Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01008 , Macrophage colony-stimulating factor 1 receptor
Gene Name CSF1R
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P07333
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01008
 
Compound ID Compound Name Compound Formula
CP0002778
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide
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C29H31N7O
 1
1
IC50 = 960 nM
   TI
   LI
   LO
   TS
CP0115223
4-[6-Methoxy-7-(3-morpholin-4-yl-propoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide
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C30H40N6O5
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0034949
4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-yl]-N-(4-propan-2-yloxyphenyl)piperazine-1-carboxamide
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C31H42N6O4
 1
1
IC50 = 3430 nM
   TI
   LI
   LO
   TS
CP0406454
4-[6-Methoxy-7-(2-piperidin-1-yl-ethoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide
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C30H40N6O4
 1
1
IC50 = 3430 nM
   TI
   LI
   LO
   TS
CP0377709
4-[6-Methoxy-7-(2-methoxy-ethoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide
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C26H33N5O5
 1
1
IC50 = 5460 nM
   TI
   LI
   LO
   TS