Compound ID |
Compound Name |
Compound Formula |
CP0389986
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl)-3-isopropoxy-4-biphenylcarboxylic acid
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|
C27H31NO4
|
1
|
1 |
EC50 = 0.19 nM
|
|
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CP0135429
|
(4R)-2-amino-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
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|
C25H28N4O2S
|
1
|
1 |
EC50 = 0.19 nM
|
|
|
CP0375142
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-3-propoxy-4-biphenylcarboxylic acid
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|
C26H30N2O4
|
1
|
1 |
EC50 = 0.51 nM
|
|
|
CP0845051
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylsulfanyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
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|
C27H33ClN2O4S2
|
1
|
1 |
EC50 = 0.68 nM
|
|
|
CP0882007
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-isobutyl-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
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|
C28H35ClN2O4S
|
1
|
1 |
EC50 = 0.88 nM
|
|
|
CP0881981
|
4'-(2-{[(2R)-2-(4-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-(cyclohexyloxy)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
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|
C30H39Cl2N3O5S
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0037154
|
(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
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|
C26H28ClNO4
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0217241
|
4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-ylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
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|
C28H34N2O6S
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0845050
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylamino)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
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|
C27H35Cl2N3O4S
|
1
|
1 |
EC50 = 1.1 nM
|
|
|
CP0372880
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(isopropylthio)biphenyl-4-carboxylic acid
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|
C26H29NO3S
|
1
|
1 |
EC50 = 1.2 nM
|
|
|
CP0418059
|
(R)-3-(cyclohexyloxy)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)biphenyl-4-carboxylic acid
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|
C28H32N2O4
|
1
|
1 |
EC50 = 1.3 nM
|
|
|
CP0900959
|
3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
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|
C29H37Cl2N3O5S
|
1
|
1 |
EC50 = 1.4 nM
|
|
|
CP0459677
|
(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-pivalamidobenzoic acid
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|
C28H31ClN2O5
|
1
|
1 |
EC50 = 1.6 nM
|
|
|
CP0504190
|
(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-(2-oxopyrrolidin-1-yl)benzoic acid
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|
C27H27ClN2O5
|
1
|
1 |
EC50 = 1.9 nM
|
|
|
CP0375139
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
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|
C27H31NO3
|
1
|
1 |
EC50 = 2.2 nM
|
|
|
CP0877318
|
4'-(2-{[(2R)-2-(4-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
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|
C27H35Cl2N3O5S
|
1
|
1 |
EC50 = 2.512 nM
|
|
|
CP0137177
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
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|
C26H29NO4
|
1
|
1 |
EC50 = 2.9 nM
|
|
|
CP0849245
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)-3-phenoxybiphenyl-4-carboxamide Hydrochloride
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|
C30H31ClN2O5S
|
1
|
1 |
EC50 = 2.9 nM
|
|
|
CP0474560
|
(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
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|
C26H31N3O3
|
1
|
1 |
EC50 = 3.2 nM
|
|
|
CP0467666
|
(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-isopropoxybenzoic acid
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|
C26H28ClNO5
|
1
|
1 |
EC50 = 3.2 nM
|
|
|
CP0375138
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-isobutyl-4-biphenylcarboxylic acid
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|
C26H31N3O3
|
1
|
1 |
EC50 = 3.2 nM
|
|
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CP0484975
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
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|
C27H31NO4
|
1
|
1 |
EC50 = 3.7 nM
|
|
|
CP0135426
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C24H26N4O2S
|
1
|
1 |
EC50 = 5 nM
|
|
|
CP0399297
|
(R)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
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|
C25H28N2O4
|
2
|
1 |
EC50 = 10 nM
|
|
|
2 |
EC50 = 11 nM
|
|
|
CP0434840
|
4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
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|
C26H32N4O5S
|
1
|
1 |
EC50 = 10 nM
|
|
|
CP0105650
|
KRP-114V
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|
C26H28N4O3
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0105651
|
(6S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide
Show/Hide
|
C24H27N5O2
|
1
|
1 |
EC50 = 22 nM
|
|
|
CP0493893
|
4-((S)-7-((R)-2-(4-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
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|
C25H24ClNO3
|
1
|
1 |
EC50 = 25 nM
|
|
|
CP0156740
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-(4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C31H27F3N4O3S2
|
1
|
1 |
EC50 = 25 nM
|
|
|
CP0288880
|
ethyl 2-[[(6S)-6-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]oxy]acetate
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|
C23H28ClNO4
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0156745
|
(2S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)propanamide
Show/Hide
|
C25H28N4O3
|
1
|
1 |
EC50 = 39 nM
|
|
|
CP0372774
|
5-[((7S)-7-{[(2R)-2-(6-Chloro-3-pyridinyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
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|
C25H25ClN2O5
|
1
|
1 |
EC50 = 46 nM
|
|
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CP0105652
|
N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)acetamide
Show/Hide
|
C24H26N4O3
|
1
|
1 |
EC50 = 47 nM
|
|
|