Brief Information of the Compound and Protein
Compound Name
2-(4-fluorophenyl)-N-methyl-2-[(5-methyl-3-pyridin-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]acetamide
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PubChem ID
CID: 168277952
Canonical SMILES
CNC(=O)C(Nc1cc(C)nc2c(cnn12)-c1ccccn1)c1ccc(F)cc1
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Compound Formula C21H19FN6O
Compound Structure
Protein Name
G-protein coupled receptor 39
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
O43194
Gene Name
GPR39
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 78 nM
   TI
   LI
   LO
   TS
2
EC50 > 27100 nM
   TI
   LI
   LO
   TS