| Compound ID |
Compound Name |
Compound Formula |
|
CP0388123
|
6-fluoro-5-methyl-3-[1-(1-methyl-4-propoxycyclohexyl)piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C23H34FN3O2
|
1
|
| 1 |
EC50 = 12.59 nM
|
|
|
|
CP0000324
|
2-acetoxyethyl(trimethyl)ammonium;bromide
Show/Hide
|
C7H16NO2+
|
2
|
| 1 |
EC50 = 19.1 nM
|
|
|
| 2 |
Ki = 9772.37 nM
|
|
|
|
CP0372671
|
6-methyl-1-[1-(1-methyl-4-propoxycyclohexyl)piperidin-4-yl]-3H-indol-2-one
Show/Hide
|
C24H36N2O2
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0416347
|
CHEMBL1223804
Show/Hide
|
C23H34N2O2
|
1
|
| 1 |
EC50 = 19.95 nM
|
|
|
|
CP0388126
|
3-[1-(4-ethoxy-1-methylcyclohexyl)piperidin-4-yl]-6-fluoro-5-methyl-1,3-benzoxazol-2-one
Show/Hide
|
C22H31FN2O3
|
1
|
| 1 |
EC50 = 50.12 nM
|
|
|
|
CP0049755
|
(R)-1-Aza-bicyclo[2.2.2]oct-3-yl-[(Z)-methoxyimino]-acetonitrile
Show/Hide
|
C10H15N3O
|
1
|
| 1 |
EC50 = 123 nM
|
|
|
|
CP0372673
|
CHEMBL1223805
Show/Hide
|
C22H32N2O2
|
1
|
| 1 |
EC50 = 125.89 nM
|
|
|
|
CP0371787
|
5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine; oxalic acid
Show/Hide
|
C14H23N3OS
|
3
|
| 1 |
EC50 = 142 nM
|
|
|
| 2 |
Ki = 9.333 nM
|
|
|
| 3 |
Ki = 15.14 nM
|
|
|
|
CP0372675
|
CHEMBL1223861
Show/Hide
|
C22H31FN2O3
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
|
CP0372676
|
CHEMBL1223862
Show/Hide
|
C22H32N2O4
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
|
CP0406096
|
CHEMBL1223940
Show/Hide
|
C23H34N2O4
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
|
CP0514870
|
CHEMBL1223939
Show/Hide
|
C23H34N2O5S
|
1
|
| 1 |
EC50 = 316.23 nM
|
|
|
|
CP0374543
|
3-[1-(4-ethoxy-1-methylcyclohexyl)piperidin-4-yl]-2-oxo-1,3-benzoxazole-5-carbonitrile
Show/Hide
|
C22H29N3O3
|
1
|
| 1 |
EC50 = 398.11 nM
|
|
|
|
CP0388124
|
3-[1-(4-methoxy-1-methylcyclohexyl)piperidin-4-yl]-5-methyl-1,3-benzoxazol-2-one
Show/Hide
|
C21H30N2O3
|
1
|
| 1 |
EC50 = 398.11 nM
|
|
|
|
CP0384743
|
Talsaclidine
Show/Hide
|
C10H15NO
|
1
|
| 1 |
EC50 = 422 nM
|
|
|
|
CP0316264
|
6-fluoro-5-methyl-3-[1-(oxan-4-yl)piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C18H24FN3O2
|
1
|
| 1 |
EC50 = 794.33 nM
|
|
|
|
CP0374547
|
3-[1-[4-(2-methoxyethoxy)-1-methylcyclohexyl]piperidin-4-yl]-2-oxo-1,3-benzoxazole-5-carbonitrile
Show/Hide
|
C23H31N3O4
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0388125
|
CHEMBL1223807
Show/Hide
|
C21H30N2O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0059332
|
1-(4-methoxybenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C17H12F3NO4
|
4
|
| 1 |
EC50 = 1100 nM
|
|
|
| 2 |
EC50 = 1160 nM
|
|
|
| 3 |
Ki = 159 nM
|
|
|
| 4 |
Ki = 1610 nM
|
|
|
|
CP0374545
|
3-[1-(4-ethoxy-1-methylcyclohexyl)piperidin-4-yl]-5-methylsulfonyl-1,3-benzoxazol-2-one
Show/Hide
|
C22H32N2O5S
|
1
|
| 1 |
EC50 = 1258.93 nM
|
|
|
|
CP0186462
|
5-methyl-3-[1-(oxan-4-yl)piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C18H25N3O2
|
1
|
| 1 |
EC50 = 1258.93 nM
|
|
|
|
CP0071482
|
1-(4-(6-fluoropyridin-2-yloxy)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H12F4N2O4
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0085573
|
3-[1-[3-(4-fluorophenoxy)propyl]piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C21H24FN3O2
|
1
|
| 1 |
EC50 = 1584.89 nM
|
|
|
|
CP0388592
|
1-(4-(pyridin-3-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H13F3N2O3
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0473885
|
1-(biphenyl-4-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H14F3NO3
|
2
|
| 1 |
EC50 = 1600 nM
|
|
|
| 2 |
EC50 = 2700 nM
|
|
|
|
CP0437592
|
1-(3-methoxybenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C17H12F3NO4
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0454184
|
5-(trifluoromethoxy)-1-(4-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C17H9F6NO3
|
1
|
| 1 |
EC50 = 1850 nM
|
|
|
|
CP0388741
|
5-(trifluoromethoxy)-1-(4-(trifluoromethoxy)benzyl)indoline-2,3-dione
Show/Hide
|
C17H9F6NO4
|
1
|
| 1 |
EC50 = 1860 nM
|
|
|
|
CP0059333
|
1-(4-phenoxybenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H14F3NO4
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
|
CP0496671
|
1-(4-bromobenzyl)-7-fluoroindoline-2,3-dione
Show/Hide
|
C15H9BrFNO2
|
1
|
| 1 |
EC50 = 1930 nM
|
|
|
|
CP0388743
|
7-chloro-1-(4-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H9ClF3NO2
|
2
|
| 1 |
EC50 = 2100 nM
|
|
|
| 2 |
EC50 = 2110 nM
|
|
|
|
CP0388590
|
1-(4-(pyrimidin-5-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3N3O3
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0388591
|
1-(4-(6-methoxypyridin-2-yloxy)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H15F3N2O5
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0403511
|
1-((6-chloropyridin-3-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C15H8ClF3N2O3
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
|
CP0488983
|
1-(biphenyl-4-ylmethyl)-6-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H14F3NO3
|
1
|
| 1 |
EC50 = 2700 nM
|
|
|
|
CP0371698
|
1-(4-(thiophen-3-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3NO3S
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0375624
|
1-(4-(thiazol-2-yloxy)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C19H11F3N2O4S
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0379379
|
1-(4-(pyridin-4-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H13F3N2O3
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0372657
|
1-((5-phenylpyridin-2-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H13F3N2O3
|
1
|
| 1 |
EC50 = 3100 nM
|
|
|
|
CP0454182
|
1-(4-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H10F3NO2
|
1
|
| 1 |
EC50 = 3190 nM
|
|
|
|
CP0473539
|
1-(4-(pyridin-2-yloxy)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H13F3N2O4
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0511757
|
1-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C17H10F3NO5
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0454200
|
7-fluoro-1-(4-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H9F4NO2
|
1
|
| 1 |
EC50 = 3260 nM
|
|
|
|
CP0454181
|
1-(2-methylbenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C17H12F3NO3
|
1
|
| 1 |
EC50 = 3280 nM
|
|
|
|
CP0494467
|
1-(4-(1-methyl-1H-pyrazol-4-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H14F3N3O3
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
|
CP0513953
|
1-(4-(6-fluoropyridin-3-yl)benzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H12F4N2O3
|
1
|
| 1 |
EC50 = 3600 nM
|
|
|
|
CP0388594
|
1-((6-phenylpyridin-3-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C21H13F3N2O3
|
1
|
| 1 |
EC50 = 3800 nM
|
|
|
|
CP0387457
|
1-((2'-methoxybiphenyl-4-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C23H16F3NO4
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0388734
|
7-chloro-1-(4-methoxybenzyl)indoline-2,3-dione
Show/Hide
|
C16H12ClNO3
|
1
|
| 1 |
EC50 = 3960 nM
|
|
|
|
CP0388593
|
1-(2,3'-bipyridin-5-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3N3O3
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0454185
|
1-(2-chlorobenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C16H9ClF3NO3
|
1
|
| 1 |
EC50 = 4070 nM
|
|
|
|
CP0113928
|
1-(4-bromobenzyl)indoline-2,3-dione
Show/Hide
|
C15H10BrNO2
|
3
|
| 1 |
EC50 = 4080 nM
|
|
|
| 2 |
EC50 = 4100 nM
|
|
|
| 3 |
EC50 = 4600 nM
|
|
|
|
CP0374358
|
5-fluoro-1-(2-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H9F4NO2
|
1
|
| 1 |
EC50 = 4090 nM
|
|
|
|
CP0372655
|
1-(2,4'-bipyridin-5-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3N3O3
|
1
|
| 1 |
EC50 = 4400 nM
|
|
|
|
CP0400848
|
1-(4-bromo-2-fluorobenzyl)-7-chloroindoline-2,3-dione
Show/Hide
|
C15H8BrClFNO2
|
1
|
| 1 |
EC50 = 4660 nM
|
|
|
|
CP0422157
|
1-[4-(6-chloro-3-pyridyl)benzyl]-5-(trifluoromethoxy)isatin;2,2,2-trifluoroacetic acid
Show/Hide
|
C21H12ClF3N2O3
|
1
|
| 1 |
EC50 = 4800 nM
|
|
|
|
CP0374546
|
CHEMBL1223938
Show/Hide
|
C23H34N2O5S
|
1
|
| 1 |
EC50 = 5011.87 nM
|
|
|
|
CP0470228
|
1-(4-methoxybenzyl)-6-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C17H12F3NO4
|
1
|
| 1 |
EC50 = 5700 nM
|
|
|
|
CP0502800
|
1-((3-fluorobiphenyl-4-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H13F4NO3
|
1
|
| 1 |
EC50 = 5900 nM
|
|
|
|
CP0454183
|
5-fluoro-1-(4-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H9F4NO2
|
1
|
| 1 |
EC50 = 7130 nM
|
|
|
|
CP0496672
|
4,7-dichloro-1-(3-methoxybenzyl)indoline-2,3-dione
Show/Hide
|
C16H11Cl2NO3
|
1
|
| 1 |
EC50 = 7150 nM
|
|
|
|
CP0437595
|
1-(4-bromo-2-fluorobenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C16H8BrF4NO3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0400206
|
2-(4-chloro-1,3-thiazol-2-yl)-N-(piperidin-4-ylmethyl)benzamide
Show/Hide
|
C16H18ClN3OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0045827
|
3-[1-(oxan-4-yl)piperidin-4-yl]-1H-benzimidazol-2-one
Show/Hide
|
C17H23N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0045829
|
3-(1-cyclohexylpiperidin-4-yl)-1H-benzimidazol-2-one
Show/Hide
|
C18H25N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0375319
|
N-benzyl-N-ethyl-1-(2-methoxyphenyl)sulfonylpiperidine-4-carboxamide
Show/Hide
|
C22H28N2O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0375320
|
N-benzyl-N-ethyl-1-(1H-imidazol-5-ylsulfonyl)piperidine-4-carboxamide
Show/Hide
|
C18H24N4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0375324
|
1-(1H-indazol-5-ylsulfonyl)-N-propan-2-yl-N-[[2-(trifluoromethyl)phenyl]methyl]piperidine-4-carboxamide
Show/Hide
|
C24H27F3N4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0375327
|
N-benzyl-N-ethyl-1-pyridin-2-ylsulfonylpiperidine-4-carboxamide
Show/Hide
|
C20H25N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379197
|
N-benzyl-N-ethyl-1-[6-(trifluoromethyl)pyridin-3-yl]sulfonylpiperidine-4-carboxamide
Show/Hide
|
C21H24F3N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379198
|
N-benzyl-N-ethyl-1-pyridin-4-ylsulfonylpiperidine-4-carboxamide
Show/Hide
|
C20H25N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0397059
|
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-benzyl-N-ethylpiperidine-4-carboxamide
Show/Hide
|
C21H24N4O3S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0413440
|
N-ethyl-N-[(4-fluorophenyl)methyl]-1-(1H-indazol-6-ylsulfonyl)piperidine-4-carboxamide
Show/Hide
|
C22H25FN4O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0413445
|
N-benzyl-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-N-ethylpiperidine-4-carboxamide
Show/Hide
|
C23H28N2O5S
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0415206
|
N-benzyl-N-ethyl-1-(5-methylthiophen-2-yl)sulfonylpiperidine-4-carboxamide
Show/Hide
|
C20H26N2O3S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0415256
|
N-benzyl-1-(3,4-dimethoxyphenyl)sulfonyl-N-ethylpiperidine-4-carboxamide
Show/Hide
|
C23H30N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0433221
|
N-benzyl-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-ethylpiperidine-4-carboxamide
Show/Hide
|
C20H27N3O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0433222
|
N-benzyl-N-ethyl-1-pyridin-3-ylsulfonylpiperidine-4-carboxamide
Show/Hide
|
C20H25N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0498636
|
N-benzyl-1-(2,3-dihydro-1,4-benzodioxin-5-ylsulfonyl)-N-ethylpiperidine-4-carboxamide
Show/Hide
|
C23H28N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0533193
|
N-benzyl-N-ethyl-1-quinolin-7-ylsulfonylpiperidine-4-carboxamide
Show/Hide
|
C24H27N3O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0533196
|
N-(2-hydroxyethyl)-1-(1H-indazol-5-ylsulfonyl)-N-[[2-(trifluoromethyl)phenyl]methyl]piperidine-4-carboxamide
Show/Hide
|
C23H25F3N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0405616
|
2-[(3R,4S)-3-hydroxyoxan-4-yl]-5-methyl-6-[[4-(1,3-oxazol-4-yl)phenyl]methyl]-3H-isoindol-1-one
Show/Hide
|
C24H24N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0500365
|
5-[[2,6-difluoro-4-(2-methylindazol-4-yl)phenyl]methyl]-1-(oxolan-2-ylmethyl)-4H-pyrrolo[3,4-c]pyrazol-6-one
Show/Hide
|
C25H23F2N5O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0557965
|
5-[[2-fluoro-4-(2-methylindazol-5-yl)phenyl]methyl]-4H-pyrrolo[3,4-d][1,3]thiazol-6-one
Show/Hide
|
C20H15FN4OS
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0423460
|
1-[N'-[3-(2-amino-4-methyl-1,3-thiazol-5-yl)propyl]carbamimidoyl]-3-pentylurea
Show/Hide
|
C14H26N6OS
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Kd = 0.2 nM
|
|
|
|
CP0543296
|
1-[(1R)-1-phenylethyl]-3-[N'-[3-(1H-1,2,4-triazol-5-yl)propyl]carbamimidoyl]urea;dihydrochloride
Show/Hide
|
C15H23Cl2N7O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Kd = 0.2 nM
|
|
|
|
CP0543300
|
1-[N'-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]carbamimidoyl]-3-benzylurea;2,2,2-trifluoroacetic acid
Show/Hide
|
C18H21F6N7O5S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Kd = 0.2 nM
|
|
|
|
CP0551746
|
1-[N'-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]carbamimidoyl]-3-pentylurea;2,2,2-trifluoroacetic acid
Show/Hide
|
C16H25F6N7O5S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
Kd = 0.2 nM
|
|
|
|
CP0374356
|
1-(4-methoxybenzyl)indoline-2,3-dione
Show/Hide
|
C16H13NO3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0400849
|
7-fluoro-1-(2-(trifluoromethyl)benzyl)indoline-2,3-dione
Show/Hide
|
C16H9F4NO2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0405390
|
1-(3,4'-bipyridin-6-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3N3O3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0473535
|
1-(3,3'-bipyridin-6-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C20H12F3N3O3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0474474
|
1-(biphenyl-3-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H14F3NO3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0511756
|
1-((3,5-difluorobiphenyl-4-yl)methyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H12F5NO3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0522119
|
1-(3-phenoxybenzyl)-5-(trifluoromethoxy)indoline-2,3-dione
Show/Hide
|
C22H14F3NO4
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0168609
|
ethyl 4-[(3R)-3-[(2-methylbenzoyl)amino]piperidin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C21H31N3O3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0392295
|
4-[2-(o-toluoylamino)ethylamino]piperidine-1-carboxylic acid ethyl ester;hydrochloride
Show/Hide
|
C18H27N3O3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0305211
|
1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
Show/Hide
|
C25H32N4O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0412637
|
1-methyl-4-[[6-(1-methylpyrazol-4-yl)pyridin-3-yl]methyl]-N-(oxan-4-yl)pyrrolo[2,3-b]pyridine-6-carboxamide
Show/Hide
|
C24H26N6O2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0673968
|
SID50106181
Show/Hide
|
C21H26INO2
|
2
|
| 1 |
IC50 = 0.32 nM
|
|
|
| 2 |
Ki = 0.48 nM
|
|
|
|
CP0040500
|
3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9-aza-tricyclo[3.3.1.0*2,4*]non-7-yl ester
Show/Hide
|
C18H24NO4+
|
2
|
| 1 |
IC50 = 2.3 nM
|
|
|
| 2 |
Ki = 0.2089 nM
|
|
|
|
CP0543679
|
(3R,4R)-N-(1,3-benzothiazol-5-yl)-1-(5-chloro-1-methylpyrazol-4-yl)sulfonyl-3-fluoropiperidine-4-carboxamide
Show/Hide
|
C17H17ClFN5O3S2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0857826
|
1-Cyclohexyl-1-phenyl-3-piperidin-1-yl-propan-1-ol hydrochloride
Show/Hide
|
C20H32ClNO
|
1
|
| 1 |
IC50 = 10.3 nM
|
|
|
|
CP0577435
|
(3R,4R)-N-(1,3-benzothiazol-5-yl)-3-fluoro-1-[(2-methyl-1,3-thiazol-5-yl)sulfonyl]piperidine-4-carboxamide
Show/Hide
|
C17H17FN4O3S3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0847735
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-p-tolyl-ethyl ester oxalic acid
Show/Hide
|
C25H29NO6
|
1
|
| 1 |
IC50 = 24.8 nM
|
|
|
|
CP0576561
|
(3R,4S)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-3-fluoro-4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidine
Show/Hide
|
C18H22FN3O3S2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0870135
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid benzyl ester hydrochloride
Show/Hide
|
C21H24ClNO2
|
1
|
| 1 |
IC50 = 42.5 nM
|
|
|
|
CP0854268
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid cyclohexyl ester oxalic acid
Show/Hide
|
C22H29NO6
|
1
|
| 1 |
IC50 = 54.1 nM
|
|
|
|
CP0869657
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-cyclohexyl-ethyl ester oxalic acid
Show/Hide
|
C24H33NO6
|
1
|
| 1 |
IC50 = 56.2 nM
|
|
|
|
CP0850038
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid octyl ester oxalic acid
Show/Hide
|
C24H35NO6
|
1
|
| 1 |
IC50 = 57.9 nM
|
|
|
|
CP0543680
|
N-(1,3-benzothiazol-5-yl)-1-pyridin-3-ylsulfonylpiperidine-4-carboxamide
Show/Hide
|
C18H18N4O3S2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0849760
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid cyclohexyl ester oxalic acid
Show/Hide
|
C22H29NO6
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0847169
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid phenethyl ester oxalic acid
Show/Hide
|
C24H27NO6
|
1
|
| 1 |
IC50 = 78.1 nM
|
|
|
|
CP0404712
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid nonyl ester
Show/Hide
|
C23H35NO2
|
1
|
| 1 |
IC50 = 85.4 nM
|
|
|
|
CP0578800
|
(2R,4S)-N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-2-methylpiperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0861085
|
1-Ethyl-4-phenyl-piperidine-3-carboxylic acid phenethyl ester oxalic acid
Show/Hide
|
C24H29NO6
|
1
|
| 1 |
IC50 = 96.8 nM
|
|
|
|
CP0579849
|
N-(1,3-benzothiazol-5-yl)-1-(6-methylpyridin-3-yl)sulfonylpiperidine-4-carboxamide
Show/Hide
|
C19H20N4O3S2
|
1
|
| 1 |
IC50 = 105 nM
|
|
|
|
CP0552044
|
N-(1,3-benzothiazol-5-yl)-1-[(3-methyl-2,3-dihydro-1-benzofuran-5-yl)sulfonyl]piperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 = 109 nM
|
|
|
|
CP0579616
|
N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)piperidine-4-carboxamide
Show/Hide
|
C21H21N3O4S2
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0845078
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid cyclohexylmethyl ester oxalic acid
Show/Hide
|
C23H31NO6
|
1
|
| 1 |
IC50 = 115.4 nM
|
|
|
|
CP0568824
|
(2R,4R)-N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-2-methylpiperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 = 134 nM
|
|
|
|
CP0878826
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid hexyl ester oxalic acid
Show/Hide
|
C22H31NO6
|
1
|
| 1 |
IC50 = 138.9 nM
|
|
|
|
CP0550426
|
N-(1,2,3-benzothiadiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)piperidine-4-carboxamide
Show/Hide
|
C20H20N4O4S2
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0859753
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 2-cyclohexyl-ethyl ester oxalic acid
Show/Hide
|
C24H33NO6
|
1
|
| 1 |
IC50 = 159.2 nM
|
|
|
|
CP0568825
|
N-(1,3-benzothiazol-5-yl)-1-(6-chloropyridin-3-yl)sulfonylpiperidine-4-carboxamide
Show/Hide
|
C18H17ClN4O3S2
|
1
|
| 1 |
IC50 = 168 nM
|
|
|
|
CP0860615
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 2-p-tolyl-ethyl ester oxalic acid
Show/Hide
|
C25H29NO6
|
1
|
| 1 |
IC50 = 190.3 nM
|
|
|
|
CP0886216
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid heptyl ester oxalic acid
Show/Hide
|
C23H33NO6
|
1
|
| 1 |
IC50 = 194.2 nM
|
|
|
|
CP0860558
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid cyclohexylmethyl ester oxalic acid
Show/Hide
|
C23H31NO6
|
1
|
| 1 |
IC50 = 214.5 nM
|
|
|
|
CP0878820
|
(3R,4R)-1-Ethyl-4-phenyl-piperidine-3-carboxylic acid hexyl ester oxalic acid
Show/Hide
|
C22H33NO6
|
1
|
| 1 |
IC50 = 222.1 nM
|
|
|
|
CP0392493
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid decyl ester
Show/Hide
|
C24H37NO2
|
1
|
| 1 |
IC50 = 235.6 nM
|
|
|
|
CP0869546
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid butyl ester oxalic acid
Show/Hide
|
C20H27NO6
|
1
|
| 1 |
IC50 = 254.9 nM
|
|
|
|
CP0914385
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 3-phenyl-propyl ester hydrochloride
Show/Hide
|
C23H28ClNO2
|
1
|
| 1 |
IC50 = 255.8 nM
|
|
|
|
CP0849749
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid butyl ester oxalic acid
Show/Hide
|
C20H27NO6
|
1
|
| 1 |
IC50 = 264.7 nM
|
|
|
|
CP0577109
|
N-(1,3-benzothiazol-5-yl)-1-(1,3-benzothiazol-6-ylsulfonyl)piperidine-4-carboxamide
Show/Hide
|
C20H18N4O3S3
|
1
|
| 1 |
IC50 = 266 nM
|
|
|
|
CP0854470
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid benzyl ester hydrochloride
Show/Hide
|
C21H24ClNO2
|
1
|
| 1 |
IC50 = 272.8 nM
|
|
|
|
CP0317131
|
(9bS)-9b-(4-chlorophenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C23H15ClF2N2O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0568251
|
N-(1,3-benzothiazol-5-yl)-1-(1,3-dimethylpyrazol-4-yl)sulfonylpiperidine-4-carboxamide
Show/Hide
|
C18H21N5O3S2
|
1
|
| 1 |
IC50 = 304 nM
|
|
|
|
CP0568826
|
(3R,4R)-N-(1,3-benzothiazol-5-yl)-1-(1,3-dimethylpyrazol-4-yl)sulfonyl-3-fluoropiperidine-4-carboxamide
Show/Hide
|
C18H20FN5O3S2
|
1
|
| 1 |
IC50 = 309 nM
|
|
|
|
CP0381434
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid nonyl ester
Show/Hide
|
C23H35NO2
|
1
|
| 1 |
IC50 = 328.6 nM
|
|
|
|
CP0914469
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid phenethyl ester oxalic acid
Show/Hide
|
C24H27NO6
|
1
|
| 1 |
IC50 = 330.9 nM
|
|
|
|
CP0056034
|
11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C19H21N5O2
|
2
|
| 1 |
IC50 = 340.6 nM
|
|
|
| 2 |
Ki = 35.48 nM
|
|
|
|
CP0860587
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid pentyl ester oxalic acid
Show/Hide
|
C21H29NO6
|
1
|
| 1 |
IC50 = 341.9 nM
|
|
|
|
CP0854465
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid pentyl ester oxalic acid
Show/Hide
|
C21H29NO6
|
1
|
| 1 |
IC50 = 374 nM
|
|
|
|
CP0914612
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid octyl ester oxalic acid
Show/Hide
|
C24H35NO6
|
1
|
| 1 |
IC50 = 400.6 nM
|
|
|
|
CP0847343
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid isobutyl ester oxalic acid
Show/Hide
|
C20H27NO6
|
1
|
| 1 |
IC50 = 407.3 nM
|
|
|
|
CP0569370
|
(3S,4S)-N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-3-methylpiperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 = 419 nM
|
|
|
|
CP0550227
|
5-[(3-acetylphenoxy)methyl]-N-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C21H21N3O4
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0845389
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 5-phenyl-pentyl ester oxalic acid
Show/Hide
|
C27H33NO6
|
1
|
| 1 |
IC50 = 472.2 nM
|
|
|
|
CP0853934
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 3-phenyl-propyl ester hydrochloride
Show/Hide
|
C23H28ClNO2
|
1
|
| 1 |
IC50 = 479.4 nM
|
|
|
|
CP0861083
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 2-(4-methoxy-phenyl)-ethyl ester oxalic acid
Show/Hide
|
C25H29NO7
|
1
|
| 1 |
IC50 = 499.7 nM
|
|
|
|
CP0405990
|
2-(3-chlorophenyl)-6-fluoro-N-[[(3R,4S)-3-methylpiperidin-4-yl]methyl]benzamide
Show/Hide
|
C20H22ClFN2O
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0861075
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid hexyl ester oxalic acid
Show/Hide
|
C22H31NO6
|
1
|
| 1 |
IC50 = 508.2 nM
|
|
|
|
CP0389547
|
[1-[6-(2,4-difluorophenoxy)pyrimidin-4-yl]piperidin-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone
Show/Hide
|
C25H24F2N4O2
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0850036
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid heptyl ester oxalic acid
Show/Hide
|
C23H33NO6
|
1
|
| 1 |
IC50 = 537.3 nM
|
|
|
|
CP0863347
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid isobutyl ester oxalic acid
Show/Hide
|
C20H27NO6
|
1
|
| 1 |
IC50 = 558.9 nM
|
|
|
|
CP0568252
|
1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-N-(2-methyl-1,3-benzothiazol-5-yl)piperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 = 594 nM
|
|
|
|
CP0889381
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid propyl ester oxalic acid
Show/Hide
|
C19H25NO6
|
1
|
| 1 |
IC50 = 602.9 nM
|
|
|
|
CP0389549
|
[1-[6-(4-chlorophenoxy)pyrimidin-4-yl]piperidin-4-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone
Show/Hide
|
C25H25ClN4O2
|
1
|
| 1 |
IC50 = 695 nM
|
|
|
|
CP0510932
|
9b-(4-fluoro-3-methoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C24H16F4N2O3
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0389544
|
3,4-dihydro-1H-isoquinolin-2-yl-[1-[6-(2-fluorophenoxy)pyrimidin-4-yl]piperidin-4-yl]methanone
Show/Hide
|
C25H25FN4O2
|
1
|
| 1 |
IC50 = 732 nM
|
|
|
|
CP0473116
|
2-(3-chloro-4-methylphenyl)-N-(piperidin-4-ylmethyl)benzamide
Show/Hide
|
C20H23ClN2O
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0849717
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 4-phenyl-butyl ester oxalic acid
Show/Hide
|
C26H31NO6
|
1
|
| 1 |
IC50 = 842 nM
|
|
|
|
CP0861084
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-(4-methoxy-phenyl)-ethyl ester oxalic acid
Show/Hide
|
C25H29NO7
|
1
|
| 1 |
IC50 = 865.9 nM
|
|
|
|
CP0523419
|
9b-(3-methoxy-4-methylphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C25H19F3N2O3
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0578801
|
N-(1,3-benzothiazol-5-yl)-1-quinolin-6-ylsulfonylpiperidine-4-carboxamide
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C22H20N4O3S2
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1
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| 1 |
IC50 = 959 nM
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CP0860435
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1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid methyl ester oxalic acid
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C17H21NO6
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1
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| 1 |
IC50 = 977.3 nM
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CP0878792
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9b-(4-chlorophenyl)-1-(3,5-difluorobenzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
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C23H15ClF2N2O2
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1
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| 1 |
IC50 = 1000 nM
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CP0545747
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9b-(1,3-benzodioxol-5-yl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C24H15F3N2O4
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1
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| 1 |
IC50 = 1000 nM
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CP0054849
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methyl-6-(S)-methyl-piperidin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one
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C22H35NO2
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2
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| 1 |
IC50 = 1016 nM
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| 2 |
Ki = 489.78 nM
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CP0456704
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4-[4-[6-(3,3-dimethylpiperidin-1-yl)pyridazin-3-yl]piperazin-1-yl]sulfonyl-3,5-dimethyl-1,2-oxazole
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C20H30N6O3S
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1
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| 1 |
IC50 = 1030 nM
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CP0409466
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9b-(1,3-benzodioxol-5-yl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C27H24N2O5
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1
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| 1 |
IC50 = 1100 nM
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CP0392206
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid decyl ester
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C24H37NO2
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1
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| 1 |
IC50 = 1114.8 nM
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CP0910088
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid propyl ester oxalic acid
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C19H25NO6
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1
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| 1 |
IC50 = 1127.9 nM
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CP0356645
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[1-[6-(2,4-difluorophenoxy)pyrimidin-4-yl]piperidin-4-yl]-(1,3-dihydroisoindol-2-yl)methanone
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C24H22F2N4O2
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1
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| 1 |
IC50 = 1130 nM
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CP0456389
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1-(3,4-difluorobenzoyl)-9b-(4-methoxy-3-methylphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C25H20F2N2O3
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1
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| 1 |
IC50 = 1200 nM
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CP0447292
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(9bS)-9b-(4-chloro-3-methylphenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C24H17ClF2N2O2
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1
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| 1 |
IC50 = 1200 nM
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CP0863310
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1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 3-cyclohexyl-propyl ester oxalic acid
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C25H35NO6
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1
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| 1 |
IC50 = 1260.5 nM
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CP0386265
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9b-(4-fluoro-3-methoxyphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C27H25FN2O4
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1
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| 1 |
IC50 = 1300 nM
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CP0413528
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1-(3,4-difluorobenzoyl)-9b-(3-methoxy-4-methylphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C25H20F2N2O3
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1
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| 1 |
IC50 = 1300 nM
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CP0508960
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9b-(1,3-benzodioxol-5-yl)-1-(3,4-difluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C24H16F2N2O4
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1
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| 1 |
IC50 = 1300 nM
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CP0566800
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9b-(4-methoxy-3-methylphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C28H28N2O4
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1
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| 1 |
IC50 = 1300 nM
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CP0859752
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1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid ethyl ester oxalic acid
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C18H23NO6
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1
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| 1 |
IC50 = 1331.2 nM
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CP0481709
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9b-(3-chloro-4-methoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C24H16ClF3N2O3
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1
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| 1 |
IC50 = 1400 nM
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CP0862779
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1-Ethyl-5-(3-pentyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-1,2,3,6-tetrahydro-pyridine oxalic acid
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C22H29N3O5
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1
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| 1 |
IC50 = 1467.3 nM
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CP0578885
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(3R,4S)-N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-3-methylpiperidine-4-carboxamide
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C22H23N3O4S2
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1
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| 1 |
IC50 = 1530 nM
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CP0847170
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 5-phenyl-pentyl ester oxalic acid
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C27H33NO6
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1
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| 1 |
IC50 = 1567.9 nM
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CP0846965
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1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid phenyl ester oxalic acid
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C22H23NO6
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1
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| 1 |
IC50 = 1568.6 nM
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CP0400210
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2-(3-chlorophenyl)-6-fluoro-N-(1,2,3,6-tetrahydropyridin-4-ylmethyl)benzamide
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C19H18ClFN2O
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1
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| 1 |
IC50 = 1584.89 nM
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CP0425773
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9b-(4-chloro-3-methoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C24H16ClF3N2O3
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1
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| 1 |
IC50 = 1600 nM
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CP0500468
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2,7-Dimethyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C23H24N2O3
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1
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| 1 |
IC50 = 1731.8 nM
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CP0579804
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1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-N-quinolin-7-ylpiperidine-4-carboxamide
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C23H23N3O4S
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1
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| 1 |
IC50 = 1802 nM
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CP0393182
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(3R,4R)-1-Ethyl-4-phenyl-piperidine-3-carboxylic acid cyclohexyl ester
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C20H29NO2
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1
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| 1 |
IC50 = 1889.3 nM
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CP0510931
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1-(4-propan-2-yloxybenzoyl)-9b-(4-propan-2-yloxyphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C29H30N2O4
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1
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| 1 |
IC50 = 1900 nM
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CP0523422
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9b-(4-chloro-3-methoxyphenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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C24H17ClF2N2O3
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1
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| 1 |
IC50 = 2000 nM
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CP0453286
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2-Methyl-9-phenoxy-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C28H26N2O4
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1
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| 1 |
IC50 = 2033.9 nM
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CP0855705
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1-Ethyl-3-(3-pentyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-1,2,3,6-tetrahydro-pyridine oxalic acid
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C22H29N3O5
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1
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| 1 |
IC50 = 2075.4 nM
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CP0376534
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1-Methyl-5-(4-methylsulfanyl-[1,2,5]thiadiazol-3-yl)-1,2,3,6-tetrahydro-pyridine; oxalic acid
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C9H13N3S2
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1
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| 1 |
IC50 = 2100 nM
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CP0578774
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2-[[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)piperidin-4-yl]methylsulfanyl]-4-methyl-1,3-thiazole
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C18H22N2O4S3
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1
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| 1 |
IC50 = 2110 nM
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CP0418169
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9b-(3-methoxy-4-methylphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C28H28N2O4
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1
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| 1 |
IC50 = 2200 nM
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CP0510933
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9b-(4-propan-2-yloxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C26H21F3N2O3
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1
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| 1 |
IC50 = 2400 nM
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CP0456388
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1-(3,4-difluorobenzoyl)-9b-(4-fluoro-3-methoxyphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C24H17F3N2O3
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1
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| 1 |
IC50 = 2700 nM
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CP0578886
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N-(1,3-benzothiazol-5-yl)-1-(5-chlorothiophen-2-yl)sulfonylpiperidine-4-carboxamide
Show/Hide
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C17H16ClN3O3S3
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1
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| 1 |
IC50 = 2803 nM
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CP0860591
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(3S,4R)-1-Ethyl-4-phenyl-piperidine-3-carboxylic acid cyclohexyl ester oxalic acid
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C22H31NO6
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1
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| 1 |
IC50 = 2971.4 nM
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CP0854016
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1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2,2-diphenyl-ethyl ester oxalic acid
Show/Hide
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C30H31NO6
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1
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| 1 |
IC50 = 3108.6 nM
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CP0579245
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3-[2-[4-[(4-chloro-1,3-benzothiazol-2-yl)oxy]piperidin-1-yl]-2-oxoethyl]-1,3-benzoxazol-2-one
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C21H18ClN3O4S
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1
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| 1 |
IC50 = 3170 nM
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CP0492431
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9b-(3-fluoro-4-methoxyphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C27H25FN2O4
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1
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| 1 |
IC50 = 3200 nM
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CP0545748
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1-(3,4-difluorobenzoyl)-9b-(4-ethoxyphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C25H20F2N2O3
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1
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| 1 |
IC50 = 3200 nM
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CP0481665
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1-(3,4-difluorobenzoyl)-9b-(3-fluoro-4-methoxyphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C24H17F3N2O3
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1
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| 1 |
IC50 = 3300 nM
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CP0566801
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9b-(3-chloro-4-methoxyphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C27H25ClN2O4
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1
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| 1 |
IC50 = 3300 nM
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CP0381598
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1-(4-fluorobenzoyl)-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C23H17FN2O2
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1
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| 1 |
IC50 = 3490 nM
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CP0886217
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 2,2-diphenyl-ethyl ester oxalic acid
Show/Hide
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C30H31NO6
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1
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| 1 |
IC50 = 3565.8 nM
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CP0383656
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid propyl ester
Show/Hide
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C24H26N2O4
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1
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| 1 |
IC50 = 3807.6 nM
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CP0451231
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2,9-Dimethyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C23H24N2O3
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1
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| 1 |
IC50 = 3884.2 nM
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CP0408846
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid methyl ester
Show/Hide
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C22H22N2O4
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1
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| 1 |
IC50 = 4093 nM
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CP0447267
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9b-(4-ethoxyphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C28H28N2O4
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1
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| 1 |
IC50 = 4100 nM
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CP0850116
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid ethyl ester oxalic acid
Show/Hide
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C18H23NO6
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1
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| 1 |
IC50 = 4169.5 nM
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CP0510618
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2-Methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C22H22N2O3
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1
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| 1 |
IC50 = 4187.1 nM
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CP0880188
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(3R,4R)-1-Ethyl-4-phenyl-piperidine-3-carboxylic acid phenethyl ester oxalic acid
Show/Hide
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C24H29NO6
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1
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| 1 |
IC50 = 4264 nM
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CP0404668
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid isopropyl ester
Show/Hide
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C24H26N2O4
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1
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| 1 |
IC50 = 4737 nM
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CP0853885
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1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 4-phenyl-butyl ester oxalic acid
Show/Hide
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C26H31NO6
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1
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| 1 |
IC50 = 5000 nM
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CP0406059
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2-(5-chloro-2-fluorophenyl)-N-(piperidin-4-ylmethyl)benzamide
Show/Hide
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C19H20ClFN2O
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1
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| 1 |
IC50 = 5011.87 nM
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CP0579396
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1-(2,4-dichloro-5-methylphenyl)sulfonyl-4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidine
Show/Hide
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C17H21Cl2N3O2S2
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1
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| 1 |
IC50 = 5440 nM
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CP0447269
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9b-(3-chloro-4-methoxyphenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C24H17ClF2N2O3
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1
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| 1 |
IC50 = 5500 nM
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CP0448496
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2-Methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid methyl ester
Show/Hide
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C21H20N2O3
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1
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| 1 |
IC50 = 5760.1 nM
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CP0448414
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9-Methoxy-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C22H22N2O4
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1
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| 1 |
IC50 = 5999.2 nM
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CP0400212
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2-(3-chlorophenyl)-6-fluoro-N-[[(3S,4R)-4-fluoro-3-methylpiperidin-4-yl]methyl]benzamide
Show/Hide
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C20H21ClF2N2O
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1
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| 1 |
IC50 = 6309.57 nM
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CP0425772
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9b-(4-chloro-3-methoxyphenyl)-1-(4-propan-2-yloxybenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
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C27H25ClN2O4
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1
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| 1 |
IC50 = 6400 nM
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CP0249049
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3-[4-(2-chlorophenyl)sulfonylpiperazin-1-yl]-6-[(2S)-2-methylpiperidin-1-yl]pyridazine
Show/Hide
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C20H26ClN5O2S
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1
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| 1 |
IC50 = 6500 nM
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CP0139207
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C23H24N2O4
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2
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| 1 |
IC50 = 7411.7 nM
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| 2 |
Ki = 3388.44 nM
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CP0037621
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(oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one
Show/Hide
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C12H18N2O
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1
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| 1 |
IC50 = 8000 nM
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CP0454447
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8-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C23H24N2O4
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1
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| 1 |
IC50 = 8211.3 nM
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CP0448197
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9-Ethoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C24H26N2O4
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1
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| 1 |
IC50 = 8624 nM
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CP0576562
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1-[3-[4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidin-1-yl]sulfonylphenyl]ethanone
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C18H23N3O3S2
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1
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| 1 |
IC50 = 8810 nM
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CP0386486
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2-(3-chlorophenyl)-N-(piperidin-4-ylmethyl)benzamide
Show/Hide
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C19H21ClN2O
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1
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| 1 |
IC50 > 10000 nM
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CP0416360
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2-(3-chlorophenyl)-N-[(3-methylpiperidin-4-yl)methyl]benzamide
Show/Hide
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C20H23ClN2O
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1
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| 1 |
IC50 > 10000 nM
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CP0849148
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1-(3,5-difluorobenzoyl)-9b-(4-fluorophenyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
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C23H15F3N2O2
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1
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| 1 |
IC50 > 10000 nM
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CP0849155
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9b-p-tolyl-1-(4-(trifluoromethyl)benzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
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C25H19F3N2O2
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1
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| 1 |
IC50 > 10000 nM
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CP0849156
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1-(4-methylbenzoyl)-9b-p-tolyl-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
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C25H22N2O2
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1
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| 1 |
IC50 > 10000 nM
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|
|
CP0849157
|
9b-p-tolyl-1-(3-(trifluoromethyl)benzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C25H19F3N2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0878791
|
9b-(4-fluorophenyl)-1-(4-(trifluoromethyl)benzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C24H16F4N2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0880197
|
1-(3,4-difluorobenzoyl)-9b-(4-fluorophenyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C23H15F3N2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0884640
|
9b-(4-fluorophenyl)-1-(4-methylbenzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C24H19FN2O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0895327
|
9b-(4-fluorophenyl)-1-(4-(trifluoromethoxy)benzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C24H16F4N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0545262
|
1-[(2,2-difluoro-1,3-benzodioxol-5-yl)sulfonyl]-4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidine
Show/Hide
|
C17H19F2N3O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0568216
|
1-(2,3-dihydro-1H-inden-5-ylsulfonyl)-4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidine
Show/Hide
|
C19H25N3O2S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0568304
|
1-(2,3-dihydro-1,4-benzodioxin-5-ylsulfonyl)-4-[(1-methylimidazol-2-yl)sulfanylmethyl]piperidine
Show/Hide
|
C18H23N3O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0569778
|
2-[[1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)pyrrolidin-3-yl]methylsulfanyl]-1-methylimidazole
Show/Hide
|
C17H21N3O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0550427
|
N-(1,3-benzothiazol-5-yl)-1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)sulfonyl]piperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0577642
|
N-(1,3-benzothiazol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylsulfonyl)-N-methylpiperidine-4-carboxamide
Show/Hide
|
C22H23N3O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0880203
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid 3-cyclohexyl-propyl ester oxalic acid
Show/Hide
|
C25H35NO6
|
1
|
| 1 |
IC50 = 10969.8 nM
|
|
|
|
CP0847050
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid methyl ester oxalic acid
Show/Hide
|
C17H21NO6
|
1
|
| 1 |
IC50 = 16901.9 nM
|
|
|
|
CP0403792
|
9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
IC50 = 17980.7 nM
|
|
|
|
CP0457513
|
8-Methyl-6,7,8,9-tetrahydro-5H-2,4-dithia-1,3,8-triaza-cyclopenta[a]naphthalene
Show/Hide
|
C9H11N3S2
|
1
|
| 1 |
IC50 = 23000 nM
|
|
|
|
CP0635477
|
(2-Carbamoyloxy-ethyl)-trimethyl-ammonium chloride
Show/Hide
|
C6H15ClN2O2
|
3
|
| 1 |
IC50 = 25200 nM
|
|
|
| 2 |
Ki = 4265.8 nM
|
|
|
| 3 |
Ki = 69183.1 nM
|
|
|
|
CP0458944
|
8,9-Dimethoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
|
C24H26N2O5
|
1
|
| 1 |
IC50 = 26644.8 nM
|
|
|
|
CP0393505
|
N-[3-oxo-3-(4-pyridin-4-ylpiperazin-1-yl)propyl]quinoline-5-sulfonamide
Show/Hide
|
C21H23N5O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0880196
|
(+)-(R)-9b-(4-chlorophenyl)-1-(3,4-difluorobenzoyl)-2,3-dihydro-1H-imidazo[2,1-a]isoindol-5(9bH)-one
Show/Hide
|
C23H15ClF2N2O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0523420
|
9b-(3-fluoro-4-methoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C24H16F4N2O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0523421
|
9b-(4-ethoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C25H19F3N2O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0566802
|
1-(3,4-difluorobenzoyl)-9b-(4-propan-2-yloxyphenyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
Show/Hide
|
C26H22F2N2O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0854472
|
1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-carboxylic acid phenyl ester oxalic acid
Show/Hide
|
C22H23NO6
|
1
|
| 1 |
IC50 = 31057 nM
|
|
|
|
CP0448346
|
8,9-Dimethoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene
Show/Hide
|
C21H22N2O3
|
1
|
| 1 |
IC50 = 43462.7 nM
|
|
|
|
CP0404049
|
8,9-Dimethoxy-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
|
C23H24N2O5
|
1
|
| 1 |
IC50 = 47361.5 nM
|
|
|
|
CP0018455
|
1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid methyl ester;hydrobromide
Show/Hide
|
C8H13NO2
|
2
|
| 1 |
IC50 = 62500 nM
|
|
|
| 2 |
Ki = 56234.13 nM
|
|
|
|
CP0382980
|
6,7,8,9-Tetrahydro-2-thia-1,3,8-triaza-cyclopenta[a]naphthalene
Show/Hide
|
C9H9N3S
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
|
CP0421075
|
1,4-Dimethyl-5-(4-methylsulfanyl-[1,2,5]thiadiazol-3-yl)-1,2,3,6-tetrahydro-pyridine
Show/Hide
|
C10H15N3S2
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
|
CP0218742
|
3,4-dihydro-1H-isoquinolin-2-yl-[1-[6-(4-ethylphenoxy)pyrimidin-4-yl]piperidin-4-yl]methanone
Show/Hide
|
C27H30N4O2
|
1
|
| 1 |
IC50 < 1500 nM
|
|
|
|
CP0666404
|
Tiotropium bromide
Show/Hide
|
C19H24BrNO5S2
|
1
|
| 1 |
Ki = 0.0266 nM
|
|
|
|
CP0889526
|
(S)-2-((2R,5S)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H32INOS
|
1
|
| 1 |
Ki = 0.1072 nM
|
|
|
|
CP0199765
|
5-[3-(3-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 0.169 nM
|
|
|
|
CP0877788
|
(S)-2-((2S,5S)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H32INOS
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0109931
|
ATROPEN
Show/Hide
|
C17H23NO3
|
4
|
| 1 |
Ki = 0.21 nM
|
|
|
| 2 |
Ki = 0.54 nM
|
|
|
| 3 |
Ki = 0.6 nM
|
|
|
| 4 |
Ki = 1.47 nM
|
|
|
|
CP0869209
|
(S)-2-((S)-2,2-diphenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H26INOS
|
1
|
| 1 |
Ki = 0.4074 nM
|
|
|
|
CP0881062
|
(R)-2-((2R,5R)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H32INOS
|
1
|
| 1 |
Ki = 0.7762 nM
|
|
|
|
CP0070586
|
Ipratropium Bromide
Show/Hide
|
C20H30BrNO3
|
1
|
| 1 |
Ki = 1.04 nM
|
|
|
|
CP0881063
|
(2R,2'R,5'R)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H29NOS
|
1
|
| 1 |
Ki = 1.202 nM
|
|
|
|
CP0858803
|
(2S,2'R,5'S)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H29NOS
|
1
|
| 1 |
Ki = 1.349 nM
|
|
|
|
CP0894757
|
(R)-2-(5-((R)-cyclohexyl(hydroxy)(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO2
|
1
|
| 1 |
Ki = 1.549 nM
|
|
|
|
CP0858907
|
(S)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 1.698 nM
|
|
|
|
CP0440619
|
1-azabicyclo[2.2.2]octan-3-yl N-[2-(4-fluorophenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C22H25FN2O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0879684
|
(S)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine Oxalate
Show/Hide
|
C21H25NO6
|
1
|
| 1 |
Ki = 1.82 nM
|
|
|
|
CP0858802
|
(2R,2'S,5'R)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H29NOS
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0877786
|
(2S,2'S,5'S)-1-methyl-2-(2-cyclohexyl-2-phenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H29NOS
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
|
CP0378654
|
1-[3-[4-[7-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]heptyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C32H47N5O2S
|
1
|
| 1 |
Ki = 2.291 nM
|
|
|
|
CP0010653
|
2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-pyrrolidin-3-yl}-2,2-diphenyl-acetamide (Darifenacin)
Show/Hide
|
C28H30N2O2
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0871074
|
(2R,5R)-2-cyclohexyl-2-phenyl-5-((dimethylamino)methyl)-1,3-oxathiolane methiodide
Show/Hide
|
C19H30INOS
|
1
|
| 1 |
Ki = 2.818 nM
|
|
|
|
CP0378646
|
1-[3-[4-[9-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]nonyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C34H51N5O2S
|
1
|
| 1 |
Ki = 2.951 nM
|
|
|
|
CP0877787
|
(2R,5'R)-1-methyl2-(2,2-diphenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H23NOS
|
1
|
| 1 |
Ki = 3.236 nM
|
|
|
|
CP0881061
|
(R)-2-((2S,5R)-2-cyclohexyl-2-phenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H32INOS
|
1
|
| 1 |
Ki = 3.236 nM
|
|
|
|
CP0439251
|
(R)-cyclohexyl-[5-[(2R)-1-methylpyrrolidin-2-yl]furan-2-yl]-phenylmethanol
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 3.311 nM
|
|
|
|
CP0869207
|
(R)-2-((R)-2,2-diphenyl-[1,3]oxathiolan-5-yl)-1,1-dimethyl-pyrrolidinium iodide
Show/Hide
|
C21H26INOS
|
1
|
| 1 |
Ki = 3.467 nM
|
|
|
|
CP0399528
|
1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2,5-thiadiazol-3-yloxy]nonane
Show/Hide
|
C25H38N6O2S2
|
1
|
| 1 |
Ki = 3.981 nM
|
|
|
|
CP0867620
|
(+/-)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 4.365 nM
|
|
|
|
CP0858902
|
(+/-)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine Oxalate
Show/Hide
|
C21H25NO6
|
1
|
| 1 |
Ki = 5.37 nM
|
|
|
|
CP0876058
|
(2S,5'S)-1-methyl 2-(2,2-diphenyl-1,3-oxathiolan-5-yl)pirrolidine
Show/Hide
|
C20H23NOS
|
1
|
| 1 |
Ki = 5.623 nM
|
|
|
|
CP0378653
|
1-[3-[4-[5-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]pentyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C30H43N5O2S
|
1
|
| 1 |
Ki = 5.623 nM
|
|
|
|
CP0405296
|
3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxyisoxazole sesquifumarate
Show/Hide
|
C11H11N3O2
|
1
|
| 1 |
Ki = 6.166 nM
|
|
|
|
CP0405687
|
cyclohexyl-[5-(1-methylpyrrolidin-2-yl)furan-2-yl]-phenylmethanol
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 7.079 nM
|
|
|
|
CP0415932
|
1-[3-[4-[11-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]undecyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C36H55N5O2S
|
1
|
| 1 |
Ki = 8.71 nM
|
|
|
|
CP0413084
|
1-azabicyclo[2.2.2]octan-3-yl N-[2-(4-methoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C23H28N2O3
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0874916
|
2-(5-(cyclohexyl(hydroxy)(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO2
|
1
|
| 1 |
Ki = 11.48 nM
|
|
|
|
CP0880938
|
(S)-2-(5-((R)-cyclohexyl(hydroxy)(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO2
|
1
|
| 1 |
Ki = 12.02 nM
|
|
|
|
CP0062485
|
4-(Diethylamino)-2-butynyl alpha-phenylcyclohexaneglycolic acid ester
Show/Hide
|
C22H31NO3
|
1
|
| 1 |
Ki = 14.13 nM
|
|
|
|
CP0858486
|
2-(5-(cyclohexyl(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO
|
1
|
| 1 |
Ki = 15.49 nM
|
|
|
|
CP0398877
|
(R)-cyclohexyl-[5-[(2S)-1-methylpyrrolidin-2-yl]furan-2-yl]-phenylmethanol
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 27.54 nM
|
|
|
|
CP0886180
|
N-(2-{2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethylcarbamoyl}-ethyl)-3,3,3-triphenyl-propionamide
Show/Hide
|
C40H52N4O3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0413078
|
(3-fluoro-4-methylphenyl)methyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H25FN2O2
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0406146
|
1-[3-[4-[13-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]tridecyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C38H59N5O2S
|
1
|
| 1 |
Ki = 30.9 nM
|
|
|
|
CP0858619
|
2-(5-benzhydrylfuran-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H26INO
|
1
|
| 1 |
Ki = 31.62 nM
|
|
|
|
CP0058613
|
CAS_132947
Show/Hide
|
C64H77N13O6
|
1
|
| 1 |
Ki = 33.88 nM
|
|
|
|
CP0847176
|
N-({2-[(1-Cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethylcarbamoyl}-methyl)-3,3,3-triphenyl-propionamide
Show/Hide
|
C39H50N4O3
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0917620
|
2-(5-(hydroxydiphenylmethyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H26INO2
|
1
|
| 1 |
Ki = 37.15 nM
|
|
|
|
CP0413081
|
1,3-benzodioxol-5-ylmethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H24N2O4
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0413083
|
(3-fluoro-4-methoxyphenyl)methyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H25FN2O3
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0413481
|
1-[3-[4-[9-[1-[3-(2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]nonyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C43H64N4O2
|
1
|
| 1 |
Ki = 48.98 nM
|
|
|
|
CP0510568
|
1-[4-(2-methylimidazol-1-yl)but-2-ynyl]pyrrolidin-2-one
Show/Hide
|
C12H15N3O
|
1
|
| 1 |
Ki = 51.29 nM
|
|
|
|
CP0388205
|
2-[5-[cyclohexyl(phenyl)methyl]furan-2-yl]-1-methylpyrrolidine
Show/Hide
|
C22H29NO
|
1
|
| 1 |
Ki = 54.95 nM
|
|
|
|
CP0849742
|
1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carboxylic acid {2-[(1-cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-ethyl}-amide
Show/Hide
|
C42H54N4O3
|
1
|
| 1 |
Ki = 58 nM
|
|
|
|
CP0413080
|
(1-methylpiperidin-4-yl) N-[2-(4-fluorophenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C21H25FN2O2
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0413082
|
(3,4-dichlorophenyl)methyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C21H22Cl2N2O2
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0413087
|
1-azabicyclo[2.2.2]octan-3-yl N-[2-(3,4-dimethoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C24H30N2O4
|
1
|
| 1 |
Ki = 65 nM
|
|
|
|
CP0416523
|
2-(3,4-dichlorophenyl)ethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H24Cl2N2O2
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0875623
|
(R)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine Oxalate
Show/Hide
|
C21H25NO6
|
1
|
| 1 |
Ki = 81.28 nM
|
|
|
|
CP0431004
|
[5-(1-methylpyrrolidin-2-yl)furan-2-yl]-diphenylmethanol
Show/Hide
|
C22H23NO2
|
1
|
| 1 |
Ki = 97.72 nM
|
|
|
|
CP0413079
|
3-(3,4-difluorophenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H26F2N2O2
|
1
|
| 1 |
Ki = 100 nM
|
|
|
|
CP0399526
|
1-[3-[4-[3-[[4-(1-methyl-3,6-dihydro-2H-pyridin-5-yl)-1,2,5-thiadiazol-3-yl]oxy]propyl]piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C28H39N5O2S
|
1
|
| 1 |
Ki = 102.33 nM
|
|
|
|
CP0439204
|
2-(5-benzhydrylfuran-2-yl)-1-methylpyrrolidine
Show/Hide
|
C22H23NO
|
1
|
| 1 |
Ki = 104.71 nM
|
|
|
|
CP0858903
|
(R)-(6,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 107.15 nM
|
|
|
|
CP0413077
|
3-(3,4-dichlorophenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H26Cl2N2O2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0416520
|
3-(3-fluoro-4-methylphenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C24H29FN2O2
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0849054
|
1-[1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carbonyl]-pyrrolidine-2-carboxylic acid (1-cyclohexylmethyl-piperidin-3-ylmethyl)-amide
Show/Hide
|
C44H56N4O3
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0440614
|
(1-methylpiperidin-3-yl) N-[2-(4-fluorophenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C21H25FN2O2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0440616
|
benzyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0469418
|
(1-methylpiperidin-4-yl) N-[2-(4-methoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C22H28N2O3
|
1
|
| 1 |
Ki = 190 nM
|
|
|
|
CP0377612
|
N-[3-[[1-(cyclohexylmethyl)piperidin-3-yl]methylamino]-3-oxopropyl]-4-(3,3,3-triphenylpropanoylamino)butanamide
Show/Hide
|
C41H54N4O3
|
1
|
| 1 |
Ki = 200 nM
|
|
|
|
CP0859758
|
6-(3,3,3-Triphenyl-propionylamino)-hexanoic acid (1-cyclohexylmethyl-piperidin-3-ylmethyl)-amide
Show/Hide
|
C40H53N3O2
|
1
|
| 1 |
Ki = 210 nM
|
|
|
|
CP0859818
|
(R)-2-(5-((S)-cyclohexyl(hydroxy)(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO2
|
1
|
| 1 |
Ki = 229.09 nM
|
|
|
|
CP0440618
|
2-(4-methoxyphenyl)ethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H28N2O3
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0416527
|
2-(1,3-benzodioxol-5-yl)ethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H26N2O4
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0440621
|
[(1R,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] N-[2-(4-methoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C24H30N2O3
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0416522
|
3-phenylpropyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H28N2O2
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0416526
|
2-phenylethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0518455
|
3-(3-fluoro-4-methoxyphenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C24H29FN2O3
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0543664
|
N-ethyl-2,2-dimethyl-N-[3-[1-[2-oxo-2-(6-oxo-5H-benzo[b][1,4]benzodiazepin-11-yl)ethyl]piperidin-4-yl]propyl]pentanamide
Show/Hide
|
C32H44N4O3
|
1
|
| 1 |
Ki = 316.23 nM
|
|
|
|
CP0413482
|
1-[3-[4-(13-hydroxytridecyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C30H50N2O2
|
1
|
| 1 |
Ki = 338.84 nM
|
|
|
|
CP0378643
|
1-[3-[4-(11-hydroxyundecyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C28H46N2O2
|
1
|
| 1 |
Ki = 346.74 nM
|
|
|
|
CP0411349
|
(1-methyl-4-phenylpiperidin-4-yl)methyl 3-(4-methoxyphenyl)propanoate
Show/Hide
|
C23H29NO3
|
1
|
| 1 |
Ki = 380 nM
|
|
|
|
CP0459315
|
(1-methylpiperidin-4-yl) N-[2-(3,4-dimethoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C23H30N2O4
|
1
|
| 1 |
Ki = 380 nM
|
|
|
|
CP0388200
|
(S)-cyclohexyl-[5-[(2R)-1-methylpyrrolidin-2-yl]furan-2-yl]-phenylmethanol
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 467.74 nM
|
|
|
|
CP0416518
|
(4-methoxyphenyl)methyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C22H26N2O3
|
1
|
| 1 |
Ki = 470 nM
|
|
|
|
CP0378256
|
ethyl 7-benzyl-6-ethyl-17-methoxy-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C31H32N2O4
|
1
|
| 1 |
Ki = 478.63 nM
|
|
|
|
CP0392367
|
prop-2-enyl 17-methoxy-7-[(4-methoxyphenyl)methyl]-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C32H32N2O5
|
1
|
| 1 |
Ki = 501.19 nM
|
|
|
|
CP0459833
|
2-(4-(pyrrolidin-1-yl)but-2-ynyl)isoxazolidin-3-one
Show/Hide
|
C11H16N2O2
|
1
|
| 1 |
Ki = 510 nM
|
|
|
|
CP0217520
|
AF-DX 384
Show/Hide
|
C27H38N6O2
|
1
|
| 1 |
Ki = 537.03 nM
|
|
|
|
CP0880166
|
2-(4-Piperidin-1-ylbut-2-yn-1-yl)isoxazolidin-3-one oxalate
Show/Hide
|
C14H20N2O6
|
1
|
| 1 |
Ki = 544 nM
|
|
|
|
CP0416519
|
(3,4-dimethoxyphenyl)methyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C23H28N2O4
|
1
|
| 1 |
Ki = 550 nM
|
|
|
|
CP0416517
|
3-(4-methoxyphenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C24H30N2O3
|
1
|
| 1 |
Ki = 640 nM
|
|
|
|
CP0393635
|
1-[3-[4-(2-phenylethyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C25H32N2O
|
1
|
| 1 |
Ki = 758.58 nM
|
|
|
|
CP0514143
|
CAS_91533
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 794.33 nM
|
|
|
|
CP0378645
|
1-[3-[4-(9-hydroxynonyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C26H42N2O2
|
1
|
| 1 |
Ki = 851.14 nM
|
|
|
|
CP0381401
|
2-(4-methoxyphenyl)ethyl 1-methyl-4-phenylpiperidine-4-carboxylate
Show/Hide
|
C22H27NO3
|
1
|
| 1 |
Ki = 870 nM
|
|
|
|
CP0860901
|
(S)-2-(5-((S)-cyclohexyl(hydroxy)(phenyl)methyl)furan-2-yl)-1,1-dimethylpyrrolidinium iodide
Show/Hide
|
C23H32INO2
|
1
|
| 1 |
Ki = 870.96 nM
|
|
|
|
CP0139206
|
Arecaidine Propargyl Ester
Show/Hide
|
C10H13NO2
|
1
|
| 1 |
Ki = 933.25 nM
|
|
|
|
CP0467303
|
(2R)-N-(1-cyclopentylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide
Show/Hide
|
C43H51F3N4O4
|
1
|
| 1 |
Ki = 940 nM
|
|
|
|
CP0390496
|
(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide
Show/Hide
|
C38H43Cl3N4O4
|
1
|
| 1 |
Ki = 950 nM
|
|
|
|
CP0378979
|
1-azabicyclo[2.2.2]octan-3-yl (3E)-3-(pyridin-2-ylmethylidene)indene-1-carboxylate
Show/Hide
|
C23H22N2O2
|
1
|
| 1 |
Ki = 977.24 nM
|
|
|
|
CP0467135
|
1-azabicyclo[2.2.2]octan-3-yl (3E)-3-(pyridin-4-ylmethylidene)indene-1-carboxylate
Show/Hide
|
C23H22N2O2
|
1
|
| 1 |
Ki = 1047.13 nM
|
|
|
|
CP0440617
|
(1-methylpiperidin-3-yl) N-[2-(4-methoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C22H28N2O3
|
1
|
| 1 |
Ki = 1050 nM
|
|
|
|
CP0404810
|
N-[[1-(cyclohexylmethyl)piperidin-3-yl]methyl]-4-[[2-(3,3,3-triphenylpropanoylamino)acetyl]amino]butanamide
Show/Hide
|
C40H52N4O3
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0377555
|
5-benzyl-17-methoxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene
Show/Hide
|
C27H26N2O2
|
1
|
| 1 |
Ki = 1122.02 nM
|
|
|
|
CP0392482
|
benzyl 17-methoxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C28H26N2O4
|
1
|
| 1 |
Ki = 1122.02 nM
|
|
|
|
CP0403333
|
1-azabicyclo[2.2.2]octan-3-yl (3E)-3-(pyridin-3-ylmethylidene)indene-1-carboxylate
Show/Hide
|
C23H22N2O2
|
1
|
| 1 |
Ki = 1230.27 nM
|
|
|
|
CP0225899
|
AQ-RA 741
Show/Hide
|
C27H37N5O2
|
1
|
| 1 |
Ki = 1258.93 nM
|
|
|
|
CP0413085
|
[(1R,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] N-[2-(3,4-dimethoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
|
C25H32N2O4
|
1
|
| 1 |
Ki = 1370 nM
|
|
|
|
CP0392351
|
ethyl 6-butyl-17-methylsulfanyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C26H30N2O3S
|
1
|
| 1 |
Ki = 1479.11 nM
|
|
|
|
CP0443229
|
(S)-cyclohexyl-[5-[(2S)-1-methylpyrrolidin-2-yl]furan-2-yl]-phenylmethanol
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 1548.82 nM
|
|
|
|
CP0394158
|
(2R)-N-(1-cyclopropylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1 -[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide
Show/Hide
|
C41H47F3N4O4
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0408072
|
(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine -2-yl)-carbonyl-N-(1-methyl-4-piperidinylmethyl)pyrrolidine-2-carboxamide
Show/Hide
|
C38H43F3N4O4
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0440620
|
3-(3,4-dimethoxyphenyl)propyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
|
C25H32N2O4
|
1
|
| 1 |
Ki = 1610 nM
|
|
|
|
CP0425298
|
ethyl 7-methyl-17-methylsulfanyl-6-propyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C26H30N2O3S
|
1
|
| 1 |
Ki = 1698.24 nM
|
|
|
|
CP0376654
|
(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-[(3R)-3-piperidinylmethyl]-pyrrolidine-2-carboxamide
Show/Hide
|
C37H41F3N4O4
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0458127
|
(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide
Show/Hide
|
C38H43F3N4O4
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0401417
|
3-(4-methoxyphenyl)-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]propanamide
Show/Hide
|
C23H30N2O2
|
1
|
| 1 |
Ki = 1810 nM
|
|
|
|
CP0858930
|
5-phenyl-3-[(4-pyrrolidin-1-ylbut-2-yn-1-yl)oxy]isoxazole methiodide
Show/Hide
|
C18H21IN2O2
|
1
|
| 1 |
Ki = 1836 nM
|
|
|
|
CP0407747
|
ethyl 6-methyl-17-methylsulfanyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C23H24N2O3S
|
1
|
| 1 |
Ki = 1949.84 nM
|
|
|
|
CP0393633
|
1-[3-(4-propylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C20H30N2O
|
1
|
| 1 |
Ki = 1949.84 nM
|
|
|
|
CP0860436
|
1-(3,3,3-Triphenyl-propionyl)-pyrrolidine-2-carboxylic acid {[(1-cyclohexylmethyl-piperidin-3-ylmethyl)-carbamoyl]-methyl}-amide
Show/Hide
|
C41H52N4O3
|
1
|
| 1 |
Ki = 2000 nM
|
|
|
|
CP0489929
|
1-[3-(4-phenylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 2041.74 nM
|
|
|
|
CP0447909
|
2-(4-methoxyphenyl)ethyl N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]carbamate
Show/Hide
|
C23H30N2O3
|
1
|
| 1 |
Ki = 2050 nM
|
|
|
|
CP0374692
|
(1-methyl-4-phenylpiperidin-4-yl)methyl 3-(3,4-dimethoxyphenyl)propanoate
Show/Hide
|
C24H31NO4
|
1
|
| 1 |
Ki = 2140 nM
|
|
|
|
CP0376946
|
prop-2-enyl 17-methoxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C24H24N2O4
|
1
|
| 1 |
Ki = 2238.72 nM
|
|
|
|
CP0404800
|
ethyl 17-methoxy-6-propyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C25H28N2O4
|
1
|
| 1 |
Ki = 2238.72 nM
|
|
|
|
CP0425884
|
2-(3,4-dimethoxyphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H27NO4
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1
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| 1 |
Ki = 2240 nM
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CP0129619
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N-[3-[2-[[(6S)-2-amino-4,5,6,7-tetrahydro-1,3-benzothiazol-6-yl]-propylamino]ethyl]-3-hydroxycyclobutyl]naphthalene-2-carboxamide
Show/Hide
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C27H34N4O2S
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1
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| 1 |
Ki = 2297 nM
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CP0459891
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ethyl 17-methylsulfanyl-6-propyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C25H28N2O3S
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1
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| 1 |
Ki = 2398.83 nM
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CP0073146
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benzyl 7-(4-cyclopentylpiperazin-1-yl)-3,4-dihydro-1H-isoquinoline-2-carboxylate
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C26H33N3O2
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1
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| 1 |
Ki = 2471 nM
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CP0376043
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(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide
Show/Hide
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C37H41Cl3N4O4
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1
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| 1 |
Ki = 2500 nM
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CP0382995
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butyl 17-methoxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C25H28N2O4
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1
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| 1 |
Ki = 2511.89 nM
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CP0409101
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ethyl 7-ethyl-17-methoxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C25H28N2O4
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1
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| 1 |
Ki = 2511.89 nM
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CP0389578
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benzyl 7-[4-(3-ethoxy-3-oxopropyl)piperazin-1-yl]-3,4-dihydro-1H-isoquinoline-2-carboxylate
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C26H33N3O4
|
1
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| 1 |
Ki = 2591 nM
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CP0431973
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(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-chlorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-((3R)-3-piperidinylmethyl)-pyrrolidine-2-carboxamide
Show/Hide
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C37H41Cl3N4O4
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1
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| 1 |
Ki = 2700 nM
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CP0390498
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(2R)-N-(1-ethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide
Show/Hide
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C39H45F3N4O4
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1
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| 1 |
Ki = 2800 nM
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CP0480403
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ethyl 6-ethyl-17-methoxy-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C24H26N2O4
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1
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| 1 |
Ki = 3090.3 nM
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CP0492196
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ethyl 6-ethyl-17-methoxy-7-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C25H28N2O4
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1
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| 1 |
Ki = 3090.3 nM
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CP0393625
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1-[3-[4-(7-hydroxyheptyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C24H38N2O2
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1
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| 1 |
Ki = 3090.3 nM
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CP0390495
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(2R)-N-(1-cyclobutylmethyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide
Show/Hide
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C42H49F3N4O4
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1
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| 1 |
Ki = 3100 nM
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CP0394494
|
Milameline
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C8H14N2O
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1
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| 1 |
Ki = 3162.28 nM
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CP0895036
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2-(2-Furyl)-1-methylpyrrolidineMethiodide
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C10H16INO
|
1
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| 1 |
Ki = 3162.28 nM
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CP0393859
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(2R)-N-(1-cyclopentyl-4-piperidinylmethyl)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)-propanoyl]pyrrolidine-2-yl)carbonylpyrrolidine-2-carboxamide
Show/Hide
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C42H49F3N4O4
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1
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| 1 |
Ki = 3200 nM
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CP0393079
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ethyl 17-methoxy-7-methyl-6-propyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C26H30N2O4
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1
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| 1 |
Ki = 3388.44 nM
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CP0413086
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2-(3,4-dimethoxyphenyl)ethyl N-(1-azabicyclo[2.2.2]octan-3-yl)-N-phenylcarbamate
Show/Hide
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C24H30N2O4
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1
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| 1 |
Ki = 3490 nM
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CP0085414
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(3aS,6R,6aS,9aR,9bR)-6-benzyl-1-methyl-3,3a,4,6,6a,7,8,9,9a,9b-decahydro-2H-benzo[de]quinolin-5-one
Show/Hide
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C20H27NO
|
1
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| 1 |
Ki = 3493 nM
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CP0067391
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(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide
Show/Hide
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C37H41F3N4O4
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1
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| 1 |
Ki = 3500 nM
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CP0411640
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1-[3-(4-pentylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
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C22H34N2O
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1
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| 1 |
Ki = 3548.13 nM
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CP0415357
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methyl 17-methoxy-6,7-dimethyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C23H24N2O4
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1
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| 1 |
Ki = 3630.78 nM
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CP0870440
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(S)-1,1-Dimethyl-2-(5-methyl-furan-2-yl)-pyrrolidinium
Show/Hide
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C11H18INO
|
1
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| 1 |
Ki = 3630.78 nM
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CP0377061
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ethyl 17-methoxy-6,7-dimethyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C24H26N2O4
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1
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| 1 |
Ki = 3715.35 nM
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CP0394502
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trimethyl-[[(2R,6S)-6-methyl-1,4-dioxan-2-yl]methyl]azanium
Show/Hide
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C9H20NO2+
|
1
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| 1 |
Ki = 3715.35 nM
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CP0116478
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1-[3-(4-benzylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C24H30N2O
|
1
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| 1 |
Ki = 3715.35 nM
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CP0848084
|
[4-(4-chloro-phenylcarbamoyloxy)-but-2-ynyl]-trimethyl-ammonium chloride
Show/Hide
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C14H18Cl2N2O2
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1
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| 1 |
Ki = 3801.89 nM
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CP0773921
|
SID50106034
Show/Hide
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C14H18Cl2N2O2
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1
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| 1 |
Ki = 3801.89 nM
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CP0423369
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(McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2-ynyl]-trimethyl-ammonium; chloride
Show/Hide
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C14H18ClN2O2+
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1
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| 1 |
Ki = 3801.89 nM
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CP0880167
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1-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]piperidine methiodide
Show/Hide
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C13H21IN2O2
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1
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| 1 |
Ki = 4116 nM
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CP0530916
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1-[2-(4-methoxyphenyl)ethyl]-3-[(1-methyl-4-phenylpiperidin-4-yl)methyl]urea
Show/Hide
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C23H31N3O2
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1
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| 1 |
Ki = 4300 nM
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CP0440615
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(1-methylpiperidin-3-yl) N-[2-(3,4-dimethoxyphenyl)ethyl]-N-phenylcarbamate
Show/Hide
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C23H30N2O4
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1
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| 1 |
Ki = 4490 nM
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CP0845388
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Cis-N,N,N-trimethyl-1-((2R,6S)-6-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
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C9H20INO2
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2
|
| 1 |
Ki = 4570.88 nM
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| 2 |
Ki = 7762.47 nM
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CP0378647
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1-[3-[4-(5-hydroxypentyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C22H34N2O2
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1
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| 1 |
Ki = 4570.88 nM
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CP0895034
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2-(5-Methyl-2-furyl)-1-methylpyrrolidine Methiodide
Show/Hide
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C11H18INO
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1
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| 1 |
Ki = 4677.35 nM
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CP0377554
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ethyl 15-chloro-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C22H21ClN2O3
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1
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| 1 |
Ki = 4786.3 nM
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CP0880168
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1-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]piperidine oxalate
Show/Hide
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C14H20N2O6
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1
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| 1 |
Ki = 5139 nM
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CP0404711
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ethyl 17-chloro-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C22H21ClN2O3
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1
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| 1 |
Ki = 5370.32 nM
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CP0474634
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ethyl 17-methoxy-6-pentyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
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C27H32N2O4
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1
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| 1 |
Ki = 5370.32 nM
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CP0232092
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1-[3-(4-butylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C21H32N2O
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1
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| 1 |
Ki = 5370.32 nM
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CP0374693
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(1-methyl-4-phenylpiperidin-4-yl)methyl N-[2-(3,4-dimethoxyphenyl)ethyl]carbamate
Show/Hide
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C24H32N2O4
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1
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| 1 |
Ki = 5410 nM
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CP0858932
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2-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]-1,2,3,4-tetrahydroisoquinoline methiodide
Show/Hide
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C17H21IN2O2
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1
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| 1 |
Ki = 5664 nM
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CP0472845
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1-[3-(4-benzylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C23H29N3O
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1
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| 1 |
Ki = 6025.6 nM
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CP0402148
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17-methoxy-6-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene
Show/Hide
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C23H22N4O3
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1
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| 1 |
Ki = 6165.95 nM
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CP0900137
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N,N-dimethyl-4-[(5-methylisoxazol-3-yl)oxy]but-2-yn-1-amine methiodide
Show/Hide
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C11H17IN2O2
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1
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| 1 |
Ki = 6310 nM
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CP0858931
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5-phenyl-3-[(4-pyrrolidin-1-ylbut-2-yn-1-yl)oxy]-isoxazole fumarate
Show/Hide
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C21H22N2O6
|
1
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| 1 |
Ki = 6885 nM
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CP0249974
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5-methylfurmethide
Show/Hide
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C9H16NO+
|
1
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| 1 |
Ki = 6918.31 nM
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CP0374691
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2-(3,4-dimethoxyphenyl)ethyl 1-methyl-4-phenylpiperidine-4-carboxylate
Show/Hide
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C23H29NO4
|
1
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| 1 |
Ki = 6950 nM
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CP0381400
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N-[2-(4-methoxyphenyl)ethyl]-1-methyl-4-phenylpiperidine-4-carboxamide
Show/Hide
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C22H28N2O2
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1
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| 1 |
Ki = 6970 nM
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CP0873039
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5-methyl-3-[(4-pyrrolidin-1-ylbut-2-yn-1-yl)oxy]isoxazole methiodide
Show/Hide
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C13H19IN2O2
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1
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| 1 |
Ki = 7514 nM
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CP0878023
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Cis-((2R*,6S*)-6-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
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C21H28INO2
|
1
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| 1 |
Ki = 7585.78 nM
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CP0393626
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1-[3-[4-(2-phenylethyl)piperazin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C24H31N3O
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1
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| 1 |
Ki = 7943.28 nM
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CP0411642
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1-[3-(4-butylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
Show/Hide
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C20H31N3O
|
1
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| 1 |
Ki = 9120.11 nM
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CP0845041
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(R)-1,1-Dimethyl-2-(5-methyl-furan-2-yl)-pyrrolidinium
Show/Hide
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C11H18INO
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1
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| 1 |
Ki = 9549.93 nM
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CP0876609
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1-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]indoline methiodide
Show/Hide
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C16H19IN2O2
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1
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| 1 |
Ki > 10000 nM
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CP0881243
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2-[4-(8-azabicyclo[3.2.1]oct-8-yl)but-2-yn-1-yl]isoxazolidin-3-one hydrochloride
Show/Hide
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C14H21ClN2O2
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1
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| 1 |
Ki > 10000 nM
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CP0881244
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2-(4-piperidin-1-ylbut-2-yn-1-yl)isoxazolidin-3-one methiodide
Show/Hide
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C13H21IN2O2
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1
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| 1 |
Ki > 10000 nM
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CP0886548
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5-methyl-3-[(4-pyrrolidin-1-ylbut-2-yn-1-yl)oxy]-isoxazole fumarate
Show/Hide
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C16H20N2O6
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1
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| 1 |
Ki > 10000 nM
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CP0886549
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2-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]-1,2,3,4-tetrahydroisoquinoline oxalate
Show/Hide
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C18H20N2O6
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1
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| 1 |
Ki > 10000 nM
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CP0894494
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1-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]indoline hydrochloride
Show/Hide
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C15H17ClN2O2
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1
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| 1 |
Ki > 10000 nM
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CP0894495
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2-[4-(3,4-dihydroisoquinolin-2(1H)-yl)but-2-yn-1-yl]isoxazolidin-3-one methiodide
Show/Hide
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C17H21IN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0897808
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N,N-dimethyl-4-[(5-methylisoxazol-3-yl)oxy]-but-2-yn-1-amine fumarate
Show/Hide
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C14H18N2O6
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1
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| 1 |
Ki > 10000 nM
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CP0897809
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8-[4-(4,5-dihydroisoxazol-3-yloxy)but-2-yn-1-yl]-8-azabicyclo[3.2.1]octane oxalate
Show/Hide
|
C16H22N2O5
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1
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| 1 |
Ki > 10000 nM
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CP0910936
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quinuclidin-3-one O-[4-(isoxazol-3-yloxy)but-2-yn-1-yl]oxime methiodide
Show/Hide
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C15H20IN3O3
|
1
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| 1 |
Ki > 10000 nM
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CP0910938
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N,N-dimethyl-4-[(5-phenylisoxazol-3-yl)oxy]but-2-yn-1-amine oxalat
Show/Hide
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C17H18N2O6
|
1
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| 1 |
Ki > 10000 nM
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CP0918257
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2-[4-(3,4-dihydroisoquinolin-2(1H)-yl)but-2-yn-1-yl]isoxazolidin-3-one oxalate
Show/Hide
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C18H20N2O6
|
1
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| 1 |
Ki > 10000 nM
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CP0920153
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2-[4-(2,3-dihydro-1H-indol-1-yl)but-2-yn-1-yl]isoxazolidin-3-one methiodide
Show/Hide
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C16H19IN2O2
|
1
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| 1 |
Ki > 10000 nM
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CP0002070
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1-(1H-Indol-3-yl)-2-propanamine
Show/Hide
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C11H14N2
|
1
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| 1 |
Ki > 10000 nM
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CP0002071
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N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-prop-2-enylprop-2-en-1-amine
Show/Hide
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C17H22N2O
|
1
|
| 1 |
Ki > 10000 nM
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CP0635067
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2-amino-6-chloro-3,4-dihydroquinazoline hydrochloride
Show/Hide
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C8H9Cl2N3
|
1
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| 1 |
Ki > 10000 nM
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CP0401297
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3-(3,4-dimethoxyphenyl)-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]propanamide
Show/Hide
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C24H32N2O3
|
1
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| 1 |
Ki > 10000 nM
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CP0431550
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1-[2-(3,4-dimethoxyphenyl)ethyl]-3-[(1-methyl-4-phenylpiperidin-4-yl)methyl]urea
Show/Hide
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C24H33N3O3
|
1
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| 1 |
Ki > 10000 nM
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CP0054519
|
(1R,12R,13S,17R,21S)-12-ethyl-18-propyl-7-(trifluoromethyl)-10,18-diazapentacyclo[11.7.1.02,11.04,9.017,21]henicosa-2(11),3,5,7,9-pentaene
Show/Hide
|
C25H31F3N2
|
1
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| 1 |
Ki > 10000 nM
|
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CP0387083
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(3aS,9bS)-3a-methyl-5-phenyl-2,3,4,9b-tetrahydro-1H-pyrrolo[2,3-c]quinoline
Show/Hide
|
C18H20N2
|
1
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| 1 |
Ki > 10000 nM
|
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CP0391120
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(1S,2R)-1-ethyl-7-methoxy-2-methyl-3,4-dihydro-1H-naphthalen-2-amine
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0391121
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(3S,4S)-4-ethyl-3,6-dimethyl-2,4-dihydrochromen-3-amine
Show/Hide
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C13H19NO
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0391154
|
(3aS,9bS)-7,9-dimethoxy-3a-methyl-2,3,4,9b-tetrahydro-1H-chromeno[3,4-b]pyrrole
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C14H19NO3
|
1
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| 1 |
Ki > 10000 nM
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CP0411059
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(3S,4S)-4-ethyl-3-methyl-1-phenyl-2,4-dihydroquinolin-3-amine
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C18H22N2
|
1
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| 1 |
Ki > 10000 nM
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CP0089021
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(+)-pilocarpine
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C11H16N2O2
|
1
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| 1 |
Ki = 10232.93 nM
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CP0373254
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(2S)-1,1-dimethyl-2-[(2S,5S)-2-methyl-1,3-oxathiolan-5-yl]pyrrolidin-1-ium
Show/Hide
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C10H20NOS+
|
1
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| 1 |
Ki = 10232.93 nM
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CP0916821
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Cis-N,N,N-Trimethyl((2R*,6S*)-6-phenyl-1,4-dioxan-2-yl)methanaminium Iodide
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C14H22INO2
|
1
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| 1 |
Ki = 10232.93 nM
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CP0462684
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(2R)-1,1-dimethyl-2-[(2S,5S)-2-methyl-1,3-oxathiolan-5-yl]pyrrolidin-1-ium
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C10H20NOS+
|
1
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| 1 |
Ki = 10715.19 nM
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CP0067390
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ethyl 6-butyl-17-methoxy-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
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C26H30N2O4
|
1
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| 1 |
Ki = 11220.18 nM
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CP0412497
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trimethyl-[[(2R,5R)-2-methyl-1,3-oxathiolan-5-yl]methyl]azanium
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C8H18NOS+
|
1
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| 1 |
Ki = 13182.57 nM
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CP0379138
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1-[3-[4-(3-hydroxypropyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
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C20H30N2O2
|
1
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| 1 |
Ki = 14454.4 nM
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CP0859714
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((2R*,5S*,6S*)-5,6-Dimethyl-1,4-dioxan-2-yl)-N,N,Ntrimethylmethanaminium iodide
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C10H22INO2
|
1
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| 1 |
Ki = 15488.17 nM
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CP0509683
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(2R)-2-(5-methylfuran-2-yl)pyrrolidine
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C9H13NO
|
1
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| 1 |
Ki = 15848.93 nM
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CP0902206
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N,N,N-Trimethyl((2R*,5S*)-5,6,6-trimethyl-1,4-dioxan-2-yl)methanaminium iodide
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C11H24INO2
|
1
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| 1 |
Ki = 16595.87 nM
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CP0497956
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2-(furan-2-yl)pyrrolidine
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C8H11NO
|
1
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| 1 |
Ki = 16595.87 nM
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CP0393421
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2-(dimethylamino)ethyl (3E)-3-(pyridin-2-ylmethylidene)indene-1-carboxylate
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C20H20N2O2
|
1
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| 1 |
Ki = 17782.79 nM
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CP0409674
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N,N-dimethyl-2-[(3E)-3-(pyridin-2-ylmethylidene)inden-1-yl]ethanamine
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C19H20N2
|
1
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| 1 |
Ki = 19054.61 nM
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CP0876494
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2-(5-Methyl-2-furyl)-pyrrolidine
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C9H13NO
|
1
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| 1 |
Ki = 19054.61 nM
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CP0376953
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N-ethyl-17-methoxy-N,6-dimethyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxamide
Show/Hide
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C24H27N3O3
|
1
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| 1 |
Ki = 19498.45 nM
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CP0895035
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(S)-2-Furan-2-yl-1,1-dimethyl-pyrrolidinium
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C10H16INO
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1
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| 1 |
Ki = 20892.96 nM
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CP0386217
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(+)-CIS-DIOXOLANE
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C8H18NO2+
|
1
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| 1 |
Ki = 21877.62 nM
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CP0898948
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2-(5-Methyl-2-furyl)-1-methylpyrrolidine
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C10H15NO
|
1
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| 1 |
Ki = 21877.62 nM
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CP0848059
|
SID855871
Show/Hide
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C8H18INO2
|
1
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| 1 |
Ki = 21877.62 nM
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CP0394497
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(2S)-1,1-dimethyl-2-[(2S,4R)-2-methyl-1,3-dioxolan-4-yl]pyrrolidin-1-ium
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C10H20NO2+
|
1
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| 1 |
Ki = 22908.68 nM
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CP0407925
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(2S)-1,1-dimethyl-2-[(2R,5R)-2-methyl-1,3-oxathiolan-5-yl]pyrrolidin-1-ium
Show/Hide
|
C10H20NOS+
|
1
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| 1 |
Ki = 23442.29 nM
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CP0910892
|
(R)-2-Furan-2-yl-1,1-dimethyl-pyrrolidinium
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C10H16INO
|
1
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| 1 |
Ki = 23442.29 nM
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CP0393627
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1-[3-(4-methylpiperidin-1-yl)propyl]-3,4-dihydroquinolin-2-one
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C18H26N2O
|
1
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| 1 |
Ki = 23988.33 nM
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CP0485774
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(2R)-1,1-dimethyl-2-[(2R,5R)-2-methyl-1,3-oxathiolan-5-yl]pyrrolidin-1-ium
Show/Hide
|
C10H20NOS+
|
1
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| 1 |
Ki = 24547.09 nM
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CP0877929
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Cis-((2R*,6S*)-6-Ethyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
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C10H22INO2
|
1
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| 1 |
Ki = 26302.68 nM
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CP0379047
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2-(dimethylamino)ethyl (3E)-3-(pyridin-4-ylmethylidene)indene-1-carboxylate
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C20H20N2O2
|
1
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| 1 |
Ki = 26915.35 nM
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CP0449315
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N,N-dimethyl-2-[(3E)-3-(pyridin-3-ylmethylidene)inden-1-yl]ethanamine
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C19H20N2
|
1
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| 1 |
Ki = 26915.35 nM
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CP0232093
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1-[3-(4-phenylpiperazin-1-yl)propyl]-3,4-dihydroquinolin-2-one
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C22H27N3O
|
1
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| 1 |
Ki = 27542.29 nM
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CP0409139
|
ethyl 6-hexyl-17-methoxy-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C28H34N2O4
|
1
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| 1 |
Ki > 28183.83 nM
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CP0431291
|
ethyl 17-hydroxy-6-methyl-12-oxa-1,7-diazapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),5,9,14(19),15,17-heptaene-5-carboxylate
Show/Hide
|
C22H22N2O4
|
1
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| 1 |
Ki > 28183.83 nM
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CP0859477
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(6,6-Dimethyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium iodide
Show/Hide
|
C10H22INO2
|
1
|
| 1 |
Ki = 28183.83 nM
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CP0447908
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N-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-4-phenylpiperidine-4-carboxamide
Show/Hide
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C23H30N2O3
|
1
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| 1 |
Ki > 30000 nM
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CP0410895
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2-(dimethylamino)ethyl (3E)-3-(pyridin-3-ylmethylidene)indene-1-carboxylate
Show/Hide
|
C20H20N2O2
|
1
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| 1 |
Ki = 30199.52 nM
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CP0474436
|
trimethyl-[[(2S,6S)-6-methyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C9H20NO2+
|
1
|
| 1 |
Ki = 30199.52 nM
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CP0372804
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(2R)-2-(furan-2-yl)pyrrolidine
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C8H11NO
|
1
|
| 1 |
Ki = 31622.78 nM
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CP0372904
|
(2R)-1-methyl-2-(5-methylfuran-2-yl)pyrrolidine
Show/Hide
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C10H15NO
|
1
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| 1 |
Ki = 31622.78 nM
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CP0895136
|
Trans-((2R*,6R*)-6-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
|
C21H28INO2
|
1
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| 1 |
Ki = 31622.78 nM
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CP0859660
|
N,N,N-Trimethyl((2R*,5R*)-5,6,6-trimethyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C11H24INO2
|
1
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| 1 |
Ki = 32359.37 nM
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CP0875624
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Trans-N,N,N-Trimethyl((2R*,6R*)-6-phenyl-1,4-dioxan-2-yl)methanaminium Iodide
Show/Hide
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C14H22INO2
|
1
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| 1 |
Ki = 33113.11 nM
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CP0455031
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(2R,3R,5R)-5-[(2S)-1,1-dimethylpyrrolidin-1-ium-2-yl]-2-methyl-1,3-oxathiolane 3-oxide;iodide
Show/Hide
|
C10H20INO2S
|
1
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| 1 |
Ki = 33884.42 nM
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CP0433872
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(2S)-1-methyl-2-(5-methylfuran-2-yl)pyrrolidine
Show/Hide
|
C10H15NO
|
1
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| 1 |
Ki = 39810.72 nM
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CP0848060
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(R)-1-(1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium iodide
Show/Hide
|
C8H18INO2
|
1
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| 1 |
Ki = 41686.94 nM
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CP0371717
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trimethyl-[[(2S,6R)-6-methyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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|
C9H20NO2+
|
1
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| 1 |
Ki = 44668.36 nM
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CP0910891
|
2-(2-Furyl)-1-methylpyrrolidine
Show/Hide
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C9H13NO
|
1
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| 1 |
Ki = 44668.36 nM
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CP0372805
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(2S)-2-(furan-2-yl)pyrrolidine
Show/Hide
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C8H11NO
|
1
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| 1 |
Ki = 47863.01 nM
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CP0374978
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(3E)-N-[2-(dimethylamino)ethyl]-N-methyl-3-(pyridin-2-ylmethylidene)indene-1-carboxamide
Show/Hide
|
C21H23N3O
|
1
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| 1 |
Ki = 52480.75 nM
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CP0412496
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(2R)-1,1-dimethyl-2-[(2S,4R)-2-methyl-1,3-dioxolan-4-yl]pyrrolidin-1-ium
Show/Hide
|
C10H20NO2+
|
1
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| 1 |
Ki = 52480.75 nM
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CP0845387
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N,N,N-Trimethyl((2R*,6S*)-5,5,6-trimethyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C11H24INO2
|
1
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| 1 |
Ki = 52480.75 nM
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CP0393373
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(3E)-N-[2-(dimethylamino)ethyl]-3-(pyridin-4-ylmethylidene)indene-1-carboxamide
Show/Hide
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C20H21N3O
|
1
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| 1 |
Ki = 53703.18 nM
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CP0405252
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(3E)-N-[2-(dimethylamino)ethyl]-N-methyl-3-(pyridin-3-ylmethylidene)indene-1-carboxamide
Show/Hide
|
C21H23N3O
|
1
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| 1 |
Ki = 53703.18 nM
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CP0377730
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(4-methylpiperazin-1-yl)-[(3E)-3-(pyridin-4-ylmethylidene)inden-1-yl]methanone
Show/Hide
|
C21H21N3O
|
1
|
| 1 |
Ki = 54954.09 nM
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CP0429992
|
(3E)-N-[2-(dimethylamino)ethyl]-3-(pyridin-2-ylmethylidene)indene-1-carboxamide
Show/Hide
|
C20H21N3O
|
1
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| 1 |
Ki = 54954.09 nM
|
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CP0859713
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(2R*,5S*)-N,N,N-Trimethyl-(5-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
1
|
| 1 |
Ki = 63095.73 nM
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CP0500729
|
(2S)-2-(furan-2-yl)-1-methylpyrrolidine
Show/Hide
|
C9H13NO
|
1
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| 1 |
Ki = 63095.73 nM
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CP0430112
|
(3E)-N-[2-(dimethylamino)ethyl]-3-(pyridin-3-ylmethylidene)indene-1-carboxamide
Show/Hide
|
C20H21N3O
|
1
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| 1 |
Ki = 66069.34 nM
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CP0916016
|
N,N,N-Trimethyl(5,5,6,6-tetramethyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C12H26INO2
|
1
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| 1 |
Ki = 66069.34 nM
|
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CP0859716
|
()-(2R,6R)-N,N,N-trimethyl(6-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
2
|
| 1 |
Ki = 67608.3 nM
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| 2 |
Ki = 87096.36 nM
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CP0465871
|
(2R)-2-(furan-2-yl)-1-methylpyrrolidine
Show/Hide
|
C9H13NO
|
1
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| 1 |
Ki = 75857.76 nM
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CP0859717
|
N,N,N-Trimethyl((2R*,6R*)-5,5,6-trimethyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C11H24INO2
|
1
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| 1 |
Ki = 83176.38 nM
|
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CP0864337
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N,N,N-trimethyl-1-((2R,5R)-5-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
1
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| 1 |
Ki = 93325.43 nM
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CP0859715
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((2R*,5R*,6S*)-5,6-Dimethyl-1,4-dioxan-2-yl)-N,N,Ntrimethylmethanaminium iodide
Show/Hide
|
C10H22INO2
|
1
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| 1 |
Ki = 97723.72 nM
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CP0859476
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((2S*,5S*,6S*)-5,6-Dimethyl-1,4-dioxan-2-yl)-N,N,Ntrimethylmethanaminium iodide
Show/Hide
|
C10H22INO2
|
1
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| 1 |
Ki > 100000 nM
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CP0868051
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(5,5-Dimethyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium iodide
Show/Hide
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C10H22INO2
|
1
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| 1 |
Ki > 100000 nM
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CP0904026
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((2R*,5S*,6R*)-5,6-Dimethyl-1,4-dioxan-2-yl)-N,N,Ntrimethylmethanaminium iodide
Show/Hide
|
C10H22INO2
|
1
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| 1 |
Ki > 100000 nM
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CP0867621
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Trans-((2R*,6R*)-6-Ethyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide
Show/Hide
|
C10H22INO2
|
1
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| 1 |
Ki > 100000 nM
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CP0407014
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(5S,2'S)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone
Show/Hide
|
C8H14N2O2
|
1
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| 1 |
Ki > 100000 nM
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CP0414425
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(5R,2'S)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone
Show/Hide
|
C8H14N2O2
|
1
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| 1 |
Ki > 100000 nM
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CP0846921
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(S)-N,N,N-trimethyl-1-(2-oxooxazolidin-5-yl)methanaminium
Show/Hide
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C7H15N2O2+
|
1
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| 1 |
Ki > 100000 nM
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CP0846922
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(S)-2-(carbamoyloxymethyl)-1,1-dimethylpyrrolidinium
Show/Hide
|
C8H17N2O2+
|
1
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| 1 |
Ki > 100000 nM
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CP0846927
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(R)-5-((dimethylamino)methyl)oxazolidin-2-one
Show/Hide
|
C6H12N2O2
|
1
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| 1 |
Ki > 100000 nM
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CP0848614
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(S)-5-((dimethylamino)methyl)-3-methyloxazolidin-2-one
Show/Hide
|
C7H14N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0856191
|
(S)-(1-methylpyrrolidin-2-yl)methyl carbamate
Show/Hide
|
C7H14N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0860582
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(R)-N,N,N-trimethyl-1-(3-methyl-2-oxooxazolidin-5-yl)methanaminium
Show/Hide
|
C8H17N2O2+
|
1
|
| 1 |
Ki > 100000 nM
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CP0861363
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(S)-N,N,N-trimethyl-1-(3-methyl-2-oxooxazolidin-5-yl)methanaminium
Show/Hide
|
C8H17N2O2+
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0866588
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(R)-N,N,N-trimethyl-1-(2-oxooxazolidin-5-yl)methanaminium
Show/Hide
|
C7H15N2O2+
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0886638
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(R)-4-((S)-1-methylpyrrolidin-2-yl)oxazolidin-2-one
Show/Hide
|
C8H14N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0902643
|
(R)-5-((dimethylamino)methyl)-3-methyloxazolidin-2-one
Show/Hide
|
C7H14N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0902877
|
(S)-5-((dimethylamino)methyl)oxazolidin-2-one
Show/Hide
|
C6H12N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0912137
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(S)-4-((S)-1-methylpyrrolidin-2-yl)oxazolidin-2-one
Show/Hide
|
C8H14N2O2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0848040
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(R)-N,N,N-Trimethyl-1-(2-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0866923
|
N,N,N-trimethyl-1-((2R,3S)-3-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
1
|
| 1 |
Ki > 100000 nM
|
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CP0913147
|
N,N,N-trimethyl-1-((2R,3R)-3-methyl-1,4-dioxan-2-yl)methanaminium iodide
Show/Hide
|
C9H20INO2
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
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CP0307921
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H26FN3O3S2
|
1
|
| 1 |
Ki > 1000 nM
|
|
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CP0467302
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(R)-N-((S)-piperidin-3-ylmethyl)-1-((S)-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-carbonyl)pyrrolidine-2-carboxamide
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C37H44N4O3
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1
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| 1 |
Ki > 5000 nM
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CP0390494
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(2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-(4-piperidinylmethyl)pyrrolidine-2-carboxamide
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C37H44N4O4
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1
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| 1 |
Ki > 5100 nM
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CP0390497
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(2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-(4-piperidinylethyl)pyrrolidine-2-carboxamide
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C38H46N4O4
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1
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| 1 |
Ki > 5100 nM
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CP0393862
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(2R)-1-[(2S,4R)-4-hydroxy-1-(3,3,3-triphenylpropanoyl)pyrrolidine-2-yl]carbonyl-N-((3R)-3-piperidinylmethyl)pyrrolidine-2-carboxamide
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C37H44N4O4
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1
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| 1 |
Ki > 5100 nM
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CP0485213
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(2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluorophenyl)propanoyl]pyrrolidine-2-yl)carbonyl-N-[1-(2-propyl)-4-piperidinylmethyl]pyrrolidine-2-carboxamide
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C34H36F3N3O4
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1
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| 1 |
Ki > 5400 nM
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CP0379517
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(2R,3S,5R)-2-methyl-5-[(2R)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0379521
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(2R,3S,5R)-5-[(2S)-1,1-dimethylpyrrolidin-1-ium-2-yl]-2-methyl-1,3-oxathiolane 3-oxide;iodide
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C10H20INO2S
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1
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| 1 |
Ki < 100000 nM
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CP0379525
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(2S,3R,5S)-2-methyl-5-[(2S)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0379526
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(2R,3R,5R)-5-[(2R)-1,1-dimethylpyrrolidin-1-ium-2-yl]-2-methyl-1,3-oxathiolane 3-oxide;iodide
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C10H20INO2S
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1
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| 1 |
Ki < 100000 nM
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CP0379527
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(2S,3S,5S)-2-methyl-5-[(2R)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0419569
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(2R,3S,5R)-5-[(2R)-1,1-dimethylpyrrolidin-1-ium-2-yl]-2-methyl-1,3-oxathiolane 3-oxide;iodide
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C10H20INO2S
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1
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| 1 |
Ki < 100000 nM
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CP0419583
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(2S,3R,5S)-2-methyl-5-[(2R)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0424750
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(2R,3R,5R)-2-methyl-5-[(2R)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0431823
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(2R,3S,5R)-2-methyl-5-[(2S)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0432602
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(2R,3R,5R)-2-methyl-5-[(2S)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0449147
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(2S,3S,5S)-2-methyl-5-[(2S)-1-methylpyrrolidin-2-yl]-1,3-oxathiolane 3-oxide
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C9H17NO2S
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1
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| 1 |
Ki < 100000 nM
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CP0461163
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(2S,3S,5S)-5-[(2S)-1,1-dimethylpyrrolidin-1-ium-2-yl]-2-methyl-1,3-oxathiolane 3-oxide;iodide
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C10H20INO2S
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1
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| 1 |
Ki < 100000 nM
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