Compound ID |
Compound Name |
Compound Formula |
CP0125632
|
((5Z,8Z)-Icosa-5,8,11,14-tetraenoylamino)-acetic acid
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|
C22H35NO3
|
3
|
1 |
EC50 = 20 nM
|
|
|
2 |
EC50 > 10000 nM
|
|
|
3 |
IC50 > 10000 nM
|
|
|
CP0422931
|
10-[2-(1H-indol-3-yl)ethyl]-1,3-dimethyl-6,7,8,9-tetrahydropurino[7,8-a][1,3]diazepine-2,4-dione
Show/Hide
|
C21H24N6O2
|
1
|
1 |
EC50 = 454 nM
|
|
|
CP0392989
|
9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C20H22N6O2
|
2
|
1 |
EC50 = 562 nM
|
|
|
2 |
IC50 = 944 nM
|
|
|
CP0045801
|
(10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tetrahydro-6H-benzo[c]chromen-1-ol
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|
C21H30O2
|
1
|
1 |
EC50 = 4610 nM
|
|
|
CP0422932
|
6-[2-(1H-indol-3-yl)ethyl]-2,4-dimethyl-7,8-dihydropurino[7,8-a]imidazole-1,3-dione
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|
C19H20N6O2
|
1
|
1 |
EC50 = 5680 nM
|
|
|
CP0048192
|
2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl)-5-(2-methyloctan-2-yl)phenol
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|
C24H40O3
|
2
|
1 |
EC50 = 5990 nM
|
|
|
2 |
IC50 = 5990 nM
|
|
|
CP0389155
|
(4Z)-2-[(4-bromophenyl)methylsulfanyl]-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-1H-imidazol-5-one
Show/Hide
|
C24H18BrClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 2290 nM
|
|
|
CP0389156
|
(4Z)-2-benzylsulfanyl-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-1H-imidazol-5-one
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|
C24H19ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0389157
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-3-methyl-2-[(4-methylphenyl)methylsulfanyl]imidazol-4-one
Show/Hide
|
C26H23ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0389159
|
(2Z)-2-[[3-[6-(4-chlorophenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C25H27ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 650 nM
|
|
|
CP0396299
|
(2Z)-2-[[3-[4-(4-chlorophenoxy)butoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C23H23ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 2380 nM
|
|
|
CP0396300
|
(2Z)-2-[[3-[6-(4-propan-2-ylphenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C28H34N2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0396303
|
(4Z)-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-(2-phenylethylsulfanyl)-1H-imidazol-5-one
Show/Hide
|
C25H21ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 4780 nM
|
|
|
CP0396304
|
(4Z)-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-fluorophenyl)methylsulfanyl]-1H-imidazol-5-one
Show/Hide
|
C24H18ClFN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0396305
|
(2Z)-2-[[3-[5-(4-chlorophenoxy)pentoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C24H25ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 1140 nM
|
|
|
CP0396306
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2,3-dihydroimidazo[2,1-b][1,3]thiazol-6-one
Show/Hide
|
C19H15ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0396308
|
(4Z)-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-methylphenyl)methylsulfanyl]-1H-imidazol-5-one
Show/Hide
|
C25H21ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0396310
|
(2Z)-2-[[3-[3-(4-chlorophenoxy)propoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C22H21ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 3250 nM
|
|
|
CP0396311
|
(2Z)-2-[[3-[6-(4-methylphenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C26H30N2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 238 nM
|
|
|
CP0396331
|
(2Z)-2-[[3-[2-(4-chlorophenoxy)ethoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C21H19ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 5000 nM
|
|
|
CP0396341
|
(4Z)-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-[(4-chlorophenyl)methylsulfanyl]-1H-imidazol-5-one
Show/Hide
|
C24H18Cl2N2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0396346
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
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|
C17H12ClNO3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0408491
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
Show/Hide
|
C17H12ClNO2S2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0408540
|
(6Z)-6-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
Show/Hide
|
C19H15ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0408541
|
(2Z)-2-[[3-[(4-fluorophenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C20H17FN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0429381
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-3-methyl-2-methylsulfanylimidazol-4-one
Show/Hide
|
C19H17ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0429382
|
(2Z)-2-[[3-[7-(4-chlorophenoxy)heptoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C26H29ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 1710 nM
|
|
|
CP0429401
|
(2Z)-2-[[3-[6-(4-ethylphenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C27H32N2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 25000 nM
|
|
|
CP0429402
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-imino-1-methylimidazolidin-4-one
Show/Hide
|
C18H16ClN3O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0429406
|
(2Z)-2-[[3-(2-phenylethoxy)phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C21H20N2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0429408
|
(2Z)-2-[[3-[6-(2-chlorophenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C25H27ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0432722
|
(2Z)-2-[[3-[(4-methylphenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C21H20N2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 3590 nM
|
|
|
CP0445929
|
(2Z)-2-[[3-[6-(2,6-dimethylphenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C27H32N2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 10000 nM
|
|
|
CP0470826
|
(2Z)-2-[[3-[(4-bromophenyl)methoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C20H17BrN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 1730 nM
|
|
|
CP0471723
|
(2Z)-2-[[3-[8-(4-chlorophenoxy)octoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C27H31ClN2O3S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 1150 nM
|
|
|
CP0471783
|
(5Z)-5-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-sulfanylideneimidazolidin-4-one
Show/Hide
|
C17H13ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 33000 nM
|
|
|
CP0471793
|
(4Z)-4-[[3-[(4-chlorophenyl)methoxy]phenyl]methylidene]-2-methylsulfanyl-1H-imidazol-5-one
Show/Hide
|
C18H15ClN2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 13800 nM
|
|
|
CP0471794
|
(2Z)-2-[[3-(3-phenylpropoxy)phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C22H22N2O2S
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 = 1490 nM
|
|
|
CP0471795
|
(2Z)-2-[[3-[6-(3-chlorophenoxy)hexoxy]phenyl]methylidene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3-one
Show/Hide
|
C25H27ClN2O3S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0085151
|
9-(4-chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C18H20ClN5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0123281
|
9-(4-chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C17H18ClN5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0378535
|
9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C24H30N6O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0378537
|
9-(4-methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C19H23N5O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0422929
|
9-ethyl-1,3-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Show/Hide
|
C12H17N5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0422930
|
6-(4-hydroxyphenyl)-2,4-dimethyl-7,8-dihydropurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C15H15N5O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0422933
|
9-(3,4-dimethoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C20H25N5O4
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0427936
|
1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione
Show/Hide
|
C18H21N5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0466255
|
4-[(1R,6R)-3-methyl-6-prop-1-en-2-ylcyclohex-2-en-1-yl]-5-pentylbenzene-1,3-diol
Show/Hide
|
C21H30O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0466257
|
1,3-dimethyl-9-pentyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Show/Hide
|
C15H23N5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0466263
|
9-(2-methoxyethyl)-1,3-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Show/Hide
|
C13H19N5O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0478985
|
9-butyl-1,3-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Show/Hide
|
C14H21N5O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0490958
|
(4Z,7S,8E,10Z,12E,14E,16R,17S)-7,16,17-trihydroxydocosa-4,8,10,12,14-pentaenoic acid
Show/Hide
|
C22H34O5
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0507518
|
9-[2-(diethylamino)ethyl]-1,3-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
Show/Hide
|
C16H26N6O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
IC50 > 10000 nM
|
|
|
CP0003146
|
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H21Cl3N4O
|
2
|
1 |
EC50 = 10100 nM
|
|
|
2 |
IC50 = 10100 nM
|
|
|
CP0659892
|
(Z)-2-(3-(4-Chlorobenzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H17ClN2O2S
|
1
|
1 |
IC50 = 279 nM
|
|
|
CP0877023
|
(Z)-2-(3-(2-Chlorobenzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H17ClN2O2S
|
1
|
1 |
IC50 = 1650 nM
|
|
|
CP0859209
|
(Z)-2-(3-(2,4-Dichlorobenzyloxy)benzylidene)-6,7-dihydro-2Himidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H16Cl2N2O2S
|
1
|
1 |
IC50 = 2550 nM
|
|
|
CP0849218
|
(Z)-2-(3-(2,4-dichlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H18Cl2N2O2S
|
1
|
1 |
IC50 = 4610 nM
|
|
|
CP0868197
|
(Z)-2-(3-(3,4-Dichlorobenzyloxy)benzylidene)-6,7-dihydro-2Himidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H16Cl2N2O2S
|
1
|
1 |
IC50 = 6160 nM
|
|
|
CP0893073
|
(Z)-3-((3-Oxo-6,7-dihydro-3H-imidazo[2,1-b][1,3]thiazin-2(5H)-ylidene)methyl)phenyl benzoate
Show/Hide
|
C20H16N2O3S
|
1
|
1 |
IC50 = 6350 nM
|
|
|
CP0893067
|
(Z)-3-((3-oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-ylidene)methyl)phenyl 4-methylbenzoate
Show/Hide
|
C22H20N2O3S
|
1
|
1 |
IC50 = 6450 nM
|
|
|
CP0898591
|
(Z)-2-(3-(2-Chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19ClN2O2S
|
1
|
1 |
IC50 = 6480 nM
|
|
|
CP0849167
|
(Z)-2-(3-(Benzyloxy)benzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C20H18N2O2S
|
1
|
1 |
IC50 = 7220 nM
|
|
|
CP0393601
|
3-benzyl-5-hydroxy-7-(2-methyloctan-2-yl)chromen-2-one
Show/Hide
|
C25H30O3
|
1
|
1 |
IC50 = 8100 nM
|
|
|
CP0374913
|
5-methoxy-3-[(3-methoxyphenyl)methyl]-7-pentylchromen-2-one
Show/Hide
|
C23H26O4
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0374915
|
3-[(4-chlorophenyl)methyl]-5-methoxy-7-pentylchromen-2-one
Show/Hide
|
C22H23ClO3
|
1
|
1 |
IC50 = 10000 nM
|
|
|
CP0375105
|
7-(1-butylcyclohexyl)-5-methoxy-3-[(2-methoxyphenyl)methyl]chromen-2-one
Show/Hide
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C28H34O4
|
1
|
1 |
IC50 > 10000 nM
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CP0375117
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3-benzyl-6-hydroxy-5,7,8-trimethylchromen-2-one
Show/Hide
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C19H18O3
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1
|
1 |
IC50 > 10000 nM
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CP0375124
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3-Benzyl-5-isopropyl-8-methylchromen-2-one
Show/Hide
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C20H20O2
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1
|
1 |
IC50 > 10000 nM
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CP0375125
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6-hydroxy-5,7,8-trimethyl-3-[(2-methylphenyl)methyl]chromen-2-one
Show/Hide
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C20H20O3
|
1
|
1 |
IC50 > 10000 nM
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CP0375127
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3-benzyl-5-methoxy-7-(2-methyloctan-2-yl)chromen-2-one
Show/Hide
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C26H32O3
|
1
|
1 |
IC50 > 10000 nM
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CP0375165
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5-methoxy-3-[(2-methoxyphenyl)methyl]-7-(2-methylnonan-2-yl)chromen-2-one
Show/Hide
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C28H36O4
|
1
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1 |
IC50 > 10000 nM
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CP0375169
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3-[(2-chlorophenyl)methyl]-5-methoxy-7-pentylchromen-2-one
Show/Hide
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C22H23ClO3
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1
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1 |
IC50 > 10000 nM
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CP0375170
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5-hydroxy-3-[(3-hydroxyphenyl)methyl]-7-pentylchromen-2-one
Show/Hide
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C21H22O4
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1
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1 |
IC50 > 10000 nM
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CP0375171
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3-[(4-fluorophenyl)methyl]-6-hydroxy-5,7,8-trimethylchromen-2-one
Show/Hide
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C19H17FO3
|
1
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1 |
IC50 >= 10000 nM
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CP0375172
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6-methoxy-3-[(2-methoxyphenyl)methyl]-5,7,8-trimethylchromen-2-one
Show/Hide
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C21H22O4
|
1
|
1 |
IC50 > 10000 nM
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CP0376853
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7-(1-butylcyclopentyl)-5-methoxy-3-[(2-methoxyphenyl)methyl]chromen-2-one
Show/Hide
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C27H32O4
|
1
|
1 |
IC50 > 10000 nM
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CP0376854
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5-hydroxy-3-[(2-methylphenyl)methyl]-7-pentylchromen-2-one
Show/Hide
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C22H24O3
|
1
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1 |
IC50 > 10000 nM
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CP0387822
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7-(1-butylcyclohexyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]chromen-2-one
Show/Hide
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C26H30O4
|
1
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1 |
IC50 >= 10000 nM
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CP0387823
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5-methoxy-3-[(2-methoxyphenyl)methyl]-7-pentylchromen-2-one
Show/Hide
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C23H26O4
|
1
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1 |
IC50 > 10000 nM
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CP0387824
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5-methoxy-3-[(2-methoxyphenyl)methyl]-7-(2-methyloctan-2-yl)chromen-2-one
Show/Hide
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C27H34O4
|
1
|
1 |
IC50 > 10000 nM
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CP0387826
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5-methoxy-3-[(2-methylphenyl)methyl]-7-pentylchromen-2-one
Show/Hide
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C23H26O3
|
1
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1 |
IC50 > 10000 nM
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CP0391309
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7-bromo-5-methoxy-3-[(3-methoxyphenyl)methyl]chromen-2-one
Show/Hide
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C18H15BrO4
|
1
|
1 |
IC50 > 10000 nM
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CP0393582
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3-Benzyl-5-methoxy-7-methylchromen-2-one
Show/Hide
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C18H16O3
|
1
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1 |
IC50 > 10000 nM
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|
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CP0393584
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3-[(2-hydroxyphenyl)methyl]-8-methyl-5-propan-2-ylchromen-2-one
Show/Hide
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C20H20O3
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0393585
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3-[(4-bromophenyl)methyl]-5-methoxy-7-pentylchromen-2-one
Show/Hide
|
C22H23BrO3
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0393598
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6-methoxy-5,7,8-trimethyl-3-[(2-methylphenyl)methyl]chromen-2-one
Show/Hide
|
C21H22O3
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0393599
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3-[(2-methoxyphenyl)methyl]-5,8-dimethylchromen-2-one
Show/Hide
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C19H18O3
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0393600
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7-(1-butylcyclopentyl)-5-hydroxy-3-[(2-hydroxyphenyl)methyl]chromen-2-one
Show/Hide
|
C25H28O4
|
1
|
1 |
IC50 >= 10000 nM
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|
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CP0393602
|
3-[(2-chlorophenyl)methyl]-5-hydroxy-7-pentylchromen-2-one
Show/Hide
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C21H21ClO3
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0393614
|
5-Isopropyl-3,8-dimethylchromen-2-one
Show/Hide
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C14H16O2
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0394936
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3-[(4-fluorophenyl)methyl]-6-methoxy-5,7,8-trimethylchromen-2-one
Show/Hide
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C20H19FO3
|
1
|
1 |
IC50 > 10000 nM
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|
|
CP0409866
|
3-benzyl-6-methoxy-5,7,8-trimethylchromen-2-one
Show/Hide
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C20H20O3
|
1
|
1 |
IC50 >= 10000 nM
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|
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CP0659851
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(Z)-2-(2,4-dimethoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0659893
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(Z)-2-(3-(4-chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19ClN2O2S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0659958
|
(Z)-2-(2-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
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C13H11ClN2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0677588
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(Z)-2-benzylidene-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
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C13H12N2OS
|
1
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1 |
IC50 > 10000 nM
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CP0692927
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(Z)-2-(2,3-Difluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
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C13H10F2N2OS
|
1
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1 |
IC50 > 10000 nM
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CP0709769
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(Z)-2-(3-(3-Chlorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
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C21H19ClN2O2S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849166
|
(Z)-2-(4-bromobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11BrN2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849168
|
(Z)-2-(4-methoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C14H14N2O2S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849169
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(Z)-2-(2,4-Difluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10F2N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849399
|
6,6-diphenyl-2,3-dihydroimidazo[2,1-b]thiazol-5(6H)-one
Show/Hide
|
C17H14N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849409
|
(Z)-2-(2-methoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C14H14N2O2S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849467
|
(Z)-2-(3-phenoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C19H16N2O2S
|
1
|
1 |
IC50 = 10000 nM
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|
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CP0849468
|
(Z)-2-(3,4-dimethoxybenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849470
|
(Z)-2-(3-nitrobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11N3O3S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849472
|
(Z)-2-(3-phenylallylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H14N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0849480
|
(Z)-3-(3-phenylallylidene)-3,5,6,7-tetrahydro-2H-imidazo[2,1-b][1,3]thiazin-2-one
Show/Hide
|
C15H14N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0849481
|
1-lysophosphatidylinositol
Show/Hide
|
C29H49O12P
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0850010
|
(Z)-2-(2,6-Dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0858888
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(Z)-2-(2,3-dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0858889
|
(Z)-2-(4-isopropylbenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C16H18N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859207
|
(Z)-2-(4-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11ClN2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859208
|
(Z)-ethyl 2-(3-((3-oxo-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-ylidene)methyl)phenoxy)acetate
Show/Hide
|
C18H20N2O4S
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859210
|
2,2-diphenyl-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C19H18N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859211
|
ethyl 5-oxo-6,6-diphenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylate
Show/Hide
|
C20H18N2O3S
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0859212
|
2,2-diphenyl-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C18H16N2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0859457
|
(Z)-2-(3-chlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11ClN2OS
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0859468
|
(Z)-2-(2,4-Dichlorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]-thiazin-3(5H)-one
Show/Hide
|
C13H10Cl2N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859481
|
(Z)-2-(biphenyl-4-ylmethylene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C20H18N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0859491
|
3,3-diphenyl-3,5,6,7-tetrahydro-2H-imidazo[2,1-b][1,3]thiazin-2-one
Show/Hide
|
C18H16N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0866547
|
ethyl 6-oxo-5,5-diphenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole-2-carboxylate
Show/Hide
|
C20H18N2O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0866629
|
3,3-diphenyl-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-2(3H)-one
Show/Hide
|
C19H18N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0866766
|
5,5-diphenyl-2,3-dihydroimidazo[2,1-b]thiazol-6(5H)-one
Show/Hide
|
C17H14N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0866767
|
(Z)-2-(1-phenylethylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C15H16N2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0867263
|
(Z)-2-(4-nitrobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11N3O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0868782
|
(Z)-2-(3-(4-Fluorobenzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H19FN2O2S
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0868783
|
(Z)-2-(4-(dimethylamino)benzylidene)-6,7-dihydro-2H-imidazo[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H17N3OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0900469
|
(Z)-2-(3-(Benzyloxy)benzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C21H20N2O2S
|
1
|
1 |
IC50 = 10000 nM
|
|
|
CP0905395
|
(Z)-2-(2-Fluorobenzylidene)-6,7-dihydro-2H-imidazo[2,1-b]-[1,3]thiazin-3(5H)-one
Show/Hide
|
C13H11FN2OS
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0916683
|
(Z)-2-(2,3-Dimethoxybenzylidene)-6,7-dihydro-2H-imidazo-[2,1-b][1,3]thiazin-3(5H)-one
Show/Hide
|
C15H16N2O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0375166
|
3-[(2-methoxyphenyl)methyl]-5-methyl-8-propan-2-ylchromen-2-one
Show/Hide
|
C21H22O3
|
1
|
1 |
IC50 = 11300 nM
|
|
|
CP0393612
|
5-hydroxy-3-[(2-hydroxyphenyl)methyl]-7-(2-methylnonan-2-yl)chromen-2-one
Show/Hide
|
C26H32O4
|
1
|
1 |
IC50 = 12500 nM
|
|
|
CP0881784
|
(Z)-2-(3-phenoxybenzylidene)-5,6,7,8-tetrahydroimidazo[2,1-b][1,3]thiazepin-3(2H)-one
Show/Hide
|
C20H18N2O2S
|
1
|
1 |
IC50 = 14100 nM
|
|
|
CP0859466
|
(Z)-3-((3-Oxo-6,7-dihydro-3H-imidazo[2,1-b][1,3]thiazin-2(5H)-ylidene)methyl)phenyl 4-chloro-benzoate
Show/Hide
|
C20H15ClN2O3S
|
1
|
1 |
IC50 = 14300 nM
|
|
|
CP0397664
|
5-hydroxy-3-[(2-hydroxyphenyl)methyl]-7-(2-methyloctan-2-yl)chromen-2-one
Show/Hide
|
C25H30O4
|
1
|
1 |
IC50 = 15900 nM
|
|
|