| Compound ID |
Compound Name |
Compound Formula |
|
CP0380668
|
N-[2-(4-ethyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C15H19N3O2
|
2
|
| 1 |
EC50 = 0.021 nM
|
|
|
| 2 |
Ki = 0.062 nM
|
|
|
|
CP0034701
|
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]acetamide
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|
C13H16N2O2
|
20
|
| 1 |
EC50 = 0.0257 nM
|
|
|
| 2 |
EC50 = 0.026 nM
|
|
|
| 3 |
EC50 = 0.098 nM
|
|
|
| 4 |
EC50 = 0.11 nM
|
|
|
| 5 |
EC50 = 1.5 nM
|
|
|
| 6 |
EC50 = 1.92 nM
|
|
|
| 7 |
EC50 = 2.2 nM
|
|
|
| 8 |
EC50 = 2.24 nM
|
|
|
| 9 |
IC50 = 0.11 nM
|
|
|
| 10 |
Ki = 0.091 nM
|
|
|
| 11 |
Ki = 0.13 nM
|
|
|
| 12 |
Ki = 0.18 nM
|
|
|
| 13 |
Ki = 0.2 nM
|
|
|
| 14 |
Ki = 0.22 nM
|
|
|
| 15 |
Ki = 0.23 nM
|
|
|
| 16 |
Ki = 0.24 nM
|
|
|
| 17 |
Ki = 0.27 nM
|
|
|
| 18 |
Ki = 0.296 nM
|
|
|
| 19 |
Ki = 0.4571 nM
|
|
|
| 20 |
Ki = 0.525 nM
|
|
|
|
CP0419698
|
US10781182, Compound IA2-121
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|
C14H18ClN3O3
|
3
|
| 1 |
EC50 = 0.035 nM
|
|
|
| 2 |
EC50 = 0.14 nM
|
|
|
| 3 |
Ki = 0.88 nM
|
|
|
|
CP0444082
|
US10781182, Compound IA2-120
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|
C15H21N3O3
|
3
|
| 1 |
EC50 = 0.036 nM
|
|
|
| 2 |
EC50 = 0.18 nM
|
|
|
| 3 |
Ki = 1.1 nM
|
|
|
|
CP0444081
|
N-[2-(2-ethoxy-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
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|
C15H19N3O3
|
3
|
| 1 |
EC50 = 0.037 nM
|
|
|
| 2 |
EC50 = 0.32 nM
|
|
|
| 3 |
Ki = 0.34 nM
|
|
|
|
CP0534080
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]acetamide
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|
C14H19N3O3
|
3
|
| 1 |
EC50 = 0.04 nM
|
|
|
| 2 |
EC50 = 0.33 nM
|
|
|
| 3 |
Ki = 0.42 nM
|
|
|
|
CP0520740
|
N-[2-(2-methoxy-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C14H17N3O3
|
3
|
| 1 |
EC50 = 0.042 nM
|
|
|
| 2 |
EC50 = 0.42 nM
|
|
|
| 3 |
Ki = 0.61 nM
|
|
|
|
CP0565247
|
N-[2-(2,6-dimethoxybenzimidazol-1-yl)ethyl]acetamide
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|
C13H17N3O3
|
3
|
| 1 |
EC50 = 0.042 nM
|
|
|
| 2 |
EC50 = 0.2 nM
|
|
|
| 3 |
Ki = 1.2 nM
|
|
|
|
CP0429924
|
N-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]acetamide
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|
C16H18N2O2
|
2
|
| 1 |
EC50 = 0.05 nM
|
|
|
| 2 |
Ki = 0.4 nM
|
|
|
|
CP0450973
|
US10781182, Compound IA2-143
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|
C13H16ClN3O3
|
3
|
| 1 |
EC50 = 0.063 nM
|
|
|
| 2 |
EC50 = 0.25 nM
|
|
|
| 3 |
Ki = 2.1 nM
|
|
|
|
CP0548271
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]butanamide
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|
C16H23N3O3
|
2
|
| 1 |
EC50 = 0.14 nM
|
|
|
| 2 |
Ki = 0.39 nM
|
|
|
|
CP0045783
|
N-[2-(5-methoxy-2-phenyl-1-benzofuran-3-yl)ethyl]acetamide
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|
C19H19NO3
|
1
|
| 1 |
EC50 = 0.17 nM
|
|
|
|
CP0178199
|
Agomelatine
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|
C15H17NO2
|
7
|
| 1 |
EC50 = 0.1995 nM
|
|
|
| 2 |
EC50 = 1.4 nM
|
|
|
| 3 |
EC50 = 1.56 nM
|
|
|
| 4 |
EC50 = 1.6 nM
|
|
|
| 5 |
Ki = 0.1 nM
|
|
|
| 6 |
Ki = 0.12 nM
|
|
|
| 7 |
Ki = 0.1202 nM
|
|
|
|
CP0393386
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-methylurea
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|
C16H19N3O2
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0429915
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]acetamide
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|
C18H21NO2
|
2
|
| 1 |
EC50 = 0.2 nM
|
|
|
| 2 |
Ki = 0.1 nM
|
|
|
|
CP0548270
|
US10781182, Compound IA2-140
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|
C14H19N3O3
|
3
|
| 1 |
EC50 = 0.233 nM
|
|
|
| 2 |
EC50 = 1.92 nM
|
|
|
| 3 |
Ki = 2.2 nM
|
|
|
|
CP0548268
|
N-[2-(6-methoxy-2-methylsulfanylbenzimidazol-1-yl)ethyl]acetamide
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|
C13H17N3O2S
|
2
|
| 1 |
EC50 = 0.24 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0372709
|
N-[2-(7-benzyl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C22H23NO2
|
2
|
| 1 |
EC50 = 0.5129 nM
|
|
|
| 2 |
Ki = 2.7 nM
|
|
|
|
CP0419697
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]cyclopropanecarboxamide
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|
C16H21N3O3
|
2
|
| 1 |
EC50 = 0.75 nM
|
|
|
| 2 |
Ki = 0.71 nM
|
|
|
|
CP0428962
|
N-[2-(2-methoxyquinolin-8-yl)ethyl]acetamide
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|
C14H16N2O2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0404133
|
N-[(1-methyl-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
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|
C14H20N2O
|
2
|
| 1 |
EC50 = 0.9 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
|
CP0429922
|
1-[(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)methyl]-3-propylurea
Show/Hide
|
C18H23N3O2
|
2
|
| 1 |
EC50 = 0.9 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0459154
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C17H19NO2
|
2
|
| 1 |
EC50 = 0.9 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0419699
|
US10781182, Compound IA2-142
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|
C15H20ClN3O3
|
3
|
| 1 |
EC50 = 0.937 nM
|
|
|
| 2 |
EC50 = 2.13 nM
|
|
|
| 3 |
Ki = 13 nM
|
|
|
|
CP0534038
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]propanamide
Show/Hide
|
C15H21N3O3
|
2
|
| 1 |
EC50 = 0.97 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0105645
|
N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]cyclopropanecarboxamide
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|
C18H17NO3
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 1.9 nM
|
|
|
|
CP0309821
|
N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]cyclopropanecarboxamide
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|
C18H17NO3
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
|
CP0413687
|
N-[(5-methoxy-1-methyl-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
Show/Hide
|
C15H22N2O2
|
2
|
| 1 |
EC50 = 1.7 nM
|
|
|
| 2 |
Ki = 0.03 nM
|
|
|
|
CP0430453
|
N-[2-[7-[4-[[3-(2-acetamidoethyl)-1-benzothiophen-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C30H34N2O4S
|
2
|
| 1 |
EC50 = 1.94 nM
|
|
|
| 2 |
Ki = 3.47 nM
|
|
|
|
CP0413688
|
N-[(1-propyl-3,4-dihydro-2H-quinolin-2-yl)methyl]acetamide
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|
C15H22N2O
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 5.8 nM
|
|
|
|
CP0410497
|
(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylurea
Show/Hide
|
C16H18N2O2
|
2
|
| 1 |
EC50 = 2 nM
|
|
|
| 2 |
Ki = 0.3 nM
|
|
|
|
CP0462764
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]butanamide
Show/Hide
|
C14H19N3O2
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0469064
|
N-[2-[7-[4-[4-[4-(hydroxymethyl)phenyl]phenoxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C31H33NO4
|
2
|
| 1 |
EC50 = 2.37 nM
|
|
|
| 2 |
Ki = 0.09 nM
|
|
|
|
CP0373460
|
N-[2-[7-[4-[[3-(2-acetamidoethyl)-1H-indol-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C30H35N3O4
|
2
|
| 1 |
EC50 = 2.38 nM
|
|
|
| 2 |
Ki = 4.04 nM
|
|
|
|
CP0400793
|
N-[2-[7-[4-[[3-(2-acetamidoethyl)-1-benzofuran-5-yl]oxy]butoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C30H34N2O5
|
2
|
| 1 |
EC50 = 2.49 nM
|
|
|
| 2 |
Ki = 1.38 nM
|
|
|
|
CP0390834
|
methyl 2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]acetate
Show/Hide
|
C31H33NO5
|
2
|
| 1 |
EC50 = 2.89 nM
|
|
|
| 2 |
Ki = 0.07 nM
|
|
|
|
CP0417995
|
N-[3-[5-methoxy-2-(3-methoxyphenyl)phenyl]propyl]propanamide
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|
C20H25NO3
|
2
|
| 1 |
EC50 = 2.94 nM
|
|
|
| 2 |
Ki = 32.7 nM
|
|
|
|
CP0425881
|
N-[2-[7-(3-propan-2-ylphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C24H27NO2
|
2
|
| 1 |
EC50 = 3.02 nM
|
|
|
| 2 |
Ki = 13 nM
|
|
|
|
CP0400791
|
2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]acetic acid
Show/Hide
|
C30H31NO5
|
2
|
| 1 |
EC50 = 3.14 nM
|
|
|
| 2 |
Ki = 9.1 nM
|
|
|
|
CP0419695
|
N-[2-(2-ethoxy-6-methoxybenzimidazol-1-yl)ethyl]cyclobutanecarboxamide
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|
C17H23N3O3
|
2
|
| 1 |
EC50 = 3.58 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0467650
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]acetamide
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|
C12H15N3O2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0405073
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C16H19NO3S
|
2
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0377934
|
N-[2-[7-(cyclohexylmethyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H29NO2
|
2
|
| 1 |
EC50 = 4.467 nM
|
|
|
| 2 |
Ki = 9.2 nM
|
|
|
|
CP0121891
|
N-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]acetamide
Show/Hide
|
C17H17NO3
|
2
|
| 1 |
EC50 = 4.6 nM
|
|
|
| 2 |
Ki = 2.8 nM
|
|
|
|
CP0406180
|
N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]acetamide
Show/Hide
|
C16H15NO3
|
2
|
| 1 |
EC50 = 4.8 nM
|
|
|
| 2 |
Ki = 4.6 nM
|
|
|
|
CP0429916
|
2-methoxy-N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]acetamide
Show/Hide
|
C18H21NO3
|
2
|
| 1 |
EC50 = 5 nM
|
|
|
| 2 |
Ki = 0.6 nM
|
|
|
|
CP0485368
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]urea
Show/Hide
|
C19H24N2O2
|
2
|
| 1 |
EC50 = 5 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
|
CP0462765
|
N-[2-(6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]propanamide
Show/Hide
|
C13H17N3O2
|
1
|
| 1 |
EC50 = 5.1 nM
|
|
|
|
CP0121948
|
N-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C19H19NO3
|
2
|
| 1 |
EC50 = 5.2 nM
|
|
|
| 2 |
Ki = 23.6 nM
|
|
|
|
CP0429921
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-methylthiourea
Show/Hide
|
C18H22N2OS
|
2
|
| 1 |
EC50 = 6 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0464195
|
N-[(1-phenyl-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
Show/Hide
|
C19H22N2O
|
2
|
| 1 |
EC50 = 6.2 nM
|
|
|
| 2 |
Ki = 1.6 nM
|
|
|
|
CP0414625
|
N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]acetamide
Show/Hide
|
C16H15NO3
|
2
|
| 1 |
EC50 = 7.7 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
|
CP0407039
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C32H40N2O4
|
2
|
| 1 |
EC50 = 7.75 nM
|
|
|
| 2 |
Ki = 0.26 nM
|
|
|
|
CP0472545
|
N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]-2-methylpropanamide
Show/Hide
|
C18H19NO3
|
2
|
| 1 |
EC50 = 8.1 nM
|
|
|
| 2 |
Ki = 158 nM
|
|
|
|
CP0396581
|
N-[3-[5-methoxy-2-[2-(3-methoxyphenyl)ethynyl]phenyl]propyl]propanamide
Show/Hide
|
C22H25NO3
|
2
|
| 1 |
EC50 = 8.38 nM
|
|
|
| 2 |
Ki = 38.2 nM
|
|
|
|
CP0414939
|
1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
Show/Hide
|
C20H26N2O2
|
2
|
| 1 |
EC50 = 9 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0409354
|
N-[3-[5-methoxy-2-[(3-methoxyphenyl)methoxy]phenyl]propyl]propanamide
Show/Hide
|
C21H27NO4
|
3
|
| 1 |
EC50 = 9.03 nM
|
|
|
| 2 |
Ki = 121 nM
|
|
|
| 3 |
Ki = 1348.96 nM
|
|
|
|
CP0400713
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]cyclopropanecarboxamide
Show/Hide
|
C34H38N2O4
|
2
|
| 1 |
EC50 = 9.1 nM
|
|
|
| 2 |
Ki = 1.07 nM
|
|
|
|
CP0121949
|
2-fluoro-N-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]acetamide
Show/Hide
|
C16H14FNO3
|
2
|
| 1 |
EC50 = 9.5 nM
|
|
|
| 2 |
Ki = 5.7 nM
|
|
|
|
CP0428961
|
1-ethyl-3-[2-(2-methoxyquinolin-8-yl)ethyl]urea
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0469375
|
1-ethyl-3-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]thiourea
Show/Hide
|
C19H24N2OS
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
Ki = 4 nM
|
|
|
|
CP0847772
|
2,2-difluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H17F2NO3
|
2
|
| 1 |
EC50 = 10.23 nM
|
|
|
| 2 |
Ki = 1.905 nM
|
|
|
|
CP0401701
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]furan-2-carboxamide
Show/Hide
|
C35H36N2O5
|
2
|
| 1 |
EC50 = 11.2 nM
|
|
|
| 2 |
Ki = 0.64 nM
|
|
|
|
CP0373463
|
N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]but-3-enamide
Show/Hide
|
C34H38N2O4
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
Ki = 0.79 nM
|
|
|
|
CP0458757
|
4-azamelatonin
Show/Hide
|
C12H15N3O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0486875
|
N-[2-(2-methoxy-5,6,7,8-tetrahydropyrido[2,3-b]indol-9-yl)ethyl]acetamide
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C16H21N3O2
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1
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| 1 |
EC50 = 16 nM
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CP0429925
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(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methylthiourea
Show/Hide
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C16H18N2OS
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2
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| 1 |
EC50 = 16 nM
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| 2 |
Ki = 6 nM
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CP0373468
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N-[2-[7-[4-[8-[2-(but-3-enoylamino)ethyl]naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]but-3-enamide
Show/Hide
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C36H40N2O4
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2
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| 1 |
EC50 = 16.1 nM
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| 2 |
Ki = 0.92 nM
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CP0396582
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N-[3-[5-methoxy-2-[2-(3-methoxyphenyl)ethyl]phenyl]propyl]propanamide
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C22H29NO3
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2
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| 1 |
EC50 = 16.3 nM
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| 2 |
Ki = 22.2 nM
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CP0454903
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1-[2-(2-methoxyquinolin-8-yl)ethyl]-3-methylurea
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C14H17N3O2
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1
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| 1 |
EC50 = 19 nM
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CP0847773
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(R)-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)propionamide
Show/Hide
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C17H21NO3
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2
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| 1 |
EC50 = 19.5 nM
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| 2 |
Ki = 3.388 nM
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CP0432632
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N-(1-phenyl-3,4-dihydro-2H-quinolin-3-yl)propanamide
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C18H20N2O
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2
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| 1 |
EC50 = 20 nM
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| 2 |
Ki = 22 nM
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CP0393387
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
Show/Hide
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C19H24N2OS
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2
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| 1 |
EC50 = 20 nM
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| 2 |
Ki = 63 nM
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CP0416460
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1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]urea
Show/Hide
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C18H22N2O2
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2
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| 1 |
EC50 = 20 nM
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| 2 |
Ki = 2 nM
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CP0083725
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N-[2-(2-benzyl-5-methoxy-1-benzofuran-3-yl)ethyl]acetamide
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C20H21NO3
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1
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| 1 |
EC50 = 21 nM
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CP0407040
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methyl 2-[6-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-2-yl]propanoate
Show/Hide
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C32H35NO5
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2
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| 1 |
EC50 = 21.7 nM
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| 2 |
Ki = 0.37 nM
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CP0400794
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2-[6-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-2-yl]propanoic acid
Show/Hide
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C31H33NO5
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2
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| 1 |
EC50 = 22 nM
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| 2 |
Ki = 1.51 nM
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CP0452012
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N-[2-(5-fluoro-1-benzothiophen-3-yl)ethyl]acetamide
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C12H12FNOS
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2
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| 1 |
EC50 = 23.8 nM
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| 2 |
Ki = 24.6 nM
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CP0214091
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But-3-enoic acid [2-(2-benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-amide
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C22H23NO3
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1
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| 1 |
EC50 = 25 nM
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CP0877970
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rac-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
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C16H18FNO3
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2
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| 1 |
EC50 = 25.12 nM
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| 2 |
Ki = 4.677 nM
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CP0402287
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4-[4-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]phenyl]benzoic acid
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C31H31NO5
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2
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| 1 |
EC50 = 26.1 nM
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| 2 |
Ki = 0.55 nM
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CP0309822
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2-fluoro-N-[(8-methoxybenzo[e][1]benzofuran-1-yl)methyl]acetamide
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C16H14FNO3
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2
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| 1 |
EC50 = 29 nM
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| 2 |
Ki = 9.9 nM
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CP0391337
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1-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]-3-propylurea
Show/Hide
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C19H24N2O2
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2
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| 1 |
EC50 = 30 nM
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| 2 |
Ki = 5 nM
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CP0413683
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N-[(1-benzyl-3,4-dihydro-2H-quinolin-2-yl)methyl]acetamide
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C19H22N2O
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2
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| 1 |
EC50 = 31 nM
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| 2 |
Ki = 45 nM
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CP0474650
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1-ethyl-3-[2-(2-methoxyquinolin-8-yl)ethyl]thiourea
Show/Hide
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C15H19N3OS
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1
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| 1 |
EC50 = 31 nM
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CP0467651
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N-[2-(3-iodo-6-methoxypyrrolo[2,3-b]pyridin-1-yl)ethyl]acetamide
Show/Hide
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C12H14IN3O2
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1
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| 1 |
EC50 = 32 nM
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CP0452656
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N-[(1-benzyl-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
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C20H24N2O
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2
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| 1 |
EC50 = 36 nM
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| 2 |
Ki = 37 nM
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CP0098513
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N-[2-[5-methoxy-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
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C21H23NO4
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2
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| 1 |
EC50 = 37 nM
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| 2 |
Ki = 27 nM
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CP0385360
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3-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylpropanamide
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C15H16N2O2
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2
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| 1 |
EC50 = 38 nM
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| 2 |
Ki = 5 nM
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CP0514069
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N-[3-[5-methoxy-2-[(3-methoxyphenyl)methyl]phenyl]propyl]propanamide
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C21H27NO3
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2
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| 1 |
EC50 = 41.6 nM
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| 2 |
Ki = 39.5 nM
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CP0400795
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methyl 4-[4-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]phenyl]benzoate
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C32H33NO5
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2
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| 1 |
EC50 = 46.2 nM
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| 2 |
Ki = 2.37 nM
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CP0381571
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5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
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C13H13N3O3
|
3
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| 1 |
EC50 = 48 nM
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| 2 |
EC50 = 326 nM
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| 3 |
Ki = 35 nM
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CP0877971
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rac-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
Show/Hide
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C17H21NO3
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2
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| 1 |
EC50 = 48.98 nM
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| 2 |
Ki = 1.349 nM
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CP0406657
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3-(2-methoxyquinolin-8-yl)-N-methylpropanamide
Show/Hide
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C14H16N2O2
|
1
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| 1 |
EC50 = 65 nM
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CP0405082
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1-ethyl-3-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]thiourea
Show/Hide
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C18H22N2OS
|
2
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| 1 |
EC50 = 70 nM
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| 2 |
Ki = 29 nM
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CP0378677
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N-[3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamide
Show/Hide
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C16H19NO3
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2
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| 1 |
EC50 = 72.44 nM
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| 2 |
Ki = 10.96 nM
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CP0400796
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N-[2-[7-[4-[8-(2-acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
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C32H36N2O4
|
3
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| 1 |
EC50 = 73 nM
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| 2 |
Ki = 0.6 nM
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| 3 |
Ki = 3.1 nM
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CP0105646
|
1-ethyl-3-[2-(8-methoxybenzo[e][1]benzofuran-1-yl)ethyl]urea
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C18H20N2O3
|
2
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| 1 |
EC50 = 75 nM
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| 2 |
Ki = 157 nM
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CP0847771
|
(R)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
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C16H18FNO3
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2
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| 1 |
EC50 = 79.43 nM
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| 2 |
Ki = 5.888 nM
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CP0454899
|
1-[2-(2-methoxyquinolin-8-yl)ethyl]-3-methylthiourea
Show/Hide
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C14H17N3OS
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1
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| 1 |
EC50 = 90 nM
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CP0436038
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N-[2-[6-methoxy-3-(2,2,2-trifluoroacetyl)pyrrolo[2,3-b]pyridin-1-yl]ethyl]acetamide
Show/Hide
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C14H14F3N3O3
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1
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| 1 |
EC50 = 93 nM
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CP0405083
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1-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]-3-propylthiourea
Show/Hide
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C20H26N2OS
|
2
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| 1 |
EC50 = 100 nM
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| 2 |
Ki = 9 nM
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CP0472476
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1-ethyl-3-[(1-methyl-3,4-dihydro-2H-quinolin-2-yl)methyl]urea
Show/Hide
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C14H21N3O
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2
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| 1 |
EC50 = 110 nM
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| 2 |
Ki = 5.3 nM
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CP0192453
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But-3-enoic acid {2-[5-methoxy-2-(3-methoxy-benzyl)-benzofuran-3-yl]-ethyl}-amide
Show/Hide
|
C23H25NO4
|
1
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| 1 |
EC50 = 138 nM
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CP0404132
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1-ethyl-3-[(5-methoxy-1-methyl-3,4-dihydro-2H-quinolin-2-yl)methyl]urea
Show/Hide
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C15H23N3O2
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2
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| 1 |
EC50 = 160 nM
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| 2 |
Ki = 5 nM
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CP0474362
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N-[(1-benzyl-5-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
Show/Hide
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C21H26N2O2
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2
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| 1 |
EC50 = 177 nM
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| 2 |
Ki = 17 nM
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CP0436558
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N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]but-3-enamide
Show/Hide
|
C20H17F2NOS2
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2
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| 1 |
EC50 = 188 nM
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| 2 |
Ki = 52.8 nM
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CP0464190
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N-[[(2R)-1-benzyl-3,4-dihydro-2H-quinolin-2-yl]methyl]acetamide
Show/Hide
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C19H22N2O
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2
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| 1 |
EC50 = 192 nM
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| 2 |
Ki = 45 nM
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CP0424931
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N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]acetamide
Show/Hide
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C18H15F2NOS2
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2
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| 1 |
EC50 = 202 nM
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| 2 |
Ki = 57 nM
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CP0381574
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3-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylpropanamide
Show/Hide
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C15H18N2O2
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2
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| 1 |
EC50 = 204 nM
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| 2 |
Ki = 2.5 nM
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CP0404128
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N-(1,2,3,4-tetrahydroquinolin-2-ylmethyl)propanamide
Show/Hide
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C13H18N2O
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2
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| 1 |
EC50 = 242 nM
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| 2 |
Ki = 13 nM
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CP0071154
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2-(5-methoxy-1H-indol-3-yl)-N,N-dimethyl-ethanamine
Show/Hide
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C13H18N2O
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2
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| 1 |
EC50 = 257 nM
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| 2 |
Ki = 210 nM
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CP0382347
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2-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylacetamide
Show/Hide
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C14H14N2O2
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2
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| 1 |
EC50 = 289 nM
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| 2 |
Ki = 14 nM
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CP0847750
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(S)-N-(1-hydroxy-3-(7-methoxynaphthalen-1-yl)propan-2-yl)propionamide
Show/Hide
|
C17H21NO3
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2
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| 1 |
EC50 = 389.05 nM
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| 2 |
Ki = 181.97 nM
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CP0431495
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1-[(1-benzyl-5-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]-3-ethylurea
Show/Hide
|
C21H27N3O2
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2
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| 1 |
EC50 = 393 nM
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| 2 |
Ki = 132 nM
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CP0072976
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N-[2-[2-(cyclohexylmethyl)-5-methoxy-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C20H27NO3
|
1
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| 1 |
EC50 = 481 nM
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CP0397791
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2-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylacetamide
Show/Hide
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C14H16N2O2
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2
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| 1 |
EC50 = 525 nM
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| 2 |
Ki = 17 nM
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CP0382351
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5-[(5-methoxy-1H-indol-3-yl)methyl]-3-methyl-1,2,4-oxadiazole
Show/Hide
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C13H13N3O2
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2
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| 1 |
EC50 = 711 nM
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| 2 |
Ki = 170 nM
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CP0413684
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1-ethyl-3-[(1-methyl-3,4-dihydro-2H-quinolin-2-yl)methyl]thiourea
Show/Hide
|
C14H21N3S
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2
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| 1 |
EC50 = 809 nM
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| 2 |
Ki = 22 nM
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CP0464194
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N-[(5-methoxy-1,2,3,4-tetrahydroquinolin-2-yl)methyl]propanamide
Show/Hide
|
C14H20N2O2
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2
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| 1 |
EC50 = 906 nM
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| 2 |
Ki = 57 nM
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CP0072131
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2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-5-methyl-1,3,4-oxadiazole
Show/Hide
|
C14H15N3O2
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2
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| 1 |
EC50 = 961 nM
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| 2 |
Ki = 709 nM
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CP0376624
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2-[(5-methoxy-1H-indol-3-yl)methyl]-5-methyl-1,3-oxazole
Show/Hide
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C14H14N2O2
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2
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| 1 |
EC50 = 989 nM
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| 2 |
Ki = 280 nM
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CP0877969
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(S)-2-fluoro-N-(3-hydroxy-2-(7-methoxynaphthalen-1-yl)propyl)acetamide
Show/Hide
|
C16H18FNO3
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2
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| 1 |
EC50 = 1047.13 nM
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| 2 |
Ki = 346.74 nM
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CP0436037
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7-azamelatonin
Show/Hide
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C12H15N3O2
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1
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| 1 |
EC50 = 1100 nM
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CP0428960
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2-(2-methoxyquinolin-8-yl)ethylurea
Show/Hide
|
C13H15N3O2
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1
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| 1 |
EC50 = 1620 nM
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CP0404129
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1-ethyl-3-(1,2,3,4-tetrahydroquinolin-2-ylmethyl)urea
Show/Hide
|
C13H19N3O
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2
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| 1 |
EC50 = 2420 nM
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| 2 |
Ki = 115 nM
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CP0452655
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1-ethyl-3-(1,2,3,4-tetrahydroquinolin-2-ylmethyl)thiourea
Show/Hide
|
C13H19N3S
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2
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| 1 |
EC50 = 2660 nM
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| 2 |
Ki = 305 nM
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CP0095846
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N-[2-[5-methoxy-2-[(4-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H23NO4
|
1
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| 1 |
EC50 > 10000 nM
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CP0100122
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N-[2-(2-benzyl-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
|
C19H19NO2
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1
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| 1 |
EC50 > 10000 nM
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CP0217078
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N-[2-[5-methoxy-2-[(2-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H23NO4
|
1
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| 1 |
EC50 > 10000 nM
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CP0297769
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N-[2-[5-ethyl-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C22H25NO3
|
1
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| 1 |
EC50 > 10000 nM
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CP0301499
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N-[2-[5-methoxy-2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-3-yl]ethyl]acetamide
Show/Hide
|
C21H20F3NO3
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1
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| 1 |
EC50 > 10000 nM
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CP0452010
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N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]propanamide
Show/Hide
|
C19H17F2NOS2
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2
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| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 226 nM
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CP0452013
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2-bromo-N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]acetamide
Show/Hide
|
C18H14BrF2NOS2
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2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 22.1 nM
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CP0406181
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N-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]acetamide
Show/Hide
|
C17H17NO3
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2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 10 nM
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CP0414626
|
N-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C19H19NO3
|
2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 73 nM
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CP0443574
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1-ethyl-3-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]urea
Show/Hide
|
C17H18N2O3
|
2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 17 nM
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CP0389225
|
N-[(1-phenyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
Show/Hide
|
C18H20N2O
|
1
|
| 1 |
EC50 > 10000 nM
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CP0389226
|
N-[(1-methyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
Show/Hide
|
C13H18N2O
|
2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 83 nM
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CP0426377
|
N-[(1-ethyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
Show/Hide
|
C14H20N2O
|
2
|
| 1 |
EC50 > 10000 nM
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| 2 |
Ki = 20 nM
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CP0432491
|
N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]ethanesulfonamide
Show/Hide
|
C17H21NO3S
|
2
|
| 1 |
EC50 = 10000 nM
|
|
|
| 2 |
Ki = 7 nM
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|
CP0389325
|
2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazole
Show/Hide
|
C13H13N3O2
|
2
|
| 1 |
EC50 > 1000 nM
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|
|
| 2 |
Ki = 570 nM
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CP0389326
|
2-[(5-methoxy-1H-indol-3-yl)methyl]-5-methyl-1,3,4-oxadiazole
Show/Hide
|
C13H13N3O2
|
2
|
| 1 |
EC50 > 1000 nM
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|
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| 2 |
Ki = 210 nM
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CP0454898
|
methyl N-[2-(2-methoxyquinolin-8-yl)ethyl]carbamate
Show/Hide
|
C14H16N2O3
|
1
|
| 1 |
EC50 > 1000 nM
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|
|
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CP0488406
|
3-(2-methoxyquinolin-8-yl)-N-methylsulfonylpropanamide
Show/Hide
|
C14H16N2O4S
|
1
|
| 1 |
EC50 > 1000 nM
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CP0372536
|
N-[2-(8-methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamide
Show/Hide
|
C19H27N3O2
|
2
|
| 1 |
IC50 = 3.14 nM
|
|
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| 2 |
Ki = 6.607 nM
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CP0795225
|
1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylaminocarbonyl)oxime
Show/Hide
|
C19H16N2O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0425880
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]propanamide
Show/Hide
|
C19H25NO2
|
1
|
| 1 |
Ki = 0.013 nM
|
|
|
|
CP0499108
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C18H23NO2
|
1
|
| 1 |
Ki = 0.024 nM
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CP0376971
|
N-[2-(4-cyclopropyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C17H21N3O2
|
1
|
| 1 |
Ki = 0.026 nM
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|
|
|
CP0521668
|
2,2,2-Trifluoro-N-[2-(7-isopropyl-1,6-dihydro-2H-indeno-[5,4-b]furan-8-yl)ethyl]acetamide
Show/Hide
|
C18H20F3NO2
|
1
|
| 1 |
Ki = 0.032 nM
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CP0441548
|
N-[2-(4-ethyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C16H21N3O2
|
1
|
| 1 |
Ki = 0.039 nM
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CP0455738
|
N-[2-(4-cyclopropyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 0.044 nM
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|
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CP0494363
|
N-[2-(2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C15H17NO2
|
1
|
| 1 |
Ki = 0.045 nM
|
|
|
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CP0422004
|
N-[2-[7-(3-methoxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 0.057 nM
|
|
|
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CP0521667
|
N-[2-(7-pyridin-3-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamide
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
Ki = 0.069 nM
|
|
|
|
CP0055675
|
2-Iodomelatonin
Show/Hide
|
C13H15IN2O2
|
1
|
| 1 |
Ki = 0.08 nM
|
|
|
|
CP0458342
|
N-[2-(4-phenyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 0.082 nM
|
|
|
|
CP0501182
|
N-[2-(4-methyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]propanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 0.083 nM
|
|
|
|
CP0384067
|
N-[2-(2,7-dimethoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C17H21NO3
|
1
|
| 1 |
Ki = 0.099 nM
|
|
|
|
CP0437994
|
N-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C20H25NO2
|
1
|
| 1 |
Ki = 0.11 nM
|
|
|
|
CP0040580
|
N-[2-(5-methoxy-1-benzofuran-3-yl)ethyl]acetamide
Show/Hide
|
C13H15NO3
|
1
|
| 1 |
Ki = 0.15 nM
|
|
|
|
CP0458343
|
N-[2-(4-methyl-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl)ethyl]acetamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0390104
|
N-[2-[4-(trifluoromethyl)-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl]ethyl]propanamide
Show/Hide
|
C15H16F3N3O2
|
1
|
| 1 |
Ki = 0.31 nM
|
|
|
|
CP0510962
|
N-[2-(2-ethoxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C18H23NO3
|
1
|
| 1 |
Ki = 0.39 nM
|
|
|
|
CP0441549
|
N-[2-[4-(trifluoromethyl)-10-oxa-5,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-3-yl]ethyl]acetamide
Show/Hide
|
C14H14F3N3O2
|
1
|
| 1 |
Ki = 0.48 nM
|
|
|
|
CP0508414
|
N-[(8-methoxy-1-methyl-2,3-dihydrocyclopenta[a]naphthalen-1-yl)methyl]methanesulfonamide
Show/Hide
|
C17H21NO3S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0047706
|
N-[3-[2-(4-phenylbutyl)-1,3-benzoxazol-7-yl]propyl]cyclopropanecarboxamide
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 0.63 nM
|
|
|
|
CP0437993
|
N-[2-[7-(thiophen-3-ylmethyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C20H21NO2S
|
1
|
| 1 |
Ki = 0.88 nM
|
|
|
|
CP0401703
|
N-[2-[7-[4-[8-[2-(cyclopropanecarbonylamino)ethyl]naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]cyclopropanecarboxamide
Show/Hide
|
C36H40N2O4
|
1
|
| 1 |
Ki = 1.01 nM
|
|
|
|
CP0499107
|
1-ethyl-3-[2-(7-propan-2-yl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]urea
Show/Hide
|
C19H26N2O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0501489
|
N-[2-[7-(2-methoxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0521669
|
N-[2-[7-(1-benzothiophen-3-yl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C23H21NO2S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0186244
|
(4-Methoxy-6,7-dihydro-5H-dibenzo[a,c]cyclohepten-6-ylmethyl)-methoxymethyl-amine
Show/Hide
|
C20H23NO2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0501488
|
N-[2-[7-(4-tert-butylphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C25H29NO2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0429929
|
methyl N-[(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)methyl]carbamate
Show/Hide
|
C17H19NO3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0474642
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]butanamide
Show/Hide
|
C16H20N2O2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0448964
|
N-[2-(2-hydroxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C16H19NO3
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0377936
|
N-[2-[7-(4-methoxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C22H23NO3
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0548970
|
N-[2-(6-hexoxy-3,4-dihydro-2H-chromen-4-yl)ethyl]acetamide
Show/Hide
|
C19H29NO3
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0475208
|
N-[[(3R,4S)-1-methyl-4-phenyl-3,4-dihydro-2H-quinolin-3-yl]methyl]propanamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0389224
|
N-[[(1S,2R)-1-phenyl-1,2,3,4-tetrahydronaphthalen-2-yl]methyl]propanamide
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0193528
|
N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C31H34N2O4
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0415638
|
N-[2-[5-(3-phenylpropoxy)-1H-indol-3-yl]ethyl]acetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
|
CP0432490
|
N-[2-(8-methoxy-2,3-dihydro-1H-cyclopenta[a]naphthalen-1-yl)ethyl]acetamide
Show/Hide
|
C18H21NO2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0509510
|
N-[2-[2-(2-hydroxyethoxy)-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C18H23NO4
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0416462
|
N-[2-(2-methoxy-8,9-dihydro-7H-cyclopenta[h]quinolin-9-yl)ethyl]acetamide
Show/Hide
|
C17H20N2O2
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0375514
|
N-[2-[7-[8-(2-acetamidoethyl)naphthalen-2-yl]naphthalen-1-yl]ethyl]acetamide
Show/Hide
|
C28H28N2O2
|
1
|
| 1 |
Ki = 5.2 nM
|
|
|
|
CP0866793
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)propionamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 5.623 nM
|
|
|
|
CP0491332
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]acetamide
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0518308
|
N-[2-(6-methoxyquinolin-4-yl)ethyl]propanamide
Show/Hide
|
C15H18N2O2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0467376
|
N-[2-(2-butoxy-7-methoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C20H27NO3
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0385096
|
N-[2-[5-(3-phenoxypropoxy)-1H-indol-3-yl]ethyl]acetamide
Show/Hide
|
C21H24N2O3
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0383358
|
N-[2-(7-methoxy-2-propoxynaphthalen-1-yl)ethyl]propanamide
Show/Hide
|
C19H25NO3
|
1
|
| 1 |
Ki = 8.1 nM
|
|
|
|
CP0381636
|
2-((S)-2-Hydroxymethylindolin-1-ylmethyl)-melatonin
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
Ki = 9.8 nM
|
|
|
|
CP0874931
|
N-[2-(8-Methoxy-2-methyl-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)ethyl]acetamide
Show/Hide
|
C17H23N3O2
|
1
|
| 1 |
Ki = 11.75 nM
|
|
|
|
CP0920948
|
N-[2-(5-Methoxy-2-{[(methyl(phenyl)amino]methyl}-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C21H25N3O2
|
1
|
| 1 |
Ki = 15.49 nM
|
|
|
|
CP0514746
|
(+/-)-2-(2-Hydroxymethylindolin-1-ylmethyl)-melatonin
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
Ki = 17.5 nM
|
|
|
|
CP0458341
|
N-[2-(2-phenyl-7,8-dihydrofuro[2,3-g]benzimidazol-1-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0487668
|
N-[2-(2-cyclopropyl-6-methoxyquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C16H19N3O2
|
1
|
| 1 |
Ki = 22.1 nM
|
|
|
|
CP0390102
|
N-[3-(3-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO2
|
1
|
| 1 |
Ki = 23.3 nM
|
|
|
|
CP0869995
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)but-3-enamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
Ki = 23.99 nM
|
|
|
|
CP0389223
|
N-[(1-phenyl-3,4-dihydronaphthalen-2-yl)methyl]propanamide
Show/Hide
|
C20H21NO
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0499033
|
(+/-)-2-(2-Hydroxymethyl-5-methoxyindolin-1-ylmethyl)-melatonin
Show/Hide
|
C24H29N3O4
|
1
|
| 1 |
Ki = 34.5 nM
|
|
|
|
CP0486386
|
N-[2-[2-[2-(dimethylamino)ethoxy]-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C20H28N2O3
|
1
|
| 1 |
Ki = 42 nM
|
|
|
|
CP0420022
|
1-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]-3-methylthiourea
Show/Hide
|
C16H16N2O2S
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0849192
|
N-(2-(2-((1H-indol-1-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclobutanecarboxamide
Show/Hide
|
C25H27N3O2
|
1
|
| 1 |
Ki = 57.54 nM
|
|
|
|
CP0114370
|
4-P-PDOT
Show/Hide
|
C19H21NO
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0389221
|
N-[(1-benzyl-3,4-dihydro-2H-quinolin-3-yl)methyl]acetamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0859463
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclopropanecarboxamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
Ki = 61.66 nM
|
|
|
|
CP0426376
|
N-[[(1R,2R)-1-phenyl-1,2,3,4-tetrahydronaphthalen-2-yl]methyl]propanamide
Show/Hide
|
C20H23NO
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0081204
|
N-[2-(11-methoxy-6,7-dihydro-5H-indolo[2,1-a][2]benzazepin-13-yl)ethyl]butanamide
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 66 nM
|
|
|
|
CP0532362
|
N-[3-(3-methoxyphenyl)propyl]propanamide
Show/Hide
|
C13H19NO2
|
1
|
| 1 |
Ki = 85.4 nM
|
|
|
|
CP0907712
|
{2-[7-Methoxy-1-(2-propionylamino-ethyl)-naphthalen-2-yloxy]-ethyl}-trimethyl-ammonium iodide
Show/Hide
|
C21H31IN2O3
|
1
|
| 1 |
Ki = 93 nM
|
|
|
|
CP0437583
|
N-[2-[2-(2-iodoethoxy)-7-methoxynaphthalen-1-yl]ethyl]propanamide
Show/Hide
|
C18H22INO3
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0921994
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)cyclobutanecarboxamide
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
Ki = 112.2 nM
|
|
|
|
CP0442981
|
N-[[(2S)-1-benzyl-3,4-dihydro-2H-quinolin-2-yl]methyl]acetamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 122 nM
|
|
|
|
CP0485220
|
N-[3-(3-methoxyphenyl)-3-naphthalen-2-ylpropyl]acetamide
Show/Hide
|
C22H23NO2
|
1
|
| 1 |
Ki = 132 nM
|
|
|
|
CP0309824
|
1-ethyl-3-[(8-methoxybenzo[e][1]benzofuran-2-yl)methyl]thiourea
Show/Hide
|
C17H18N2O2S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0431523
|
N-[[1-(2-phenylethyl)-3,4-dihydro-2H-quinolin-2-yl]methyl]acetamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 171 nM
|
|
|
|
CP0867260
|
N-(2-(2-((1H-indol-1-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
Ki = 181.97 nM
|
|
|
|
CP0430666
|
N-[3-(2-ethoxy-5-methoxyphenyl)propyl]acetamide
Show/Hide
|
C14H21NO3
|
1
|
| 1 |
Ki = 183 nM
|
|
|
|
CP0404130
|
N-[(1-benzyl-6-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
Ki = 186 nM
|
|
|
|
CP0105647
|
1-ethyl-3-[2-(8-methoxybenzo[e][1]benzofuran-2-yl)ethyl]urea
Show/Hide
|
C18H20N2O3
|
1
|
| 1 |
Ki = 210 nM
|
|
|
|
CP0514689
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]propanamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 210 nM
|
|
|
|
CP0442980
|
N-[(1-benzyl-7-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamide
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
Ki = 214 nM
|
|
|
|
CP0375021
|
(E)-N-[3-(3-methoxyphenyl)-3-phenyl-2-propenyl]acetamide
Show/Hide
|
C18H19NO2
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0479258
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0524750
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]prop-2-enamide
Show/Hide
|
C19H15F2NOS2
|
1
|
| 1 |
Ki = 236 nM
|
|
|
|
CP0432631
|
N-[[1-(2-phenylethyl)-3,4-dihydro-2H-quinolin-3-yl]methyl]acetamide
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
Ki = 246 nM
|
|
|
|
CP0947476
|
N-(2-(2-((3,4-dihydroisoquinolin-2(1H)-yl)methyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
Ki = 251.19 nM
|
|
|
|
CP0447593
|
N-[3-(4-hydroxy-3-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO3
|
1
|
| 1 |
Ki = 257 nM
|
|
|
|
CP0914470
|
N-[2-(2-{[(4-Chlorophenyl)(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C21H24ClN3O2
|
1
|
| 1 |
Ki = 257.04 nM
|
|
|
|
CP0921467
|
N-[2-(2-Methyl-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)ethyl]butanamide
Show/Hide
|
C18H25N3O
|
1
|
| 1 |
Ki = 257.04 nM
|
|
|
|
CP0486794
|
5-[(E)-2-(7-methoxynaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C15H12N2O3
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0488698
|
N-[3-(5-methoxy-2-phenylmethoxyphenyl)propyl]propanamide
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 263 nM
|
|
|
|
CP0849416
|
N-(2-(2-(isoindolin-2-ylmethyl)-5-methoxy-1H-indol-3-yl)ethyl)acetamide
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
Ki = 281.84 nM
|
|
|
|
CP0452657
|
N-[(1-benzyl-3,4-dihydro-2H-quinolin-2-yl)methyl]cyclopropanecarboxamide
Show/Hide
|
C21H24N2O
|
1
|
| 1 |
Ki = 291 nM
|
|
|
|
CP0381637
|
N-[2-(7-methoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14,16,18-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C23H25N3O2
|
2
|
| 1 |
Ki = 316.23 nM
|
|
|
| 2 |
Ki = 319.3 nM
|
|
|
|
CP0513018
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]butanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 320 nM
|
|
|
|
CP0464196
|
N-[2-(1-benzyl-3,4-dihydro-2H-quinolin-2-yl)ethyl]propanamide
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
Ki = 326 nM
|
|
|
|
CP0447591
|
N-[3-(2-hydroxy-5-methoxyphenyl)propyl]acetamide
Show/Hide
|
C12H17NO3
|
1
|
| 1 |
Ki = 379 nM
|
|
|
|
CP0470465
|
N-[3-(5-methoxy-2-propoxyphenyl)propyl]acetamide
Show/Hide
|
C15H23NO3
|
1
|
| 1 |
Ki = 400 nM
|
|
|
|
CP0473011
|
N-(1,2,3,4-tetrahydroquinolin-3-ylmethyl)acetamide
Show/Hide
|
C12H16N2O
|
1
|
| 1 |
Ki = 430 nM
|
|
|
|
CP0452109
|
N-[3-[5-methoxy-2-[(3-methoxyphenyl)methoxy]phenyl]propyl]acetamide
Show/Hide
|
C20H25NO4
|
1
|
| 1 |
Ki = 441 nM
|
|
|
|
CP0404131
|
1-ethyl-3-[(5-methoxy-1,2,3,4-tetrahydroquinolin-2-yl)methyl]urea
Show/Hide
|
C14H21N3O2
|
1
|
| 1 |
Ki = 480 nM
|
|
|
|
CP0514682
|
N-[2-[6-methoxy-2-(3-methoxyphenyl)quinazolin-4-yl]ethyl]acetamide
Show/Hide
|
C20H21N3O3
|
1
|
| 1 |
Ki = 500 nM
|
|
|
|
CP0547557
|
N-[2-(6-methoxyquinazolin-4-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C15H17N3O2
|
1
|
| 1 |
Ki = 549 nM
|
|
|
|
CP0258343
|
3-(cyclobutylmethyl)-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C18H21N3O3
|
1
|
| 1 |
Ki = 550 nM
|
|
|
|
CP0511802
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-methyl-1,3,4-oxadiazol-2-amine
Show/Hide
|
C14H16N4O2
|
1
|
| 1 |
Ki = 550 nM
|
|
|
|
CP0413686
|
N-[(1-benzyl-3,4-dihydro-2H-quinolin-2-yl)methyl]cyclobutanecarboxamide
Show/Hide
|
C22H26N2O
|
1
|
| 1 |
Ki = 633 nM
|
|
|
|
CP0422156
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-(3-phenylpropyl)-1,3,4-oxadiazol-2-one
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
Ki = 690 nM
|
|
|
|
CP0399886
|
N-[2-[(1R,3R)-7-methoxy-3-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]ethyl]cyclobutanecarboxamide
Show/Hide
|
C24H29NO2
|
1
|
| 1 |
Ki = 797 nM
|
|
|
|
CP0504561
|
N-[3-(5-methoxy-2-phenylmethoxyphenyl)propyl]acetamide
Show/Hide
|
C19H23NO3
|
1
|
| 1 |
Ki = 879 nM
|
|
|
|
CP0432630
|
N-(1-benzyl-3,4-dihydro-2H-quinolin-3-yl)propanamide
Show/Hide
|
C19H22N2O
|
1
|
| 1 |
Ki = 892 nM
|
|
|
|
CP0514684
|
N-[2-(6-methoxy-2-phenylquinazolin-4-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki = 896 nM
|
|
|
|
CP0452008
|
N-[2-[5-fluoro-2-(4-fluorophenyl)sulfanyl-1-benzothiophen-3-yl]ethyl]cyclobutanecarboxamide
Show/Hide
|
C21H19F2NOS2
|
1
|
| 1 |
Ki = 915 nM
|
|
|
|
CP0474655
|
N-[2-(3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4,6,8,10,14,16,18-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C22H23N3O
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0844959
|
N-[2-(2-{[Ethyl(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C17H25N3O2
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0558328
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]butanamide
Show/Hide
|
C15H19N3O2
|
1
|
| 1 |
Ki = 1140 nM
|
|
|
|
CP0430665
|
N-[3-(5-methoxy-2-phenylmethoxyphenyl)propyl]butanamide
Show/Hide
|
C21H27NO3
|
1
|
| 1 |
Ki = 1172 nM
|
|
|
|
CP0400307
|
N-[3-(2,5-dimethoxyphenyl)propyl]acetamide
Show/Hide
|
C13H19NO3
|
1
|
| 1 |
Ki = 1280 nM
|
|
|
|
CP0920290
|
N-[2-(2-{[(Benzyl(methyl)amino]methyl}-5-methoxy-1H-indol-3-yl)ethyl]acetamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
Ki = 1288.25 nM
|
|
|
|
CP0111066
|
N-[[1-[(4-chlorophenyl)methyl]-4-methoxyindol-2-yl]methyl]propanamide
Show/Hide
|
C20H21ClN2O2
|
1
|
| 1 |
Ki = 1290 nM
|
|
|
|
CP0452111
|
N-[3-[3-methoxy-4-[(3-methoxyphenyl)methoxy]phenyl]propyl]acetamide
Show/Hide
|
C20H25NO4
|
1
|
| 1 |
Ki = 1460 nM
|
|
|
|
CP0514683
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]propanamide
Show/Hide
|
C14H17N3O2
|
1
|
| 1 |
Ki = 1470 nM
|
|
|
|
CP0094726
|
N-[2-(7,17-dimethoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14(19),15,17-heptaen-10-yl)ethyl]acetamide
Show/Hide
|
C24H27N3O3
|
2
|
| 1 |
Ki = 1800 nM
|
|
|
| 2 |
Ki = 1819.7 nM
|
|
|
|
CP0430669
|
N-[3-[5-methoxy-2-(pyridin-2-ylmethoxy)phenyl]propyl]acetamide
Show/Hide
|
C18H22N2O3
|
1
|
| 1 |
Ki = 1840 nM
|
|
|
|
CP0470444
|
N-[3-(3-methoxy-4-phenylmethoxyphenyl)propyl]propanamide
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 2010 nM
|
|
|
|
CP0552037
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]acetamide
Show/Hide
|
C13H15N3O2
|
1
|
| 1 |
Ki = 2110 nM
|
|
|
|
CP0400306
|
N-[3-[5-methoxy-2-[(4-methoxyphenyl)methoxy]phenyl]propyl]acetamide
Show/Hide
|
C20H25NO4
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0452009
|
4-chloro-N-(2-(5-fluoro-2-(4-fluorophenylthio)benzo[b]thiophen-3-yl)ethyl)butanamide
Show/Hide
|
C20H18ClF2NOS2
|
1
|
| 1 |
Ki = 2860 nM
|
|
|
|
CP0430667
|
N-[3-[5-methoxy-2-(2-phenylethoxy)phenyl]propyl]acetamide
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 2930 nM
|
|
|
|
CP0424907
|
N-[2-(7-methoxyphthalazin-1-yl)ethyl]cyclopropanecarboxamide
Show/Hide
|
C15H17N3O2
|
1
|
| 1 |
Ki = 3020 nM
|
|
|
|
CP0914471
|
N-[2-(9-Methoxy-2-methyl-2,3,4,5-tetrahydro-1H-[1,4]diazepino[1,2-a]indol-11-yl)ethyl]acetamide
Show/Hide
|
C18H25N3O2
|
1
|
| 1 |
Ki = 5623.41 nM
|
|
|
|
CP0036921
|
3-HYDROXYTYRAMINE HYDROCHLORIDE
Show/Hide
|
C8H11NO2
|
1
|
| 1 |
Ki = 7100 nM
|
|
|
|
CP0477491
|
N-[3-(3-methoxy-4-phenylmethoxyphenyl)propyl]acetamide
Show/Hide
|
C19H23NO3
|
1
|
| 1 |
Ki = 8980 nM
|
|
|
|
CP0404134
|
N-[[1-[2-(methylamino)-2-oxoethyl]-3,4-dihydro-2H-quinolin-2-yl]methyl]propanamide
Show/Hide
|
C16H23N3O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0442978
|
N-[(5-methoxyquinolin-2-yl)methyl]propanamide
Show/Hide
|
C14H16N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0317553
|
3-(cyclopentylmethyl)-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C19H23N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0362932
|
5-[(E)-2-(7-methoxy-3,4-dihydronaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C15H14N2O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0487632
|
3-hexyl-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C19H25N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0511803
|
3-heptyl-5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-one
Show/Hide
|
C20H27N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0549637
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-propyl-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H19N3O3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0487667
|
N-ethyl-4-(6-methoxyquinazolin-4-yl)piperazine-1-carboxamide
Show/Hide
|
C16H21N5O2
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0547558
|
N-[2-[(6-methoxyquinazolin-4-yl)amino]ethyl]acetamide
Show/Hide
|
C13H16N4O2
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0547559
|
cyclopropyl-[4-(6-methoxyquinazolin-4-yl)piperazin-1-yl]methanone
Show/Hide
|
C17H20N4O2
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
|
CP0509534
|
N-[2-[7-(2-propan-2-yloxyphenyl)-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl]ethyl]acetamide
Show/Hide
|
C24H27NO3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0376970
|
N-[2-(11-phenyl-5-oxa-1,10-diazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraen-12-yl)ethyl]acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0258344
|
5-[(E)-2-(5-methoxy-1H-indol-3-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C13H11N3O3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0478995
|
(E)-3-(5-methoxy-1H-indol-3-yl)-N-prop-2-ynylprop-2-enamide
Show/Hide
|
C15H14N2O2
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0487486
|
5-[(E)-2-(5-methoxy-1H-indol-3-yl)ethenyl]-3-prop-2-ynyl-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H13N3O3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0549638
|
(E)-3-(5-methoxy-1H-indol-3-yl)-N-prop-2-enylprop-2-enamide
Show/Hide
|
C15H16N2O2
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0869937
|
5-[1-(5-Methoxy-1H-indol-3-yl)propan-2-yl]-1,3,4-oxadiazol-2(3H)-one
Show/Hide
|
C14H15N3O3
|
1
|
| 1 |
Ki > 100 nM
|
|
|
|
CP0897694
|
6-Methoxy-1-methyl-4-(2-propionylamino-ethyl)-quinolinium iodide
Show/Hide
|
C16H21IN2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0919223
|
4-(2-Acetylamino-ethyl)-6-methoxy-1-methyl-quinolinium iodide
Show/Hide
|
C15H19IN2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0376623
|
5-[(5-methoxy-1H-indol-3-yl)methyl]-3H-1,3,4-oxadiazole-2-thione
Show/Hide
|
C12H11N3O2S
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0381569
|
5-[(5-methoxy-1H-indol-3-yl)methyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C12H11N3O3
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0381570
|
3-[(5-methoxy-1H-indol-3-yl)methyl]-4-methyl-1H-1,2,4-triazol-5-one
Show/Hide
|
C13H14N4O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0398233
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3H-1,3,4-oxadiazole-2-thione
Show/Hide
|
C13H13N3O2S
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0398249
|
4-ethyl-3-[(5-methoxy-1H-indol-3-yl)methyl]-1H-1,2,4-triazole-5-thione
Show/Hide
|
C14H16N4OS
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0401209
|
N-ethyl-5-[(5-methoxy-1H-indol-3-yl)methyl]-1,3,4-thiadiazol-2-amine
Show/Hide
|
C14H16N4OS
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0415040
|
2-[2-(5-methoxy-1H-indol-3-yl)ethyl]-5-methyl-1,3-oxazole
Show/Hide
|
C15H16N2O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0433770
|
3-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-methyl-1H-1,2,4-triazol-5-one
Show/Hide
|
C14H16N4O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0449128
|
4-ethyl-3-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1H-1,2,4-triazole-5-thione
Show/Hide
|
C15H18N4OS
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0482626
|
5-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-methyl-1,2,4-oxadiazole
Show/Hide
|
C14H15N3O2
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0428520
|
1-ethyl-3-[(5-methoxy-1,2,3,4-tetrahydroquinolin-2-yl)methyl]thiourea
Show/Hide
|
C14H21N3OS
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
|
CP0558022
|
5-[(E)-2-(6,7-dimethoxynaphthalen-1-yl)ethenyl]-3H-1,3,4-oxadiazol-2-one
Show/Hide
|
C16H14N2O4
|
1
|
| 1 |
Ki > 1000 nM
|
|
|
