Brief Information of the Compound and Protein
Compound Name
7,7-dimethyl-N-[3-(4-methylphenyl)pentan-3-yl]-2,5-diphenyl-5,6-dihydro-4H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
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PubChem ID
CID: 136188844
Canonical SMILES
CCC(CC)(NC(=O)c1c2NC(CC(C)(C)n2nc1-c1ccccc1)c1ccccc1)c1ccc(C)cc1
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Compound Formula C33H38N4O
Compound Structure
Protein Name
Extracellular calcium-sensing receptor
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Ion receptor (family C GPCR)
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Calcium sensing receptor
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Calcium sensing receptor
Uniprot ID
P41180
Gene Name
CASR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 81 nM
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