Brief Information of the Compound and Protein
Compound Name
rac-N-[1-Ethyl-1-(4-methylphenyl)propyl]-2,7,7-trimethyl-5-phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide hydrochloride
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PubChem ID
CID: 136030615
Canonical SMILES
CCC(CC)(NC(=O)c1c(C)nn2c1NC(c1ccccc1)CC2(C)C)c1ccc(C)cc1.Cl
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Compound Formula C28H37ClN4O
Compound Structure
Protein Name
Extracellular calcium-sensing receptor
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Ion receptor (family C GPCR)
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Calcium sensing receptor
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Calcium sensing receptor
Uniprot ID
P41180
Gene Name
CASR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 4.1 nM
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