| Compound ID |
Compound Name |
Compound Formula |
|
CP0414285
|
6-bromo-8-[(3-fluoro-4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H11BrFNO6
|
2
|
| 1 |
EC50 = 4.37 nM
|
|
|
| 2 |
Ki = 1.64 nM
|
|
|
|
CP0389123
|
6-bromo-8-[(2-fluoro-4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H11BrFNO6
|
2
|
| 1 |
EC50 = 4.45 nM
|
|
|
| 2 |
Ki = 1.37 nM
|
|
|
|
CP0379959
|
6-bromo-8-[(2,6-difluoro-4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H10BrF2NO6
|
2
|
| 1 |
EC50 = 5.54 nM
|
|
|
| 2 |
Ki = 0.589 nM
|
|
|
|
CP0379961
|
6-chloro-8-[(2-fluoro-4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H11ClFNO6
|
2
|
| 1 |
EC50 = 6.06 nM
|
|
|
| 2 |
Ki = 1.92 nM
|
|
|
|
CP0395599
|
6-bromo-8-[(2-chloro-4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H11BrClNO6
|
3
|
| 1 |
EC50 = 11.1 nM
|
|
|
| 2 |
EC50 = 14.7 nM
|
|
|
| 3 |
Ki = 1.12 nM
|
|
|
|
CP0380136
|
6-bromo-8-[(2,4-dichlorobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H8BrCl2NO5
|
3
|
| 1 |
EC50 = 16.4 nM
|
|
|
| 2 |
EC50 = 34.6 nM
|
|
|
| 3 |
Ki = 0.938 nM
|
|
|
|
CP0397174
|
6-chloro-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12ClNO6
|
3
|
| 1 |
EC50 = 16.8 nM
|
|
|
| 2 |
EC50 = 28.6 nM
|
|
|
| 3 |
Ki = 5.5 nM
|
|
|
|
CP0395591
|
8-[(2,4-dichlorobenzoyl)amino]-6-fluoro-4-oxochromene-2-carboxylic acid
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|
C17H8Cl2FNO5
|
2
|
| 1 |
EC50 = 20.5 nM
|
|
|
| 2 |
Ki = 4.12 nM
|
|
|
|
CP0389119
|
6-bromo-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12BrNO6
|
2
|
| 1 |
EC50 = 22.1 nM
|
|
|
| 2 |
Ki = 5.18 nM
|
|
|
|
CP0395598
|
6-bromo-8-[(4-chlorobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H9BrClNO5
|
3
|
| 1 |
EC50 = 25.1 nM
|
|
|
| 2 |
EC50 = 40.5 nM
|
|
|
| 3 |
Ki = 4.79 nM
|
|
|
|
CP0395586
|
6-bromo-8-[(3,4-dichlorobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H8BrCl2NO5
|
3
|
| 1 |
EC50 = 25.1 nM
|
|
|
| 2 |
EC50 = 27.2 nM
|
|
|
| 3 |
Ki = 2.18 nM
|
|
|
|
CP0413804
|
6-methoxy-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C19H15NO7
|
2
|
| 1 |
EC50 = 25.5 nM
|
|
|
| 2 |
Ki = 20.5 nM
|
|
|
|
CP0505056
|
8-[(4-methoxybenzoyl)amino]-6-methyl-4-oxochromene-2-carboxylic acid
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|
C19H15NO6
|
2
|
| 1 |
EC50 = 37.7 nM
|
|
|
| 2 |
Ki = 42.8 nM
|
|
|
|
CP0285587
|
2-[2-[4-[(4-chlorophenyl)-phenyl-methyl]piperazino]ethoxy]ethanol
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|
C23H16O6
|
3
|
| 1 |
EC50 = 50 nM
|
|
|
| 2 |
EC50 = 1200 nM
|
|
|
| 3 |
Ki = 11.5 nM
|
|
|
|
CP0381004
|
8-(1,3-benzodioxole-5-carbonylamino)-6-bromo-4-oxochromene-2-carboxylic acid
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|
C18H10BrNO7
|
3
|
| 1 |
EC50 = 59.9 nM
|
|
|
| 2 |
EC50 = 128 nM
|
|
|
| 3 |
Ki = 15 nM
|
|
|
|
CP0380130
|
8-[(3,4-dichlorobenzoyl)amino]-6-fluoro-4-oxochromene-2-carboxylic acid
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|
C17H8Cl2FNO5
|
3
|
| 1 |
EC50 = 106 nM
|
|
|
| 2 |
EC50 = 117 nM
|
|
|
| 3 |
Ki = 11.5 nM
|
|
|
|
CP0380113
|
ethyl 6-fluoro-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylate
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|
C20H16FNO6
|
2
|
| 1 |
EC50 = 112 nM
|
|
|
| 2 |
Ki = 198 nM
|
|
|
|
CP0395601
|
6-fluoro-8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12FNO6
|
3
|
| 1 |
EC50 = 112 nM
|
|
|
| 2 |
EC50 = 143 nM
|
|
|
| 3 |
Ki = 25.4 nM
|
|
|
|
CP0380115
|
6-bromo-8-[(5-methoxypyridine-2-carbonyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H11BrN2O6
|
2
|
| 1 |
EC50 = 144 nM
|
|
|
| 2 |
Ki = 56.8 nM
|
|
|
|
CP0404055
|
8-benzamido-6-bromo-4-oxochromene-2-carboxylic acid
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|
C17H10BrNO5
|
2
|
| 1 |
EC50 = 303 nM
|
|
|
| 2 |
Ki = 81.6 nM
|
|
|
|
CP0395595
|
8-[(4-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H13NO6
|
3
|
| 1 |
EC50 = 346 nM
|
|
|
| 2 |
EC50 = 472 nM
|
|
|
| 3 |
Ki = 221 nM
|
|
|
|
CP0378851
|
2-[4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]phenoxy]acetic acid
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|
C12H9NO5S
|
2
|
| 1 |
EC50 = 349 nM
|
|
|
| 2 |
Ki = 50.8 nM
|
|
|
|
CP0395588
|
8-[(2,3-dichlorobenzoyl)amino]-6-fluoro-4-oxochromene-2-carboxylic acid
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|
C17H8Cl2FNO5
|
3
|
| 1 |
EC50 = 382 nM
|
|
|
| 2 |
EC50 = 873 nM
|
|
|
| 3 |
Ki = 119 nM
|
|
|
|
CP0395733
|
6-bromo-8-[(4-cyanobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H9BrN2O5
|
2
|
| 1 |
EC50 = 399 nM
|
|
|
| 2 |
Ki = 148 nM
|
|
|
|
CP0389127
|
8-benzamido-6-chloro-4-oxochromene-2-carboxylic acid
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|
C17H10ClNO5
|
2
|
| 1 |
EC50 = 430 nM
|
|
|
| 2 |
Ki = 138 nM
|
|
|
|
CP0389124
|
6-bromo-8-[(3,4-dimethoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C19H14BrNO7
|
2
|
| 1 |
EC50 = 628 nM
|
|
|
| 2 |
Ki = 228 nM
|
|
|
|
CP0380116
|
6-bromo-8-[(4-ethoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C19H14BrNO6
|
2
|
| 1 |
EC50 = 634 nM
|
|
|
| 2 |
Ki = 98.4 nM
|
|
|
|
CP0378849
|
8-[(4-bromobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H10BrNO5
|
3
|
| 1 |
EC50 = 678 nM
|
|
|
| 2 |
EC50 = 804 nM
|
|
|
| 3 |
Ki = 233 nM
|
|
|
|
CP0395590
|
6-bromo-8-[(3-methylbenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12BrNO5
|
3
|
| 1 |
EC50 = 699 nM
|
|
|
| 2 |
EC50 = 842 nM
|
|
|
| 3 |
Ki = 128 nM
|
|
|
|
CP0380137
|
6-chloro-8-[(3-methylbenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12ClNO5
|
2
|
| 1 |
EC50 = 1220 nM
|
|
|
| 2 |
Ki = 250 nM
|
|
|
|
CP0748604
|
5-[3-(2-carboxy-4-oxo-4H-5-chromenyloxy)-2-hydroxypropoxy]-4-oxo-4H-2-chromenecarboxylic acid (sodium) (disodium cromoglycate)
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|
C23H14Na2O11
|
1
|
| 1 |
EC50 = 1260 nM
|
|
|
|
CP0397194
|
4-oxo-8-(quinoline-2-carbonylamino)chromene-2-carboxylic acid
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|
C20H12N2O5
|
2
|
| 1 |
EC50 = 1340 nM
|
|
|
| 2 |
Ki = 691 nM
|
|
|
|
CP0395602
|
8-[(4-methylbenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H13NO5
|
2
|
| 1 |
EC50 = 1380 nM
|
|
|
| 2 |
Ki = 697 nM
|
|
|
|
CP0395600
|
6-chloro-8-[(4-nitrobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H9ClN2O7
|
2
|
| 1 |
EC50 = 1710 nM
|
|
|
| 2 |
Ki = 183 nM
|
|
|
|
CP0037172
|
3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0]nona-1,3,6-trien-5-one
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|
C13H13N5O2
|
3
|
| 1 |
EC50 = 1960 nM
|
|
|
| 2 |
EC50 = 2240 nM
|
|
|
| 3 |
Ki = 401 nM
|
|
|
|
CP0395587
|
8-(cyclohexanecarbonylamino)-4-oxochromene-2-carboxylic acid
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|
C17H17NO5
|
2
|
| 1 |
EC50 = 4200 nM
|
|
|
| 2 |
Ki = 3580 nM
|
|
|
|
CP0381006
|
8-(naphthalene-2-carbonylamino)-4-oxochromene-2-carboxylic acid
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|
C21H13NO5
|
2
|
| 1 |
EC50 = 4670 nM
|
|
|
| 2 |
Ki = 714 nM
|
|
|
|
CP0397173
|
8-benzamido-4-oxochromene-2-carboxylic acid
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|
C17H11NO5
|
2
|
| 1 |
EC50 = 4910 nM
|
|
|
| 2 |
Ki = 3290 nM
|
|
|
|
CP0397175
|
8-[(3-methylbenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H13NO5
|
2
|
| 1 |
EC50 = 5440 nM
|
|
|
| 2 |
Ki = 4780 nM
|
|
|
|
CP0381000
|
8-[(3-nitrobenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H10N2O7
|
2
|
| 1 |
EC50 = 6970 nM
|
|
|
| 2 |
Ki = 4390 nM
|
|
|
|
CP0395596
|
4-oxo-8-[(2-phenylacetyl)amino]chromene-2-carboxylic acid
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|
C18H13NO5
|
2
|
| 1 |
EC50 = 8960 nM
|
|
|
| 2 |
Ki = 2720 nM
|
|
|
|
CP0070834
|
3,3''''-methylenebis(4-hydroxy-coumarin
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|
C19H12O6
|
2
|
| 1 |
EC50 = 9780 nM
|
|
|
| 2 |
Ki = 39 nM
|
|
|
|
CP0066118
|
4-chloro-2-[(furan-2-ylmethyl)amino]-5-sulfamoylbenzoic acid
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|
C12H11ClN2O5S
|
2
|
| 1 |
EC50 = 11200 nM
|
|
|
| 2 |
Ki = 3270 nM
|
|
|
|
CP0395597
|
8-amino-6-bromo-4-oxochromene-2-carboxylic acid
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|
C10H6BrNO4
|
2
|
| 1 |
EC50 = 12600 nM
|
|
|
| 2 |
Ki = 3010 nM
|
|
|
|
CP0380135
|
4-oxo-8-(propanoylamino)chromene-2-carboxylic acid
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|
C13H11NO5
|
2
|
| 1 |
EC50 = 13400 nM
|
|
|
| 2 |
Ki = 6770 nM
|
|
|
|
CP0395589
|
4-oxo-8-[[4-(trifluoromethyl)benzoyl]amino]chromene-2-carboxylic acid
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|
C18H10F3NO5
|
2
|
| 1 |
EC50 = 15500 nM
|
|
|
| 2 |
Ki = 10300 nM
|
|
|
|
CP0374969
|
8-[(3-methoxy-3-oxopropanoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C14H11NO7
|
2
|
| 1 |
EC50 = 20200 nM
|
|
|
| 2 |
Ki = 18600 nM
|
|
|
|
CP0378850
|
8-acetamido-4-oxochromene-2-carboxylic acid
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|
C12H9NO5
|
2
|
| 1 |
EC50 = 24100 nM
|
|
|
| 2 |
Ki = 18500 nM
|
|
|
|
CP0084320
|
CAS_4394-00-7
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|
C13H9F3N2O2
|
2
|
| 1 |
EC50 = 30800 nM
|
|
|
| 2 |
Ki = 3610 nM
|
|
|
|
CP0049039
|
4-hydroxyquinoline-2-carboxylic acid
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|
C10H7NO3
|
1
|
| 1 |
EC50 = 39200 nM
|
|
|
|
CP0380101
|
8-nitro-4-oxochromene-2-carboxylic acid
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|
C10H5NO6
|
2
|
| 1 |
EC50 = 46300 nM
|
|
|
| 2 |
Ki = 13600 nM
|
|
|
|
CP0208524
|
2-hydroxy-4-({4-[5-(2-methyl-3-phenyl-2-propen-1-ylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]butanoyl}amino)benzoic acid
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|
C24H22N2O5S2
|
2
|
| 1 |
IC50 = 522 nM
|
|
|
| 2 |
Ki = 8.76 nM
|
|
|
|
CP0856570
|
SID99309109
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|
C17H19F2N5O2S
|
2
|
| 1 |
IC50 = 574 nM
|
|
|
| 2 |
Ki = 42.2 nM
|
|
|
|
CP0868920
|
6-Bromo-8-(4-[3H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic acid
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|
C18H12BrNO6
|
4
|
| 1 |
Kd = 5.27 nM
|
|
|
| 2 |
Kd = 5.65 nM
|
|
|
| 3 |
Kd = 5.92 nM
|
|
|
| 4 |
Kd = 115 nM
|
|
|
|
CP0381005
|
6-bromo-8-[(6-methoxypyridine-3-carbonyl)amino]-4-oxochromene-2-carboxylic acid
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|
C17H11BrN2O6
|
1
|
| 1 |
Ki = 25.7 nM
|
|
|
|
CP0397163
|
6-bromo-8-[(2-methoxybenzoyl)amino]-4-oxochromene-2-carboxylic acid
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|
C18H12BrNO6
|
1
|
| 1 |
Ki = 331 nM
|
|
|
|
CP0382598
|
2-[3-cyano-5-(3,4-dichlorophenyl)-4,5-dimethylfuran-2-ylidene]propanedinitrile
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|
C16H9Cl2N3O
|
1
|
| 1 |
Ki = 655 nM
|
|
|
|
CP0082759
|
CROMOLYN
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|
C23H16O11
|
1
|
| 1 |
Ki = 2340 nM
|
|
|
|
CP0411386
|
8-[[4-(cyclopropylmethoxy)benzoyl]amino]-4-oxochromene-2-carboxylic acid
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|
C21H17NO6
|
1
|
| 1 |
Ki = 3710 nM
|
|
|
|
CP0381003
|
4-oxo-8-[(4-propoxybenzoyl)amino]chromene-2-carboxylic acid
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|
C20H17NO6
|
1
|
| 1 |
Ki = 8060 nM
|
|
|
|
CP0033053
|
(4S)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acid
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|
C11H8N2O3S2
|
1
|
| 1 |
Ki = 9860 nM
|
|
|
