| Compound ID |
Compound Name |
Compound Formula |
|
CP0478164
|
4-{5-chloro-1'-[(2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
Show/Hide
|
C22H18ClFN2O5
|
2
|
| 1 |
EC50 = 2200 nM
|
|
|
| 2 |
Ki = 1759 nM
|
|
|
|
CP0505209
|
4-{5-chloro-1'-[(4-chlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
Show/Hide
|
C22H18Cl2N2O5
|
2
|
| 1 |
EC50 = 5600 nM
|
|
|
| 2 |
Ki = 758 nM
|
|
|
|
CP0385506
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]pentanamide
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|
C21H22FN5O3
|
2
|
| 1 |
IC50 = 2.8 nM
|
|
|
| 2 |
Ki = 2 nM
|
|
|
|
CP0389705
|
2-[1-[4-(1H-indole-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
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|
C27H19N3O4
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
IC50 = 3.5 nM
|
|
|
|
CP0524697
|
2-[1-[4-[(3-chlorobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C25H17ClN2O4
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0387883
|
2-[1-[4-[(4-chlorobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C25H17ClN2O4
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0113938
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]-2-phenylacetamide
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|
C23H20FN5O3S
|
2
|
| 1 |
IC50 = 3.7 nM
|
|
|
| 2 |
Ki = 0.9 nM
|
|
|
|
CP0551799
|
2-[1-[4-[2-(3,4-dichlorophenyl)ethylcarbamoyl]benzoyl]isoquinolin-4-yl]acetic acid
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|
C27H20Cl2N2O4
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0420654
|
2-[1-[4-(1-benzofuran-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
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|
C27H18N2O5
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0386064
|
2-[1-[4-(naphthalene-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
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|
C29H20N2O4
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0476029
|
2-[1-[4-[[(E)-3-(3,4-dichlorophenyl)prop-2-enoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C27H18Cl2N2O4
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0519814
|
2-[1-[4-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C26H17F3N2O4
|
1
|
| 1 |
IC50 = 4.9 nM
|
|
|
|
CP0420653
|
2-[1-[4-[(4-methylbenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C26H20N2O4
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
|
CP0387881
|
2-[1-[4-[(3,4-dichlorophenyl)methylamino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H18Cl2N2O3
|
1
|
| 1 |
IC50 = 6.1 nM
|
|
|
|
CP0386062
|
2-[1-[4-[[4-(dimethylamino)benzoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C27H23N3O4
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0387882
|
2-[1-[4-[(3,4-dichlorophenyl)methoxycarbonylamino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C26H18Cl2N2O5
|
1
|
| 1 |
IC50 = 6.7 nM
|
|
|
|
CP0154904
|
2-[4-chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
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|
C20H19ClO5S
|
3
|
| 1 |
IC50 = 7 nM
|
|
|
| 2 |
IC50 = 32 nM
|
|
|
| 3 |
Ki = 2 nM
|
|
|
|
CP0549646
|
2-[1-[4-[(4-methoxybenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C26H20N2O5
|
1
|
| 1 |
IC50 = 7.3 nM
|
|
|
|
CP0380031
|
2-[1-[4-[2-(4-chlorophenyl)ethylcarbamoyl]benzoyl]isoquinolin-4-yl]acetic acid
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|
C27H21ClN2O4
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
|
CP0420652
|
2-[1-[4-[(4-cyanobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C26H17N3O4
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
|
CP0387884
|
2-[1-(4-benzamidobenzoyl)isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H18N2O4
|
1
|
| 1 |
IC50 = 7.9 nM
|
|
|
|
CP0395103
|
2-[4-chloro-2-[2-(2-fluoro-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H16ClFO5S
|
3
|
| 1 |
IC50 = 8 nM
|
|
|
| 2 |
IC50 = 28 nM
|
|
|
| 3 |
Ki = 3.4 nM
|
|
|
|
CP0551800
|
2-[1-[4-[(4-chlorophenyl)carbamoyl]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H17ClN2O4
|
1
|
| 1 |
IC50 = 8.2 nM
|
|
|
|
CP0424092
|
(S)-2-(4-chloro-2-((4-(2-(4-fluorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H24ClFN2O4
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0498085
|
2-[4-chloro-2-[[(3S)-4-[2-(4-chlorophenyl)acetyl]-3-methylpiperazin-1-yl]methyl]phenoxy]acetic acid
Show/Hide
|
C22H24Cl2N2O4
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0484520
|
2-[1-[4-[(4-nitrobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
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|
C25H17N3O6
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0290305
|
2-(5-chloro-3'-cyanobiphenyl-2-yloxy)acetic acid
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|
C15H10ClNO3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0409058
|
2-[1-[4-[(3,4-dichlorophenyl)carbamoyl]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H16Cl2N2O4
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0415476
|
N-[3-chloro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methoxyphenyl)methyl]pentanamide
Show/Hide
|
C20H22ClN5O2
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 3.6 nM
|
|
|
|
CP0447086
|
(S)-2-(2-((4-(benzylsulfonyl)-3-methylpiperazin-1-yl)methyl)-4-chlorophenyl)acetic acid
Show/Hide
|
C21H25ClN2O4S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0386063
|
2-[1-[4-[[4-(trifluoromethoxy)benzoyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C26H17F3N2O5
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0555896
|
2-[1-[4-[3-(4-chlorophenyl)propoxy]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C27H22ClNO4
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0531041
|
2-[1-[4-[2-(4-chlorophenyl)ethoxy]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C26H20ClNO4
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0498086
|
(S)-2-(4-chloro-2-((4-(phenylsulfonyl)-3-propylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H27ClN2O5S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0387887
|
2-[1-[4-[3-(3,4-dichlorophenyl)propanoylamino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C27H20Cl2N2O4
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0549647
|
2-[1-[4-[(3,4-dichlorophenyl)carbamoylamino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H17Cl2N3O4
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0409056
|
2-[1-[4-(cyclohexanecarbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H24N2O4
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0392650
|
2-[1-[4-[(4-phenoxybenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C31H22N2O5
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0432735
|
2-[1-[4-[[2-(3,4-dichlorophenyl)acetyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C26H18Cl2N2O4
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0399932
|
(S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0399934
|
(S)-2-(4-chloro-2-((4-(2-(2-chlorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H24Cl2N2O4
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0506025
|
2-(2-((4-(benzylsulfonyl)piperazin-1-yl)methyl)-4-chlorophenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0522682
|
2-[4-chloro-2-[[(3S)-4-[2-(4-chlorophenyl)acetyl]-3-methylpiperazin-1-yl]methyl]phenyl]acetic acid
Show/Hide
|
C22H24Cl2N2O3
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0392651
|
2-[1-[4-[(4-phenylbenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C31H22N2O4
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0424657
|
2-{5-chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,5'-dione}acetic acid
Show/Hide
|
C24H20ClN3O5
|
2
|
| 1 |
IC50 = 19 nM
|
|
|
| 2 |
Ki = 3.8 nM
|
|
|
|
CP0056577
|
2-[1-[4-[(3,4-dichlorobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H16Cl2N2O4
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0139382
|
N-[3-chloro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]pentanamide
Show/Hide
|
C20H19ClF3N5O2
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0386065
|
2-[1-[4-[(2-cyclohexylacetyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C26H26N2O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0435032
|
2-{5-chloro-1'-[(5-methyl-3-phenyl-1,2-oxazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C24H18ClN3O6
|
2
|
| 1 |
IC50 = 21 nM
|
|
|
| 2 |
Ki = 7.6 nM
|
|
|
|
CP0489856
|
2-[1-[4-[[2-(1-adamantyl)acetyl]amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C30H30N2O4
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0485747
|
2-{5-chloro-1'-[(3-methyl-5-phenyl-1,2-oxazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C24H18ClN3O6
|
2
|
| 1 |
IC50 = 23 nM
|
|
|
| 2 |
Ki = 5.3 nM
|
|
|
|
CP0399653
|
2-[1-[4-[2-(4-chlorophenyl)ethylcarbamoyl]benzoyl]isoquinolin-4-yl]oxyacetic acid
Show/Hide
|
C27H21ClN2O5
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0378230
|
2-[1-(4-chlorophenyl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
Show/Hide
|
C17H13ClFNO4S
|
2
|
| 1 |
IC50 = 26 nM
|
|
|
| 2 |
Ki = 29 nM
|
|
|
|
CP0500985
|
(S)-2-(4-chloro-2-((3-methyl-4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H25ClN2O4
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0447088
|
(S)-2-(4-chloro-2-((4-(2-(3-chlorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H24Cl2N2O4
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0164558
|
2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl)biphenyl-2-yloxy)acetic acid
Show/Hide
|
C18H17F3O5S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0297983
|
2-[4-chloro-2-[2-(3-chlorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C16H10Cl2O3
|
5
|
| 1 |
IC50 = 29 nM
|
|
|
| 2 |
IC50 = 104 nM
|
|
|
| 3 |
IC50 = 114 nM
|
|
|
| 4 |
IC50 = 1200 nM
|
|
|
| 5 |
Ki = 29 nM
|
|
|
|
CP0502399
|
2-(1-(4-cyano-3-ethoxyphenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C19H17N3O5S
|
2
|
| 1 |
IC50 = 31 nM
|
|
|
| 2 |
Ki = 43 nM
|
|
|
|
CP0447087
|
(S)-2-(4-chloro-2-((3-ethyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C21H25ClN2O5S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0906028
|
rac-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0484522
|
2-[1-[4-(naphthalene-1-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C29H20N2O4
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0066158
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C18H15F4N5O
|
2
|
| 1 |
IC50 = 37 nM
|
|
|
| 2 |
Ki = 5.7 nM
|
|
|
|
CP0054111
|
2-[2-methyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C18H18N2O4S
|
3
|
| 1 |
IC50 = 37 nM
|
|
|
| 2 |
Kd = 15.14 nM
|
|
|
| 3 |
Ki = 36 nM
|
|
|
|
CP0380963
|
2-[1-[4-[(3,4-dichlorophenyl)methoxy]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H17Cl2NO4
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0425641
|
(S)-2-(4-chloro-2-((4-(2-(4-chlorophenyl)-2-methylpropanoyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C24H28Cl2N2O4
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0404910
|
2-(1-(4-chloro-3-cyanophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C17H12ClN3O4S
|
2
|
| 1 |
IC50 = 41 nM
|
|
|
| 2 |
Ki = 35 nM
|
|
|
|
CP0391849
|
2-[1-(2,5-dichlorophenyl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
Show/Hide
|
C17H12Cl2FNO4S
|
2
|
| 1 |
IC50 = 44 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0409057
|
2-[1-[4-[(2-chlorobenzoyl)amino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C25H17ClN2O4
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0133932
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-3-methyl-N-[(4-methylsulfonylphenyl)methyl]butanamide
Show/Hide
|
C20H22FN5O3S
|
2
|
| 1 |
IC50 = 46 nM
|
|
|
| 2 |
Ki = 3.2 nM
|
|
|
|
CP0435033
|
2-{5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H13Cl2FN2O5
|
2
|
| 1 |
IC50 = 48 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0505203
|
2-(5-chloro-1'-{[2-(3-chlorophenyl)-1,3-thiazol-4-yl]methyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione)acetic acid
Show/Hide
|
C23H15Cl2N3O5S
|
2
|
| 1 |
IC50 = 48 nM
|
|
|
| 2 |
Ki = 24 nM
|
|
|
|
CP0566214
|
2-[1-[4-(pyridine-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C24H17N3O4
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0387885
|
2-[1-[4-(cyclopropanecarbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C22H18N2O4
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0153959
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]cyclopentanecarboxamide
Show/Hide
|
C21H22FN5O3S
|
2
|
| 1 |
IC50 = 57 nM
|
|
|
| 2 |
Ki = 5.4 nM
|
|
|
|
CP0245256
|
2-(1-(3,4-difluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C16H12F2N2O4S
|
2
|
| 1 |
IC50 = 60 nM
|
|
|
| 2 |
Ki = 31 nM
|
|
|
|
CP0420584
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(3-methoxyphenyl)methyl]propanamide
Show/Hide
|
C18H18FN5O2
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2
|
| 1 |
IC50 = 64 nM
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| 2 |
Ki = 8.2 nM
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CP0160937
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2-[(3R)-5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C20H13Cl2FN2O5
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2
|
| 1 |
IC50 = 66 nM
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| 2 |
Ki = 5.3 nM
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CP0489810
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2-[1-[4-(1,3-thiazole-4-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
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C22H15N3O4S
|
1
|
| 1 |
IC50 = 67 nM
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CP0447089
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2-[2-[[4-(benzenesulfonyl)-2-methylpiperazin-1-yl]methyl]-4-chlorophenoxy]acetic acid
Show/Hide
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C20H23ClN2O5S
|
1
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| 1 |
IC50 = 71 nM
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CP0432066
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2-{5-chloro-1'-[(3,5-dichlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C20H13Cl3N2O5
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2
|
| 1 |
IC50 = 82 nM
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| 2 |
Ki = 36 nM
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CP0530736
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2-[1-[4-(pyridine-4-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
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C24H17N3O4
|
1
|
| 1 |
IC50 = 83 nM
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CP0169760
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N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(3-hydroxyphenyl)methyl]propanamide
Show/Hide
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C17H16FN5O2
|
2
|
| 1 |
IC50 = 85 nM
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| 2 |
Ki = 26 nM
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CP0503269
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2-(2-((4-(benzylsulfonyl)-1,4-diazepan-1-yl)methyl)-4-chlorophenoxy)acetic acid
Show/Hide
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C21H25ClN2O5S
|
1
|
| 1 |
IC50 = 89 nM
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CP0503954
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2-(1-(4-fluoro-3-methoxyphenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C17H15FN2O5S
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2
|
| 1 |
IC50 = 91 nM
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| 2 |
Ki = 56 nM
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CP0377112
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2-(1-(3-cyano-4-fluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C17H12FN3O4S
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2
|
| 1 |
IC50 = 101 nM
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| 2 |
Ki = 36 nM
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CP0109477
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2-[(3R)-5-chloro-1'-[(3-chlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C20H14Cl2N2O5
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2
|
| 1 |
IC50 = 107 nM
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| 2 |
Ki = 23 nM
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CP0529890
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2-{5-chloro-1'-[(3-chlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C20H14Cl2N2O5
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2
|
| 1 |
IC50 = 122 nM
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| 2 |
Ki = 68 nM
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CP0379870
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2-[2-methyl-1-[(4-nitrophenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C17H15N3O4
|
2
|
| 1 |
IC50 = 143 nM
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| 2 |
Ki = 147 nM
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CP0438204
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2-[2-methyl-1-[[4-(trifluoromethylsulfonyl)phenyl]methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C18H15F3N2O4S
|
2
|
| 1 |
IC50 = 147 nM
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| 2 |
Ki = 208 nM
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CP0201722
|
2-(4-chloro-2-cycloheptylphenoxy)acetic acid
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C15H19ClO3
|
2
|
| 1 |
IC50 = 148 nM
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| 2 |
Ki = 59 nM
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CP0259564
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2-[5-fluoro-2-methyl-1-(4-methylsulfonylphenyl)sulfonylindol-3-yl]acetic acid
Show/Hide
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C18H16FNO6S2
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2
|
| 1 |
IC50 = 158 nM
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| 2 |
Ki = 68 nM
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CP0503860
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2-[5-fluoro-1-(4-fluorophenyl)sulfonyl-2-methylindol-3-yl]acetic acid
Show/Hide
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C17H13F2NO4S
|
2
|
| 1 |
IC50 = 158 nM
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| 2 |
Ki = 71 nM
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CP0435034
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2-{5-chloro-1'-[(4-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H14ClFN2O5
|
2
|
| 1 |
IC50 = 182 nM
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| 2 |
Ki = 96 nM
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CP0405110
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2-[2-[(4-benzoyl-3-methylpiperazin-1-yl)methyl]-4-chlorophenoxy]acetic acid
Show/Hide
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C21H23ClN2O4
|
1
|
| 1 |
IC50 = 199 nM
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CP0380962
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2-[1-[4-[2-(4-chlorophenyl)ethylcarbamoyl]benzoyl]isoquinolin-4-yl]-2-methylpropanoic acid
Show/Hide
|
C29H25ClN2O4
|
1
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| 1 |
IC50 = 200 nM
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CP0511333
|
2-[2-[[4-(benzenesulfonyl)piperazin-1-yl]methyl]-4-chlorophenoxy]acetic acid
Show/Hide
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C19H21ClN2O5S
|
1
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| 1 |
IC50 = 201 nM
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CP0048953
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(R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydrocarbazol-9-yl)propanoic acid
Show/Hide
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C21H21FN2O4S
|
3
|
| 1 |
IC50 = 210 nM
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| 2 |
IC50 = 461 nM
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| 3 |
Ki = 73 nM
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CP0476028
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2-[1-[4-[(3,4-dichlorobenzoyl)-methylamino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
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C26H18Cl2N2O4
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1
|
| 1 |
IC50 = 210 nM
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CP0405206
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2-{5-chloro-1'-[(2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H14ClFN2O5
|
2
|
| 1 |
IC50 = 212 nM
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| 2 |
Ki = 37 nM
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CP0485749
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2-{5-chloro-1'-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C19H16ClN3O6
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2
|
| 1 |
IC50 = 220 nM
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| 2 |
Ki = 51 nM
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CP0054115
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2-[2-methyl-1-[(4-methylsulfinylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C18H18N2O3S
|
2
|
| 1 |
IC50 = 233 nM
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| 2 |
Ki = 249 nM
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CP0427740
|
2-{5-chloro-1'-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C18H14ClN3O5S
|
2
|
| 1 |
IC50 = 236 nM
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|
| 2 |
Ki = 38 nM
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CP0473220
|
(R)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 240 nM
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CP0476027
|
2-[1-[4-(pyrimidine-2-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C23H16N4O4
|
1
|
| 1 |
IC50 = 290 nM
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CP0373094
|
2-{5-chloro-1'-[(2,3-difluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H13ClF2N2O5
|
2
|
| 1 |
IC50 = 296 nM
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|
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| 2 |
Ki = 25 nM
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CP0506218
|
2-(1-(3-chloro-4-fluorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C16H12ClFN2O4S
|
2
|
| 1 |
IC50 = 311 nM
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| 2 |
Ki = 158 nM
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CP0391851
|
2-[5-fluoro-1-(4-methoxyphenyl)sulfonyl-2-methylindol-3-yl]acetic acid
Show/Hide
|
C18H16FNO5S
|
2
|
| 1 |
IC50 = 318 nM
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|
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| 2 |
Ki = 299 nM
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CP0555897
|
2-[1-[4-(pyridazine-3-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C23H16N4O4
|
1
|
| 1 |
IC50 = 322 nM
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CP0420655
|
2-[1-(4-acetamidobenzoyl)isoquinolin-4-yl]acetic acid
Show/Hide
|
C20H16N2O4
|
1
|
| 1 |
IC50 = 330 nM
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CP0387886
|
2-[1-[4-[(3,4-dichlorophenyl)sulfonylamino]benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C24H16Cl2N2O5S
|
1
|
| 1 |
IC50 = 340 nM
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CP0498416
|
2-(1-(3,4-dichlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C16H12Cl2N2O4S
|
2
|
| 1 |
IC50 = 354 nM
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| 2 |
Ki = 52 nM
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CP0380032
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2-[1-[4-(oxane-4-carbonylamino)benzoyl]isoquinolin-4-yl]acetic acid
Show/Hide
|
C24H22N2O5
|
1
|
| 1 |
IC50 = 400 nM
|
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CP0103498
|
2-{1'-benzyl-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H15ClN2O5
|
2
|
| 1 |
IC50 = 418 nM
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| 2 |
Ki = 196 nM
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CP0209430
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2-[1-[(4-chlorophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C17H15ClN2O2
|
2
|
| 1 |
IC50 = 484 nM
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| 2 |
Ki = 149 nM
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CP0511435
|
2-(2-{[(3S)-4-(benzylsulfonyl)-3-methylpiperazin-1-yl]methyl}-4-chlorophenyl)-N-(methylsulfonyl)acetamide
Show/Hide
|
C22H28ClN3O5S2
|
1
|
| 1 |
IC50 = 486 nM
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CP0461748
|
2-(2-((4-(phenylsulfonyl)piperazin-1-yl)methyl)-4-(trifluoromethyl)phenoxy)acetic acid
Show/Hide
|
C20H21F3N2O5S
|
1
|
| 1 |
IC50 = 517 nM
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CP0473222
|
3-(4-Chloro-2-{[(3S)-3-methyl-4-(phenylacetyl)piperazin-1-yl]methyl}phenyl)propanoic acid
Show/Hide
|
C23H27ClN2O3
|
1
|
| 1 |
IC50 = 547 nM
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CP0054113
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2-[1-[(4-cyanophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C18H15N3O2
|
2
|
| 1 |
IC50 = 554 nM
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| 2 |
Ki = 379 nM
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CP0054110
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2-(1-(4-chlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C16H13ClN2O4S
|
2
|
| 1 |
IC50 = 565 nM
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| 2 |
Ki = 103 nM
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CP0498276
|
2-[5-fluoro-1-(3-fluorophenyl)sulfonyl-2-methylindol-3-yl]acetic acid
Show/Hide
|
C17H13F2NO4S
|
2
|
| 1 |
IC50 = 639 nM
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| 2 |
Ki = 225 nM
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CP0456427
|
2-(1-butylsulfonyl-5-fluoro-2-methylindol-3-yl)acetic acid
Show/Hide
|
C15H18FNO4S
|
2
|
| 1 |
IC50 = 842 nM
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| 2 |
Ki = 634 nM
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CP0378076
|
(1-Benzenesulfonyl-5-fluoro-2-methyl-1H-indol-3-yl)-acetic acid
Show/Hide
|
C17H14FNO4S
|
2
|
| 1 |
IC50 = 987 nM
|
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|
| 2 |
Ki = 250 nM
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CP0405109
|
2-(4-chloro-2-((4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C21H23ClN2O4
|
1
|
| 1 |
IC50 = 1082 nM
|
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CP0503270
|
(S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)-2-methylpropanoic acid
Show/Hide
|
C22H27ClN2O5S
|
1
|
| 1 |
IC50 = 1442 nM
|
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CP0446446
|
2-[5-fluoro-2-methyl-1-(4-methylphenyl)sulfonylindol-3-yl]acetic acid
Show/Hide
|
C18H16FNO4S
|
2
|
| 1 |
IC50 = 2184 nM
|
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| 2 |
Ki = 457 nM
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CP0503271
|
2-(4-chloro-2-(((3S,5R)-3,5-dimethyl-4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C23H27ClN2O4
|
1
|
| 1 |
IC50 = 3840 nM
|
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CP0473223
|
2-(4-chloro-2-((4-(phenylsulfonyl)-1,4-diazepan-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 4093 nM
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CP0485411
|
2-[1-(1,2-dimethylimidazol-4-yl)sulfonyl-5-fluoro-2-methylindol-3-yl]acetic acid
Show/Hide
|
C16H16FN3O4S
|
2
|
| 1 |
IC50 > 10000 nM
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| 2 |
Ki = 2979 nM
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CP0081955
|
Fevipiprant
Show/Hide
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C19H17F3N2O4S
|
2
|
| 1 |
Kd = 1.023 nM
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| 2 |
Ki = 4 nM
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CP0090559
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2-[1-[(2-chloro-4-ethylsulfonylphenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C19H19ClN2O4S
|
2
|
| 1 |
Kd = 1.905 nM
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| 2 |
Ki = 6 nM
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CP0323455
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2-[2-methyl-1-[(4-methylsulfonylphenyl)methyl]indol-3-yl]acetic acid
Show/Hide
|
C19H19NO4S
|
2
|
| 1 |
Kd = 25.12 nM
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| 2 |
Ki = 19 nM
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CP0490654
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2-[(3S)-4-(4-chlorophenyl)sulfanyl-7-fluoro-2,3-dihydro-1H-pyrrolo[1,2-a]indol-3-yl]acetic acid
Show/Hide
|
C19H15ClFNO2S
|
1
|
| 1 |
Ki = 0.8 nM
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CP0431188
|
2-[4-chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]propanoic acid
Show/Hide
|
C21H21ClO5S
|
1
|
| 1 |
Ki = 1.2 nM
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CP0382535
|
2-[2-[2-(4-acetamido-2-methyl-5-propylsulfonylphenyl)ethynyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C22H22ClNO6S
|
1
|
| 1 |
Ki = 1.3 nM
|
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|
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CP0456485
|
2-[4-chloro-2-[2-[2-methyl-5-(2-methylpiperidin-1-yl)sulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C23H24ClNO5S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0387495
|
2-[4-chloro-2-[2-(2-chloro-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H16Cl2O5S
|
1
|
| 1 |
Ki = 2.1 nM
|
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|
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CP0550743
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]benzamide
Show/Hide
|
C22H18FN5O3S
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
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CP0133930
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethyl)phenyl]methyl]pentanamide
Show/Hide
|
C20H19F4N5O
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
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CP0550744
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-3-(4-methylphenyl)-N-[(4-methylsulfonylphenyl)methyl]propanamide
Show/Hide
|
C25H24FN5O3S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
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CP0475661
|
2-[4-chloro-2-[2-(2-chloro-5-propan-2-ylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H16Cl2O5S
|
1
|
| 1 |
Ki = 2.9 nM
|
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CP0418994
|
2-[4-chloro-2-[2-[2-methyl-5-(2-methylpropylsulfonyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H21ClO5S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0432740
|
2-[4-chloro-2-[2-(2-fluoro-5-propylsulfonylphenyl)ethynyl]phenoxy]propanoic acid
Show/Hide
|
C20H18ClFO5S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0410379
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(3-methoxyphenyl)methyl]pentanamide
Show/Hide
|
C20H22FN5O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0550741
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methoxyphenyl)methyl]pentanamide
Show/Hide
|
C20H22FN5O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
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CP0506094
|
2-[4-chloro-2-[2-[5-(dimethylsulfamoyl)-2-fluorophenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H15ClFNO5S
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0169837
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]propanamide
Show/Hide
|
C18H18FN5O3S
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0495444
|
2-[4-chloro-2-[2-(3-methylsulfinylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C17H13ClO4S
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0392176
|
2-[4-chloro-2-[2-(2-fluoro-5-methylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C17H12ClFO5S
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0410377
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
|
C21H22FN5O3
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0400876
|
2-[4-chloro-2-[2-[2-methyl-5-(propan-2-ylsulfamoyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H20ClNO5S
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0456483
|
2-[4-chloro-2-[2-[5-(diethylsulfamoyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H22ClNO5S
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0499401
|
2-[4-chloro-2-[2-(2-chloro-5-methylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C17H12Cl2O5S
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0520268
|
2-[4-chloro-2-[2-[4-(2-chlorophenyl)-3-methylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C23H16Cl2O5S
|
1
|
| 1 |
Ki = 3.5 nM
|
|
|
|
CP0393378
|
2-[4-chloro-2-[2-(2-methyl-5-morpholin-4-ylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H20ClNO6S
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0456416
|
2-[4-chloro-2-[2-[5-(2-methoxyethylsulfamoyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H20ClNO6S
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0387496
|
2-[4-chloro-2-[2-[2-methyl-5-[methyl(propan-2-yl)sulfamoyl]phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H22ClNO5S
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0427437
|
2-[4-chloro-2-[2-(2-fluoro-5-propan-2-ylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H16ClFO5S
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0410380
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]pyridine-3-carboxamide
Show/Hide
|
C21H17FN6O3S
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0081954
|
2-[1-[(2-chloro-4-methylsulfonylphenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C18H17ClN2O4S
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0387497
|
2-[4-chloro-2-[2-[5-[2-methoxyethyl(methyl)sulfamoyl]-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H22ClNO6S
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0456484
|
2-[4-chloro-2-[2-[2-methyl-5-[methyl(2-methylpropyl)sulfamoyl]phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C22H24ClNO5S
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0427150
|
2-[4-chloro-2-[2-(4-propylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H16ClNO3
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0459329
|
2-[4-chloro-2-[2-[5-(ethylsulfamoyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H18ClNO5S
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0139383
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[3-(trifluoromethoxy)phenyl]methyl]pentanamide
Show/Hide
|
C20H19F4N5O2
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
|
CP0476266
|
2-[4-chloro-2-[2-(5-methylsulfonyl-2-propan-2-ylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H19ClO5S
|
1
|
| 1 |
Ki = 4.6 nM
|
|
|
|
CP0495977
|
2-[4-chloro-2-[2-[4-(2-methylpropyl)pyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H18ClNO3
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
|
CP0502868
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]butanamide
Show/Hide
|
C20H20FN5O3
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
|
CP0382594
|
2-[4-chloro-2-[2-(3-methylsulfonyl-4-phenylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C23H17ClO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0387449
|
2-[4-chloro-2-[2-[5-(dimethylsulfamoyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H18ClNO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0392175
|
2-[4-chloro-2-[2-(2-methyl-5-methylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H15ClO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0401043
|
2-[3-[2-[[cyclopropanecarbonyl(ethyl)amino]methyl]-4-(5-methoxypyridin-2-yl)phenyl]-4-methoxyphenyl]acetic acid
Show/Hide
|
C28H30N2O5
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0418996
|
2-[2-[2-(5-benzylsulfonyl-2-methylphenyl)ethynyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C24H19ClO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0432585
|
2-[2-[2-[5-(tert-butylsulfamoyl)-2-methylphenyl]ethynyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C21H22ClNO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0523751
|
2-[4-chloro-2-[2-(2-methyl-5-piperidin-1-ylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C22H22ClNO5S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0416091
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethylsulfonyl)phenyl]methyl]propanamide
Show/Hide
|
C18H15F4N5O3S
|
1
|
| 1 |
Ki = 5.2 nM
|
|
|
|
CP0509741
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]-3-methylbutanamide
Show/Hide
|
C21H22FN5O3
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0392177
|
2-[2-[2-[5-(benzenesulfonyl)-2-methylphenyl]ethynyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C23H17ClO5S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0461787
|
2-[4-chloro-2-[2-(2-methyl-5-propan-2-ylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H19ClO5S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0123607
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(3-propan-2-yloxyphenyl)methyl]propanamide
Show/Hide
|
C20H22FN5O2
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
|
CP0066163
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]propanamide
Show/Hide
|
C18H15F4N5O2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0382533
|
2-[4-chloro-2-[2-[4-(4-methoxyphenyl)-3-methylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C24H19ClO6S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0463234
|
2-[4-chloro-2-[2-[2-methyl-5-(2-phenylethylsulfonyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C25H21ClO5S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0475227
|
2-[4-cyano-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H19NO5S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0112127
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
|
C21H23N5O3
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0424659
|
2-[5'-chloro-1-[(5-methyl-3-phenyl-1,2-oxazol-4-yl)methyl]-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C23H17ClN4O6
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0445485
|
2-[1-[[4-ethylsulfonyl-2-(trifluoromethyl)phenyl]methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C20H19F3N2O4S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0432885
|
N-(1-benzofuran-2-ylmethyl)-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
|
C21H20FN5O2
|
1
|
| 1 |
Ki = 7.1 nM
|
|
|
|
CP0432881
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methoxyphenyl)methyl]propanamide
Show/Hide
|
C18H18FN5O2
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0066159
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethoxy)phenyl]methyl]pentanamide
Show/Hide
|
C20H19F4N5O2
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0382534
|
2-[4-chloro-2-[2-[4-(3-methoxyphenyl)-3-methylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C24H19ClO6S
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0392178
|
2-[4-chloro-2-[2-[5-(3-hydroxypropylsulfonyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H19ClO6S
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0505975
|
2-[4-chloro-2-[2-(5-methylsulfonyl-2-propylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H19ClO5S
|
1
|
| 1 |
Ki = 8.6 nM
|
|
|
|
CP0520243
|
2-[4-chloro-2-[2-(5-ethylsulfonyl-2-methylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H17ClO5S
|
1
|
| 1 |
Ki = 8.6 nM
|
|
|
|
CP0392174
|
2-[4-chloro-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H17ClO5S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0427151
|
2-[4-chloro-2-[2-[3-(2-hydroxyethylsulfonyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H15ClO6S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0456565
|
2-[2-[2-(3-propylsulfonylphenyl)ethynyl]-4-(trifluoromethyl)phenoxy]acetic acid
Show/Hide
|
C20H17F3O5S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0463236
|
2-[4-chloro-2-[2-[2-methyl-5-(methylsulfamoyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H16ClNO5S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0415474
|
N-[(3-ethynylphenyl)methyl]-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
|
C21H20FN5O
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0542406
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
|
C19H18FN5O3
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0394532
|
2-{5-chloro-1'-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C22H20ClN3O6
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0390764
|
2-[4-cyano-2-[2-(5-methylsulfonyl-2-propan-2-ylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H19NO5S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0391011
|
2-[4-chloro-2-[2-(5,5-dioxodibenzothiophen-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C22H13ClO5S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0401044
|
2-[2-[2-(2-chlorophenyl)ethynyl]-4-(trifluoromethyl)phenoxy]acetic acid
Show/Hide
|
C17H10ClF3O3
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0505929
|
2-[2-[2-(3-propylsulfonylphenyl)ethynyl]-3-thiophen-2-ylphenoxy]acetic acid
Show/Hide
|
C23H20O5S2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0470516
|
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]butanamide
Show/Hide
|
C20H21N5O3
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0373107
|
2-[(3R)-5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,5'-dione]acetic acid
Show/Hide
|
C20H15Cl2FN2O4
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0524931
|
2-[(3S)-5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,5'-dione]acetic acid
Show/Hide
|
C20H15Cl2FN2O4
|
2
|
| 1 |
Ki = 13 nM
|
|
|
| 2 |
Ki = 683 nM
|
|
|
|
CP0382595
|
2-[4-chloro-2-[2-[4-(4-chlorophenyl)-3-methylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C23H16Cl2O5S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0482210
|
2-[4-chloro-2-[2-[3-(dimethylsulfamoyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H16ClNO5S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0525014
|
2-[2-[2-(2-tert-butyl-1,1,3-trioxo-1,2-benzothiazol-6-yl)ethynyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C21H18ClNO6S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0395105
|
2-[4-chloro-2-[2-(3-methylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C17H13ClO5S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0494026
|
2-[(4S)-5'-chloro-1-[(5-chloro-2-fluorophenyl)methyl]-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C19H12Cl2FN3O5
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0523749
|
2-[4-chloro-2-[2-[4-(3-chlorophenyl)-3-methylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C23H16Cl2O5S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0566443
|
2-[5'-chloro-3-methyl-2,2',5-trioxo-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]spiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C23H17ClN4O5S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0525027
|
2-[4-chloro-2-[2-(4-methyl-1-oxidopyridin-1-ium-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C16H12ClNO4
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0415478
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-2-methyl-N-[(4-methylsulfonylphenyl)methyl]propanamide
Show/Hide
|
C19H20FN5O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0550745
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]pyridine-4-carboxamide
Show/Hide
|
C21H17FN6O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0459218
|
2-[2-[2-(3-propylsulfonylphenyl)ethynyl]-3-thiophen-3-ylphenoxy]acetic acid
Show/Hide
|
C23H20O5S2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0470515
|
N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-(naphthalen-2-ylmethyl)pentanamide
Show/Hide
|
C23H22FN5O
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0394818
|
2-[4-chloro-2-[2-[5-(methanesulfonamido)pyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C16H13ClN2O5S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0395108
|
2-[3-phenyl-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C25H22O5S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0520245
|
2-[4-chloro-2-[2-[5-(2-hydroxyethylsulfonyl)-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C19H17ClO6S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0210131
|
2-(2-cyclohexyl-4-(trifluoromethyl)phenoxy)acetic acid
Show/Hide
|
C15H17F3O3
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0513855
|
2-{5-chloro-1'-[(3-chloro-5-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H13Cl2FN2O5
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0513856
|
2-{5-chloro-1'-[(2,5-difluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H13ClF2N2O5
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0461782
|
2-[4-cyano-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C20H17NO5S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0505954
|
2-[4-chloro-2-[2-(3-methoxy-2,2-dimethyl-1,1-dioxo-3H-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C21H19ClO6S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0525028
|
2-[4-chloro-2-[2-[2-methyl-5-(4-methylpiperazin-1-yl)sulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C22H23ClN2O5S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0393375
|
2-[4-chloro-2-[2-[2-fluoro-4-(methoxymethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H14ClFO4
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0550742
|
N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-hydroxyphenyl)methyl]propanamide
Show/Hide
|
C17H16FN5O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0109471
|
2-[(3R)-5-chloro-1'-[(2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
|
C20H14ClFN2O5
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0433274
|
2-[4-chloro-2-[2-(1,1-dioxo-2,3-dihydro-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C18H13ClO5S
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1
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| 1 |
Ki = 23 nM
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CP0484561
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2-[2-[2-(2-chlorophenyl)ethynyl]-4-cyanophenoxy]acetic acid
Show/Hide
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C17H10ClNO3
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1
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| 1 |
Ki = 24 nM
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CP0505933
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2-[4-chloro-2-[2-[2-(trifluoromethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H10ClF3O3
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1
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| 1 |
Ki = 24 nM
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CP0395104
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2-[4-chloro-2-[2-(4-methylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H12ClNO3
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1
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| 1 |
Ki = 25 nM
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CP0433273
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2-[4-chloro-2-[2-(1,1-dioxo-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C18H11ClO5S
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1
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| 1 |
Ki = 25 nM
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CP0433275
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2-[4-chloro-2-[2-(3-methoxy-2,2,3-trimethyl-1,1-dioxo-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C22H21ClO6S
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1
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| 1 |
Ki = 25 nM
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CP0266551
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2-[4-chloro-2-[2-(2-chlorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H10Cl2O3
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1
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| 1 |
Ki = 28 nM
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CP0390880
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2-[4-chloro-2-[2-[3-(3-hydroxypropylsulfonyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C19H17ClO6S
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1
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| 1 |
Ki = 28 nM
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CP0432741
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2-[4-chloro-2-[2-[2-fluoro-4-(hydroxymethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H12ClFO4
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1
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| 1 |
Ki = 28 nM
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CP0525015
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2-[4-chloro-2-[2-(3-hydroxy-2,2,3-trimethyl-1,1-dioxo-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C21H19ClO6S
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1
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| 1 |
Ki = 28 nM
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CP0509733
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N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-[(4-methylsulfonylphenyl)methyl]oxane-4-carboxamide
Show/Hide
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C21H22FN5O4S
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1
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| 1 |
Ki = 28 nM
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CP0424658
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2-[5'-chloro-1-[(5-chloro-2-fluorophenyl)methyl]-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C19H12Cl2FN3O5
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1
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| 1 |
Ki = 28 nM
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CP0147599
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2-[1-[[2,4-bis(trifluoromethyl)phenyl]methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C19H14F6N2O2
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1
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| 1 |
Ki = 29 nM
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CP0503079
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2-[4-chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]butanoic acid
Show/Hide
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C22H23ClO5S
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1
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| 1 |
Ki = 30 nM
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CP0393371
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2-[4-chloro-2-[2-(2,2-dimethyl-1,1,3-trioxo-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C20H15ClO6S
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1
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| 1 |
Ki = 31 nM
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CP0246918
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2-[2-methyl-1-[(2-methyl-4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C19H20N2O4S
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1
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| 1 |
Ki = 31 nM
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CP0248457
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2-[2-methyl-1-[[4-methylsulfonyl-3-(trifluoromethyl)phenyl]methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C19H17F3N2O4S
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1
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| 1 |
Ki = 31 nM
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CP0427736
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2-{5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,5'-dione}acetic acid
Show/Hide
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C20H15Cl2FN2O4
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1
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| 1 |
Ki = 32 nM
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CP0520267
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2-[4-chloro-2-[2-(3-hydroxy-2,2-dimethyl-1,1-dioxo-3H-1-benzothiophen-6-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C20H17ClO6S
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1
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| 1 |
Ki = 33 nM
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CP0140521
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2-[(4S)-5'-chloro-1-[(5-chloro-2-fluorophenyl)methyl]-3-methyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C20H14Cl2FN3O5
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1
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| 1 |
Ki = 35 nM
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CP0478153
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2-{5-chloro-1'-[(3,5-difluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C20H13ClF2N2O5
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1
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| 1 |
Ki = 37 nM
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CP0392179
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2-[4-chloro-2-[2-[5-(dimethylsulfamoyl)pyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H15ClN2O5S
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1
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| 1 |
Ki = 37 nM
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CP0450684
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N-(naphthalen-2-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
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C23H23N5O
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1
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| 1 |
Ki = 39 nM
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CP0427149
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2-[4-chloro-2-[2-[2-fluoro-3-(hydroxymethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H12ClFO4
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1
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| 1 |
Ki = 41 nM
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CP0461409
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2-[4-chloro-2-[2-[5-(dimethylsulfamoyl)-2-methylpyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
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C18H17ClN2O5S
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1
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| 1 |
Ki = 41 nM
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CP0524904
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2-[4-chloro-2-[2-(5-morpholin-4-ylsulfonylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C19H17ClN2O6S
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1
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| 1 |
Ki = 41 nM
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CP0542405
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N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C19H19N5O3
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1
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| 1 |
Ki = 42 nM
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CP0435020
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2-{5-chloro-1'-[(2-chloro-5-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C20H13Cl2FN2O5
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1
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| 1 |
Ki = 43 nM
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CP0523750
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2-[4-chloro-2-[2-(4-hexylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C21H22ClNO3
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1
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| 1 |
Ki = 43 nM
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CP0525016
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2-[4-chloro-2-[2-[3-methylsulfonyl-4-[4-(trifluoromethyl)phenyl]phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C24H16ClF3O5S
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1
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| 1 |
Ki = 43 nM
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CP0520269
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2-[1-[2-(3-propylsulfonylphenyl)ethynyl]naphthalen-2-yl]oxyacetic acid
Show/Hide
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C23H20O5S
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1
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| 1 |
Ki = 44 nM
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CP0416073
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N-[(3-methoxyphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
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C20H23N5O2
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1
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| 1 |
Ki = 44 nM
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CP0470517
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N-[2,4-difluoro-5-(2H-tetrazol-5-yl)phenyl]-N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pentanamide
Show/Hide
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C21H21F2N5O3
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1
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| 1 |
Ki = 45 nM
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CP0372522
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2-[4-chloro-2-[2-[4-(diethylcarbamoyl)-3-propan-2-ylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C24H26ClNO6S
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1
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| 1 |
Ki = 46 nM
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CP0482209
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2-[4-chloro-2-[2-(2-fluorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H10ClFO3
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1
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| 1 |
Ki = 47 nM
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CP0106923
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2-[6-ethyl-2-methyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C20H22N2O4S
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1
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| 1 |
Ki = 47 nM
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CP0506312
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2-(2-methyl-1-(4-nitrophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C16H13N3O6S
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1
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| 1 |
Ki = 48 nM
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CP0495937
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2-[4-chloro-2-[2-[3-(methylsulfonylmethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C18H15ClO5S
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1
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| 1 |
Ki = 48 nM
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CP0010057
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2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl-1H-indol-3-yl}acetic acid
Show/Hide
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C19H16ClNO4
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2
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| 1 |
Ki = 50 nM
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| 2 |
Ki = 8000 nM
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CP0066161
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N-[(4-methoxyphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
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C20H23N5O2
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1
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| 1 |
Ki = 50 nM
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CP0248458
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2-[1-[(4-ethylsulfonylphenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C19H20N2O4S
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1
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| 1 |
Ki = 50 nM
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CP0495936
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2-[4-chloro-2-[2-[3-(dimethylcarbamoyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C19H16ClNO4
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1
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| 1 |
Ki = 52 nM
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CP0467402
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2-[4-chloro-2-[2-[3-(methanesulfonamido)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H14ClNO5S
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1
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| 1 |
Ki = 54 nM
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CP0484562
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2-[3-(2,4-dimethyl-1,3-thiazol-5-yl)-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C24H23NO5S2
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1
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| 1 |
Ki = 54 nM
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CP0516323
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2-(5-chloro-1'-{[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione)acetic acid
Show/Hide
|
C23H15Cl2N3O5S
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1
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| 1 |
Ki = 55 nM
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CP0393374
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2-[3-chloro-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C19H17ClO5S
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1
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| 1 |
Ki = 55 nM
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CP0520248
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2-[4-chloro-2-[2-[4-(dimethylcarbamoyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C19H16ClNO4
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1
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| 1 |
Ki = 55 nM
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CP0443960
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N-[3-fluoro-5-(2H-tetrazol-5-yl)phenyl]-N-(quinolin-2-ylmethyl)propanamide
Show/Hide
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C20H17FN6O
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1
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| 1 |
Ki = 56 nM
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CP0461784
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2-[4-chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]pentanoic acid
Show/Hide
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C23H25ClO5S
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1
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| 1 |
Ki = 57 nM
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CP0390878
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2-[4-chloro-2-[2-(4-chlorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H10Cl2O3
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1
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| 1 |
Ki = 60 nM
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CP0432586
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2-[4-chloro-2-[2-(5-methylsulfonylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H12ClNO5S
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1
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| 1 |
Ki = 60 nM
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CP0382596
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2-[4-chloro-2-[2-[4-(dimethylcarbamoyl)-3-propan-2-ylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C22H22ClNO6S
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1
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| 1 |
Ki = 65 nM
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CP0433276
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2-[4-fluoro-2-[2-(3-propylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C19H17FO5S
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1
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| 1 |
Ki = 65 nM
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CP0506254
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N-[(4-methylsulfonylphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C18H19N5O3S
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1
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| 1 |
Ki = 69 nM
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CP0373089
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2-[(3R)-5-chloro-1'-[(3-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
|
C21H17ClN2O6
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1
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| 1 |
Ki = 72 nM
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CP0495976
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2-[4-chloro-2-[2-[2-fluoro-5-(methoxymethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C18H14ClFO4
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1
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| 1 |
Ki = 72 nM
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CP0081956
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2-[2,6-dimethyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C19H20N2O4S
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1
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| 1 |
Ki = 72 nM
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CP0427148
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2-[4-chloro-2-[2-[2-fluoro-5-(hydroxymethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H12ClFO4
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1
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| 1 |
Ki = 73 nM
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CP0328153
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(S)-2-(4-chloro-2-cyclohexylphenoxy)propanoic acid
Show/Hide
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C15H19ClO3
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1
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| 1 |
Ki = 75 nM
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CP0505200
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2-[(3R)-1'-benzyl-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
|
C20H15ClN2O5
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1
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| 1 |
Ki = 81 nM
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CP0311206
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2-(4-bromo-2-cyclohexylphenoxy)acetic acid
Show/Hide
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C14H17BrO3
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1
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| 1 |
Ki = 83 nM
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CP0520246
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2-[4-chloro-2-[2-(4-methylsulfonylphenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C17H13ClO5S
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1
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| 1 |
Ki = 86 nM
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CP0147600
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2-[2-methyl-1-[(4-propan-2-ylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C20H22N2O4S
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1
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| 1 |
Ki = 86 nM
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CP0456493
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2-[4-chloro-2-[2-[4-(morpholine-4-carbonyl)-3-propan-2-ylsulfonylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C24H24ClNO7S
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1
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| 1 |
Ki = 87 nM
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CP0478146
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2-{5-chloro-1'-[(3,4-difluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H13ClF2N2O5
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1
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| 1 |
Ki = 89 nM
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CP0309152
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2-(4-chloro-2-(1-methylcyclohexyl)phenoxy)acetic acid
Show/Hide
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C15H19ClO3
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1
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| 1 |
Ki = 90 nM
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CP0522139
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2-[4-chloro-2-[2-[3-(trifluoromethyl)phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H10ClF3O3
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1
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| 1 |
Ki = 92 nM
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CP0424660
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2-[5'-chloro-1-[(1,3-diphenylpyrazol-4-yl)methyl]-3-methyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C29H22ClN5O5
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1
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| 1 |
Ki = 96 nM
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CP0309153
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(3-cyclohexyl-4'-fluoro-biphenyl-4-yloxy)-acetic acid
Show/Hide
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C20H21FO3
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1
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| 1 |
Ki = 99 nM
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CP0505965
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2-[4-chloro-2-[2-(2,4-difluorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H9ClF2O3
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1
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| 1 |
Ki = 101 nM
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CP0459328
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2-[4-chloro-2-(2-phenylethynyl)phenoxy]acetic acid
Show/Hide
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C16H11ClO3
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1
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| 1 |
Ki = 108 nM
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CP0542924
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2-[1-[(3,4-dichlorophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C17H14Cl2N2O2
|
1
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| 1 |
Ki = 109 nM
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CP0066160
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N-[3-(2H-tetrazol-5-yl)phenyl]-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C18H16F3N5O
|
1
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| 1 |
Ki = 110 nM
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CP0482094
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2-[(4S)-5'-chloro-1-[(5-chloro-2-fluorophenyl)methyl]-2,2',5-trioxo-3-propylspiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C22H18Cl2FN3O5
|
1
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| 1 |
Ki = 110 nM
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CP0566442
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2-[5'-chloro-3-methyl-1-[(5-methyl-3-phenyl-1,2-oxazol-4-yl)methyl]-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
|
C24H19ClN4O6
|
1
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| 1 |
Ki = 110 nM
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CP0539703
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2-{5-chloro-1'-[(4-chlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H14Cl2N2O5
|
1
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| 1 |
Ki = 115 nM
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CP0390879
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2-[4-chloro-2-(2-pyridin-3-ylethynyl)phenoxy]acetic acid
Show/Hide
|
C15H10ClNO3
|
1
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| 1 |
Ki = 117 nM
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CP0418998
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2-[4-chloro-2-[2-[3-[methyl(methylsulfonyl)amino]phenyl]ethynyl]phenoxy]acetic acid
Show/Hide
|
C18H16ClNO5S
|
1
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| 1 |
Ki = 122 nM
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CP0416074
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N-(1,3-benzodioxol-5-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
|
C18H17N5O3
|
1
|
| 1 |
Ki = 130 nM
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CP0470512
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N-[(3-ethynylphenyl)methyl]-N-[2-fluoro-5-(2H-tetrazol-5-yl)phenyl]acetamide
Show/Hide
|
C18H14FN5O
|
1
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| 1 |
Ki = 140 nM
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CP0427743
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2-{5-chloro-1'-[(4-phenoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C26H19ClN2O6
|
1
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| 1 |
Ki = 143 nM
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CP0495934
|
2-[4-chloro-2-[2-(2-methylpyridin-3-yl)ethynyl]phenoxy]acetic acid
Show/Hide
|
C16H12ClNO3
|
1
|
| 1 |
Ki = 143 nM
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CP0447845
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2-[2-methyl-1-[[4-(trifluoromethyl)phenyl]methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C18H15F3N2O2
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1
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| 1 |
Ki = 145 nM
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CP0201721
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2-(4-chloro-2-cyclopentylphenoxy)acetic acid
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C13H15ClO3
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1
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| 1 |
Ki = 150 nM
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CP0315423
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2-(4-chloro-2-cyclohexylphenoxy)acetic acid
Show/Hide
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C14H17ClO3
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1
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| 1 |
Ki = 154 nM
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CP0422076
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2-{5-chloro-1'-[(3-fluoro-4-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C21H16ClFN2O6
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1
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| 1 |
Ki = 154 nM
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CP0427744
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2-{5-chloro-1'-[(3-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C21H17ClN2O6
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1
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| 1 |
Ki = 169 nM
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CP0427147
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2-[4-chloro-2-[2-(5-chlorothiophen-2-yl)ethynyl]phenoxy]acetic acid
Show/Hide
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C14H8Cl2O3S
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1
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| 1 |
Ki = 183 nM
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CP0467398
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2-[4-chloro-2-[2-(2-methoxyphenyl)ethynyl]phenoxy]acetic acid
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C17H13ClO4
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1
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| 1 |
Ki = 190 nM
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CP0427739
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2-(5-chloro-1'-{[5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione)acetic acid
Show/Hide
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C23H17ClN4O7
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1
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| 1 |
Ki = 212 nM
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CP0066157
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N-[3-(2H-tetrazol-5-yl)phenyl]-N-[[3-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
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C18H16F3N5O
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1
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| 1 |
Ki = 220 nM
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CP0415475
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N-[(4-methoxyphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C18H19N5O2
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1
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| 1 |
Ki = 220 nM
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CP0349972
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2-(4-cyano-2-cyclohexylphenoxy)acetic acid
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C15H17NO3
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1
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| 1 |
Ki = 230 nM
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CP0412552
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2-{5-chloro-1'-[(2-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C21H17ClN2O6
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1
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| 1 |
Ki = 233 nM
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CP0441090
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2-[2-[[4-chloro-2-(1,2-oxazol-5-yl)phenoxy]methyl]phenoxy]acetic acid
Show/Hide
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C18H14ClNO5
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1
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| 1 |
Ki = 247 nM
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CP0484563
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2-[4-chloro-2-[2-(2-fluoro-5-propylsulfonylphenyl)ethynyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C21H20ClFO5S
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1
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| 1 |
Ki = 260 nM
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CP0426682
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2-[(4S)-5'-chloro-1-[(5-chloro-2-fluorophenyl)methyl]-3-ethyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C21H16Cl2FN3O5
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1
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| 1 |
Ki = 260 nM
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CP0435022
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2-[5-chloro-1'-(2-phenylethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C21H17ClN2O5
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1
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| 1 |
Ki = 267 nM
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CP0554499
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2-[1-[(3-chlorophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C17H15ClN2O2
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1
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| 1 |
Ki = 270 nM
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CP0471155
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2-[1-[(3,4-difluorophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C17H14F2N2O2
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1
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| 1 |
Ki = 278 nM
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CP0462755
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2-[5'-chloro-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C22H21ClN4O6
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1
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| 1 |
Ki = 280 nM
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CP0524692
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2-(2-methyl-1-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C16H14N2O4S
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1
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| 1 |
Ki = 282 nM
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CP0533191
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2-[2-[2-(2-chlorophenyl)ethynyl]-4-methylphenoxy]acetic acid
Show/Hide
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C17H13ClO3
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1
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| 1 |
Ki = 283 nM
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CP0400686
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2-[4-chloro-2-[2-[5-[3-(dimethylamino)propyl-methylsulfamoyl]-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C23H27ClN2O5S
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1
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| 1 |
Ki = 287 nM
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CP0520266
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2-[4-chloro-2-[2-[5-(2-hydroxyethylsulfamoyl)pyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H15ClN2O6S
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1
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| 1 |
Ki = 301 nM
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CP0507927
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2-[(3S)-5-chloro-1'-[(5-chloro-2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C20H13Cl2FN2O5
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1
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| 1 |
Ki = 302 nM
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CP0519728
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2-[2-methyl-1-[(4-methylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C18H18N2O2
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1
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| 1 |
Ki = 302 nM
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CP0157437
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2-(2-cyclohexylphenoxy)acetic acid
Show/Hide
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C14H18O3
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1
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| 1 |
Ki = 311 nM
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CP0435019
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2-[5-chloro-1'-(furan-3-ylmethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C18H13ClN2O6
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1
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| 1 |
Ki = 318 nM
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CP0517468
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N-(isoquinolin-6-ylmethyl)-N-[3-(2H-tetrazol-5-yl)phenyl]pentanamide
Show/Hide
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C22H22N6O
|
1
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| 1 |
Ki = 330 nM
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CP0542586
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2-[2-methyl-6-[[2-(propylcarbamoyl)phenoxy]methyl]phenoxy]acetic acid
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C20H23NO5
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1
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| 1 |
Ki = 333 nM
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CP0315424
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2-(2-cyclohexyl-4-methylphenoxy)acetic acid
Show/Hide
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C15H20O3
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1
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| 1 |
Ki = 353 nM
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CP0394565
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2-[5-chloro-1'-(1-phenylethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C21H17ClN2O5
|
1
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| 1 |
Ki = 356 nM
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CP0406725
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2-[4-chloro-2-methyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C18H17ClN2O4S
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1
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| 1 |
Ki = 356 nM
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CP0410378
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N-[(3-methoxyphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C18H19N5O2
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1
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| 1 |
Ki = 360 nM
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CP0495935
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2-[4-chloro-2-[2-[5-[2-(dimethylamino)ethyl-methylsulfamoyl]-2-methylphenyl]ethynyl]phenoxy]acetic acid
Show/Hide
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C22H25ClN2O5S
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1
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| 1 |
Ki = 369 nM
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CP0497381
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2-(1-(3-chlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C16H13ClN2O4S
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1
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| 1 |
Ki = 377 nM
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CP0459324
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2-[4-chloro-2-[2-[5-[methyl(methylsulfonyl)amino]pyridin-3-yl]ethynyl]phenoxy]acetic acid
Show/Hide
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C17H15ClN2O5S
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1
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| 1 |
Ki = 378 nM
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CP0549623
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2-[5'-chloro-1-[(2-fluorophenyl)methyl]-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C19H13ClFN3O5
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1
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| 1 |
Ki = 390 nM
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CP0549718
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2-[5'-chloro-1-[(2,5-difluorophenyl)methyl]-3-methyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C20H14ClF2N3O5
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1
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| 1 |
Ki = 390 nM
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CP0427737
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2-[5-chloro-1'-(1,3-oxazol-2-ylmethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C17H12ClN3O6
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1
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| 1 |
Ki = 438 nM
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CP0467222
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2-(2-cyclohexyl-4-fluorophenoxy)acetic acid
Show/Hide
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C14H17FO3
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1
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| 1 |
Ki = 446 nM
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CP0460790
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2-[5'-chloro-3-methyl-2,2',5-trioxo-1-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]spiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C20H19ClN4O5S
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1
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| 1 |
Ki = 490 nM
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CP0416361
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2-[2-[(2-methylquinolin-8-yl)oxymethyl]phenoxy]acetic acid
Show/Hide
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C19H17NO4
|
1
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| 1 |
Ki = 492 nM
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CP0505202
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2-{5-chloro-1'-[(5-cyclopropyl-1,3,4-thiadiazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C19H15ClN4O5S
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1
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| 1 |
Ki = 497 nM
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CP0379871
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2-[1-[(4-methoxyphenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C18H18N2O3
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1
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| 1 |
Ki = 504 nM
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CP0499400
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2-[4-chloro-2-[2-(2-methyl-5-propylsulfonylphenyl)ethynyl]phenoxy]-4-methylpentanoic acid
Show/Hide
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C24H27ClO5S
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1
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| 1 |
Ki = 515 nM
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CP0416363
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2-[2-[(5-chloro-2-methylphenoxy)methyl]phenoxy]acetic acid
Show/Hide
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C16H15ClO4
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1
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| 1 |
Ki = 520 nM
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CP0494063
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2-[1-[(3-bromophenyl)methyl]-3,5-diethylpyrazol-4-yl]acetic acid
Show/Hide
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C16H19BrN2O2
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1
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| 1 |
Ki = 563 nM
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CP0549230
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2-[3,5-diethyl-1-(naphthalen-2-ylmethyl)pyrazol-4-yl]acetic acid
Show/Hide
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C20H22N2O2
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1
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| 1 |
Ki = 574 nM
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CP0432884
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N-[(3-methylphenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C18H19N5O
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1
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| 1 |
Ki = 580 nM
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CP0541839
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2-(1-benzyl-2-methylpyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C17H16N2O2
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1
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| 1 |
Ki = 588 nM
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CP0525264
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2-[2-[(2-cyclopropyl-4-fluorophenoxy)methyl]phenoxy]acetic acid
Show/Hide
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C18H17FO4
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1
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| 1 |
Ki = 591 nM
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CP0529887
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2-[5-chloro-1'-(1H-indol-3-ylmethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C22H16ClN3O5
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1
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| 1 |
Ki = 596 nM
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CP0418993
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2-[4-chloro-2-(2-pyridin-4-ylethynyl)phenoxy]acetic acid
Show/Hide
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C15H10ClNO3
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1
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| 1 |
Ki = 601 nM
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CP0498415
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2-(2-methyl-1-tosyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C17H16N2O4S
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1
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| 1 |
Ki = 619 nM
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CP0470513
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N-[3-(2H-tetrazol-5-yl)phenyl]-N-(thiophen-2-ylmethyl)pentanamide
Show/Hide
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C17H19N5OS
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1
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| 1 |
Ki = 620 nM
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CP0515588
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2-[1-[(2,5-dichlorophenyl)methyl]-3,5-diethylpyrazol-4-yl]acetic acid
Show/Hide
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C16H18Cl2N2O2
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1
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| 1 |
Ki = 623 nM
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CP0540767
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2-[1-[(2-chlorophenyl)methyl]-2-methylpyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C17H15ClN2O2
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1
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| 1 |
Ki = 624 nM
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CP0416365
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2-[3,5-diethyl-4-(naphthalen-2-ylmethyl)pyrazol-1-yl]acetic acid
Show/Hide
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C20H22N2O2
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1
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| 1 |
Ki = 631 nM
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CP0485751
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2-{1'-benzyl-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,5'-dione}acetic acid
Show/Hide
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C20H17ClN2O4
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1
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| 1 |
Ki = 702 nM
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CP0478160
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2-{1'-benzyl-5-fluoro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C20H15FN2O5
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1
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| 1 |
Ki = 712 nM
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CP0090560
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2-[5-bromo-2-methyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C18H17BrN2O4S
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1
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| 1 |
Ki = 735 nM
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CP0403126
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2-{5-chloro-1'-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C22H17ClN2O5
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1
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| 1 |
Ki = 747 nM
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CP0456494
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2-[2-[2-(2-chlorophenyl)ethynyl]phenoxy]acetic acid
Show/Hide
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C16H11ClO3
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1
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| 1 |
Ki = 747 nM
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CP0424661
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2-[1-(1,3-benzothiazol-2-ylmethyl)-5'-chloro-3-methyl-2,2',5-trioxospiro[imidazolidine-4,3'-indole]-1'-yl]acetic acid
Show/Hide
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C21H15ClN4O5S
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1
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| 1 |
Ki = 750 nM
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CP0525265
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2-[5-(2-phenyl-1,3-thiazole-4-carbonyl)-6,7-dihydro-4H-imidazo[4,5-c]pyridin-1-yl]acetic acid
Show/Hide
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C18H16N4O3S
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1
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| 1 |
Ki = 752 nM
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CP0435028
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4-[5-chloro-1'-(prop-2-en-1-yl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]butanoic acid
Show/Hide
|
C18H17ClN2O5
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1
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| 1 |
Ki = 769 nM
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CP0321150
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2-(2-cyclohexyl-4-methoxyphenoxy)acetic acid
Show/Hide
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C15H20O4
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1
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| 1 |
Ki = 782 nM
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CP0371641
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3-(4-chloro-2-cyclohexylphenoxy)propanoic acid
Show/Hide
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C15H19ClO3
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1
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| 1 |
Ki = 799 nM
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CP0434995
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2-[(3S)-5-chloro-1'-[(3-chlorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C20H14Cl2N2O5
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1
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| 1 |
Ki = 870 nM
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CP0500618
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2-[(3S)-5-chloro-1'-[(2-fluorophenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
|
C20H14ClFN2O5
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1
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| 1 |
Ki = 926 nM
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CP0517469
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N-[(2-fluorophenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C17H16FN5O
|
1
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| 1 |
Ki = 950 nM
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CP0436483
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4-{5-chloro-1'-[(4-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
Show/Hide
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C23H21ClN2O6
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1
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| 1 |
Ki = 960 nM
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CP0500996
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2-[2-methyl-1-(pyridin-3-ylmethyl)pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C16H15N3O2
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1
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| 1 |
Ki = 1060 nM
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CP0388114
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2-[4-chloro-2-(2-pyridin-2-ylethynyl)phenoxy]acetic acid
Show/Hide
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C15H10ClNO3
|
1
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| 1 |
Ki = 1120 nM
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CP0506217
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2-(1-(4-chloro-3-(trifluoromethyl)phenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
|
C17H12ClF3N2O4S
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1
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| 1 |
Ki = 1171 nM
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CP0536780
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2-[(3S)-5-chloro-1'-[(3-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C21H17ClN2O6
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1
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| 1 |
Ki = 1172 nM
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CP0432883
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N-[(4-fluorophenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
|
C17H16FN5O
|
1
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| 1 |
Ki = 1200 nM
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CP0422075
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2-{5-chloro-1'-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C21H16ClN5O5
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1
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| 1 |
Ki = 1300 nM
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CP0242029
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2-[2,5-dimethyl-1-[(4-methylsulfonylphenyl)methyl]pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
|
C19H20N2O4S
|
1
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| 1 |
Ki = 1335 nM
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CP0427738
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2-{1'-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
|
C20H19ClN4O6
|
1
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| 1 |
Ki = 1338 nM
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CP0432882
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N-[(3-fluorophenyl)methyl]-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
Show/Hide
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C17H16FN5O
|
1
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| 1 |
Ki = 1400 nM
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CP0436485
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2-[5-chloro-1'-(2-methoxyethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
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C16H15ClN2O6
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1
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| 1 |
Ki = 1448 nM
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CP0505966
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2-[4-chloro-2-[2-(1-methylimidazol-2-yl)ethynyl]phenoxy]acetic acid
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C14H11ClN2O3
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1
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| 1 |
Ki = 1470 nM
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CP0435021
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2-{5-chloro-1'-[(4-methanesulfonylphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
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C21H17ClN2O7S
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1
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| 1 |
Ki = 1506 nM
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CP0536835
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1'-benzyl-5-chloro-1-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione
Show/Hide
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C20H15ClN6O3
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1
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| 1 |
Ki = 1536 nM
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CP0536836
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4-{1'-benzyl-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
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C22H19ClN2O5
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1
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| 1 |
Ki = 1660 nM
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CP0435910
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N-benzyl-N-[3-(2H-tetrazol-5-yl)phenyl]propanamide
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C17H17N5O
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1
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| 1 |
Ki = 1800 nM
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CP0288742
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4-(4-chloro-2-cyclohexylphenoxy)butanoic acid
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C16H21ClO3
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1
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| 1 |
Ki = 1990 nM
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CP0536781
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2-[(3S)-1'-benzyl-5-chloro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]acetic acid
Show/Hide
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C20H15ClN2O5
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1
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| 1 |
Ki = 2044 nM
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CP0513854
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2-{5-chloro-1'-[(5-methyl-3-phenyl-1,2-oxazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2'-dione}acetic acid
Show/Hide
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C24H20ClN3O5
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2
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| 1 |
Ki = 2200 nM
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| 2 |
Ki = 2237 nM
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CP0490097
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2-[2-methyl-1-(pyridin-4-ylmethyl)pyrrolo[2,3-b]pyridin-3-yl]acetic acid
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C16H15N3O2
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1
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| 1 |
Ki = 2230 nM
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CP0216457
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(R)-2-(4-chloro-2-cyclohexylphenoxy)propanoic acid
Show/Hide
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C15H19ClO3
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1
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| 1 |
Ki = 2250 nM
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CP0439275
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2-(1-(4-methoxyphenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C17H16N2O5S
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1
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| 1 |
Ki = 2619 nM
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CP0516327
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2-{1'-benzyl-5-methoxy-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C21H18N2O6
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1
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| 1 |
Ki = 2741 nM
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CP0490096
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2-[2-methyl-1-(pyridin-2-ylmethyl)pyrrolo[2,3-b]pyridin-3-yl]acetic acid
Show/Hide
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C16H15N3O2
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1
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| 1 |
Ki = 2940 nM
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CP0497382
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2-(1-(2-chlorophenylsulfonyl)-2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetic acid
Show/Hide
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C16H13ClN2O4S
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1
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| 1 |
Ki = 3220 nM
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CP0194852
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methyl 2-(4-chloro-2-cyclohexylphenoxy)acetate
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C15H19ClO3
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1
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| 1 |
Ki = 3280 nM
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CP0000254
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(Z)-2-(3-(4-(methylthio)benzylidene)-6-fluoro-2-methyl-3H-inden-1-yl)acetic acid
Show/Hide
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C20H17FO2S
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1
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| 1 |
Ki = 3500 nM
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CP0394202
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2-{5-fluoro-1'-[(2-methoxyethoxy)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C17H17FN2O7
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1
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| 1 |
Ki = 3829 nM
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CP0478156
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4-[5-fluoro-1'-(prop-2-en-1-yl)-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione]butanoic acid
Show/Hide
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C18H17FN2O5
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1
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| 1 |
Ki = 4131 nM
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CP0407993
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4-{1'-benzyl-5-fluoro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
Show/Hide
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C22H19FN2O5
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1
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| 1 |
Ki = 4174 nM
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CP0435992
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2-[3-[2,3-dihydro-1,4-benzodioxin-6-ylmethyl(pentanoyl)amino]phenyl]acetic acid
Show/Hide
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C22H25NO5
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1
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| 1 |
Ki = 4300 nM
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CP0373103
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2-{5-chloro-1'-[(dimethylcarbamoyl)methyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C17H16ClN3O6
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1
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| 1 |
Ki = 4669 nM
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CP0459325
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2-[2-[2-(2-chlorophenyl)ethynyl]-5-fluorophenoxy]acetic acid
Show/Hide
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C16H10ClFO3
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1
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| 1 |
Ki = 4780 nM
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CP0136016
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2-(2-allyl-4-chlorophenoxy)acetic acid
Show/Hide
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C11H11ClO3
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1
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| 1 |
Ki = 5130 nM
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CP0435026
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2-{5-chloro-1'-methyl-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C14H11ClN2O5
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1
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| 1 |
Ki = 7615 nM
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CP0432886
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3-[(3-methoxyphenyl)methyl-pentanoylamino]benzoic acid
Show/Hide
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C20H23NO4
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1
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| 1 |
Ki = 8000 nM
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CP0373100
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4-{5-fluoro-1'-methyl-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}butanoic acid
Show/Hide
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C16H15FN2O5
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1
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| 1 |
Ki = 8903 nM
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CP0094725
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((4-chloro-o-tolyl)oxy)acetic acid,
Show/Hide
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C9H9ClO3
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1
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| 1 |
Ki > 10000 nM
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CP0221441
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2-(4-chloro-2-cyclohexylphenoxy)-N-(methylsulfonyl)acetamide
Show/Hide
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C15H20ClNO4S
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1
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| 1 |
Ki > 10000 nM
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CP0307487
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2-(4-chloro-2-cyclohexylphenoxy)ethanol
Show/Hide
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C14H19ClO2
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1
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| 1 |
Ki > 10000 nM
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CP0315425
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5-((4-chloro-2-cyclohexylphenoxy)methyl)-1H-tetrazole
Show/Hide
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C14H17ClN4O
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1
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| 1 |
Ki > 10000 nM
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CP0407997
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1'-benzyl-5-chloro-1-methyl-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione
Show/Hide
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C19H15ClN2O3
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1
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| 1 |
Ki = 11629 nM
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CP0435030
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Spiro-indolinone analogue, 51
Show/Hide
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C22H19ClN2O5
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1
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| 1 |
Ki > 30000 nM
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CP0529891
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2-{1'-[(dimethylcarbamoyl)methyl]-5-fluoro-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2,2',5'-trione}acetic acid
Show/Hide
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C17H16FN3O6
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1
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| 1 |
Ki > 30000 nM
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