Brief Information of the Compound and Protein
Compound Name
9b-(4-chloro-3-methoxyphenyl)-1-(3,4,5-trifluorobenzoyl)-2,3-dihydroimidazo[2,1-a]isoindol-5-one
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PubChem ID
CID: 118719491
Canonical SMILES
COc1cc(ccc1Cl)C12N(CCN1C(=O)c1ccccc21)C(=O)c1cc(F)c(F)c(F)c1
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Compound Formula C24H16ClF3N2O3
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08912
Gene Name
CHRM5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1600 nM
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