
IC50 = 5 nM
|
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CP0539344
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-(4-methoxybenzyl)phenyl)-6-(fluoromethyl)-5-methoxytetrahydro-2H-pyran-3,4-diol
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C21H24ClFO5
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1
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| 1 |
IC50 = 5.1 nM
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CP0466042
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
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C20H19ClFNO6S
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1
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| 1 |
IC50 = 5.35 nM
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CP0484167
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(2S,3R,4R,5S,6R)-2-(4-Chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-(2-methoxyethoxy)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H26ClNO8S
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1
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| 1 |
IC50 = 5.55 nM
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CP0424909
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-(hydroxymethyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO7S
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1
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| 1 |
IC50 = 5.81 nM
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CP0436618
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(2S,3R,4R,5S,6R)-2-(4-chloro-2-(hydroxymethyl)-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO6S2
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1
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| 1 |
IC50 = 5.88 nM
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CP0429577
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxy-3-fluorophenyl)methyl]phenyl]-1-methoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C22H24ClFO7
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1
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| 1 |
IC50 = 5.9 nM
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CP0469920
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(1R,2S,3R,4R,5S)-5-[4-chloro-3-[[4-(2-cyclopropyloxyethoxy)phenyl]methyl]phenyl]-1-(difluoromethoxy)-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C25H27ClF2O8
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1
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| 1 |
IC50 = 5.9 nM
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CP0546248
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[[4-[(3S)-oxolan-3-yl]oxyphenyl]methyl]phenyl]-1-methoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C24H27ClO8
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1
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| 1 |
IC50 = 5.9 nM
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CP0462917
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(2S,3R,4R,5S,6R)-2-(4-Chloro-5-((5-(4-fluorophenyl)thiazol-2-yl)methyl)-2-methoxyphenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
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C23H23ClFNO6S
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1
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| 1 |
IC50 = 6.08 nM
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CP0504580
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(2S,3R,4R,5S,6R)-2-(4-Fluoro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H20FNO6S
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1
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| 1 |
IC50 = 6.11 nM
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CP0504579
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(2S,3R,4R,5S,6R)-2-(4-Bromo-3-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C20H20BrNO5S2
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1
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| 1 |
IC50 = 6.36 nM
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CP0430362
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(6S,7R,8R,9S)-6-(3-(4-methoxybenzyl)-4-methylphenyl)-2,5-dioxaspiro[3.5]nonane-7,8,9-triol
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C22H26O6
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1
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| 1 |
IC50 = 6.6 nM
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CP0552373
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxy-3-fluorophenyl)methyl]phenyl]-1-propan-2-yloxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C24H28ClFO7
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1
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| 1 |
IC50 = 6.8 nM
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CP0465083
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6-chloro-4-((5-(5-chloropyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-8-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
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C19H13Cl2F3N6O4
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1
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| 1 |
IC50 = 7 nM
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CP0566048
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6-chloro-8-nitro-4-((5-(5-(trifluoromethyl)pyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C20H13ClF6N6O4
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1
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| 1 |
IC50 = 7 nM
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CP0373640
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(2S,3R,4S,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-methyltetrahydro-2H-pyran-3,4,5-triol
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C20H20ClNO5S
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1
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| 1 |
IC50 = 7.01 nM
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CP0326093
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H19ClN2O6S
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1
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| 1 |
IC50 = 7.03 nM
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CP0502875
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(2S,3R,4R,5S,6R)-2-(4-Fluoro-3-((5-(thiazol-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H20FNO5S2
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1
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| 1 |
IC50 = 7.36 nM
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CP0462914
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(2S,3R,4R,5S,6R)-2-(4-Chloro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)-2-methoxyphenyl)-6-(hydroxymethyl)tetrahydro-2Hpyran-3,4,5-triol
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C21H22ClNO7S
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1
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| 1 |
IC50 = 7.37 nM
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CP0137894
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(2S,3R,4R,5S,6R)-2-[3-(1-benzothiophen-2-ylmethyl)-4-fluorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H21FO5S
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1
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| 1 |
IC50 = 7.4 nM
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CP0578804
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[6-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-inden-4-yl]oxane-3,4,5-triol
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C23H28O6
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1
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| 1 |
IC50 = 7.44 nM
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CP0487898
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-propylphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C23H28O6
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1
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| 1 |
IC50 = 7.5 nM
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CP0512462
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-ethoxy-5e((5-(4-fluorophenyl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H25ClFNO6S
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1
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| 1 |
IC50 = 7.55 nM
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CP0524621
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US9315438, Compound represented by formula (III)
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C25H29ClO6
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1
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| 1 |
IC50 = 7.83 nM
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CP0504722
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(5S,6R,7R,8S)-5-(3-(4-methoxybenzyl)-4-methylphenyl)-4-oxaspiro[2.5]octane-6,7,8-triol
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C22H26O5
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1
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| 1 |
IC50 = 7.9 nM
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CP0542523
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(2S,3R,4R,5S,6R)-2-[3-(azulen-2-ylmethyl)-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C23H23ClO5
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1
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| 1 |
IC50 = 7.9 nM
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CP0486628
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4-((5-(benzyloxymethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-6,8-dichloro-2H-benzo[b][1,4]oxazin-3(4H)-one
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C22H19Cl2F3N4O3
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1
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| 1 |
IC50 = 8 nM
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CP0566049
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6,8-dimethyl-4-((5-((1R,2R)-2-phenylcyclopropyl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C25H28N4O2
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1
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| 1 |
IC50 = 8 nM
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CP0479552
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1-(beta-D-Glucopyranosyl)-4-methyl-3-(5-(4-fluorophenyl)-2-thiazolylmethyl)-benzene
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C23H24FNO6S
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1
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| 1 |
IC50 = 8.1 nM
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CP0502873
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pentyloxy)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H28ClNO6S
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1
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| 1 |
IC50 = 8.2 nM
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CP0527963
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(2R,3R,4S,5S,6R)-2-[4-[(4-ethoxyphenyl)methyl]-5-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C20H26O6S
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1
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| 1 |
IC50 = 8.73 nM
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CP0465381
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(2S,3R,4R,5S,6R)-2-[5-(azulen-2-ylmethyl)-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C23H24O6
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1
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| 1 |
IC50 = 8.9 nM
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CP0474215
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6,8-dichloro-4-((5-(4-chlorophenethyl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C22H21Cl3N4O2
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3
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 16 nM
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| 3 |
IC50 = 40 nM
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CP0507600
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-methoxyphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C21H24O7
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1
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| 1 |
IC50 = 9.1 nM
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CP0516856
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(2S,3R,4R,5S,6R)-2-(3-((5-(biphenyl-4-yl)thiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C28H26ClNO5S
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1
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| 1 |
IC50 = 9.31 nM
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CP0478482
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(difluoromethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H18ClF2NO5S
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1
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| 1 |
IC50 = 9.55 nM
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CP0414952
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(1S,3'R,4'S,5'S,6'R)-6-(4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H26O7
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1
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| 1 |
IC50 = 9.6 nM
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CP0381803
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-cyclopentylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H26ClNO5S
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1
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| 1 |
IC50 = 9.71 nM
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CP0489167
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(2S,3R,4R,5S,6R)-2-(3-((5-(Furan-2-yl)thiazol-2-yl)methyl)-4-(trifluoromethyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H20F3NO6S
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1
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| 1 |
IC50 = 9.73 nM
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CP0390358
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(2S,3R,4R,5S,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H22O6S
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1
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| 1 |
IC50 = 9.8 nM
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CP0294225
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6,8-dichloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C22H18Cl3F3N4O2
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3
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 19 nM
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| 3 |
IC50 = 20 nM
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CP0438199
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6,8-dichloro-4-((5-(2-methylthiazol-4-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C18H14Cl2F3N5O2S
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1
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| 1 |
IC50 = 10 nM
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CP0566050
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(R)-6,8-dimethyl-4-((4-propyl-5-(1,2,3,4-tetrahydronaphthalen-2-yl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C26H30N4O2
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1
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| 1 |
IC50 = 10 nM
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CP0524872
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(2S,3R,4R,5S,6R)-2-(2-(Allyloxymethyl)-4-chloro-5-((5-(thiophen-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H26ClNO6S2
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1
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| 1 |
IC50 = 10 nM
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CP0262485
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(2S,3R,4R,5S,6R)-2-[3-[(4-ethylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H26O5
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1
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| 1 |
IC50 = 10 nM
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CP0564201
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(2S,3R,4R,5S,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-4-chloro-2-hydroxyphenyl]-5-fluoro-6-(hydroxymethyl)-5-methyloxane-3,4-diol
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C22H22ClFO5S
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1
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| 1 |
IC50 = 10.2 nM
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CP0498684
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-propylphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H25ClO5S
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1
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| 1 |
IC50 = 10.3 nM
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CP0434151
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-phenylfuran-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H23ClN2O6S
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1
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| 1 |
IC50 = 10.6 nM
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CP0538847
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(fluoromethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H19ClFNO5S
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1
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| 1 |
IC50 = 10.6 nM
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CP0493414
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[[4-(2-cyclopropyloxyethoxy)phenyl]methyl]phenyl]-1-methoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C25H29ClO8
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1
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| 1 |
IC50 = 10.8 nM
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CP0514776
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(methylthio)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C16H19ClN2O5S2
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1
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| 1 |
IC50 = 10.9 nM
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CP0367612
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(2S,3R,4R,5S,6R)-2-(3-((6-(1,3,4-thiadiazol-2-yl)pyridazin-3-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H19ClN4O5S
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1
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| 1 |
IC50 = 11.4 nM
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CP0502872
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(2S,3R,4R,5S,6R)-2-(3-((5-Allylthiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H22ClNO5S
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1
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| 1 |
IC50 = 11.5 nM
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CP0499316
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(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[4-[(4-methoxyphenyl)methyl]-5-methylthiophen-2-yl]oxane-3,4,5-triol
Show/Hide
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C19H24O6S
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1
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| 1 |
IC50 = 11.5 nM
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CP0501568
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-propan-2-yloxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H25ClO6S
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1
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| 1 |
IC50 = 11.9 nM
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CP0417976
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H25ClO5
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1
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| 1 |
IC50 = 12 nM
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CP0136282
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6,8-dimethyl-4-((4-propyl-5-(pyridin-2-yl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C21H23N5O2
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1
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| 1 |
IC50 = 12 nM
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CP0494447
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6,8-dichloro-4-[[5-(2-phenylcyclopropyl)-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-1,4-benzoxazin-3-one
Show/Hide
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C23H19Cl2F3N4O2
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1
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| 1 |
IC50 = 12 nM
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CP0519966
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(2S,3R,4R,5S,6R)-2-[5-[(4-ethoxyphenyl)methyl]-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H26O7
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1
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| 1 |
IC50 = 12.17 nM
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CP0509946
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-propoxythiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H24ClNO6S
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1
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| 1 |
IC50 = 12.4 nM
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CP0524069
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-heptylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H32ClNO5S
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1
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| 1 |
IC50 = 12.4 nM
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CP0503145
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(2R,3R,4S,5S,6R)-2-[3-bromo-5-[(4-ethylphenyl)methyl]-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H25BrO5S
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1
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| 1 |
IC50 = 12.4 nM
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CP0503286
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-methylsulfanylphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C18H21ClO5S2
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1
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| 1 |
IC50 = 12.8 nM
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CP0371971
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6,8-dichloro-4-((5-(pyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C19H14Cl2F3N5O2
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1
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| 1 |
IC50 = 13 nM
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CP0511772
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6,8-dichloro-4-((5-(2,3-dihydro-1H-inden-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C23H19Cl2F3N4O2
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1
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| 1 |
IC50 = 13 nM
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CP0459335
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(2S,3R,4R,5S,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-2-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C22H24O6S
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1
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| 1 |
IC50 = 13 nM
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CP0490725
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-pentylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H28ClNO5S
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1
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| 1 |
IC50 = 13.3 nM
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CP0508236
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-phenylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C22H22ClNO5S
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1
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| 1 |
IC50 = 13.3 nM
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CP0516852
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-chlorothiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H19Cl2NO5S2
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1
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| 1 |
IC50 = 13.3 nM
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CP0424910
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(2S,3R,4R,5S,6R)-2-(2,4-Dichloro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H19Cl2NO6S
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1
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| 1 |
IC50 = 13.3 nM
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CP0522901
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(methylthio)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C18H21ClN2O5S
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1
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| 1 |
IC50 = 13.4 nM
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CP0503823
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((S)-1-hydroxyethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO6S
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1
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| 1 |
IC50 = 13.5 nM
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CP0394828
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(1R,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-methylsulfanyl-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C22H25ClO6S
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1
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| 1 |
IC50 = 13.9 nM
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CP0529084
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(6S,7R,8R,9S)-6-[3-(4-Ethyl-benzyl)-4-methyl-phenyl]-2,2-dioxo-5-oxa-2lambda*6*-thia-spiro[3.5]nonane-7,8,9-triol
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C23H28O6S
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1
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| 1 |
IC50 = 14 nM
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CP0526586
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(2S,3R,4R,5S,6R)-2-(3-((5-(1,3,4-Thiadiazol-2-yl)thiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C18H18ClN3O5S2
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1
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| 1 |
IC50 = 14 nM
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CP0494448
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6,8-dichloro-4-[[5-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-1,4-benzoxazin-3-one
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C24H21Cl2F3N4O2
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1
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| 1 |
IC50 = 14 nM
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CP0460714
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(2S,3R,4R,5S,6R)-2-[3-(1-benzothiophen-2-ylmethyl)-4-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C22H24O6S
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1
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| 1 |
IC50 = 14 nM
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CP0536035
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(2S,3R,4R,5S,6R)-2-[3-(azulen-2-ylmethyl)-4-fluorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C23H23FO5
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1
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| 1 |
IC50 = 14 nM
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CP0453506
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[[4-(trifluoromethyl)phenyl]methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C21H21F3O6
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1
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| 1 |
IC50 = 14.2 nM
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CP0293282
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C19H19ClN2O5S2
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1
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| 1 |
IC50 = 14.4 nM
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CP0453507
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(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[[4-(trifluoromethoxy)phenyl]methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C21H21F3O7
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1
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| 1 |
IC50 = 14.5 nM
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CP0544080
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(2R,3S,4R,5R,6S)-2-(Hydroxymethyl)-6-(3-((5-(thiophen-3-yl)thiazol-2-yl)methyl)-4-(trifluoromethyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
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C22H21F3O5S2
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1
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| 1 |
IC50 = 14.6 nM
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CP0396637
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(2S,3R,4R,5S,6R)-2-[5-(azulen-2-ylmethyl)-2-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C24H26O6
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1
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| 1 |
IC50 = 16 nM
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CP0509572
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(2S,3R,4R,5S,6R)-2-(2-(Allyloxymethyl)-4-chloro-5-((5-(thiophen-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C24H26ClNO6S2
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1
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| 1 |
IC50 = 16.2 nM
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CP0173163
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-phenyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H21ClN2O5S
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1
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| 1 |
IC50 = 16.6 nM
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CP0509944
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-ethylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C18H22ClNO5S
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1
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| 1 |
IC50 = 16.7 nM
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CP0453323
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(3S,3'R,4'S,5'S,6'R)-5-[(4-chlorophenyl)methyl]-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C20H21ClO6
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1
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| 1 |
IC50 = 16.8 nM
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CP0315450
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(pentyloxy)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H29ClN2O6
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1
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| 1 |
IC50 = 17 nM
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CP0523809
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1-(beta-D-Glucopyranosyl)-3-(5-ethyl-2-thienylmethyl)benzene
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C19H24O6S
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1
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| 1 |
IC50 = 17 nM
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CP0465380
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(2S,3R,4R,5S,6R)-2-[3-(azulen-2-ylmethyl)-4-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C24H26O6
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1
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| 1 |
IC50 = 17 nM
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CP0226251
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(hexyloxy)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C23H31ClN2O6
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1
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| 1 |
IC50 = 17.3 nM
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CP0487489
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(2S,3R,4R,6R)-2-[5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-hydroxy-4-methoxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
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C22H24F2O7
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1
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| 1 |
IC50 = 17.3 nM
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CP0373297
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(2S,3R,4R,5S,6R)-2-(2-(allyloxymethyl)-4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H26ClNO7S
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1
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| 1 |
IC50 = 17.5 nM
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CP0188822
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H19ClN2O6S
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1
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| 1 |
IC50 = 17.7 nM
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CP0514778
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(5-chlorothiophen-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H18Cl2N2O5S2
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1
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| 1 |
IC50 = 18.2 nM
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CP0478483
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(methylthiomethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO5S2
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1
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| 1 |
IC50 = 18.6 nM
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CP0504577
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-ethoxythiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C18H22ClNO6S
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1
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| 1 |
IC50 = 18.8 nM
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CP0516855
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pentylthio)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H28ClNO5S2
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1
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| 1 |
IC50 = 18.9 nM
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CP0516854
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(2S,3R,4R,5S,6R)-2-(3-((5-butoxythiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H26ClNO6S
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1
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| 1 |
IC50 = 19.6 nM
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CP0375471
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)-2-(hydroxymethyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H22ClNO7S
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1
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| 1 |
IC50 = 20.5 nM
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CP0522289
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((S)-1-hydroxybut-3-enyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H24ClNO6S
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1
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| 1 |
IC50 = 20.8 nM
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CP0501852
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(2S,3R,4S,6S)-2-(4-chloro-3-(4-methoxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4-diol
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C20H23ClO5
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1
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| 1 |
IC50 = 21 nM
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CP0464981
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N-[6-chloro-4-[[5-[2-(4-chlorophenyl)ethyl]-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-3-oxo-1,4-benzoxazin-8-yl]-N-methylsulfonylmethanesulfonamide
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C24H24Cl2F3N5O6S2
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1
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| 1 |
IC50 = 21 nM
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CP0527240
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(2R,3R,4S,5S,6R)-2-[4-[[5-(4-fluorophenyl)thiophen-2-yl]methyl]-5-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C22H23FO5S2
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1
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| 1 |
IC50 = 21.1 nM
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CP0380473
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-fluorophenyl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H21ClFNO5S
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1
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| 1 |
IC50 = 21.2 nM
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CP0504916
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)-2-propoxyphenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H26ClNO7S
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1
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| 1 |
IC50 = 21.6 nM
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CP0326096
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiazol-4-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C18H18ClN3O5S2
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1
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| 1 |
IC50 = 21.8 nM
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CP0498707
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6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-8-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C22H18Cl2F3N5O4
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1
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| 1 |
IC50 = 22 nM
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CP0397650
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(2S,3R,4R,5S,6R)-2-[3-(azulen-2-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C23H24O5
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1
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| 1 |
IC50 = 22 nM
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CP0394827
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(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxy-3-fluorophenyl)methyl]phenyl]-1-ethoxy-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
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C23H26ClFO7
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1
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| 1 |
IC50 = 22.3 nM
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CP0502876
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(2S,3R,4R,5S,6R)-2-(3-((5-(Furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H21NO6S
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1
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| 1 |
IC50 = 22.6 nM
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CP0490988
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(6S,7R,8R,9S)-6-(4-chloro-3-(4-methoxybenzyl)phenyl)-2,5-dioxaspiro[3.5]nonane-7,8,9-triol
Show/Hide
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C21H23ClO6
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1
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| 1 |
IC50 = 23 nM
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CP0371970
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6,8-dichloro-4-((5-(4-chlorophenyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H14Cl3F3N4O2
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1
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| 1 |
IC50 = 23 nM
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CP0410030
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(methoxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H22ClNO6S
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1
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| 1 |
IC50 = 23.5 nM
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CP0522288
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((R)-1-hydroxyethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H22ClNO6S
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1
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| 1 |
IC50 = 23.8 nM
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CP0483769
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(2S,3R,4R,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-2-hydroxy-4-methoxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C22H22F2O6S
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1
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| 1 |
IC50 = 24.1 nM
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CP0527242
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(2R,3R,4S,5S,6R)-2-[5-[(4-ethylphenyl)methyl]-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H26O5S
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1
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| 1 |
IC50 = 24.8 nM
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CP0513941
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US8541380, 23
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C24H27ClN2O5S
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1
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| 1 |
IC50 = 24.9 nM
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CP0381805
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-cyclohexylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H28ClNO5S
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1
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| 1 |
IC50 = 25.4 nM
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CP0575756
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(2S,3R,4R,6R)-2-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-hydroxy-4-methoxyphenyl]-5,5-difluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C22H24F2O8
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1
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| 1 |
IC50 = 26.3 nM
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CP0529847
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(2S,3R,4R,5S,6R)-2-(4-Chloro-2-fluoro-5-((5-(4-fluorophenyl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H20ClF2NO5S
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1
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| 1 |
IC50 = 27.4 nM
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CP0530537
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(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[5-methyl-4-[(4-prop-2-enoxyphenyl)methyl]thiophen-2-yl]oxane-3,4,5-triol
Show/Hide
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C21H26O6S
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1
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| 1 |
IC50 = 27.5 nM
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CP0416344
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1-(beta-D-Glucopyranosyl)-4-chloro-3-(2-ethyl-5-pyridylmethyl)benzene
Show/Hide
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C20H24ClNO6
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1
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| 1 |
IC50 = 28 nM
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CP0547988
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(1R,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-pyridin-2-ylsulfanyl-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
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C26H26ClNO6S
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1
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| 1 |
IC50 = 28.4 nM
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CP0520792
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(2R,3R,4S,5S,6R)-2-[5-[(4-ethylphenyl)methyl]-3,4-dimethylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H28O5S
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1
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| 1 |
IC50 = 29.3 nM
|
|
|
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CP0516132
|
(3S,3'R,4'S,5'S,6'R)-6'-(hydroxymethyl)-5-[(4-hydroxyphenyl)methyl]spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
|
C20H22O7
|
1
|
| 1 |
IC50 = 29.9 nM
|
|
|
|
CP0465196
|
6-chloro-4-((5-(4-chlorophenethyl)-4-(cyclopropylmethyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C23H22Cl2N4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0466105
|
4-((4-butyl-5-(4-chlorophenethyl)-4H-1,2,4-triazol-3-yl)methyl)-6-chloro-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C23H24Cl2N4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0490441
|
(2S,3R,4R,5S,6R)-2-[3-(1-benzothiophen-2-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H22O5S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0173162
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pyridin-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H20ClN3O5S
|
1
|
| 1 |
IC50 = 30.3 nM
|
|
|
|
CP0522290
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((2-hydroxyethoxy)methyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H24ClNO7S
|
1
|
| 1 |
IC50 = 30.9 nM
|
|
|
|
CP0524070
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(ethylthio)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C18H22ClNO5S2
|
1
|
| 1 |
IC50 = 30.9 nM
|
|
|
|
CP0547987
|
(1S,2S,3R,4R,5S)-5-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-1-(2-hydroxyethoxy)-6,8-dioxabicyclo[3.2.1]octane-2,3,4-triol
Show/Hide
|
C23H27ClO8
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0527004
|
(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(ethylthiomethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H24ClNO5S2
|
1
|
| 1 |
IC50 = 31.9 nM
|
|
|
|
CP0447423
|
(6S,7R,8R,9S)-6-(4-chloro-3-(4-ethoxybenzyl)phenyl)-2,5-dioxaspiro[3.5]nonane-7,8,9-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0488883
|
1-(beta-D-Glucopyranosyl)-4-chloro-3-(1-phenyl-1H-pyrazol-4-ylmethyl)benzene
Show/Hide
|
C22H23ClN2O6
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0478537
|
(2S,3R,4R,5S,6R)-2-(2-(But-3-enyloxy)-4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H26ClNO7S
|
1
|
| 1 |
IC50 = 32.8 nM
|
|
|
|
CP0499419
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-hydroxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H21ClO6
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0508832
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-ethoxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H23ClO6S
|
1
|
| 1 |
IC50 = 34.6 nM
|
|
|
|
CP0395144
|
8-amino-6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C22H20Cl2F3N5O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0188825
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-methylpyridin-4-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H22ClN3O5S
|
1
|
| 1 |
IC50 = 36.4 nM
|
|
|
|
CP0526587
|
2-((5-(Furan-2-yl)thiazol-2-yl)methyl)-4-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-tetrahydro-2H-pyran-2-yl)benzonitrile
Show/Hide
|
C21H20N2O6S
|
1
|
| 1 |
IC50 = 36.7 nM
|
|
|
|
CP0513205
|
(2S,3R,4R,5S,6R)-2-(2-(Allyloxymethyl)-4-chloro-5-((5-(furan-3-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H26ClNO7S
|
1
|
| 1 |
IC50 = 38.7 nM
|
|
|
|
CP0536034
|
(2S,3R,4R,5S,6R)-2-[5-(azulen-2-ylmethyl)-2-fluorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H23FO5
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0507678
|
6-chloro-4-((5-(4-chlorophenethyl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C22H22Cl2N4O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0462811
|
6-chloro-8-nitro-4-((5-(pyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C19H14ClF3N6O4
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0293372
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-ethoxypyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H23ClN2O6
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0224177
|
(2S,3R,4R,5S,6R)-2-(3-((5-(Benzo[b]thiophen-2-yl)-1,3,4-thiadiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C23H21ClN2O5S2
|
1
|
| 1 |
IC50 = 44.5 nM
|
|
|
|
CP0488146
|
N-[[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]methyl]-N-methylbenzamide
Show/Hide
|
C28H30ClNO6
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0524312
|
US8541380, 21
Show/Hide
|
C20H20ClN3O5S
|
1
|
| 1 |
IC50 = 45.3 nM
|
|
|
|
CP0450847
|
(2S,3R,4R,5S,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-2-fluorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H21FO5S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0520791
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-ethylsulfanylphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H23ClO5S2
|
1
|
| 1 |
IC50 = 48.4 nM
|
|
|
|
CP0523649
|
(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(1-hydroxycyclopropyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H22ClNO6S
|
1
|
| 1 |
IC50 = 48.9 nM
|
|
|
|
CP0494410
|
(2R,3R,4S,5S,6R)-2-[5-[(4-ethylphenyl)methyl]-3-methoxy-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H28O6S
|
1
|
| 1 |
IC50 = 49.5 nM
|
|
|
|
CP0458752
|
(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[4-[(4-hydroxyphenyl)methyl]-5-methylthiophen-2-yl]oxane-3,4,5-triol
Show/Hide
|
C18H22O6S
|
1
|
| 1 |
IC50 = 50.2 nM
|
|
|
|
CP0489165
|
ethyl 2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-1,3-thiazole-5-carboxylate
Show/Hide
|
C19H22ClNO7S
|
1
|
| 1 |
IC50 = 50.3 nM
|
|
|
|
CP0509945
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-isopropylthiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H24ClNO5S
|
1
|
| 1 |
IC50 = 51.4 nM
|
|
|
|
CP0471519
|
(5R,7S,8R,9R,10S)-7-(3-(4-ethylbenzyl)-4-methylphenyl)-1,6-dioxaspiro[4.5]decane-8,9,10-triol
Show/Hide
|
C24H30O5
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0429135
|
US8541380, 20
Show/Hide
|
C20H20ClN3O5S
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0528834
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-prop-2-enoxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C20H23ClO6S
|
1
|
| 1 |
IC50 = 54.6 nM
|
|
|
|
CP0501309
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((R)-1-hydroxyallyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H22ClNO6S
|
1
|
| 1 |
IC50 = 54.8 nM
|
|
|
|
CP0380476
|
(2S,3R,4R,5S,6R)-2-(4-Cyclopropyl-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C23H25NO6S
|
1
|
| 1 |
IC50 = 54.8 nM
|
|
|
|
CP0511801
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-((S)-1-hydroxyallyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H22ClNO6S
|
1
|
| 1 |
IC50 = 54.9 nM
|
|
|
|
CP0455124
|
5-(4-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)methyl)benzylcarbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate
Show/Hide
|
C52H50ClN3O10
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0524071
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(propylthio)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H24ClNO5S2
|
1
|
| 1 |
IC50 = 56.4 nM
|
|
|
|
CP0498708
|
methyl 6-chloro-4-[[5-[2-(4-chlorophenyl)ethyl]-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-3-oxo-1,4-benzoxazine-8-carboxylate
Show/Hide
|
C24H21Cl2F3N4O4
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0503144
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-cyclopentyloxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H27ClO6S
|
1
|
| 1 |
IC50 = 57.2 nM
|
|
|
|
CP0376550
|
(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-methylfuran-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H21ClN2O6S
|
1
|
| 1 |
IC50 = 58.3 nM
|
|
|
|
CP0475799
|
(2S,3R,4R,5S,6R)-2-(3-((5-(Butylthio)thiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H26ClNO5S2
|
1
|
| 1 |
IC50 = 58.7 nM
|
|
|
|
CP0382875
|
(3S,4R,5R,6S)-6-(4-chloro-3-(4-methoxybenzyl)phenyl)-2,2-bis(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H25ClO7
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0486627
|
6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carbonitrile
Show/Hide
|
C23H18Cl2F3N5O2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0508654
|
(2S,3S,4R,5R,6S)-methyl 6-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylate
Show/Hide
|
C21H20ClNO7S
|
1
|
| 1 |
IC50 = 59.1 nM
|
|
|
|
CP0458753
|
(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[4-methyl-5-[(4-propylphenyl)methyl]thiophen-2-yl]oxane-3,4,5-triol
Show/Hide
|
C21H28O5S
|
1
|
| 1 |
IC50 = 59.8 nM
|
|
|
|
CP0498720
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-methylphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C18H21ClO5S
|
1
|
| 1 |
IC50 = 60.2 nM
|
|
|
|
CP0490831
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(furan-3-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H21ClN2O6
|
1
|
| 1 |
IC50 = 61.3 nM
|
|
|
|
CP0206473
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(furan-2-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H21ClN2O6
|
1
|
| 1 |
IC50 = 64.3 nM
|
|
|
|
CP0206474
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(pyridin-3-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H22ClN3O5
|
1
|
| 1 |
IC50 = 64.9 nM
|
|
|
|
CP0528833
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-propoxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C20H25ClO6S
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
|
CP0523648
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(ethoxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H24ClNO6S
|
1
|
| 1 |
IC50 = 68.7 nM
|
|
|
|
CP0379746
|
(2R,3S,4R,5R,6S)-2-((1H-tetrazol-1-yl)methyl)-6-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H20ClN5O5S
|
1
|
| 1 |
IC50 = 68.9 nM
|
|
|
|
CP0375880
|
(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[5-[(4-methoxyphenyl)methyl]-4-methylthiophen-2-yl]oxane-3,4,5-triol
Show/Hide
|
C19H24O6S
|
1
|
| 1 |
IC50 = 68.9 nM
|
|
|
|
CP0513065
|
(2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-[4-methyl-5-[(4-methylphenyl)methyl]thiophen-2-yl]oxane-3,4,5-triol
Show/Hide
|
C19H24O5S
|
1
|
| 1 |
IC50 = 69.6 nM
|
|
|
|
CP0438221
|
6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C22H19Cl2F3N4O2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0410800
|
(2S,3R,4R,5S,6R)-2-[5-[(4-ethylphenyl)methyl]-1H-pyrrol-3-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H25NO5
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0548192
|
(2S,3R,4R,5S,6R)-2-[5-(azulen-2-ylmethyl)-2-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H23ClO5
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0528754
|
(2R,3R,4S,5S,6R)-2-[5-chloro-4-[[4-(2-ethoxyethoxy)phenyl]methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H27ClO7S
|
1
|
| 1 |
IC50 = 70.7 nM
|
|
|
|
CP0224181
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-propoxypyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H25ClN2O6
|
1
|
| 1 |
IC50 = 70.8 nM
|
|
|
|
CP0435141
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(ethylthio)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C19H23ClN2O5S
|
1
|
| 1 |
IC50 = 71.3 nM
|
|
|
|
CP0469070
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(thiophen-2-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H21ClN2O5S
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1
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| 1 |
IC50 = 71.4 nM
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CP0435951
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(2R,3R,4S,5S,6R)-2-[5-[(4-ethoxyphenyl)methyl]-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C20H26O6S
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1
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| 1 |
IC50 = 71.4 nM
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CP0524315
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((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-(pyridin-4-yl)thiazol-5-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxylmethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H21ClN4O5S2
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1
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| 1 |
IC50 = 72.6 nM
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CP0524494
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6,8-dichloro-4-((5-((4-chlorophenoxy)methyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C21H16Cl3F3N4O3
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1
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| 1 |
IC50 = 73 nM
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CP0428906
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(2S,3R,4R,5S,6R)-2-[3-(1-benzothiophen-2-ylmethyl)-4-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H22O6S
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1
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| 1 |
IC50 = 75 nM
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CP0326016
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(thiophen-3-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H21ClN2O5S
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1
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| 1 |
IC50 = 75.4 nM
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CP0226252
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(tetrahydro-2H-pyran-4-yloxy)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C22H27ClN2O7
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1
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| 1 |
IC50 = 77.6 nM
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CP0504960
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4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-6-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one
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C21H21ClN4O2S
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1
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| 1 |
IC50 = 80 nM
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CP0175182
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(isoquinolin-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C24H22ClN3O5S
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1
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| 1 |
IC50 = 81.6 nM
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CP0082632
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(2S,3R,4R,5S,6R)-2-(3-((6-(benzo[d][1,3]dioxol-5-yl)pyridazin-3-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C24H23ClN2O7
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1
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| 1 |
IC50 = 82.7 nM
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CP0503284
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-methoxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C18H21ClO6S
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1
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| 1 |
IC50 = 86.5 nM
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CP0527241
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(2R,3R,4S,5S,6R)-2-[5-[(4-tert-butylphenyl)methyl]-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C22H30O5S
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1
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| 1 |
IC50 = 88.3 nM
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CP0512504
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6,8-dichloro-4-[[5-(2-phenylpropyl)-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-1,4-benzoxazin-3-one
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C23H21Cl2F3N4O2
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1
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| 1 |
IC50 = 89 nM
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CP0538848
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(2-hydroxypropan-2-yl)tetrahydro-2H-pyran-3,4,5-triol
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C22H24ClNO6S
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1
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| 1 |
IC50 = 89.5 nM
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CP0378176
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6-bromo-4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C20H18BrClN4O2S
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1
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| 1 |
IC50 = 90 nM
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CP0527961
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[[5-(4-fluorophenyl)thiophen-2-yl]methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H20ClFO5S2
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1
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| 1 |
IC50 = 91.3 nM
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CP0428905
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(2S,3R,4R,5S,6R)-2-[5-(1-benzothiophen-2-ylmethyl)-2-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H21ClO5S
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1
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| 1 |
IC50 = 92 nM
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CP0528835
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(2R,3R,4S,5S,6R)-2-[4-[(4-but-2-ynoxyphenyl)methyl]-5-chlorothiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H23ClO6S
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1
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| 1 |
IC50 = 94 nM
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CP0488148
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3-(3-((4-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)methyl)benzyl)(methyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C42H45BClF2N3O7
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1
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| 1 |
IC50 = 95 nM
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CP0381170
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(6-methylpyridin-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClN3O5S
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1
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| 1 |
IC50 = 97.4 nM
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CP0541196
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(2S,3R,4R,5S,6R)-2-[3-(azulen-6-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C23H24O5
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1
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| 1 |
IC50 = 99 nM
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CP0459334
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[5-[(4-methoxyphenyl)methyl]thiophen-3-yl]oxane-3,4,5-triol
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C18H22O6S
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1
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| 1 |
IC50 = 100 nM
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CP0506435
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24-[({6-[4-({2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl}methyl)phenoxy]hexyl}carbamoyl)methyl]-5,5,27,27-tetramethyl-16-oxa-12,20-diazaheptacyclo[15.11.0.0^{3,15}.0^{4,12}.0^{6,11}.0^{20,28}.0^{21,26}]octacosa-1(28),2,4(12),6(11),7,9,21(26),22,24-nonaen-12-ylium-8-sulfonate
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C56H64ClN3O11S
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1
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| 1 |
IC50 = 102 nM
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CP0173165
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C25H25ClN2O7
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1
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| 1 |
IC50 = 103 nM
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CP0224179
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US8541380, 22
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C22H23ClN2O5S
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1
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| 1 |
IC50 = 103 nM
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CP0226247
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-methylfuran-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C20H21ClN2O6S
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1
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| 1 |
IC50 = 106 nM
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CP0522291
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(2R,3S,4R,5R,6S)-2-((2H-tetrazol-2-yl)methyl)-6-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H20ClN5O5S
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1
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| 1 |
IC50 = 106 nM
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CP0490828
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(2S,3R,4R,5S,6R)-2-(3-((6-butoxypyridazin-3-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H27ClN2O6
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1
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| 1 |
IC50 = 109 nM
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CP0082631
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-isopropoxypyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H25ClN2O6
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1
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| 1 |
IC50 = 110 nM
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CP0502997
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1-((2S,3S,4R,5R,6S)-6-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-3,4,5-trihydroxytetrahydro-2H-pyran-2-yl)propan-1-one
Show/Hide
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C22H22ClNO6S
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1
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| 1 |
IC50 = 110 nM
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CP0465085
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6-chloro-3-oxo-4-((5-(pyridin-2-yl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carbonitrile
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C20H14ClF3N6O2
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1
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| 1 |
IC50 = 110 nM
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CP0514188
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(cyclohexyloxy)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H29ClN2O6
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1
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| 1 |
IC50 = 111 nM
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CP0501223
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-prop-2-ynoxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H21ClO6S
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1
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| 1 |
IC50 = 111 nM
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CP0503285
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[[4-(2-methoxyethoxy)phenyl]methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H25ClO7S
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1
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| 1 |
IC50 = 115 nM
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CP0487897
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4-[[(3S,3'R,4'S,5'S,6'R)-3',4',5'-trihydroxy-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-5-yl]methyl]benzonitrile
Show/Hide
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C21H21NO6
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1
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| 1 |
IC50 = 117.9 nM
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CP0224178
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((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(1-methyl-1Hpyrrol-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H22ClN3O5S
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1
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| 1 |
IC50 = 119 nM
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CP0502870
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(2S,3R,4R,5S,6R)-2-(3-((5-Butylthiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H26ClNO5S
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1
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| 1 |
IC50 = 119 nM
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CP0403129
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24-[({4-[4-({2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl}methyl)phenoxy]butyl}(methyl)carbamoyl)methyl]-5,5,27,27-tetramethyl-16-oxa-12,20-diazaheptacyclo[15.11.0.0^{3,15}.0^{4,12}.0^{6,11}.0^{20,28}.0^{21,26}]octacosa-1(28),2,4(12),6(11),7,9,21(26),22,24-nonaen-12-ylium-8-sulfonate
Show/Hide
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C55H62ClN3O11S
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1
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| 1 |
IC50 = 122 nM
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CP0513943
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-heptyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H31ClN2O5S
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1
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| 1 |
IC50 = 122 nM
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CP0480791
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(3S,3'R,4'S,5'S,6'R)-5-[(4-fluorophenyl)methyl]-6'-(hydroxymethyl)spiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
Show/Hide
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C20H21FO6
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1
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| 1 |
IC50 = 122.7 nM
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CP0455125
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3-(3-(4-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)methyl)benzylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
Show/Hide
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C41H43BClF2N3O7
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1
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| 1 |
IC50 = 123 nM
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CP0513944
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-chlorophenyl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H20Cl2N2O5S
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1
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| 1 |
IC50 = 126 nM
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CP0403130
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24-[({4-[4-({2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl}methyl)phenoxy]butyl}(ethyl)carbamoyl)methyl]-5,5,27,27-tetramethyl-16-oxa-12,20-diazaheptacyclo[15.11.0.0^{3,15}.0^{4,12}.0^{6,11}.0^{20,28}.0^{21,26}]octacosa-1(28),2,4(12),6(11),7,9,21(26),22,24-nonaen-12-ylium-8-sulfonate
Show/Hide
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C56H64ClN3O11S
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1
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| 1 |
IC50 = 131 nM
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CP0255698
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-ethylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H23ClN2O5
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1
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| 1 |
IC50 = 131 nM
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CP0502861
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(2S,3R,4R,5S,6R)-2-(2-(2-(1H-1,2,4-triazol-1-yl)ethoxy)-4-chloro-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H25ClN4O7S
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1
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| 1 |
IC50 = 131 nM
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CP0226254
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-pentylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H29ClN2O5
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1
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| 1 |
IC50 = 134 nM
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CP0501853
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(2S,3R,4R,5R,6R)-2-(3-(4-ethylbenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H28O5
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1
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| 1 |
IC50 = 139 nM
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CP0471518
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(2R,3S,4S,5R,6S)-6-(4-chloro-3-(4-methoxybenzyl)phenyl)-2-(hydroxymethyl)-5-methoxytetrahydro-2H-pyran-3,4-diol
Show/Hide
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C21H25ClO6
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1
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| 1 |
IC50 = 140 nM
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CP0504581
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2-((5-(Thiophen-3-yl)thiazol-2-yl)methyl)-4-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)-tetrahydro-2H-pyran-2-yl)benzonitrile
Show/Hide
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C21H20N2O5S2
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1
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| 1 |
IC50 = 140 nM
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CP0508833
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[(4-hydroxyphenyl)methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C17H19ClO6S
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1
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| 1 |
IC50 = 140 nM
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CP0431378
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24-[({4-[4-({2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl}methyl)phenoxy]butyl}carbamoyl)methyl]-5,5,27,27-tetramethyl-16-oxa-12,20-diazaheptacyclo[15.11.0.0^{3,15}.0^{4,12}.0^{6,11}.0^{20,28}.0^{21,26}]octacosa-1(28),2,4(12),6(11),7,9,21(26),22,24-nonaen-12-ylium-8-sulfonate
Show/Hide
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C54H60ClN3O11S
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1
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| 1 |
IC50 = 145 nM
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CP0226250
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-methoxy-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C16H19ClN2O6S
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1
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| 1 |
IC50 = 146 nM
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CP0500949
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3-(3-(6-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)hexylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
Show/Hide
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C39H47BClF2N3O7
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1
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| 1 |
IC50 = 148 nM
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CP0478567
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6-chloro-4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H18Cl2N4O2S
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1
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| 1 |
IC50 = 150 nM
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CP0495420
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8-chloro-4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H18Cl2N4O2S
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1
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| 1 |
IC50 = 150 nM
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CP0459551
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5-((4-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)methyl)benzyl)(methyl)carbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate
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C53H52ClN3O10
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1
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| 1 |
IC50 = 154 nM
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CP0473785
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3-(3-((4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butyl)(methyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
Show/Hide
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C38H45BClF2N3O7
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1
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| 1 |
IC50 = 155 nM
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CP0188824
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C16H16ClF3N2O5S
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1
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| 1 |
IC50 = 155 nM
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CP0538849
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(tosylmethyl)tetrahydro-2H-pyran-3,4,5-triol
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C27H26ClNO7S2
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1
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| 1 |
IC50 = 156 nM
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CP0438220
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6-chloro-4-((5-(4-chlorophenethyl)-4-isobutyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C23H24Cl2N4O2
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1
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| 1 |
IC50 = 160 nM
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CP0528836
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(2R,3R,4S,5S,6R)-2-[5-chloro-4-[[4-(oxolan-3-yloxy)phenyl]methyl]thiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H25ClO7S
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1
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| 1 |
IC50 = 162 nM
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CP0082633
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(5-methylthiophen-2-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C22H23ClN2O5S
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1
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| 1 |
IC50 = 168 nM
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CP0383398
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(phenylethynyl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C25H23ClN2O5
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1
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| 1 |
IC50 = 176 nM
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CP0401966
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-methoxybenzyl)phenyl)-6-(hydroxymethyl)-5-methoxytetrahydro-2H-pyran-3,4-diol
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C21H25ClO6
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1
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| 1 |
IC50 = 180 nM
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CP0498760
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4-((5-(4-chlorophenethyl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C23H22ClF3N4O2
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1
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| 1 |
IC50 = 180 nM
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CP0514777
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pyridazin-4-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C19H19ClN4O5S
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1
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| 1 |
IC50 = 190 nM
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CP0188826
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-chloropyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C17H18Cl2N2O5
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1
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| 1 |
IC50 = 202 nM
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CP0459547
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3-(3-(3-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)propylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C36H41BClF2N3O7
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1
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| 1 |
IC50 = 203 nM
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CP0388227
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3-(3-(8-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)octylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C41H51BClF2N3O7
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1
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| 1 |
IC50 = 205 nM
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CP0326099
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-propyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C18H23ClN2O5S
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1
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| 1 |
IC50 = 214 nM
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CP0435143
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-phenylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C23H23ClN2O5
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1
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| 1 |
IC50 = 222 nM
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CP0514155
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-propylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H25ClN2O5
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1
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| 1 |
IC50 = 237 nM
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CP0487899
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(3S,3'R,4'S,5'S,6'R)-5-[(4-ethylphenyl)methyl]-6'-(hydroxymethyl)-6-phenylspiro[1H-2-benzofuran-3,2'-oxane]-3',4',5'-triol
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C28H30O6
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1
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| 1 |
IC50 = 240.8 nM
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CP0381171
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(2S,3R,4R,5S,6R)-2-(3-((5-(Benzofuran-2-yl)-1,3,4-thiadiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H21ClN2O6S
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1
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| 1 |
IC50 = 249 nM
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CP0488305
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4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C21H18ClF3N4O2S
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1
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| 1 |
IC50 = 250 nM
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CP0241842
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-methylisoxazol-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C19H20ClN3O6S
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1
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| 1 |
IC50 = 257 nM
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CP0326018
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-isopropylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H25ClN2O5
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1
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| 1 |
IC50 = 259 nM
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CP0459549
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3-(3-(4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C37H43BClF2N3O7
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1
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| 1 |
IC50 = 267 nM
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CP0173166
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(4-fluorophenyl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C23H22ClFN2O5
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1
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| 1 |
IC50 = 272 nM
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CP0545813
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US9315438, Compound represented by formula (V)
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C25H29ClO6
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1
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| 1 |
IC50 = 281.83 nM
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CP0941704
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-((methyl(7-nitrobenzo[c][1,2,5]oxadiazol-4-yl)amino)methyl)benzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C27H27ClN4O8
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1
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| 1 |
IC50 = 286 nM
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CP0505751
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-methylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C18H21ClN2O5
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1
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| 1 |
IC50 = 293 nM
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CP0455139
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3-(3-((2-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)ethyl)(methyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C36H41BClF2N3O7
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1
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| 1 |
IC50 = 315 nM
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CP0455138
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5-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)benzyl)(methyl)carbamoyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
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C42H36ClNO11
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1
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| 1 |
IC50 = 350 nM
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CP0226253
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(3-methoxyphenyl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C24H25ClN2O6
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1
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| 1 |
IC50 = 351 nM
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CP0513942
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-pentyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C20H27ClN2O5S
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1
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| 1 |
IC50 = 353 nM
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CP0255699
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(2S,3R,4R,5S,6R)-2-(3-((6-butylpyridazin-3-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H27ClN2O5
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1
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| 1 |
IC50 = 356 nM
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CP0502588
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5-(5-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)pentanoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate
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C48H49ClN2O10
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1
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| 1 |
IC50 = 370 nM
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CP0378174
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4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]thiazin-3(4H)-one
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C21H18ClF3N4OS2
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1
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| 1 |
IC50 = 370 nM
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CP0381169
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(2S,3R,4R,5S,6R)-2-(3-((5-Butyl-1,3,4-thiadiazol-2-yl)methyl)-4-chlorophenyl)-6-(hydroxymethyl)-tetrahydro-2Hpyran-3,4,5-triol
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C19H25ClN2O5S
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1
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| 1 |
IC50 = 379 nM
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CP0388148
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3-(3-(2-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)ethylamino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
Show/Hide
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C35H39BClF2N3O7
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1
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| 1 |
IC50 = 420 nM
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CP0459548
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3-(3-((3-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)propyl)(methyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
Show/Hide
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C37H43BClF2N3O7
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1
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| 1 |
IC50 = 430 nM
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CP0466103
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7-chloro-4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H18Cl2N4O2S
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1
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| 1 |
IC50 = 430 nM
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CP0188828
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-isobutoxypyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H27ClN2O6
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1
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| 1 |
IC50 = 435 nM
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CP0326098
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-cyclopentyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C20H25ClN2O5S
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1
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| 1 |
IC50 = 445 nM
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CP0504769
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(2R,3R,4S,5S,6R)-2-[5-[(4-chlorophenyl)methyl]-4-methylthiophen-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C18H21ClO5S
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1
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| 1 |
IC50 = 451 nM
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CP0501311
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(2R,3S,4R,5R,6S)-2-((1H-1,2,4-triazol-1-yl)methyl)-6-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H21ClN4O5S
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1
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| 1 |
IC50 = 471 nM
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CP0462810
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6,8-dichloro-4-((5-(2-methyl-2-phenylpropyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C24H23Cl2F3N4O2
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1
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| 1 |
IC50 = 480 nM
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CP0412555
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N-[[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]methyl]benzamide
Show/Hide
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C27H28ClNO6
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1
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| 1 |
IC50 = 495 nM
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CP0519333
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7-bromo-4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C20H18BrClN4O2S
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1
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| 1 |
IC50 = 520 nM
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CP0514775
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US8541380, 24
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C21H27ClN2O5S
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1
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| 1 |
IC50 = 542 nM
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CP0321796
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((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(quinolin-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H22ClN3O5S
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1
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| 1 |
IC50 = 562 nM
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CP0490439
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(2S,3R,4R,5S,6R)-2-[6-[(4-ethylphenyl)methyl]pyridin-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C20H25NO5
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1
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| 1 |
IC50 = 610 nM
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CP0293371
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(6-methylpyridin-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H22ClN3O5S
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1
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| 1 |
IC50 = 638 nM
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CP0466104
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4-((5-(4-chlorophenethyl)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C22H20ClF3N4O2
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1
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| 1 |
IC50 = 640 nM
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CP0490448
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(2S,3R,4R,5S,6R)-2-[3-(1,3-benzothiazol-2-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C20H21NO5S
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1
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| 1 |
IC50 = 650 nM
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CP0464982
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6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-8-(methylsulfonyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
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C23H21Cl2F3N4O4S
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1
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| 1 |
IC50 = 660 nM
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CP0508411
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(2S,3R,4R,5S,6R)-2-[3-(1-benzofuran-2-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H22O6
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1
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| 1 |
IC50 = 675 nM
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CP0326022
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-morpholinopyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H26ClN3O6
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1
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| 1 |
IC50 = 700 nM
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CP0326094
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-chlorothiophen-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H18Cl2N2O5S2
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1
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| 1 |
IC50 = 712 nM
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CP0941501
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(2S,3R,4R,5S,6R)-2-(4-chloro-2-(2-(dimethylamino)ethoxy)-5-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol trifluoroacetic acid salt
Show/Hide
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C26H30ClF3N2O9S
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1
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| 1 |
IC50 = 713 nM
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CP0284847
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2,2,2-trifluoroethyl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C17H18ClF3N2O5S
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1
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| 1 |
IC50 = 758 nM
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CP0463873
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-methylthiophen-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H21ClN2O5S2
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1
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| 1 |
IC50 = 762 nM
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CP0326020
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-isobutylpyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H27ClN2O5
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1
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| 1 |
IC50 = 811 nM
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CP0506434
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5-(5-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)pentanoyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
Show/Hide
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C44H39ClO12
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1
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| 1 |
IC50 = 835 nM
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CP0459550
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3-(3-((4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butyl)(propyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C40H49BClF2N3O7
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1
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| 1 |
IC50 = 850 nM
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CP0470817
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1-(beta-D-Glucopyranosyl)-3-(5-ethyl-2-furylmethyl)benzene
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C19H24O7
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1
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| 1 |
IC50 = 920 nM
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CP0463934
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(2S,3R,4R,5S,6R)-2-[3-[(1-benzylazulen-2-yl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C30H30O5
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1
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| 1 |
IC50 = 970 nM
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CP0501851
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(2R,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylbenzyloxy)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C23H30O6
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1
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| 1 |
IC50 = 1000 nM
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CP0504284
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(pyrrolidin-1-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H26ClN3O5
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1
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| 1 |
IC50 = 1040 nM
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CP0378175
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4-((5-(4-chlorobenzylthio)-4-cyclopropyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]thiazin-3(4H)-one
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C22H18ClF3N4OS2
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1
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| 1 |
IC50 = 1100 nM
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CP0515864
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US9315438, Compound represented by formula (IV)
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C25H29ClO6
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1
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| 1 |
IC50 = 1110.95 nM
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CP0505754
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(2S,3R,4R,5S,6R)-2-[3-[(6-anilinopyridazin-3-yl)methyl]-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C23H24ClN3O5
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1
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| 1 |
IC50 = 1140 nM
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CP0425966
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4-((5-(4-chlorobenzylthio)-4-isopropyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]thiazin-3(4H)-one
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C22H20ClF3N4OS2
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1
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| 1 |
IC50 = 1200 nM
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CP0514774
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(2R,3S,4R,5R)-2-(Hydroxymethyl)-6-(3-((5-(pyridin-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-tetrahydro-2H-pyran-3,4,5-triol
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C20H21N3O5S
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1
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| 1 |
IC50 = 1230 nM
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CP0466100
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4-((5-(4-chlorobenzylthio)-4-methyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]thiazin-3(4H)-one
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C20H16ClF3N4OS2
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1
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| 1 |
IC50 = 1400 nM
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CP0524311
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(2R,3S,4R,5R)-2-(Hydroxymethyl)-6-(3-((5-phenyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22N2O5S
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1
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| 1 |
IC50 = 1420 nM
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CP0501310
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(2S,3R,4R,5S,6S)-2-(4-chloro-3-((5-(furan-2-yl)thiazol-2-yl)methyl)phenyl)-6-(methylsulfonylmethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO7S2
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1
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| 1 |
IC50 = 1450 nM
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CP0321747
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-methyl-6-(methylthio)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C19H23ClN2O5S
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1
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| 1 |
IC50 = 1520 nM
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CP0498041
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3-(3-((4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butyl)(isopropyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C40H49BClF2N3O7
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1
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| 1 |
IC50 = 1570 nM
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CP0456340
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6-chloro-4-((5-(4-chlorophenethyl)-4-cyclopropyl-4H-1,2,4-triazol-3-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
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C22H20Cl2N4O2
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1
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| 1 |
IC50 = 1580 nM
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CP0255696
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(5-methyloxazol-2-yl)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClN3O6
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1
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| 1 |
IC50 = 1710 nM
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CP0390808
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(phenylthio)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C23H23ClN2O5S
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1
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| 1 |
IC50 = 1870 nM
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CP0403128
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3-(3-((4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butyl)(isobutyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C41H51BClF2N3O7
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1
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| 1 |
IC50 = 2000 nM
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CP0518875
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(2S,3R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,5-diol
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C22H28O4
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1
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| 1 |
IC50 = 2000 nM
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CP0501620
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4-((5-(4-chlorobenzylthio)-4-ethyl-4H-1,2,4-triazol-3-yl)methyl)-6-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
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C20H18ClN5O4S
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1
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| 1 |
IC50 = 2100 nM
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CP0466101
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4-((5-(4-chlorobenzylthio)-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)-6-(trifluoromethyl)-2H-benzo[b][1,4]thiazin-3(4H)-one
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C25H18ClF3N4OS2
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1
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| 1 |
IC50 = 2110 nM
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CP0526131
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(2S,3R,4R,5S,6R)-2-[3-(1,3-benzoxazol-2-ylmethyl)phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C20H21NO6
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1
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| 1 |
IC50 = 2300 nM
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CP0438913
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(3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-chlorobenzyl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C22H22Cl2N2O5S
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1
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| 1 |
IC50 = 2390 nM
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CP0890958
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-((7-nitrobenzo[c][1,2,5]oxadiazol-4-ylamino)methyl)benzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C26H25ClN4O8
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1
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| 1 |
IC50 = 2400 nM
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CP0521418
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(1-methyl-1Hindazol-3-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H23ClN4O5S
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1
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| 1 |
IC50 = 3280 nM
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CP0382871
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(2S,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C22H28O5
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1
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| 1 |
IC50 = 3700 nM
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CP0508410
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(2S,3R,4R,5S,6R)-2-[6-[(4-ethylphenyl)methyl]pyrazin-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C19H24N2O5
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1
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| 1 |
IC50 = 4900 nM
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CP0373531
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(6S,7R,8R,9S)-6-(3-(4-ethylbenzyl)-4-methylphenyl)-5-oxa-2-azaspiro[3.5]nonane-7,8,9-triol
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C23H29NO4
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1
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| 1 |
IC50 = 5100 nM
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CP0395151
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6-chloro-4-((5-(3-methylpyridin-2-yl)-4-propyl-4H-1,2,4-triazol-3-yl)methyl)-8-nitro-2H-benzo[b][1,4]oxazin-3(4H)-one
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C20H19ClN6O4
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1
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| 1 |
IC50 = 5100 nM
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CP0397738
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(2S,3R,4R,5S,6R)-2-[3-[(1-ethylazulen-2-yl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C25H28O5
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1
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| 1 |
IC50 = 5200 nM
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CP0450846
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[3-[(1-methylindol-2-yl)methyl]phenyl]oxane-3,4,5-triol
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C22H25NO5
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1
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| 1 |
IC50 = 6300 nM
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CP0513940
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C18H24N2O5S
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1
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| 1 |
IC50 = 6910 nM
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CP0498040
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5-(6-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)benzylamino)-6-oxohexylcarbamoyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
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C47H45ClN2O12
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1
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| 1 |
IC50 = 8000 nM
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CP0502726
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N-[6-chloro-4-[[5-[2-(4-chlorophenyl)ethyl]-4-(3,3,3-trifluoropropyl)-1,2,4-triazol-3-yl]methyl]-3-oxo-1,4-benzoxazin-8-yl]acetamide
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C24H22Cl2F3N5O3
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1
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| 1 |
IC50 = 9800 nM
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CP0504721
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(2R,3S,4R,6R)-6-(3-(4-ethylbenzyl)-4-methylphenyl)-2-(hydroxymethyl)tetrahydro-2H-pyran-3,4-diol
Show/Hide
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C22H28O4
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1
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| 1 |
IC50 > 10000 nM
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CP0495872
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((4,5-dimethyl-6-(methylthio)pyridazin-3-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H25ClN2O5S
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1
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| 1 |
IC50 = 10000 nM
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CP0526785
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(2S,3R,4R,5S,6R)-2-(4-chloro-3-((4-methylphthalazin-1-yl)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H23ClN2O5
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1
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| 1 |
IC50 = 10000 nM
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CP0381168
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(3R,4R,5S,6R)-2-(3-((5-tert-Butyl-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H26N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0434150
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(3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-(4-chlorophenyl)propan-2-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H26Cl2N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0514779
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((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-ethyl-5-methylisoxazol-4-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C21H24ClN3O6S
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1
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| 1 |
IC50 > 10000 nM
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CP0521420
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(2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3,5-dimethylisoxazol-4-yl)-1,3,4-thiadiazol-2-yl)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C20H22ClN3O6S
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1
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| 1 |
IC50 > 10000 nM
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CP0544079
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2-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)thiazole-5-carboxylic acid
Show/Hide
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C17H18ClNO7S
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1
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| 1 |
IC50 > 10000 nM
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CP0498486
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6-chloro-4-((5-(4-chlorophenethyl)-4-(3,3,3-trifluoropropyl)-4H-1,2,4-triazol-3-yl)methyl)-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazine-8-carboxylic acid
Show/Hide
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C23H19Cl2F3N4O4
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1
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| 1 |
IC50 = 10000 nM
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CP0459546
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5-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)benzylcarbamoyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
Show/Hide
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C41H34ClNO11
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1
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| 1 |
IC50 = 11000 nM
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CP0397737
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1-[2-[[3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]azulen-1-yl]ethanone
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C25H26O6
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1
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| 1 |
IC50 = 12000 nM
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CP0474979
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5-(6-((4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzyl)benzyl)(methyl)amino)-6-oxohexylcarbamoyl)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
Show/Hide
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C48H47ClN2O12
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1
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| 1 |
IC50 = 15050 nM
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CP0463933
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[3-[(3-methylazulen-1-yl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
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C24H26O5
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1
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| 1 |
IC50 = 44000 nM
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CP0428903
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[3-(pyrazin-2-ylmethyl)phenyl]oxane-3,4,5-triol
Show/Hide
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C17H20N2O5
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1
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| 1 |
IC50 > 100000 nM
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CP0450320
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[3-[(1-methylbenzimidazol-2-yl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
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C21H24N2O5
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1
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| 1 |
IC50 > 100000 nM
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CP0490440
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[3-(pyridin-2-ylmethyl)phenyl]oxane-3,4,5-triol
Show/Hide
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C18H21NO5
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1
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| 1 |
IC50 > 100000 nM
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