General Information of the Compound
Compound ID
CP0506075
Compound Name
(2R)-1-(2-Chloro-4-(difluoromethoxy)phenylsulfonyl)-4-(4-fluoro-2-(trifluoromethyl)phenyl)-2-methylpiperazine
    Show/Hide
Structure
Formula
C19H17ClF6N2O3S
Molecular Weight
502.864
Canonical SMILES
C[C@@H]1CN(CCN1S(=O)(=O)c1ccc(OC(F)F)cc1Cl)c1ccc(F)cc1C(F)(F)F
    Show/Hide
InChI
InChI=1S/C19H17ClF6N2O3S/c1-11-10-27(16-4-2-12(21)8-14(16)19(24,25)26)6-7-28(11)32(29,30)17-5-3-13(9-15(17)20)31-18(22)23/h2-5,8-9,11,18H,6-7,10H2,1H3/t11-/m1/s1
    Show/Hide
InChIKey
QFVTWMNHGWAXOC-LLVKDONJSA-N
Physicochemical Property
logP
4.9987
Rotatable Bonds
5
Heavy Atom Count
32
Polar Areas
49.85
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
4
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 44248455
SID: 85282168
ChEMBL ID
CHEMBL550554
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01109, 11-beta-hydroxysteroid dehydrogenase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
Protein ID: PT01107, 11-beta-hydroxysteroid dehydrogenase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 18 nM
   TI
   LI
   LO
   TS