Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3,4-dihydro-1H-isoquinolin-2-yl-[1-[6-(2-fluorophenoxy)pyrimidin-4-yl]piperidin-4-yl]methanone
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 PubChem ID
CID: 137655063
Canonical SMILES
Fc1ccccc1Oc1cc(ncn1)N1CCC(CC1)C(=O)N1CCc2ccccc2C1
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Compound Formula C25H25FN4O2
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08912
Gene Name
CHRM5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 732 nM
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