| Compound ID |
Compound Name |
Compound Formula |
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CP0130814
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C33H50N12O4
|
1
|
| 1 |
Ki = 0.81 nM
|
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CP0512633
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(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(diaminomethylideneamino)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C32H49N15O4
|
1
|
| 1 |
Ki = 0.83 nM
|
|
|
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CP0528191
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(2S,3S)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]-3-methylpentanamide
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|
C34H52N12O4
|
1
|
| 1 |
Ki = 0.84 nM
|
|
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CP0457399
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C37H50N12O4
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
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CP0506636
|
(2S)-6-amino-N-[(4-carbamimidoylphenyl)methyl]-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]-3-methylbutanoyl]amino]hexanamide
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|
C33H50N10O4
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
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CP0428275
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C37H50N12O5
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0375110
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C34H53N15O4
|
1
|
| 1 |
Ki = 3 nM
|
|
|
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CP0507962
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(2S)-N-[(2S)-3-amino-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C31H47N13O4
|
1
|
| 1 |
Ki = 3 nM
|
|
|
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CP0527378
|
(2S)-6-amino-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]hexanamide
Show/Hide
|
C34H53N13O4
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
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CP0473546
|
(2S)-6-amino-2-[[(2S)-3-amino-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]propanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]hexanamide
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|
C31H47N11O4
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
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CP0528900
|
(2S)-N-[(2R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C31H46N12O4S
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
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CP0376045
|
(2S)-N-[(2S,3R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C32H48N12O5
|
1
|
| 1 |
Ki = 6 nM
|
|
|
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CP0512634
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C34H48N14O4
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
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CP0513820
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C39H51N13O4
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
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CP0501244
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
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|
C33H50N12O4S
|
1
|
| 1 |
Ki = 9.7 nM
|
|
|
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CP0425432
|
(2S)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]-4-methylpentanamide
Show/Hide
|
C34H52N12O4
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0505324
|
(2S)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]pentanediamide
Show/Hide
|
C33H49N13O5
|
1
|
| 1 |
Ki = 13 nM
|
|
|
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CP0471604
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C31H46N12O4
|
1
|
| 1 |
Ki = 19 nM
|
|
|
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CP0534797
|
(2S)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-2-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]butanediamide
Show/Hide
|
C32H47N13O5
|
1
|
| 1 |
Ki = 23 nM
|
|
|
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CP0527379
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C31H46N12O5
|
1
|
| 1 |
Ki = 24 nM
|
|
|
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CP0506633
|
(2S)-N-[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]pyrrolidine-2-carboxamide
Show/Hide
|
C33H48N12O4
|
1
|
| 1 |
Ki = 37 nM
|
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CP0457400
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(2S)-N-[2-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-2-oxoethyl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C30H44N12O4
|
1
|
| 1 |
Ki = 40 nM
|
|
|
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CP0457404
|
(4S)-5-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]-5-oxopentanoic acid
Show/Hide
|
C33H48N12O6
|
1
|
| 1 |
Ki = 102 nM
|
|
|
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CP0506634
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(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-methylamino]-3-methyl-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C34H52N12O4
|
1
|
| 1 |
Ki = 142 nM
|
|
|
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CP0431722
|
(2S)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-5-(carbamoylamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C33H49N11O5
|
1
|
| 1 |
Ki = 238 nM
|
|
|
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CP0527185
|
(2S)-6-amino-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-2-[(2-phenylacetyl)amino]hexanamide
Show/Hide
|
C33H50N10O4
|
1
|
| 1 |
Ki = 285 nM
|
|
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CP0428276
|
(3S)-4-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-[[(2S)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]-4-oxobutanoic acid
Show/Hide
|
C32H46N12O6
|
1
|
| 1 |
Ki = 405 nM
|
|
|
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CP0512635
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benzyl N-[(5S)-6-[[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-6-oxo-5-[(2-phenylacetyl)amino]hexyl]carbamate
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|
C41H56N10O6
|
1
|
| 1 |
Ki = 702 nM
|
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CP0512638
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(2R)-N-[(2S)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C33H50N12O4
|
1
|
| 1 |
Ki = 970 nM
|
|
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CP0457406
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(2S)-N-[(2R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C33H50N12O4
|
1
|
| 1 |
Ki = 1110 nM
|
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CP0512636
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(2S)-N-[(2R)-1-[[(2S)-1-[(4-carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanamide
Show/Hide
|
C31H46N12O4
|
1
|
| 1 |
Ki = 1385 nM
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CP0501245
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(2S)-2-[[(2S)-2-acetamido-3-methylbutanoyl]amino]-N-[(4-carbamimidoylphenyl)methyl]-5-(diaminomethylideneamino)pentanamide
Show/Hide
|
C21H34N8O3
|
1
|
| 1 |
Ki = 2390 nM
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CP0528192
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(2S)-5-(diaminomethylideneamino)-2-[[(2R)-5-(diaminomethylideneamino)-2-[(2-phenylacetyl)amino]pentanoyl]amino]pentanoic acid
Show/Hide
|
C20H32N8O4
|
1
|
| 1 |
Ki = 3200 nM
|
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CP0468839
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(2S)-N-[(4-carbamimidoylphenyl)methyl]-5-(diaminomethylideneamino)-2-[[(2R)-5-(diaminomethylideneamino)-2-[[(2S)-3-methyl-2-[(2-phenylacetyl)amino]butanoyl]amino]pentanoyl]amino]pentanamide
Show/Hide
|
C33H50N12O4
|
1
|
| 1 |
Ki = 7340 nM
|
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