Brief Information of the Compound and Protein
Compound Name
8,9-Dimethoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene
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PubChem ID
CID: 44302793
Canonical SMILES
COc1cc2CCN3Cc4c(OC3c2cc1OC)ccc1[nH]c(C)cc41
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Compound Formula C21H22N2O3
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08912
Gene Name
CHRM5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 43462.7 nM
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