| Compound ID |
Compound Name |
Compound Formula |
|
CP0057612
|
[(8R,9S,13S,14S)-13-methyl-17-oxo-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-yl] sulfamate
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|
C18H23NO4S
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
IC50 = 30 nM
|
|
|
|
CP0090287
|
[2-(1-adamantyl)-4-oxochromen-6-yl] sulfamate
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|
C19H21NO5S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0124667
|
[2-(1-adamantyl)-4-oxothiochromen-6-yl] sulfamate
Show/Hide
|
C19H21NO4S2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0306019
|
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxylic acid
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|
C20H20O3S
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0268929
|
4-(4-Bromo-2,5-dichloro-thiophene-3-sulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C15H19BrCl2N2O5S2
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0257149
|
4-(3,5-Bis-trifluoromethyl-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C19H22F6N2O5S
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0279787
|
4-(3,5-Dichloro-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C17H22Cl2N2O5S
|
1
|
| 1 |
IC50 = 1260 nM
|
|
|
|
CP0083400
|
[(1R,5S)-8-[[3,5-bis(trifluoromethyl)phenyl]sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C24H22F6N2O5S
|
1
|
| 1 |
IC50 = 1890 nM
|
|
|
|
CP0275823
|
8-[N-(4-chlorophenylsulfonamido)-carbonyl amino]-8-azabicyclo[3.2.1]oct-3-yl 2-phenylacetate
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|
C22H24ClN3O5S
|
1
|
| 1 |
IC50 = 3840 nM
|
|
|
|
CP0100227
|
[(1S,5R)-8-[2-(4-chlorophenyl)sulfonylacetyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
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|
C23H24ClNO5S
|
1
|
| 1 |
IC50 = 4320 nM
|
|
|
|
CP0178399
|
[(1R,5S)-8-[(4-bromophenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C22H23BrN2O5S
|
1
|
| 1 |
IC50 = 6150 nM
|
|
|
|
CP0061865
|
[(1R,5S)-8-[(4-chlorophenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C22H23ClN2O5S
|
2
|
| 1 |
IC50 = 6270 nM
|
|
|
| 2 |
IC50 = 6720 nM
|
|
|
|
CP0083806
|
[(1S,5R)-8-[[4-(trifluoromethyl)phenyl]sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C23H23F3N2O5S
|
1
|
| 1 |
IC50 = 7470 nM
|
|
|
|
CP0207559
|
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid
Show/Hide
|
C20H20O4
|
1
|
| 1 |
IC50 = 9400 nM
|
|
|
|
CP0111687
|
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C17H23ClN2O5S
|
1
|
| 1 |
IC50 = 9800 nM
|
|
|
|
CP0245139
|
4-(2,6-Dichloro-benzenesulfonylaminocarbonyl)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C17H22Cl2N2O5S
|
1
|
| 1 |
IC50 = 9900 nM
|
|
|
|
CP0175644
|
[(1R,5S)-8-[(4-chlorobenzoyl)carbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C23H23ClN2O4
|
1
|
| 1 |
IC50 = 10400 nM
|
|
|
|
CP0285303
|
4-(4-Chloro-benzenesulfonylaminocarbonyl)-piperazine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C16H22ClN3O5S
|
1
|
| 1 |
IC50 = 12000 nM
|
|
|
|
CP0132984
|
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-oxo-acetic acid
Show/Hide
|
C21H20O5
|
1
|
| 1 |
IC50 = 12300 nM
|
|
|
|
CP0177917
|
[1-[(4-chlorophenyl)sulfonylcarbamoyl]-4-cyanopiperidin-4-yl] 2-phenylacetate
Show/Hide
|
C21H20ClN3O5S
|
1
|
| 1 |
IC50 = 24500 nM
|
|
|
|
CP0244557
|
[(1S,5R)-8-(benzenesulfonylcarbamoyl)-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C22H24N2O5S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0285030
|
[1-[(4-chlorophenyl)sulfonylcarbamoyl]piperidin-4-yl] 2-phenylacetate
Show/Hide
|
C20H21ClN2O5S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0068080
|
2-Adamantan-1-yl-6-(2-hydroxy-acetyl)-chromen-4-one
Show/Hide
|
C21H22O4
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0068081
|
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid methyl ester
Show/Hide
|
C21H22O4
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0077442
|
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carbaldehyde
Show/Hide
|
C20H20O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0077444
|
(2-Adamantan-1-yl-4-oxo-4H-chromen-6-yl)-acetic acid
Show/Hide
|
C21H22O4
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0277392
|
2-Adamantan-1-yl-4-oxo-4H-chromene-6-carboxylic acid amide
Show/Hide
|
C20H21NO3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0281838
|
2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carbonitrile
Show/Hide
|
C20H19NOS
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0037702
|
[(1S,5R)-8-[(4-methylphenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C23H26N2O5S
|
1
|
| 1 |
IC50 = 37100 nM
|
|
|
|
CP0050738
|
[(1R,5S)-8-[(4-fluorophenyl)sulfonylcarbamoyl]-8-azabicyclo[3.2.1]octan-3-yl] 2-phenylacetate
Show/Hide
|
C22H23FN2O5S
|
1
|
| 1 |
IC50 = 39200 nM
|
|
|
|
CP0256733
|
2-Adamantan-1-yl-6-hydroxymethyl-chromen-4-one
Show/Hide
|
C20H22O3
|
1
|
| 1 |
IC50 ~ 30000 nM
|
|
|
