Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT02505 , Beta-1 adrenergic receptor
Gene Name ADRB1
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P18090
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT02505
 
Compound ID Compound Name Compound Formula
CP0378899
125I-CYP
   Show/Hide
C16H20IN3O2
 3
1
Kd = 0.0631 nM
   TI
   LI
   LO
   TS
2
Kd = 0.07943 nM
   TI
   LI
   LO
   TS
3
Kd = 0.3162 nM
   TI
   LI
   LO
   TS
CP0378898
CAS_155346
   Show/Hide
C16H21N3O2
 5
1
Ki = 0.03981 nM
   TI
   LI
   LO
   TS
2
Ki = 0.05012 nM
   TI
   LI
   LO
   TS
3
Ki = 0.1259 nM
   TI
   LI
   LO
   TS
4
Ki = 0.3162 nM
   TI
   LI
   LO
   TS
5
Ki = 316.23 nM
   TI
   LI
   LO
   TS
CP0378904
2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy}propyl)amino]ethoxy}benzamide; methanesulfonic acid
   Show/Hide
C23H25F3N4O5
 5
1
Ki = 1.259 nM
   TI
   LI
   LO
   TS
2
Ki = 1.995 nM
   TI
   LI
   LO
   TS
3
Ki = 7.943 nM
   TI
   LI
   LO
   TS
4
Ki = 794.33 nM
   TI
   LI
   LO
   TS
5
Ki = 10000 nM
   TI
   LI
   LO
   TS
CP0041613
Anapriline
   Show/Hide
C16H21NO2
 5
1
Ki = 3.162 nM
   TI
   LI
   LO
   TS
2
Ki = 10 nM
   TI
   LI
   LO
   TS
3
Ki = 31.62 nM
   TI
   LI
   LO
   TS
4
Ki = 39.81 nM
   TI
   LI
   LO
   TS
5
Ki = 199.53 nM
   TI
   LI
   LO
   TS
CP0075426
(-)-3-morpholino-4-(3-tert-butylamino-2-hydroxypropoxy)-1,2,5-thiadiazole
   Show/Hide
C13H24N4O3S
 5
1
Ki = 3.162 nM
   TI
   LI
   LO
   TS
2
Ki = 7.943 nM
   TI
   LI
   LO
   TS
3
Ki = 15.85 nM
   TI
   LI
   LO
   TS
4
Ki = 31.62 nM
   TI
   LI
   LO
   TS
5
Ki = 630.96 nM
   TI
   LI
   LO
   TS
CP0427117
LK-204-545
   Show/Hide
C25H32N4O6
 5
1
Ki = 7.943 nM
   TI
   LI
   LO
   TS
2
Ki = 63.1 nM
   TI
   LI
   LO
   TS
3
Ki = 79.43 nM
   TI
   LI
   LO
   TS
4
Ki = 100 nM
   TI
   LI
   LO
   TS
5
Ki = 79432.82 nM
   TI
   LI
   LO
   TS
CP0886363
(S)-1-(3,4-dimethoxyphenethylamino)-3-(4-(2-ethoxyethoxy)phenoxy)propan-2-ol
   Show/Hide
C23H33NO6
 5
1
Ki = 50.12 nM
   TI
   LI
   LO
   TS
2
Ki = 79.43 nM
   TI
   LI
   LO
   TS
3
Ki = 100 nM
   TI
   LI
   LO
   TS
4
Ki = 794.33 nM
   TI
   LI
   LO
   TS
5
Ki = 12589.25 nM
   TI
   LI
   LO
   TS
CP0048177
(2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylamino)-3-[4-(2-methoxyethyl)phenoxy]propan-2-ol
   Show/Hide
C15H25NO3
 4
1
Ki = 398.11 nM
   TI
   LI
   LO
   TS
2
Ki = 630.96 nM
   TI
   LI
   LO
   TS
3
Ki = 2511.89 nM
   TI
   LI
   LO
   TS
4
Ki = 5011.87 nM
   TI
   LI
   LO
   TS