Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01746 , 5-hydroxytryptamine receptor 7
Gene Name HTR7
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P32305
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01746
 
Compound ID Compound Name Compound Formula
CP0395135
(R)-2-(4-Fluoro-phenyl)-2-{1-[3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-ylamino}-ethanol
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C26H31FN6O
 1
1
IC50 = 540 nM
   TI
   LI
   LO
   TS
CP0096286
(R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidin-1-ylsulfonyl)phenol
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C18H28N2O3S
 1
1
Ki = 1.26 nM
   TI
   LI
   LO
   TS
CP0074093
(R)-2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)-2a,3,4,5-tetrahydrobenzo[cd]indol-2(1H)-one
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C26H30N2O
 1
1
Ki = 3.31 nM
   TI
   LI
   LO
   TS
CP0100452
(R)-6-Methyl-11-phenyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline
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C23H21N
 1
1
Ki = 9.78 nM
   TI
   LI
   LO
   TS
CP0207579
(R)-11-(2,6-Dimethoxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline
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C25H25NO2
 1
1
Ki = 13 nM
   TI
   LI
   LO
   TS
CP0062900
(1S,5aR)-6-methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ylamine
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C18H18N2
 1
1
Ki = 18 nM
   TI
   LI
   LO
   TS
CP0156235
3,N-Dimethyl-N-[(R)-1-methyl-3-(4-methyl-piperidin-1-yl)-propyl]-benzenesulfonamide
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C18H30N2O2S
 1
1
Ki = 31.6 nM
   TI
   LI
   LO
   TS
CP0497908
(R)-2-(6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-benzene-1,3-diol
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C23H21NO2
 1
1
Ki = 36.2 nM
   TI
   LI
   LO
   TS
CP0044066
(R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline
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C17H17N
 1
1
Ki = 88 nM
   TI
   LI
   LO
   TS
CP0042751
(6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol;hydrate;hydrochloride
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C17H17NO2
 1
1
Ki = 188 nM
   TI
   LI
   LO
   TS
CP0492308
(R)-Trifluoro-methanesulfonic acid 2-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-3-trifluoromethanesulfonyloxy-phenyl ester
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C25H19F6NO6S2
 1
1
Ki = 708 nM
   TI
   LI
   LO
   TS