Compound ID |
Compound Name |
Compound Formula |
CP0385472
|
(1R,2R)-N-[(2S,3S)-2-amino-3-methylpentyl]-N-[4-(4-propylphenyl)phenyl]-2-pyridin-2-ylcyclopropane-1-carboxamide
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|
C30H37N3O
|
1
|
1 |
EC50 = 50 nM
|
|
|
CP0579787
|
(2S)-N-[(1S)-2-(5-amino-1,3,4-oxadiazol-2-yl)-1-[4-(2-methylpentoxy)phenyl]ethyl]-2-phenylpropanamide
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|
C25H32N4O3
|
1
|
1 |
EC50 = 59 nM
|
|
|
CP0572976
|
(2S)-N-[(1R)-2-(methylamino)-1-[4-(2-methylpentoxy)phenyl]-2-oxoethyl]-2-phenylpropanamide
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|
C24H32N2O3
|
1
|
1 |
EC50 = 295 nM
|
|
|
CP0385442
|
(2S)-N-[(1R)-2-amino-1-[4-(2-methylpentoxy)phenyl]ethyl]-2-phenylpropanamide
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|
C23H32N2O2
|
1
|
1 |
EC50 = 414 nM
|
|
|
CP0558121
|
(2S)-N-[(R)-(5-methyl-1,3,4-oxadiazol-2-yl)-[4-(2-methylpentoxy)phenyl]methyl]-2-phenylpropanamide
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|
C25H31N3O3
|
1
|
1 |
EC50 = 525 nM
|
|
|
CP0507405
|
(2S)-N-[(1R)-1-[4-(cyclobutylmethoxy)phenyl]-2-oxo-2-(1,3-thiazol-2-ylmethylamino)ethyl]-2-phenylpropanamide
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|
C26H29N3O3S
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0465025
|
(2R)-2-[4-(2-methylpentoxy)phenyl]-2-[[(2S)-2-phenylpropanoyl]amino]acetic acid
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|
C23H29NO4
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0465028
|
methyl (2R)-2-[[2-(4-cyanophenyl)acetyl]amino]-2-[4-(2-methylpentoxy)phenyl]acetate
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|
C24H28N2O4
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0565313
|
methyl (2R)-2-(2-cyclohexylpropanoylamino)-2-[4-(2-methylpentoxy)phenyl]acetate
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|
C24H37NO4
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0466089
|
(2S)-N-[(1R)-2-hydroxy-1-[4-[(1-methylcyclobutyl)methoxy]phenyl]ethyl]-2-phenylpropanamide
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|
C23H29NO3
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0466158
|
(2S)-N-[(1R)-2-hydroxy-1-[4-(spiro[2.3]hexan-5-ylmethoxy)phenyl]ethyl]-2-phenylpropanamide
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|
C24H29NO3
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0558135
|
(2S)-N-[(1R)-1-[4-[(3,3-dimethylcyclobutyl)methoxy]phenyl]-2-hydroxyethyl]-2-phenylpropanamide
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|
C24H31NO3
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0558136
|
(2S)-N-[(1R)-2-(azetidin-3-ylmethylamino)-1-[4-(2-methylpentoxy)phenyl]-2-oxoethyl]-2-phenylpropanamide
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|
C27H37N3O3
|
1
|
1 |
EC50 > 10000 nM
|
|
|