| Compound ID |
Compound Name |
Compound Formula |
|
CP0332383
|
[(1S,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] 3,5-dichlorobenzoate
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|
C15H17Cl2NO2
|
1
|
| 1 |
IC50 = 6.9 nM
|
|
|
|
CP0022161
|
CAS_40796-97-2
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|
C15H17Cl2NO2
|
1
|
| 1 |
IC50 = 6.9 nM
|
|
|
|
CP0795225
|
1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylaminocarbonyl)oxime
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|
C19H16N2O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0510682
|
3-methyl-4-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-1H-pyridazin-6-one
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|
C19H25N3O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0078124
|
5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-2-pyridin-2-ylpyridazin-3-one
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|
C23H26N4O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0499752
|
6-methyl-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-2-pyridin-2-ylpyridazin-3-one
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|
C24H28N4O2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0418405
|
2-(6-methylpyridin-2-yl)-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyridazin-3-one
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|
C24H28N4O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0508912
|
2-methyl-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyridazin-3-one
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|
C19H25N3O2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0046463
|
3-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-1H-pyridazin-6-one
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|
C18H23N3O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0431282
|
2,6-dimethyl-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyridazin-3-one
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|
C20H27N3O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0431283
|
2-(3-methylpyridin-2-yl)-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyridazin-3-one
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|
C24H28N4O2
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0499754
|
5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-2-propan-2-ylpyridazin-3-one
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|
C21H29N3O2
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0397274
|
4-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-1H-pyridazin-6-one
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|
C18H23N3O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0418406
|
6-methyl-2-(3-methylpyridin-2-yl)-5-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyridazin-3-one
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|
C25H30N4O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0456828
|
4-[4-[3-(azepan-1-yl)propoxy]phenyl]-3-methyl-1H-pyridazin-6-one
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|
C20H27N3O2
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0495133
|
5-[4-[3-(azepan-1-yl)propoxy]phenyl]-2-pyridin-2-ylpyridazin-3-one
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|
C24H28N4O2
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0517440
|
5-[4-(3-piperidin-1-ylpropoxy)phenyl]-2-pyridin-2-ylpyridazin-3-one
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|
C23H26N4O2
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0459851
|
3-methyl-4-[4-(3-piperidin-1-ylpropoxy)phenyl]-1H-pyridazin-6-one
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|
C19H25N3O2
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0416894
|
5-[4-[3-(azepan-1-yl)propoxy]phenyl]-2-methylpyridazin-3-one
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|
C20H27N3O2
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0416895
|
2,6-dimethyl-5-[4-(3-piperidin-1-ylpropoxy)phenyl]pyridazin-3-one
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|
C20H27N3O2
|
1
|
| 1 |
Ki = 8.9 nM
|
|
|
|
CP0418409
|
5-[4-[3-[(2S)-2-methylpyrrolidin-1-yl]propoxy]phenyl]-2-pyridin-2-ylpyridazin-3-one
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|
C23H26N4O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0418408
|
2-methyl-5-[4-(3-piperidin-1-ylpropoxy)phenyl]pyridazin-3-one
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|
C19H25N3O2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0391333
|
4-[4-(3-piperidin-1-ylpropoxy)phenyl]-1H-pyridazin-6-one
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|
C18H23N3O2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
