| Compound ID |
Compound Name |
Compound Formula |
|
CP0135429
|
(4R)-2-amino-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
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|
C25H28N4O2S
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0424777
|
(S)-6-(4-(2-(3-(3-(2-cyclopropylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
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|
C31H37N5O5
|
1
|
| 1 |
EC50 = 6.8 nM
|
|
|
|
CP0437372
|
(S)-6-(4-(2-(2-hydroxy-3-(3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
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|
C27H31N5O5
|
1
|
| 1 |
EC50 = 24.5 nM
|
|
|
|
CP0135426
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
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|
C24H26N4O2S
|
1
|
| 1 |
EC50 = 27.6 nM
|
|
|
|
CP0409669
|
(S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
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|
C32H39N5O5
|
1
|
| 1 |
EC50 = 28.7 nM
|
|
|
|
CP0105650
|
KRP-114V
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|
C26H28N4O3
|
2
|
| 1 |
EC50 = 86 nM
|
|
|
| 2 |
EC50 = 122 nM
|
|
|
|
CP0156745
|
(2S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)propanamide
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|
C25H28N4O3
|
2
|
| 1 |
EC50 = 245 nM
|
|
|
| 2 |
EC50 = 531 nM
|
|
|
|
CP0105651
|
(6S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide
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|
C24H27N5O2
|
1
|
| 1 |
EC50 = 434 nM
|
|
|
|
CP0105652
|
N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)acetamide
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|
C24H26N4O3
|
2
|
| 1 |
EC50 = 615 nM
|
|
|
| 2 |
EC50 = 1064 nM
|
|
|
|
CP0156740
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-(4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)benzenesulfonamide
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|
C31H27F3N4O3S2
|
1
|
| 1 |
EC50 = 3400 nM
|
|
|
