| Compound ID |
Compound Name |
Compound Formula |
|
CP0567871
|
4-N-[(2-chlorophenyl)methyl]-2-N-methyl-6-pyridin-2-ylpyrimidine-2,4-diamine
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|
C17H16ClN5
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0067898
|
N-[3-chloro-4-[[[2-(methylamino)-6-pyridin-2-ylpyrimidin-4-yl]amino]methyl]phenyl]methanesulfonamide
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|
C18H19ClN6O2S
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0544591
|
N-[(4-fluorophenyl)methyl]-5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-amine
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|
C19H16FN5
|
2
|
| 1 |
EC50 = 15 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0544592
|
4-N-cyclohexyl-2-N-methyl-6-pyridin-2-ylpyrimidine-2,4-diamine
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|
C16H21N5
|
2
|
| 1 |
EC50 = 16 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0572896
|
5-methyl-7-(2-phenylpyrrolidin-1-yl)-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidine
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|
C22H21N5
|
2
|
| 1 |
EC50 = 17 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0542984
|
N-methyl-4-phenoxy-6-pyridin-2-ylpyrimidin-2-amine
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|
C16H14N4O
|
2
|
| 1 |
EC50 = 23 nM
|
|
|
| 2 |
EC50 = 481 nM
|
|
|
|
CP0569067
|
N-[2-(4-fluorophenyl)propan-2-yl]-5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-amine
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|
C21H20FN5
|
2
|
| 1 |
EC50 = 63 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0545070
|
2-(4-fluorophenyl)-N-methyl-2-[(5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]acetamide
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|
C21H19FN6O
|
2
|
| 1 |
EC50 = 78 nM
|
|
|
| 2 |
EC50 > 27100 nM
|
|
|
|
CP0965297
|
2-(1-amino-2-(1H-imidazol-5-yl)ethyl)-6-phenylquinazolin-4(3H)-one
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|
C19H17N5O
|
2
|
| 1 |
EC50 = 251 nM
|
|
|
| 2 |
EC50 > 50000 nM
|
|
|
|
CP0576719
|
2-N-cyclohexyl-4-N-methyl-6-pyridin-2-ylpyrimidine-2,4-diamine
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|
C16H21N5
|
2
|
| 1 |
EC50 = 487 nM
|
|
|
| 2 |
EC50 > 31600 nM
|
|
|
|
CP0968151
|
2-(1-amino-3-(benzyloxy)propyl)-6-(1-methyl-1H-pyrazol-4-yl)quinazolin-4(3H)-one
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|
C22H23N5O2
|
2
|
| 1 |
EC50 = 641 nM
|
|
|
| 2 |
EC50 > 50000 nM
|
|
|
|
CP0569877
|
2-[3-(cyclobutylmethyl)-4-oxophthalazin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
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|
C21H22N4O2
|
2
|
| 1 |
EC50 = 4040 nM
|
|
|
| 2 |
EC50 > 50000 nM
|
|
|
|
CP0055399
|
6-[4-[(6-chloroimidazo[1,2-a]pyridin-2-yl)methyl]piperazin-1-yl]pyridine-3-carbonitrile
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|
C18H17ClN6
|
1
|
| 1 |
EC50 = 6250 nM
|
|
|
|
CP0550002
|
5-methyl-7-(3-phenylpyrrolidin-1-yl)-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidine
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|
C22H21N5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0568569
|
5-methyl-3-pyridin-2-yl-7-(2-pyridin-3-ylpyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine
Show/Hide
|
C21H20N6
|
1
|
| 1 |
EC50 > 27100 nM
|
|
|
|
CP0571680
|
N-[1-(4-fluorophenyl)ethyl]-5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-amine
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|
C20H18FN5
|
1
|
| 1 |
EC50 > 27100 nM
|
|
|
|
CP0577232
|
1-(5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)-5-phenylpyrrolidin-2-one
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|
C22H19N5O
|
2
|
| 1 |
EC50 > 27100 nM
|
|
|
| 2 |
EC50 > 31600 nM
|
|
|
|
CP0006743
|
4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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|
C16H19NO3S
|
1
|
| 1 |
EC50 > 50118.72 nM
|
|
|
