| Compound ID |
Compound Name |
Compound Formula |
|
CP0418063
|
CAS_81447-78-1
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|
C11H12Cl2N2O
|
2
|
| 1 |
EC50 = 1.38 nM
|
|
|
| 2 |
Ki = 69.18 nM
|
|
|
|
CP0087650
|
2-[1-[2-(cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C15H20N2O
|
2
|
| 1 |
EC50 = 1.995 nM
|
|
|
| 2 |
Ki = 275.42 nM
|
|
|
|
CP0157934
|
2-[(1S)-1-[2-(cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C15H20N2O
|
2
|
| 1 |
EC50 = 1.995 nM
|
|
|
| 2 |
Ki = 275.42 nM
|
|
|
|
CP0416730
|
5-chloro-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylsulfanylaniline
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|
C11H14ClN3S
|
2
|
| 1 |
EC50 = 2.818 nM
|
|
|
| 2 |
Ki = 169.82 nM
|
|
|
|
CP0425305
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-fluoro-2-methylsulfanylaniline
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|
C11H14FN3S
|
2
|
| 1 |
EC50 = 5.623 nM
|
|
|
| 2 |
Ki = 114.82 nM
|
|
|
|
CP0874395
|
(4,5-Dihydro-1H-imidazol-2-ylmethyl)-(2-methylsulfanyl-phenyl)-amine hydrochloride
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|
C11H16ClN3S
|
2
|
| 1 |
EC50 = 5.623 nM
|
|
|
| 2 |
Ki = 144.54 nM
|
|
|
|
CP0417504
|
2-[(1S)-1-(2-thiophen-3-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C15H16N2OS
|
2
|
| 1 |
EC50 = 6.31 nM
|
|
|
| 2 |
Ki = 125.89 nM
|
|
|
|
CP0420934
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylsulfanyl-5-(trifluoromethyl)aniline
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|
C12H14F3N3S
|
2
|
| 1 |
EC50 = 7.943 nM
|
|
|
| 2 |
Ki = 602.56 nM
|
|
|
|
CP0479149
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-methyl-2-methylsulfanylaniline
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|
C12H17N3S
|
2
|
| 1 |
EC50 = 8.913 nM
|
|
|
| 2 |
Ki = 199.53 nM
|
|
|
|
CP0386170
|
2-[1-(2-cyclopentylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C16H22N2O
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 26.92 nM
|
|
|
|
CP0378482
|
(R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C17H17N3O3
|
3
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 257.04 nM
|
|
|
| 3 |
Ki = 363.08 nM
|
|
|
|
CP0202947
|
2-[1-(2-bromophenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C11H13BrN2O
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 281.84 nM
|
|
|
|
CP0451982
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-fluoro-2-methylsulfanylaniline
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|
C11H14FN3S
|
2
|
| 1 |
EC50 = 15.85 nM
|
|
|
| 2 |
Ki = 218.78 nM
|
|
|
|
CP0413599
|
2-[(1S)-1-(2-phenylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C17H18N2O
|
2
|
| 1 |
EC50 = 18.62 nM
|
|
|
| 2 |
Ki = 302 nM
|
|
|
|
CP0423440
|
2-[1-(2-cyclohexylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C17H24N2O
|
2
|
| 1 |
EC50 = 20.89 nM
|
|
|
| 2 |
Ki = 77.62 nM
|
|
|
|
CP0380684
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylaniline
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|
C11H15N3
|
1
|
| 1 |
EC50 = 21.88 nM
|
|
|
|
CP0419106
|
2-[1-(2-propylphenyl)ethoxy]-4,5-dihydro-1H-imidazole
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|
C14H20N2O
|
2
|
| 1 |
EC50 = 25.12 nM
|
|
|
| 2 |
Ki = 147.91 nM
|
|
|
|
CP0157932
|
2-[(1S)-1-(2-prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 25.12 nM
|
|
|
| 2 |
Ki = 70.79 nM
|
|
|
|
CP0435288
|
3-[2-[(1R)-1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenol
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|
C17H18N2O2
|
2
|
| 1 |
EC50 = 25.12 nM
|
|
|
| 2 |
Ki = 31.62 nM
|
|
|
|
CP0372608
|
2-[1-(2,6-diethylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C15H22N2O
|
2
|
| 1 |
EC50 = 27.54 nM
|
|
|
| 2 |
Ki = 275.42 nM
|
|
|
|
CP0376911
|
2-[1-(2,6-dimethylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C13H18N2O
|
2
|
| 1 |
EC50 = 27.54 nM
|
|
|
| 2 |
Ki = 251.19 nM
|
|
|
|
CP0899588
|
(4,5-Dihydro-1H-imidazol-2-ylmethyl)-(2-ethylsulfanyl-phenyl)-amine hydrochloride
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|
C12H18ClN3S
|
2
|
| 1 |
EC50 = 28.18 nM
|
|
|
| 2 |
Ki = 269.15 nM
|
|
|
|
CP0845500
|
(4,5-Dihydro-1H-imidazol-2-ylmethyl)-(2-isopropylsulfanyl-phenyl)-amine hydrochloride
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|
C13H20ClN3S
|
2
|
| 1 |
EC50 = 28.18 nM
|
|
|
| 2 |
Ki = 165.96 nM
|
|
|
|
CP0157938
|
2-[(1S)-1-(2-cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 35.48 nM
|
|
|
| 2 |
Ki = 63.1 nM
|
|
|
|
CP0372449
|
3-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]pyridine
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|
C16H17N3O
|
3
|
| 1 |
EC50 = 39.81 nM
|
|
|
| 2 |
EC50 = 50.12 nM
|
|
|
| 3 |
Ki = 64.57 nM
|
|
|
|
CP0402735
|
2-[1-(2-cyclopropylphenyl)ethoxy]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 39.81 nM
|
|
|
| 2 |
Ki = 79.43 nM
|
|
|
|
CP0110358
|
2-[1-(2-cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 39.81 nM
|
|
|
| 2 |
Ki = 79.43 nM
|
|
|
|
CP0378483
|
3-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenol
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|
C17H18N2O2
|
2
|
| 1 |
EC50 = 46.77 nM
|
|
|
| 2 |
Ki = 17.78 nM
|
|
|
|
CP0110365
|
2-[1-(2-cyclopropyloxyphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O2
|
2
|
| 1 |
EC50 = 47.86 nM
|
|
|
| 2 |
Ki = 676.08 nM
|
|
|
|
CP0157930
|
2-[1-(2-prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 50.12 nM
|
|
|
| 2 |
Ki = 85.11 nM
|
|
|
|
CP0419107
|
2-[1-(2-prop-2-enylphenyl)ethoxy]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 50.12 nM
|
|
|
| 2 |
Ki = 85.11 nM
|
|
|
|
CP0387342
|
2-[1-[2,6-bis(prop-2-enyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C17H22N2O
|
2
|
| 1 |
EC50 = 56.23 nM
|
|
|
| 2 |
Ki = 128.82 nM
|
|
|
|
CP0333694
|
2-[1-(2-phenylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C17H18N2O
|
2
|
| 1 |
EC50 = 57.54 nM
|
|
|
| 2 |
Ki = 199.53 nM
|
|
|
|
CP0041905
|
2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2)
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|
C9H9Cl2N3
|
3
|
| 1 |
EC50 = 57.54 nM
|
|
|
| 2 |
Ki = 9.333 nM
|
|
|
| 3 |
Ki = 30 nM
|
|
|
|
CP0437316
|
2-[1-(2-thiophen-2-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C15H16N2OS
|
2
|
| 1 |
EC50 = 58.88 nM
|
|
|
| 2 |
Ki = 72.44 nM
|
|
|
|
CP0373586
|
2-[1-[2-(3-fluorophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C17H17FN2O
|
2
|
| 1 |
EC50 = 60.26 nM
|
|
|
| 2 |
Ki = 16.98 nM
|
|
|
|
CP0430994
|
2-[1-(2-methylphenyl)ethoxy]-4,5-dihydro-1H-imidazole
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|
C12H16N2O
|
2
|
| 1 |
EC50 = 63.1 nM
|
|
|
| 2 |
Ki = 269.15 nM
|
|
|
|
CP0376827
|
2-[1-(2,6-diphenylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C23H22N2O
|
2
|
| 1 |
EC50 = 79.43 nM
|
|
|
| 2 |
Ki = 630.96 nM
|
|
|
|
CP0427126
|
2-[1-(2-thiophen-3-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C15H16N2OS
|
2
|
| 1 |
EC50 = 93.33 nM
|
|
|
| 2 |
Ki = 131.83 nM
|
|
|
|
CP0437314
|
N-[1-(4,5-dihydro-1H-imidazol-2-yl)ethyl]-2-phenylaniline
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|
C17H19N3
|
2
|
| 1 |
EC50 = 93.33 nM
|
|
|
| 2 |
Ki = 707.95 nM
|
|
|
|
CP0375447
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-4-fluoro-2-methylsulfanylaniline
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|
C11H14FN3S
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
Ki = 218.78 nM
|
|
|
|
CP0378487
|
2-[1-[2-(3-nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C17H17N3O3
|
3
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
EC50 = 158.49 nM
|
|
|
| 3 |
Ki = 234.42 nM
|
|
|
|
CP0435289
|
2-[(1R)-1-(2-thiophen-3-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C15H16N2OS
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
Ki = 316.23 nM
|
|
|
|
CP0376829
|
2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]benzaldehyde
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|
C12H14N2O2
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
Ki = 8709.64 nM
|
|
|
|
CP0387610
|
2-[1-(2-ethylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C13H18N2O
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
Ki = 288.4 nM
|
|
|
|
CP0403607
|
2-[1-(2-propan-2-yloxyphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H20N2O2
|
2
|
| 1 |
EC50 = 100 nM
|
|
|
| 2 |
Ki = 398.11 nM
|
|
|
|
CP0378484
|
2-[(1R)-1-(2-phenylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C17H18N2O
|
2
|
| 1 |
EC50 = 112.2 nM
|
|
|
| 2 |
Ki = 977.24 nM
|
|
|
|
CP0372603
|
2-[1-(2-prop-1-en-2-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C14H18N2O
|
2
|
| 1 |
EC50 = 114.82 nM
|
|
|
| 2 |
Ki = 602.56 nM
|
|
|
|
CP0380686
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-propylaniline
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|
C13H19N3
|
1
|
| 1 |
EC50 = 114.82 nM
|
|
|
|
CP0851097
|
2-[1-(4,5-Dihydro-1H-imidazol-2-yl)-ethoxy]-benzaldehyde Oxime
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|
C12H15N3O2
|
2
|
| 1 |
EC50 = 125.89 nM
|
|
|
| 2 |
Ki = 912.01 nM
|
|
|
|
CP0157942
|
2-[(1R)-1-(2-cyclopropylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C14H18N2O
|
2
|
| 1 |
EC50 = 125.89 nM
|
|
|
| 2 |
Ki = 125.89 nM
|
|
|
|
CP0385262
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-phenylaniline
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|
C16H17N3
|
1
|
| 1 |
EC50 = 147.91 nM
|
|
|
|
CP0431035
|
2-[(2-propylphenyl)methoxy]-4,5-dihydro-1H-imidazole
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|
C13H18N2O
|
2
|
| 1 |
EC50 = 154.88 nM
|
|
|
| 2 |
Ki = 489.78 nM
|
|
|
|
CP0380685
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-prop-2-enylaniline
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|
C13H17N3
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
|
CP0390643
|
2-[1-(2-chlorophenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C11H13ClN2O
|
2
|
| 1 |
EC50 = 165.96 nM
|
|
|
| 2 |
Ki = 489.78 nM
|
|
|
|
CP0087659
|
2-[(1R)-1-(2-prop-2-enylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C14H18N2O
|
2
|
| 1 |
EC50 = 186.21 nM
|
|
|
| 2 |
Ki = 177.83 nM
|
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|
|
CP0456784
|
1-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]ethanone
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|
C13H16N2O2
|
2
|
| 1 |
EC50 = 199.53 nM
|
|
|
| 2 |
Ki = 7413.1 nM
|
|
|
|
CP0380687
|
(2-Chloro-phenyl)-(4,5-dihydro-1H-imidazol-2-ylmethyl)-amine
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|
C10H12ClN3
|
1
|
| 1 |
EC50 = 223.87 nM
|
|
|
|
CP0391376
|
2-[1-(2-methylsulfonylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C12H16N2O3S
|
2
|
| 1 |
EC50 = 316.23 nM
|
|
|
| 2 |
Ki = 3801.89 nM
|
|
|
|
CP0087658
|
2-[(1R)-1-[2-(cyclopropylmethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C15H20N2O
|
2
|
| 1 |
EC50 = 316.23 nM
|
|
|
| 2 |
Ki = 234.42 nM
|
|
|
|
CP0427125
|
2-[1-[2-(2-methylphenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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|
C18H20N2O
|
2
|
| 1 |
EC50 = 363.08 nM
|
|
|
| 2 |
Ki = 234.42 nM
|
|
|
|
CP0044542
|
2-(2-Cyclopropyl-phenoxymethyl)-4,5-dihydro-1H-imidazole
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|
C13H16N2O
|
2
|
| 1 |
EC50 = 398.11 nM
|
|
|
| 2 |
Ki = 549.54 nM
|
|
|
|
CP0391378
|
2-[1-(2-propan-2-ylphenoxy)ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C14H20N2O
|
2
|
| 1 |
EC50 = 398.11 nM
|
|
|
| 2 |
Ki = 457.09 nM
|
|
|
|
CP0402493
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-fluoro-6-methylsulfonylaniline
Show/Hide
|
C11H14FN3O2S
|
2
|
| 1 |
EC50 = 446.68 nM
|
|
|
| 2 |
Ki = 691.83 nM
|
|
|
|
CP0461287
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-fluoro-2-methylsulfonylaniline
Show/Hide
|
C11H14FN3O2S
|
2
|
| 1 |
EC50 = 501.19 nM
|
|
|
| 2 |
Ki = 257.04 nM
|
|
|
|
CP0427124
|
3-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]aniline
Show/Hide
|
C17H19N3O
|
2
|
| 1 |
EC50 = 501.19 nM
|
|
|
| 2 |
Ki = 309.03 nM
|
|
|
|
CP0379033
|
(E)-1-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]-N-methoxymethanimine
Show/Hide
|
C13H17N3O2
|
2
|
| 1 |
EC50 = 501.19 nM
|
|
|
| 2 |
Ki = 3090.3 nM
|
|
|
|
CP0400831
|
2-[1-(2-ethenoxyphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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|
C13H16N2O2
|
1
|
| 1 |
EC50 = 630.96 nM
|
|
|
|
CP0378486
|
2-[(1S)-1-[2-(3-nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C17H17N3O3
|
2
|
| 1 |
EC50 = 741.31 nM
|
|
|
| 2 |
Ki = 537.03 nM
|
|
|
|
CP0396660
|
2-[phenyl-(2-phenylphenoxy)methyl]-4,5-dihydro-1H-imidazole
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|
C22H20N2O
|
2
|
| 1 |
EC50 = 776.25 nM
|
|
|
| 2 |
Ki = 204.17 nM
|
|
|
|
CP0409992
|
5-chloro-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylsulfonylaniline
Show/Hide
|
C11H14ClN3O2S
|
2
|
| 1 |
EC50 = 794.33 nM
|
|
|
| 2 |
Ki = 4786.3 nM
|
|
|
|
CP0039930
|
(-)-arterenol
Show/Hide
|
C8H11NO3
|
1
|
| 1 |
EC50 = 794.33 nM
|
|
|
|
CP0387574
|
2-(5-phenyl-2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole
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C17H16N2O2
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2
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| 1 |
EC50 = 794.33 nM
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| 2 |
Ki = 831.76 nM
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CP0376832
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2-[1-[2-(trifluoromethyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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C12H13F3N2O
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2
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| 1 |
EC50 = 794.33 nM
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| 2 |
Ki = 977.24 nM
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CP0441664
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2-[1-[2-(4-methylphenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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C18H20N2O
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2
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| 1 |
EC50 = 831.76 nM
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| 2 |
Ki = 251.19 nM
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CP0423441
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(E)-1-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]-N-ethoxymethanimine
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C14H19N3O2
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2
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| 1 |
EC50 = 1000 nM
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| 2 |
Ki = 338.84 nM
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CP0375544
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-methyl-2-methylsulfonylaniline
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C12H17N3O2S
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2
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| 1 |
EC50 = 1122.02 nM
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| 2 |
Ki < 5011.87 nM
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CP0373596
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2-[1-[2-(3-methylphenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
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C18H20N2O
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2
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| 1 |
EC50 = 1584.89 nM
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| 2 |
Ki = 245.47 nM
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CP0394131
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NS-49
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C9H13FN2O3S
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1
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| 1 |
EC50 = 1995.26 nM
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CP0464188
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-fluoro-2-methylsulfonylaniline
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C11H14FN3O2S
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2
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| 1 |
EC50 = 1995.26 nM
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| 2 |
Ki < 5011.87 nM
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CP0475547
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3-[2-[(1S)-1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenol
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C17H18N2O2
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2
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| 1 |
EC50 = 2511.89 nM
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| 2 |
Ki = 112.2 nM
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CP0427121
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2-[3-(2-phenylphenyl)oxiran-2-yl]-4,5-dihydro-1H-imidazole
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C17H16N2O
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2
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| 1 |
EC50 = 2691.53 nM
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| 2 |
Ki = 6456.54 nM
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CP0402731
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2-[(2-methylphenyl)methoxy]-4,5-dihydro-1H-imidazole
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C11H14N2O
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2
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| 1 |
EC50 = 2884.03 nM
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| 2 |
Ki = 501.19 nM
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CP0916328
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(4,5-Dihydro-1H-imidazol-2-ylmethyl)-(2-methanesulfonyl-phenyl)-amine hydrochloride
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C11H16ClN3O2S
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2
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| 1 |
EC50 = 3162.28 nM
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| 2 |
Ki < 5011.87 nM
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CP0423434
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2-(5-phenyl-2,3-dihydro-1,4-benzodioxin-3-yl)-4,5-dihydro-1H-imidazole
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C17H16N2O2
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2
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| 1 |
EC50 = 3162.28 nM
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| 2 |
Ki = 691.83 nM
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CP0386168
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(E)-1-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]-N-phenylmethoxymethanimine
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C19H21N3O2
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2
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| 1 |
EC50 = 3548.13 nM
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| 2 |
Ki = 676.08 nM
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CP0431046
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-ethylsulfonylaniline
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C12H17N3O2S
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2
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| 1 |
EC50 = 5011.87 nM
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| 2 |
Ki = 2511.89 nM
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CP0432293
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-1,1-dioxo-3,4-dihydro-2H-thiochromen-8-amine
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C13H17N3O2S
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2
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| 1 |
EC50 = 6309.57 nM
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| 2 |
Ki = 2691.53 nM
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CP0376836
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2-[1-(2-methoxyphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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C12H16N2O2
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2
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| 1 |
EC50 = 9772.37 nM
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| 2 |
Ki = 831.76 nM
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CP0376906
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2-[1-(2-ethoxyphenoxy)ethyl]-4,5-dihydro-1H-imidazole
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C13H18N2O2
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2
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| 1 |
EC50 = 10000 nM
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| 2 |
Ki = 758.58 nM
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CP0392166
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylsulfonyl-5-(trifluoromethyl)aniline
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C12H14F3N3O2S
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2
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| 1 |
EC50 < 10000 nM
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| 2 |
Ki < 5011.87 nM
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CP0404420
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4-chloro-N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-methylsulfonylaniline
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C11H14ClN3O2S
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2
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| 1 |
EC50 < 10000 nM
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| 2 |
Ki = 3981.07 nM
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CP0397746
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N-(4,5-dihydro-1H-imidazol-1-ium-2-ylmethyl)-2-methylsulfinylaniline;chloride
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C11H16ClN3OS
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2
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| 1 |
EC50 < 10000 nM
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| 2 |
Ki < 5011.87 nM
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CP0404419
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-2-propan-2-ylsulfonylaniline
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C13H19N3O2S
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2
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| 1 |
EC50 < 10000 nM
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| 2 |
Ki < 5011.87 nM
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CP0406394
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-4-fluoro-2-methylsulfonylaniline
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C11H14FN3O2S
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2
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| 1 |
EC50 < 10000 nM
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| 2 |
Ki < 5011.87 nM
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CP0509938
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-7-iodo-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H20IN3O2
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1
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| 1 |
IC50 = 0.6166 nM
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CP0480554
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7-bromo-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H20BrN3O2
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1
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| 1 |
IC50 = 0.6918 nM
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CP0506685
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-9-methoxy-2-methylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O3
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1
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| 1 |
IC50 = 0.7079 nM
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CP0380435
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7-chloro-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H20ClN3O2
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1
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| 1 |
IC50 = 0.7244 nM
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CP0375211
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2,6,8-trimethylpyrido[1,2-a]pyrimidin-4-one
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C24H25N3O2
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1
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| 1 |
IC50 = 0.8511 nM
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CP0430308
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2,6-dimethylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O2
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1
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| 1 |
IC50 = 1.072 nM
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CP0462778
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2,8-dimethylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O2
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1
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| 1 |
IC50 = 1.202 nM
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CP0398443
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2,7-dimethylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O2
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1
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| 1 |
IC50 = 1.288 nM
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CP0375207
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2,9-dimethylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O2
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1
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| 1 |
IC50 = 1.318 nM
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CP0409638
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7,9-dichloro-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H19Cl2N3O2
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1
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| 1 |
IC50 = 1.349 nM
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CP0479963
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-9-hydroxy-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H21N3O3
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1
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| 1 |
IC50 = 1.622 nM
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CP0437587
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LUSAPERIDONE
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C22H21N3O2
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1
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| 1 |
IC50 = 1.698 nM
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CP0503149
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3-[2-(6-chloro-3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H20ClN3O2
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1
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| 1 |
IC50 = 2.239 nM
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CP0375044
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2-benzyl-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]pyrido[1,2-a]pyrimidin-4-one
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C28H25N3O2
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1
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| 1 |
IC50 = 2.692 nM
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CP0373529
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9-chloro-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methyl-7-(trifluoromethyl)pyrido[1,2-a]pyrimidin-4-one
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C23H19ClF3N3O2
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1
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| 1 |
IC50 = 3.631 nM
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CP0380633
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3-[3-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)propyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C23H23N3O2
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1
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| 1 |
IC50 = 6.607 nM
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CP0467592
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3-[2-(3,4-dihydro-1H-[1]benzothiolo[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H21N3OS
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1
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| 1 |
IC50 = 14.13 nM
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CP0375053
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3-[2-(8-chloro-3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
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C22H20ClN3O2
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1
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| 1 |
IC50 = 27.54 nM
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CP0037622
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2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole
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C11H12N2O2
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2
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| 1 |
IC50 = 53.7 nM
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| 2 |
Ki = 17.78 nM
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CP0408409
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3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-7,8-dimethoxy-2-methylpyrido[1,2-a]pyrimidin-4-one
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C24H25N3O4
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1
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| 1 |
IC50 = 57.54 nM
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CP0030044
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(+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-triaza-tribenzo[a,c,e]cycloheptene
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C17H19N3
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1
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| 1 |
IC50 = 199.53 nM
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CP0456177
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2-(tert-butylamino)-N-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)nicotinamide
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C26H37N5O3
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2
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| 1 |
Ki = 0.5 nM
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| 2 |
Ki = 30.5 nM
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CP0069692
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(+)-yohimbine
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C21H26N2O3
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3
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| 1 |
Ki = 0.5 nM
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| 2 |
Ki = 0.8 nM
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| 3 |
Ki = 0.88 nM
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CP0485691
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6-butoxy-N-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)picolinamide
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C26H36N4O4
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2
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| 1 |
Ki = 0.6 nM
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| 2 |
Ki = 3.8 nM
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CP0077862
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4-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-butyric acid benzyl ester
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C31H37N3O4
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1
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| 1 |
Ki = 0.65 nM
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CP0423436
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(+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)-4,5-dihydro-1H-imidazole
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C12H14N2O3
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1
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| 1 |
Ki = 0.7943 nM
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CP0439786
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2-butoxy-N-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)nicotinamide
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C26H36N4O4
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2
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| 1 |
Ki = 0.8 nM
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| 2 |
Ki = 4.8 nM
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CP0445292
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2-(3-cyanophenoxy)-N-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)nicotinamide
Show/Hide
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C29H31N5O4
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2
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| 1 |
Ki = 0.8 nM
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| 2 |
Ki = 1.9 nM
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CP0071147
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(S)-N-{2-[4-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-[1,4]diazepan-1-yl]-ethyl}-2-phenoxy-nicotinamide
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C28H32N4O4
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2
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| 1 |
Ki = 0.9 nM
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| 2 |
Ki = 1.9 nM
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CP0436189
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benzyl N-[3-[[(1S,15R,18S,19R)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carbonyl]amino]propyl]carbamate
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C31H38N4O4
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1
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| 1 |
Ki = 1.1 nM
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CP0434857
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1-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-4-((3-(2-phenoxypyridin-3-yl)-1,2,4-oxadiazol-5-yl)methyl)-1,4-diazepane
Show/Hide
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C28H29N5O4
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2
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| 1 |
Ki = 1.7 nM
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| 2 |
Ki = 1.9 nM
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CP0307921
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N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
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C24H26FN3O3S2
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1
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| 1 |
Ki = 1.9 nM
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CP0399322
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1-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-4-(2-((2-phenoxypyridin-3-yl)methoxy)ethyl)-1,4-diazepane
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C28H33N3O4
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2
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| 1 |
Ki = 2.5 nM
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| 2 |
Ki = 6.8 nM
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CP0512008
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tert-butyl N-[3-[[(1S,15R,18S,19R)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carbonyl]amino]propyl]carbamate
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C28H40N4O4
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1
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| 1 |
Ki = 2.8 nM
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CP0399323
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N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)piperazin-1-yl]ethyl]-2-phenoxypyridine-3-carboxamide
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C27H30N4O4
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1
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| 1 |
Ki = 3 nM
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CP0541624
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4-[((1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carbonyl)-amino]-butyric acid
Show/Hide
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C24H31N3O4
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1
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| 1 |
Ki = 3 nM
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CP0464670
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2-(4,5-dihydro-1H-imidazol-2-yl)-1-(3-methoxyphenyl)-1-(4-methylphenyl)hydrazine
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C17H20N4O
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1
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| 1 |
Ki = 3.8 nM
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CP0439781
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N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]-2-phenoxypyridine-3-carboxamide
Show/Hide
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C28H32N4O4
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2
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| 1 |
Ki = 5 nM
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| 2 |
Ki = 25 nM
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CP0510294
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methyl 2-[[2-[[(1S,15R,18S,19R)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carbonyl]amino]acetyl]amino]acetate
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C25H32N4O5
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1
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| 1 |
Ki = 5.2 nM
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CP0448055
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methyl 2-[[(1S,15R,18S,19R)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carbonyl]amino]acetate
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C23H29N3O4
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1
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| 1 |
Ki = 8 nM
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CP0436188
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1N-{3-[2-hydroxy-(1R,2S,4aR,13bS)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]b-carbolin-1-ylcarboxamido]propyl}-2-hydroxy-(1S,2R,4aS,13bR,14aR)-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydroisoquino[3,2-a]
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C43H54N6O4
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1
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| 1 |
Ki = 8.5 nM
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CP0397609
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AGN-193080
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C12H16N4O
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1
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| 1 |
Ki = 8.9 nM
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CP0498527
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(R)-N-(2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)ethyl)-2-phenoxynicotinamide
Show/Hide
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C28H32N4O4
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1
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| 1 |
Ki = 9.2 nM
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CP0056760
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CHEBI:8862
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C10H16N2O
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1
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| 1 |
Ki = 12.59 nM
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CP0485217
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3-[N'-(4,5-Dihydro-1H-imidazol-2-yl)-N-p-tolyl-hydrazino]-phenol
Show/Hide
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C16H18N4O
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1
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| 1 |
Ki = 12.8 nM
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CP0388308
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N-[2-[4-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl]pyridine-3-carboxamide
Show/Hide
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C22H28N4O3
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1
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| 1 |
Ki = 15.7 nM
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CP0406514
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(1H-Imidazol-2-yl)-(5-methyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-amine
Show/Hide
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C12H13N3O2
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1
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| 1 |
Ki = 19 nM
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CP0453218
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(1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carboxylic acid
Show/Hide
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C20H24N2O3
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1
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| 1 |
Ki = 19 nM
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CP0046852
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1-Benzyl-4-chroman-2-ylmethyl-piperazine
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C21H26N2O
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2
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| 1 |
Ki = 19.6 nM
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| 2 |
Ki = 21.1 nM
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CP0439785
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1-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-4-(2-methoxyphenyl)piperazine
Show/Hide
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C20H24N2O3
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2
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| 1 |
Ki = 23 nM
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| 2 |
Ki = 33 nM
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CP0083828
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N-(4,5-dihydro-1H-imidazol-2-yl)-5-methylquinoxalin-6-amine
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C12H13N5
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1
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| 1 |
Ki = 27 nM
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CP0443901
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Aminoclonidine, p
Show/Hide
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C9H10Cl2N4
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1
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| 1 |
Ki = 30 nM
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CP0108416
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(+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole
Show/Hide
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C13H16N2
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1
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| 1 |
Ki = 30.9 nM
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CP0392123
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(1R,2S,4aR,13bS)-2-Hydroxy-1,2,3,4,4a,5,7,8,13,13b,14,14a-dodecahydro-indolo[2',3':3,4]pyrido[1,2-b]isoquinoline-1-carboxylic acid (3-amino-propyl)-amide
Show/Hide
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C23H32N4O2
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1
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| 1 |
Ki = 32 nM
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CP0041550
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BRIMONIDINE
Show/Hide
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C11H10BrN5
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1
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| 1 |
Ki = 44 nM
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CP0066123
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6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimethyl-phenol;hydrochloride
Show/Hide
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C16H24N2O
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1
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| 1 |
Ki = 58.88 nM
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CP0386169
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2-[phenoxy(phenyl)methyl]-4,5-dihydro-1H-imidazole
Show/Hide
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C16H16N2O
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1
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| 1 |
Ki = 64.57 nM
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CP0072943
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3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphenyl)amino]phenol;methanesulfonic acid
Show/Hide
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C17H19N3O
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1
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| 1 |
Ki = 80.3 nM
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CP0373564
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(4-tert-Butyl-3-methoxy-2,6-dimethyl-phenyl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C16H23N3O
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1
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| 1 |
Ki = 88 nM
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CP0410535
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AGN-192172
Show/Hide
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C12H17N5
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1
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| 1 |
Ki = 120 nM
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CP0379280
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2-[3-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]propoxy]benzamide
Show/Hide
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C28H30N4O4S
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1
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| 1 |
Ki = 190 nM
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CP0376585
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(1H-Imidazol-2-yl)-(5-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-amine
Show/Hide
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C12H14N4O
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1
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| 1 |
Ki = 230 nM
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CP0396661
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2-(3-methoxy-5-phenyl-2H-1,4-benzodioxin-3-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C18H18N2O3
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1
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| 1 |
Ki = 245.47 nM
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CP0387572
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2-(1-phenoxyethyl)-4,5-dihydro-1H-imidazole
Show/Hide
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C11H14N2O
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1
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| 1 |
Ki = 263.03 nM
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CP0439228
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2-(1-phenylethoxy)-4,5-dihydro-1H-imidazole
Show/Hide
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C11H14N2O
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1
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| 1 |
Ki = 263.03 nM
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CP0402484
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(5-tert-Butyl-4-methoxy-2-methyl-phenyl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C15H21N3O
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1
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| 1 |
Ki = 290 nM
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CP0373590
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2-[1-[2-(4-nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
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C17H17N3O3
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1
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| 1 |
Ki = 302 nM
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CP0428121
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4-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenol
Show/Hide
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C17H18N2O2
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1
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| 1 |
Ki = 331.13 nM
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CP0402335
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(1H-Imidazol-2-yl)-(5-methyl-quinoxalin-6-yl)-amine
Show/Hide
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C12H11N5
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1
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| 1 |
Ki = 340 nM
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CP0373437
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(1H-Benzoimidazol-5-yl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C10H9N5
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1
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| 1 |
Ki = 400 nM
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CP0506536
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(1H-Imidazol-2-yl)-(4-methoxy-2-methyl-phenyl)-amine
Show/Hide
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C11H13N3O
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1
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| 1 |
Ki = 512 nM
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CP0397965
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N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-methoxy-2-methylsulfanylaniline
Show/Hide
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C12H17N3OS
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1
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| 1 |
Ki = 602.56 nM
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CP0854701
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1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate Monohydrate
Show/Hide
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C22H30BrN3O7S2
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1
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| 1 |
Ki = 619 nM
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CP0373585
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2-[1-(2-phenylphenyl)sulfanylethyl]-4,5-dihydro-1H-imidazole
Show/Hide
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C17H18N2S
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1
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| 1 |
Ki = 707.95 nM
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CP0453117
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(2,6-Dichloro-phenyl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C9H7Cl2N3
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1
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| 1 |
Ki = 1100 nM
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CP0373587
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2-[1-[2-(2-nitrophenyl)phenoxy]ethyl]-4,5-dihydro-1H-imidazole
Show/Hide
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C17H17N3O3
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1
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| 1 |
Ki = 1230.27 nM
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CP0373584
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2-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]pyridine
Show/Hide
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C16H17N3O
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1
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| 1 |
Ki = 1258.93 nM
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CP0423442
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2-(6-phenyl-2,3-dihydro-1,4-benzodioxin-3-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C17H16N2O2
|
1
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| 1 |
Ki = 1258.93 nM
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CP0373597
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4-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]pyridine
Show/Hide
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C16H17N3O
|
1
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| 1 |
Ki = 1445.44 nM
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CP0375168
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(3,4-Dimethoxy-2-methyl-phenyl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C12H15N3O2
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1
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| 1 |
Ki = 1500 nM
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CP0423443
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2-(6-phenyl-2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C17H16N2O2
|
1
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| 1 |
Ki = 1584.89 nM
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CP0373595
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2-[2-[1-(4,5-dihydro-1H-imidazol-2-yl)ethoxy]phenyl]phenol
Show/Hide
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C17H18N2O2
|
1
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| 1 |
Ki = 1621.81 nM
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CP0135923
|
CHEBI:6956
Show/Hide
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C23H30N2O4
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1
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| 1 |
Ki = 2320 nM
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CP0380658
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(2-Bromo-phenyl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C9H8BrN3
|
1
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| 1 |
Ki = 2400 nM
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CP0853864
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(4,5-Dihydro-1H-imidazol-2-ylmethyl)-[2-(propane-1-sulfonyl)-phenyl]-amine hydrochloride
Show/Hide
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C13H20ClN3O2S
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1
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| 1 |
Ki = 2630.27 nM
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CP0427122
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2-[3-(2-phenylphenyl)oxiran-2-yl]-4,5-dihydro-1H-imidazole;hydrochloride
Show/Hide
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C17H17ClN2O
|
1
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| 1 |
Ki = 4265.8 nM
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CP0421105
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N-(2-chlorophenyl)-3,4-dihydro-2H-pyrrol-5-amine
Show/Hide
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C10H11ClN2
|
1
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| 1 |
Ki = 5011.87 nM
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CP0387054
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N-(2,6-dichlorophenyl)-5-methyl-4,5-dihydro-1H-imidazol-2-amine
Show/Hide
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C10H11Cl2N3
|
1
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| 1 |
Ki = 5754.4 nM
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CP0373591
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5-[1-(2-phenylphenoxy)ethyl]-3,4-dihydro-2H-pyrrole
Show/Hide
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C18H19NO
|
1
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| 1 |
Ki = 5888.44 nM
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CP0442626
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2-[1-(2-phenylphenoxy)ethyl]-4,5-dihydro-1,3-oxazole
Show/Hide
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C17H17NO2
|
1
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| 1 |
Ki = 5888.44 nM
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CP0405369
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2-(6,6-diphenyl-1,4-dioxan-2-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C19H20N2O2
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1
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| 1 |
Ki = 6165.95 nM
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CP0402201
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2-(5,5-diphenyl-1,4-dioxan-2-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C19H20N2O2
|
1
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| 1 |
Ki = 7413.1 nM
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CP0453851
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(1H-Imidazol-2-yl)-quinoxalin-6-yl-amine
Show/Hide
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C11H9N5
|
1
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| 1 |
Ki = 8800 nM
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CP0392952
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(5-Bromo-quinoxalin-6-yl)-(1H-imidazol-2-yl)-amine
Show/Hide
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C11H8BrN5
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1
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| 1 |
Ki > 10000 nM
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CP0372845
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2-[(2R,6S)-6-phenyl-1,4-dioxan-2-yl]-4,5-dihydro-1H-imidazole
Show/Hide
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C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0387839
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2-[(2R,6R)-6-phenyl-1,4-dioxan-2-yl]-4,5-dihydro-1H-imidazole
Show/Hide
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C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0391979
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2-[(2R,5S)-5-phenyl-1,4-dioxan-2-yl]-4,5-dihydro-1H-imidazole
Show/Hide
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C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0399099
|
2-[(2S,5R)-5-phenyl-1,4-dioxan-2-yl]-4,5-dihydro-1H-imidazole
Show/Hide
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C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0418816
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2-[(2R,5R)-5-phenyl-1,4-dioxan-2-yl]-4,5-dihydro-1H-imidazole
Show/Hide
|
C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0666295
|
rac-trans-2-(5-Phenyl-1,4-dioxan-2-yl)-4,5-dihydro-1H-imidazole
Show/Hide
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C13H16N2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0410228
|
N-(dicyclopropylmethyl)-4-methyl-4,5-dihydro-1,3-oxazol-2-amine
Show/Hide
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C11H18N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0421104
|
US9303019, 13
Show/Hide
|
C11H13ClN2
|
1
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| 1 |
Ki > 10000 nM
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CP0497542
|
N-(2-chloro-4-iodophenyl)-2-methyl-3,4-dihydro-2H-pyrrol-5-amine
Show/Hide
|
C11H12ClIN2
|
1
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| 1 |
Ki > 10000 nM
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CP0151467
|
1-Benzyl-4-chroman-3-ylmethyl-piperazine
Show/Hide
|
C21H26N2O
|
1
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| 1 |
Ki > 500 nM
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CP0456864
|
N-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-methoxy-2-methylsulfonylaniline
Show/Hide
|
C12H17N3O3S
|
1
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| 1 |
Ki < 5011.87 nM
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CP0373588
|
2-[1-(2-phenylphenoxy)ethyl]-4,5-dihydro-1,3-thiazole
Show/Hide
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C17H17NOS
|
1
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| 1 |
Ki < 10000 nM
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