Compound ID |
Compound Name |
Compound Formula |
CP0241330
|
(3S)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[4-(2H-tetrazol-5-yl)phenyl]pyrrolidin-3-amine;hydrochloride
Show/Hide
|
C23H25ClN6
|
1
|
1 |
EC50 = 17 nM
|
|
|
CP0556762
|
3-(1,3-benzothiazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H32N4O2S
|
1
|
1 |
EC50 = 20 nM
|
|
|
CP0562885
|
3-(4-chloro-1,3-benzothiazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H31ClN4O2S
|
1
|
1 |
EC50 = 20 nM
|
|
|
CP0527464
|
1-(3,3-diphenylpropyl)-3-[5-(methanesulfonamido)-1,3-benzothiazol-2-yl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N5O4S2
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0538035
|
1-(3,3-diphenylpropyl)-3-[6-(methanesulfonamido)-1,3-benzothiazol-2-yl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N5O4S2
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0540610
|
1-(3,3-diphenylpropyl)-3-(6-methyl-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O2S
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0562884
|
1-(3,3-diphenylpropyl)-3-(4-methoxy-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O3S
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0560881
|
1-(3,3-diphenylpropyl)-3-(6-methoxy-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O3S
|
1
|
1 |
EC50 = 40 nM
|
|
|
CP0068452
|
N-(2-hydroxyethyl)-4-[(3S)-3-[[(1R)-1-naphthalen-1-ylethyl]amino]pyrrolidin-1-yl]benzamide;dihydrochloride
Show/Hide
|
C25H31Cl2N3O2
|
1
|
1 |
EC50 = 50 nM
|
|
|
CP0438406
|
methyl 3-[[3,3-diphenylpropyl(3-piperazin-1-ylpropyl)carbamoyl]amino]benzoate
Show/Hide
|
C31H38N4O3
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0540359
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(1,3-oxazol-5-yl)phenyl]urea
Show/Hide
|
C31H34N4O3
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0540451
|
1-(3,3-diphenylpropyl)-3-[3-(2-methyltetrazol-5-yl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N7O2
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0456155
|
3-(6-chloro-1,3-benzothiazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H31ClN4O2S
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0510075
|
3-(1H-benzimidazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H33N5O2
|
1
|
1 |
EC50 = 60 nM
|
|
|
CP0344214
|
AMG-073
Show/Hide
|
C22H22F3N
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0372293
|
(R)-3-(2-chlorophenyl)-N-(1-(3-methoxyphenyl)ethyl)propan-1-amine
Show/Hide
|
C18H22ClNO
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0375144
|
1-(3,3-diphenylpropyl)-3-(6-methylsulfonyl-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O4S2
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0375146
|
3-(5-chloro-1,3-benzoxazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H31ClN4O3
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0411395
|
3-(4,6-dimethylpyridin-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H36N4O2
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0538036
|
1-(3,3-diphenylpropyl)-3-[6-(hydroxymethyl)-1,3-benzothiazol-2-yl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O3S
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0912861
|
TECALCET HYDROCHLORIDE
Show/Hide
|
C18H23Cl2NO
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0538037
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[6-(trifluoromethoxy)-1,3-benzothiazol-2-yl]urea
Show/Hide
|
C30H31F3N4O3S
|
1
|
1 |
EC50 = 90 nM
|
|
|
CP0249035
|
2-[4-[(3S)-3-[[(1R)-1-naphthalen-1-ylethyl]amino]pyrrolidin-1-yl]phenyl]acetic acid;dihydrochloride
Show/Hide
|
C24H28Cl2N2O2
|
1
|
1 |
EC50 = 93 nM
|
|
|
CP0438416
|
methyl 3-[[3,3-diphenylpropyl-[3-(4-methylpiperazin-1-yl)propyl]carbamoyl]amino]benzoate
Show/Hide
|
C32H40N4O3
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0553416
|
methyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C30H35N3O4
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0524021
|
2-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]-1,3-benzothiazole-6-carboxylic acid
Show/Hide
|
C30H32N4O4S
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0319457
|
(3S)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[4-(trifluoromethoxy)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2O
|
1
|
1 |
EC50 = 120 nM
|
|
|
CP0499207
|
1-(3,3-diphenylpropyl)-3-(3-methylsulfanylphenyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H35N3O2S
|
1
|
1 |
EC50 = 130 nM
|
|
|
CP0423408
|
1-(3,3-diphenylpropyl)-3-[3-(3-methyl-1,2-oxazol-5-yl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C32H36N4O3
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0435701
|
3-[3-(1,3-benzothiazol-2-yl)phenyl]-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C35H36N4O2S
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0438415
|
propan-2-yl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C32H39N3O4
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0444703
|
1-(3,3-diphenylpropyl)-3-[3-(furan-2-yl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C32H35N3O3
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0451201
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-(3-propanoylphenyl)urea
Show/Hide
|
C31H37N3O3
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0524682
|
2-hydroxyethyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C31H37N3O5
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0540447
|
methyl 3-[[3,3-diphenylpropyl(3-morpholin-4-ylpropyl)carbamoyl]amino]benzoate
Show/Hide
|
C31H37N3O4
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0536484
|
1-(3,3-diphenylpropyl)-3-(1-methylbenzimidazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N5O2
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0850747
|
CINACALCET HYDROCHLORIDE
Show/Hide
|
C22H23ClF3N
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0149670
|
(3R)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethoxy)phenyl]piperidin-3-amine;dihydrochloride
Show/Hide
|
C24H27Cl2F3N2O
|
1
|
1 |
EC50 = 190 nM
|
|
|
CP0442098
|
1-(3,3-diphenylpropyl)-3-[3-(1-methyltetrazol-5-yl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N7O2
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0442099
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-(3-pyridin-3-ylphenyl)urea
Show/Hide
|
C33H36N4O2
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0442101
|
benzyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C36H39N3O4
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0449539
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(trifluoromethoxy)phenyl]urea
Show/Hide
|
C29H32F3N3O3
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0499205
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-(3-phenylphenyl)urea
Show/Hide
|
C34H37N3O2
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0380832
|
N-[2-(dimethylamino)ethyl]-2-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]-1,3-benzothiazole-6-carboxamide
Show/Hide
|
C34H42N6O3S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0411393
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[4-(1,3-thiazol-2-yl)pyrimidin-2-yl]urea
Show/Hide
|
C29H32N6O2S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0489147
|
ethyl 2-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]-1,3-benzothiazole-6-carboxylate
Show/Hide
|
C32H36N4O4S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0527023
|
1-(3,3-diphenylpropyl)-3-(5-methyl-1,2-oxazol-3-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C26H32N4O3
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0538034
|
1-(3,3-diphenylpropyl)-3-(6-fluoro-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H31FN4O2S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0273212
|
(3R)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[4-(trifluoromethoxy)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2O
|
1
|
1 |
EC50 = 230 nM
|
|
|
CP0758372
|
4-((S)-3-((R)-1-(naphthalen-1-yl)ethylamino)pyrrolidin-1-yl)benzoic acid hydrochloride
Show/Hide
|
C23H25ClN2O2
|
1
|
1 |
EC50 = 290 nM
|
|
|
CP0382868
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(1,3-thiazol-2-yl)phenyl]urea
Show/Hide
|
C31H34N4O2S
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0382869
|
3-[3-(dimethylamino)phenyl]-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H38N4O2
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0423409
|
1-(3,3-diphenylpropyl)-3-(3-methoxyphenyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H35N3O3
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0442100
|
tert-butyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C33H41N3O4
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0524022
|
3-(1-benzylbenzimidazol-2-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C36H39N5O2
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0560915
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-(1,3-thiazol-2-yl)urea
Show/Hide
|
C25H30N4O2S
|
1
|
1 |
EC50 = 300 nM
|
|
|
CP0396501
|
(3R)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2O
|
1
|
1 |
EC50 = 320 nM
|
|
|
CP0499206
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(trifluoromethylsulfanyl)phenyl]urea
Show/Hide
|
C29H32F3N3O2S
|
1
|
1 |
EC50 = 350 nM
|
|
|
CP0149664
|
(3R)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]piperidin-3-amine;dihydrochloride
Show/Hide
|
C24H27Cl2F3N2
|
1
|
1 |
EC50 = 380 nM
|
|
|
CP0423049
|
1-(3,3-diphenylpropyl)-3-[3-(methoxymethyl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H37N3O3
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0435706
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(trifluoromethylsulfonyl)phenyl]urea
Show/Hide
|
C29H32F3N3O4S
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0499208
|
methyl 4-[3-[3,3-diphenylpropyl-[(3-methoxycarbonylphenyl)carbamoyl]amino]propyl]piperazine-1-carboxylate
Show/Hide
|
C33H40N4O5
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0524681
|
4,4,5,5,5-pentafluoropentyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C34H38F5N3O4
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0526530
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C29H32F3N3O2
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0411394
|
1-(3,3-diphenylpropyl)-3-(4-methoxy-6-methylpyrimidin-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C28H35N5O3
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0468889
|
methyl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]thiophene-2-carboxylate
Show/Hide
|
C28H33N3O4S
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0241329
|
(3R)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2
|
1
|
1 |
EC50 = 430 nM
|
|
|
CP0439132
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-pyrazin-2-ylurea
Show/Hide
|
C26H31N5O2
|
1
|
1 |
EC50 = 450 nM
|
|
|
CP0149668
|
(3S)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethyl)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2
|
1
|
1 |
EC50 = 450 nM
|
|
|
CP0524680
|
3-(3-acetylphenyl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H35N3O3
|
1
|
1 |
EC50 = 550 nM
|
|
|
CP0435703
|
3-[3-(1H-benzimidazol-2-ylamino)phenyl]-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C35H38N6O2
|
1
|
1 |
EC50 = 600 nM
|
|
|
CP0560882
|
1-(3,3-diphenylpropyl)-3-(4-methyl-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C30H34N4O2S
|
1
|
1 |
EC50 = 600 nM
|
|
|
CP0217341
|
(3S)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethoxy)phenyl]piperidin-3-amine;dihydrochloride
Show/Hide
|
C24H27Cl2F3N2O
|
1
|
1 |
EC50 = 600 nM
|
|
|
CP0322097
|
(3S)-N-[(1R)-1-naphthalen-1-ylethyl]-1-[3-(trifluoromethoxy)phenyl]pyrrolidin-3-amine;dihydrochloride
Show/Hide
|
C23H25Cl2F3N2O
|
1
|
1 |
EC50 = 600 nM
|
|
|
CP0435705
|
3-(3-cyanophenyl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H32N4O2
|
1
|
1 |
EC50 = 800 nM
|
|
|
CP0540445
|
1-(3,3-diphenylpropyl)-3-[3-(hydroxymethyl)phenyl]-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H35N3O3
|
1
|
1 |
EC50 = 800 nM
|
|
|
CP0553405
|
1-(3,3-diphenylpropyl)-3-(3-methylsulfinylphenyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H35N3O3S
|
1
|
1 |
EC50 = 800 nM
|
|
|
CP0553417
|
methyl 3-[[3,3-diphenylpropyl-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]carbamoyl]amino]benzoate
Show/Hide
|
C30H34N2O5
|
1
|
1 |
EC50 = 800 nM
|
|
|
CP0195373
|
3,3-diphenyl-N-(1-phenylethyl)-1-propanamine;hydrochloride
Show/Hide
|
C23H25N
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0472577
|
3,3-dimethylbutan-2-yl 3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoate
Show/Hide
|
C35H45N3O4
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0517840
|
1-(3,3-diphenylpropyl)-3-(3-methylsulfonylphenyl)-1-(2-morpholin-4-ylethyl)urea
Show/Hide
|
C29H35N3O4S
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0526529
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-[3-(2H-tetrazol-5-ylamino)phenyl]urea
Show/Hide
|
C29H34N8O2
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0439133
|
1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)-3-pyridin-3-ylurea
Show/Hide
|
C27H32N4O2
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1
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1 |
EC50 = 1000 nM
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CP0527463
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1-(3,3-diphenylpropyl)-3-(6-ethoxy-1,3-benzothiazol-2-yl)-1-(2-morpholin-4-ylethyl)urea
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C31H36N4O3S
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1
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1 |
EC50 = 1000 nM
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CP0319455
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4-[(3S)-3-[[(1R)-1-naphthalen-1-ylethyl]amino]piperidin-1-yl]benzoic acid;dihydrochloride
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C24H28Cl2N2O2
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1
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1 |
EC50 = 1100 nM
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CP0540452
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methyl 3-[[3,3-diphenylpropyl(2-methylpropyl)carbamoyl]amino]benzoate
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C28H32N2O3
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1
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1 |
EC50 = 1500 nM
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CP0536486
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3-(3,4-dimethyl-1,2-oxazol-5-yl)-1-(3,3-diphenylpropyl)-1-(2-morpholin-4-ylethyl)urea
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C27H34N4O3
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1
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1 |
EC50 = 1700 nM
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CP0423410
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methyl 2-chloro-5-(3,3-diphenylpropylcarbamoylamino)benzoate
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C24H23ClN2O3
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1
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1 |
EC50 = 2000 nM
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CP0487710
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methyl 3-[[benzyl(3,3-diphenylpropyl)carbamoyl]amino]benzoate
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C31H30N2O3
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1
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1 |
EC50 = 2000 nM
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CP0500044
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methyl 3-(3,3-diphenylpropylcarbamoylamino)benzoate
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C24H24N2O3
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1
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1 |
EC50 = 2000 nM
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CP0540446
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3-[[3,3-diphenylpropyl(2-morpholin-4-ylethyl)carbamoyl]amino]benzoic acid
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C29H33N3O4
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1
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1 |
EC50 = 2000 nM
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CP0423051
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ethyl 4-(3,3-diphenylpropylcarbamoylamino)benzoate
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C25H26N2O3
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1
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1 |
EC50 = 3000 nM
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CP0521689
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1-[4-chloro-3-(trifluoromethyl)phenyl]-3-(3,3-diphenylpropyl)urea
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C23H20ClF3N2O
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1
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1 |
EC50 = 3000 nM
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CP0442103
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1-(3-chlorophenyl)-3-(3,3-diphenylpropyl)urea
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C22H21ClN2O
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1
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1 |
EC50 = 4000 nM
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CP0499211
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1-[(2-chlorophenyl)methyl]-3-(3,3-diphenylpropyl)urea
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C23H23ClN2O
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1
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1 |
EC50 = 4000 nM
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CP0516992
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1-(4-chlorophenyl)-3-(3,3-diphenylpropyl)urea
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C22H21ClN2O
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1
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1 |
EC50 = 4000 nM
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CP0526531
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1-(3,3-diphenylpropyl)-3-p-tolylurea
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C23H24N2O
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1
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1 |
EC50 = 4000 nM
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CP0554445
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1-(3,3-diphenylpropyl)-3-(4-phenylphenyl)urea
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C28H26N2O
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1
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1 |
EC50 = 4000 nM
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CP0423412
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1-(2-chlorophenyl)-3-(3,3-diphenylpropyl)urea
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C22H21ClN2O
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1
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1 |
EC50 = 6000 nM
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CP0444704
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1-(3,3-diphenylpropyl)-3-[(1R)-1-phenylethyl]urea
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C24H26N2O
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1
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1 |
EC50 = 6000 nM
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CP0499232
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1-(3,3-diphenylpropyl)-3-(3-methoxyphenyl)urea
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C23H24N2O2
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1
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1 |
EC50 = 8000 nM
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CP0111371
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4-[(3R)-3-[[(1R)-1-naphthalen-1-ylethyl]amino]pyrrolidin-1-yl]benzoic acid;dihydrochloride
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C23H26Cl2N2O2
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1
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1 |
EC50 = 8800 nM
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CP0442102
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methyl 3-[[2-cyclohexylethyl(3,3-diphenylpropyl)carbamoyl]amino]benzoate
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C32H38N2O3
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1
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1 |
EC50 = 10000 nM
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CP0499230
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methyl 3-[3,3-diphenylpropylcarbamoyl(2-morpholin-4-ylethyl)amino]benzoate
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C30H35N3O4
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1
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1 |
EC50 = 10000 nM
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CP0423087
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1-(3,3-diphenylpropyl)-3-(4-methoxyphenyl)urea
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C23H24N2O2
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1
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1 |
EC50 = 15000 nM
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CP0423411
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1-(3,3-diphenylpropyl)-3-(3-phenylphenyl)urea
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C28H26N2O
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1
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1 |
EC50 = 15000 nM
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CP0554444
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1-(3,3-diphenylpropyl)-3-[(4-methoxyphenyl)methyl]urea
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C24H26N2O2
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1
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1 |
EC50 = 15000 nM
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CP0500043
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3-(3,3-diphenylpropylcarbamoylamino)benzoic acid
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C23H22N2O3
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1
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1 |
EC50 = 20000 nM
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CP0913530
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(5R)-N-[1-Ethyl-1-(4-ethylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide p-toluenesulfonate
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C36H46N4O4S
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1
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1 |
IC50 = 0.94 nM
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CP0906026
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(5R)-N-[1-Ethyl-1-(4-isopropylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
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C30H41ClN4O
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1
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1 |
IC50 = 1.7 nM
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CP0918956
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(5R)-N-[1-(3-Chloro-4-methoxyphenyl)-1-ethylpropyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
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C28H36Cl2N4O2
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1
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1 |
IC50 = 1.7 nM
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CP0863386
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(5R)-N-[1-Ethyl-1-(4-methoxyphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
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C28H37ClN4O2
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1
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1 |
IC50 = 2 nM
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CP0918958
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(5R)-N-{1-[4-(Benzyloxy)phenyl]-1-ethylpropyl}-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
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C34H41ClN4O2
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1
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1 |
IC50 = 2.2 nM
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CP0903131
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(5R)-(-)-N-[1-Ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide Hydrochloride
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C27H35ClN4O
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1
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1 |
IC50 = 2.3 nM
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CP0870813
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(5R)-N-(1-Ethyl-1-phenylpropyl)-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo-[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C27H35ClN4O
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1
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1 |
IC50 = 2.3 nM
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CP0921786
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(5R)-N-[1-Ethyl-1-(4-methylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C28H37ClN4O
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1
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1 |
IC50 = 2.4 nM
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CP0935207
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(5R)-N-[1-(4-Ethoxyphenyl)-1-ethylpropyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
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C29H39ClN4O2
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1
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1 |
IC50 = 3 nM
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CP0522570
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7,7-dimethyl-5-phenyl-N-(3-phenylpentan-3-yl)-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
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C26H32N4O
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1
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1 |
IC50 = 3.4 nM
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CP0425591
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7,7-Dimethyl-N-{1-methyl-1-[4-(trifluoromethyl)phenyl]ethyl}-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C25H27F3N4O
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1
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1 |
IC50 = 3.5 nM
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CP0863388
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rac-N-[1-Ethyl-1-(4-methylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C28H37ClN4O
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1
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1 |
IC50 = 4.1 nM
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CP0913531
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(5R)-N-[1-Ethyl-1-(4-ethylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C29H39ClN4O
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1
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1 |
IC50 = 4.2 nM
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CP0502630
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7,7-Dimethyl-5-phenyl-N-{1-propyl-1-[4-(trifluoromethyl)phenyl]-butyl}-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C29H35F3N4O
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1
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1 |
IC50 = 4.4 nM
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CP0878392
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(5R)-N-[1-Ethyl-1-(3-fluoro-4-methoxyphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C28H36ClFN4O2
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1
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1 |
IC50 = 4.6 nM
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CP0906027
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rac-N-[1-Ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-2-(methylthio)-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
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C28H37ClN4OS
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1
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1 |
IC50 = 4.7 nM
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CP0447101
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(5R)-N-[1-(4-Acetylphenyl)-1-ethylpropyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide
Show/Hide
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C29H36N4O2
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1
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1 |
IC50 = 4.8 nM
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CP0918198
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rac-N-[1-Ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide Hydrochloride
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C27H35ClN4O
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1
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1 |
IC50 = 4.9 nM
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CP0509359
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ethyl 4-[3-[(7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]pentan-3-yl]benzoate
Show/Hide
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C29H36N4O3
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1
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1 |
IC50 = 5.2 nM
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CP0500556
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7,7-dimethyl-N-[3-(4-methylphenyl)pentan-3-yl]-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C27H34N4O
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1
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1 |
IC50 = 5.5 nM
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CP0871617
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rac-N-[1-Ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-2-propyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C30H41ClN4O
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1
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1 |
IC50 = 6 nM
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CP0935208
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(5R)-N-[1-(4-Chloro-3-methoxyphenyl)-1-ethylpropyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C28H36Cl2N4O2
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1
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1 |
IC50 = 6.1 nM
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CP0500557
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N-[3-(4-methoxyphenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C27H34N4O2
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1
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1 |
IC50 = 6.6 nM
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CP0942096
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rac-2-Ethyl-N-[1-ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C29H39ClN4O
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1
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1 |
IC50 = 6.7 nM
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CP0425593
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N-[3-(4-fluorophenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C26H31FN4O
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1
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1 |
IC50 = 7.3 nM
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CP0502472
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N-[3-(4-chlorophenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C26H31ClN4O
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1
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1 |
IC50 = 7.4 nM
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CP0513056
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7,7-dimethyl-5-phenyl-N-[3-[4-(trifluoromethyl)phenyl]pentan-3-yl]-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C27H31F3N4O
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1
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1 |
IC50 = 7.6 nM
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CP0525453
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7,7-dimethyl-5-phenyl-N-[3-(4-phenylmethoxyphenyl)pentan-3-yl]-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C33H38N4O2
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1
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1 |
IC50 = 8.5 nM
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CP0487298
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(5S)-N-(1-adamantyl)-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C25H32N4O
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1
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1 |
IC50 = 10 nM
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CP0930851
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rac-2-Butyl-N-[1-ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C31H43ClN4O
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1
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1 |
IC50 = 11 nM
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CP0936043
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(5R)-N-[1-(3,4-Dimethoxyphenyl)-1-ethylpropyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C29H39ClN4O3
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1
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1 |
IC50 = 11 nM
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CP0949748
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(5R)-N-[1-Ethyl-1-(4-fluoro-3-methoxyphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C28H36ClFN4O2
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1
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1 |
IC50 = 11 nM
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CP0472184
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[4-[3-[(7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]pentan-3-yl]phenyl] propanoate
Show/Hide
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C29H36N4O3
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1
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1 |
IC50 = 12 nM
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CP0502473
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N-[3-(2-fluorophenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C26H31FN4O
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1
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1 |
IC50 = 12 nM
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CP0503292
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(5R)-N-{1-Ethyl-1-[4-(1-hydroxyethyl)phenyl]propyl}-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide
Show/Hide
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C29H38N4O2
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1
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1 |
IC50 = 13 nM
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CP0523680
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4-(1-{[(7,7-Dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-yl)carbonyl]amino}-1-ethylpropyl)benzyl Acetate
Show/Hide
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C29H36N4O3
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1
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1 |
IC50 = 14 nM
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CP0500555
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N-[3-(3-chlorophenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C26H31ClN4O
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1
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1 |
IC50 = 17 nM
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CP0438171
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7,7-dimethyl-5-phenyl-N-[5-[4-(trifluoromethyl)phenyl]nonan-5-yl]-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C31H39F3N4O
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1
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1 |
IC50 = 23 nM
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CP0512374
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N-[3-(3-fluorophenyl)pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C26H31FN4O
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1
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1 |
IC50 = 25 nM
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CP0425592
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N-[2,4-dimethyl-3-[4-(trifluoromethyl)phenyl]pentan-3-yl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C29H35F3N4O
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1
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1 |
IC50 = 30 nM
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CP0512375
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4-(1-{[(7,7-Dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-yl)carbonyl]-amino}-1-ethylpropyl)phenyl Acetate
Show/Hide
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C28H34N4O3
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1
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1 |
IC50 = 31 nM
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CP0918950
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(5S)-(+)-N-[1-Ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide Hydrochloride
Show/Hide
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C27H35ClN4O
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1
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1 |
IC50 = 31 nM
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CP0863431
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(5S)-N-[1-Ethyl-1-(4-methylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C28H37ClN4O
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1
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1 |
IC50 = 31 nM
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CP0425589
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(5S,7R)-N-(1-adamantyl)-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C24H27F3N4O
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1
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1 |
IC50 = 40 nM
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CP0942097
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rac-2-Benzyl-N-[1-ethyl-1-(4-methylphenyl)propyl]-7,7-dimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidine-3-carboxamide hydrochloride
Show/Hide
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C34H41ClN4O
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1
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1 |
IC50 = 45 nM
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CP0504661
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(5S,7S)-N-(1-adamantyl)-7-methyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C24H30N4O
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1
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1 |
IC50 = 76 nM
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CP0509934
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7,7-dimethyl-N-[3-(4-methylphenyl)pentan-3-yl]-2,5-diphenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C33H38N4O
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1
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1 |
IC50 = 81 nM
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CP0425802
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1-Adamantyl-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo-[1,5-a]-pyrimidine-3-carboxylate
Show/Hide
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C24H26F3N3O2
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1
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1 |
IC50 = 97 nM
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CP0533446
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(5S,7R)-N-(1-adamantyl)-5-(2-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C24H26ClF3N4O
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1
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1 |
IC50 = 110 nM
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CP0487299
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N-[dicyclohexyl-[4-(trifluoromethyl)phenyl]methyl]-7,7-dimethyl-5-phenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
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C35H43F3N4O
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1
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1 |
IC50 = 150 nM
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CP0406895
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(5S,7R)-N-(1-adamantyl)-5-(3-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C24H26ClF3N4O
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1
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1 |
IC50 = 320 nM
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CP0525450
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4-[1-Ethyl-1-({[(5R)-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]-pyrimidin-3-yl]carbonyl}amino)-propyl]benzoic acid
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C28H34N4O3
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1
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1 |
IC50 = 320 nM
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CP0472183
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(5S,7R)-N-benzhydryl-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C27H23F3N4O
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1
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1 |
IC50 = 380 nM
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CP0387085
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(5S,7R)-N-(1-adamantyl)-5-(furan-2-yl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C22H25F3N4O2
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1
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1 |
IC50 = 400 nM
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CP0919640
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N-(1-Adamantyl)-7,7-dimethyl-5-phenyl-4,7-dihydropyrazolo[1,5-a]pyrimid-ine-3-carboxamide
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C25H30N4O
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1
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1 |
IC50 = 580 nM
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CP0533447
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(5S,7R)-N-(1-adamantyl)-5,7-diphenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C29H32N4O
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1
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1 |
IC50 = 700 nM
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CP0425590
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(5S,7R)-5-phenyl-7-(trifluoromethyl)-N-(4-(trifluoromethyl)benzyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C22H18F6N4O
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1
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1 |
IC50 = 2900 nM
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CP0425806
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(5S)-N-(1-adamantyl)-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C23H28N4O
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1
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1 |
IC50 = 5300 nM
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CP0398073
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(5S,7R)-N-(1-adamantyl)-5-(4-chlorophenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C24H26ClF3N4O
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1
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1 |
IC50 > 10000 nM
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CP0398074
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(5S,7R)-N-(1-adamantyl)-5-(4-ethylphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C26H31F3N4O
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1
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1 |
IC50 > 10000 nM
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CP0406896
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(5R,7R)-N-(1-adamantyl)-5-methyl-7-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C24H30N4O
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1
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1 |
IC50 > 10000 nM
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CP0425803
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(5S,7R)-N-(1-adamantyl)-4-methyl-5-phenyl-7-(trifluoromethyl)-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
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C25H29F3N4O
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1
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1 |
IC50 > 10000 nM
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CP0425804
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N-[[(5S,7R)-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]methyl]adamantan-1-amine
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C24H29F3N4
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1
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1 |
IC50 > 10000 nM
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CP0425805
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(5S,7R)-N-(1-adamantyl)-5-tert-butyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C22H31F3N4O
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1
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1 |
IC50 > 10000 nM
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CP0425807
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N-(1-adamantyl)-5-phenyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
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C24H23F3N4O
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1
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1 |
IC50 > 10000 nM
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CP0505444
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(7R)-N-(1-adamantyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C18H23F3N4O
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1
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1 |
IC50 > 10000 nM
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CP0508055
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(5S,7R)-N-(1-adamantyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C25H29F3N4O2
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1
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1 |
IC50 > 10000 nM
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CP0524105
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(5S,7R)-N-(1-adamantyl)-5-pyridin-3-yl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
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C23H26F3N5O
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1
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1 |
IC50 > 10000 nM
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CP0533445
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N-[(5S,7R)-5-phenyl-7-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]adamantane-1-carboxamide
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C24H27F3N4O
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1
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1 |
IC50 > 10000 nM
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