| Compound ID |
Compound Name |
Compound Formula |
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
4
|
| 1 |
IC50 = 0.25 nM
|
|
|
| 2 |
IC50 = 0.47 nM
|
|
|
| 3 |
Ki = 0.17 nM
|
|
|
| 4 |
Ki = 0.8 nM
|
|
|
|
CP0371722
|
N-(cyclopropylmethyl)-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C27H31F3N4O2S
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0419082
|
N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26F3N3O2S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0371727
|
N-(cyclopropylmethyl)-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C27H34N4O3S
|
1
|
| 1 |
IC50 = 12.3 nM
|
|
|
|
CP0396954
|
(9S)-N-(diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide
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|
C18H17N3O2
|
2
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0086696
|
N-(diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide;hydrochloride
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|
C18H18ClN3O2
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0259093
|
N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0430836
|
N-(cyclohexylmethyl)-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C30H40N4O3S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0510369
|
N-(cyclopropylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C26H31FN4O2S
|
1
|
| 1 |
IC50 = 35.3 nM
|
|
|
|
CP0233824
|
4-Methoxy-N-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0379299
|
(9R)-N-(diaminomethylidene)spiro[fluorene-9,2'-oxolane]-2-carboxamide
Show/Hide
|
C18H17N3O2
|
2
|
| 1 |
IC50 = 41 nM
|
|
|
| 2 |
Ki = 5.1 nM
|
|
|
|
CP0501817
|
4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C20H26FN3O3S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0430831
|
N-(cyclopropylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C27H32FN3O2S
|
1
|
| 1 |
IC50 = 49.6 nM
|
|
|
|
CP0501827
|
N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H26FN3O2S
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0664572
|
N-(Diaminomethylene)-9-hydroxy-9-methyl-9Hfluorene-2-carboxamide hydrochloride
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|
C16H16ClN3O2
|
2
|
| 1 |
IC50 = 59 nM
|
|
|
| 2 |
Ki = 4.3 nM
|
|
|
|
CP0401996
|
N-(cyclohexylmethyl)-4-nitro-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C26H36N4O4S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0419080
|
4-Methoxy-N-{3-[4-(m-trifluoromethylphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H26F3N3O3S
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0452722
|
N-(cyclopropylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C24H32FN3O3S
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0419078
|
4-Methoxy-N-{3-[4-(3,4-dichlorophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C20H25Cl2N3O3S
|
1
|
| 1 |
IC50 = 103 nM
|
|
|
|
CP0459682
|
4-Methoxy-N-{3-[4-(m-trifluoromethylphenyl)-piperazin-1-yl]-1-methyl-propyl}-benzenesulfonamide
Show/Hide
|
C22H28F3N3O3S
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0528543
|
N-(cyclohexylmethyl)-4-fluoro-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C26H36FN3O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0426880
|
N-(cyclopropylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]naphthalene-2-sulfonamide
Show/Hide
|
C27H33N3O2S
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0492831
|
N-(cyclopropylmethyl)-4-methoxy-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C24H33N3O3S
|
1
|
| 1 |
IC50 = 121 nM
|
|
|
|
CP0373060
|
N-[3-[4-(3,4-dichlorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H25Cl2N3O2S
|
1
|
| 1 |
IC50 = 124 nM
|
|
|
|
CP0463951
|
N-(cyclopropylmethyl)-4-methoxy-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C25H32F3N3O3S
|
1
|
| 1 |
IC50 = 124 nM
|
|
|
|
CP0503083
|
N-[3-[4-(2-fluorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H26FN3O2S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0507696
|
N-(cyclopropylmethyl)-4-fluoro-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C23H30FN3O2S
|
1
|
| 1 |
IC50 = 147 nM
|
|
|
|
CP0447686
|
N-(cyclopropylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]naphthalene-1-sulfonamide
Show/Hide
|
C27H33N3O2S
|
1
|
| 1 |
IC50 = 152 nM
|
|
|
|
CP0497110
|
N-(cyclohexylmethyl)-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C30H37F3N4O2S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0430832
|
N-(cyclohexylmethyl)-4-methoxy-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C28H41N3O4S
|
1
|
| 1 |
IC50 = 172 nM
|
|
|
|
CP0373571
|
N-(cyclopropylmethyl)-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C28H35N3O3S
|
1
|
| 1 |
IC50 = 188 nM
|
|
|
|
CP0514881
|
N-(cyclohexylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]naphthalene-1-sulfonamide
Show/Hide
|
C30H39N3O2S
|
1
|
| 1 |
IC50 = 195 nM
|
|
|
|
CP0519870
|
N-[3-[4-(3-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O3S
|
1
|
| 1 |
IC50 = 223 nM
|
|
|
|
CP0528429
|
4-Methoxy-N-{3-[4-(o-fluorophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C20H26FN3O3S
|
1
|
| 1 |
IC50 = 289 nM
|
|
|
|
CP0415115
|
N-(cyclopropylmethyl)-4-methoxy-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C25H35N3O4S
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0497111
|
N-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butan-2-yl]naphthalene-2-sulfonamide
Show/Hide
|
C25H31N3O3S
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0373410
|
N-(cyclopropylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C24H30F3N3O2S
|
1
|
| 1 |
IC50 = 334 nM
|
|
|
|
CP0526777
|
4-Methoxy-N-{3-[4-(m-methoxyphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 = 339 nM
|
|
|
|
CP0469927
|
N-(cyclopropylmethyl)-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C28H32F3N3O2S
|
1
|
| 1 |
IC50 = 342 nM
|
|
|
|
CP0371728
|
N-[4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]butan-2-yl]naphthalene-2-sulfonamide
Show/Hide
|
C25H28F3N3O2S
|
1
|
| 1 |
IC50 = 363 nM
|
|
|
|
CP0526807
|
4-Methoxy-N-{3-[4-(p-fluorophenyl)-piperazin-1-yl]-1-methyl-propyl}-benzenesulfonamide
Show/Hide
|
C21H28FN3O3S
|
1
|
| 1 |
IC50 = 373 nM
|
|
|
|
CP0531993
|
4-Methoxy-N-[3-(4-phenyl-piperazin-1-yl)-1-methyl-propyl]-benzenesulfonamide
Show/Hide
|
C21H29N3O3S
|
1
|
| 1 |
IC50 = 377 nM
|
|
|
|
CP0383383
|
4-Methoxy-N-{3-[4-(p-trifluoromethylphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H26F3N3O3S
|
1
|
| 1 |
IC50 = 384 nM
|
|
|
|
CP0430833
|
N-(cyclohexylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]quinoline-8-sulfonamide
Show/Hide
|
C29H38N4O2S
|
1
|
| 1 |
IC50 = 419 nM
|
|
|
|
CP0371721
|
N-(cyclohexylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C29H37FN4O2S
|
1
|
| 1 |
IC50 = 442 nM
|
|
|
|
CP0502602
|
N-(cyclohexylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C27H36F3N3O2S
|
1
|
| 1 |
IC50 = 456 nM
|
|
|
|
CP0419077
|
N-[3-(4-benzylpiperazin-1-yl)propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 476 nM
|
|
|
|
CP0415113
|
N-(cyclopropylmethyl)-4-nitro-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C23H30N4O4S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0430835
|
N-(cyclohexylmethyl)-N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C31H41N3O3S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0419036
|
N,N-dimethyl-2-(3-naphthalen-1-ylsulfonylpyrrolo[2,3-b]pyridin-1-yl)ethanamine
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 = 511 nM
|
|
|
|
CP0510686
|
N-[4-[4-(4-fluorophenyl)piperazin-1-yl]butan-2-yl]naphthalene-2-sulfonamide
Show/Hide
|
C24H28FN3O2S
|
1
|
| 1 |
IC50 = 526 nM
|
|
|
|
CP0410116
|
3-[methyl-[4-(4-phenylpiperazin-1-yl)butyl]amino]phenol
Show/Hide
|
C21H29N3O
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0459683
|
N-[3-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26F3N3O2S
|
1
|
| 1 |
IC50 = 567 nM
|
|
|
|
CP0502603
|
N-(cyclohexylmethyl)-4-methoxy-N-[3-(4-phenylpiperazin-1-yl)propyl]benzenesulfonamide
Show/Hide
|
C27H39N3O3S
|
1
|
| 1 |
IC50 = 567 nM
|
|
|
|
CP0501825
|
4-Methoxy-N-{3-[4-(o-methoxyphenyl)-piperazin-1-yl]-1-methyl-propyl}-benzen sulfonamide
Show/Hide
|
C22H31N3O4S
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0373567
|
N-[4-(4-phenylpiperazin-1-yl)butan-2-yl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 657 nM
|
|
|
|
CP0373407
|
N-(cyclohexylmethyl)-4-methoxy-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C28H38F3N3O3S
|
1
|
| 1 |
IC50 = 678 nM
|
|
|
|
CP0501826
|
N-[3-(4-phenylpiperazin-1-yl)propyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H27N3O2S
|
1
|
| 1 |
IC50 = 681 nM
|
|
|
|
CP0373566
|
N-(cyclopropylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]quinoline-8-sulfonamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
IC50 = 749 nM
|
|
|
|
CP0502301
|
N-(cyclohexylmethyl)-N-[3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C31H38F3N3O2S
|
1
|
| 1 |
IC50 = 888 nM
|
|
|
|
CP0528428
|
4-Methoxy-N-[3-(4-benzyl-piperazin-1-yl)-propyl]-benzenesulfonamide
Show/Hide
|
C20H27N3O2S
|
1
|
| 1 |
IC50 = 949 nM
|
|
|
|
CP0510691
|
N-(cyclohexylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C27H38FN3O3S
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0405688
|
2-[3-(3-chlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H18ClN3O2S
|
1
|
| 1 |
IC50 = 1217 nM
|
|
|
|
CP0477664
|
N-(cyclohexylmethyl)-N-[3-(4-phenylpiperazin-1-yl)propyl]naphthalene-2-sulfonamide
Show/Hide
|
C30H39N3O2S
|
1
|
| 1 |
IC50 = 1236 nM
|
|
|
|
CP0439248
|
2-{3-[(3-Chlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
|
C15H14ClN3O2S
|
1
|
| 1 |
IC50 = 1362 nM
|
|
|
|
CP0447670
|
N-(cyclohexylmethyl)-N-[3-[4-(4-fluorophenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C30H38FN3O2S
|
1
|
| 1 |
IC50 = 1508 nM
|
|
|
|
CP0492830
|
N-(cyclohexylmethyl)-N-[3-[4-(3,4-dichlorophenyl)piperazin-1-yl]propyl]quinoline-8-sulfonamide
Show/Hide
|
C29H36Cl2N4O2S
|
1
|
| 1 |
IC50 = 2296 nM
|
|
|
|
CP0504691
|
N-[3-[4-(4-methoxyphenyl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O3S
|
1
|
| 1 |
IC50 = 3241 nM
|
|
|
|
CP0380100
|
2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H18FN3O2S
|
1
|
| 1 |
IC50 = 4764 nM
|
|
|
|
CP0419079
|
4-Methoxy-N-{3-[4-(p-methoxyphenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 = 9314 nM
|
|
|
|
CP0418521
|
4-Methoxy-N-{3-[4-(p-nitrophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C20H26N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0491989
|
4-Methoxy-N-[3-(4-phenyl-piperazin-1-yl)-propyl]-benzenesulfonamide
Show/Hide
|
C20H27N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0492153
|
Benzyl-4-(4-methoxyphenyl sulfonylaminopropyl)-piperazine-1-carboxylate
Show/Hide
|
C22H29N3O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0528427
|
4-Methoxy-N-{3-[4-(furan-2-yl-methanoyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C19H25N3O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0529541
|
4-Methoxy-N-{3-[4-(4-acetophenyl)-piperazin-1-yl]-propyl}-benzenesulfonamide
Show/Hide
|
C22H29N3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0795225
|
1-(3-Thiophen-2-yl-phenyl)-ethanone, O-(phenylaminocarbonyl)oxime
Show/Hide
|
C19H16N2O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0170456
|
3-chloro-1-(4-fluoro benzenesulfonyl)-5-(4-methylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C20H21ClFN3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0212171
|
1-(2-Bromo benzenesulfonyl)-5-(4-ethylpiperazin-1-yl-methyl)-1H-indole
Show/Hide
|
C21H24BrN3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0424416
|
2-[3-(Phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C15H15N3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0150364
|
2,8-Dimethyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H22N2
|
1
|
| 1 |
Ki = 0.2089 nM
|
|
|
|
CP0237538
|
2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C21H24N2
|
1
|
| 1 |
Ki = 0.2512 nM
|
|
|
|
CP0405600
|
5-fluoro-3-[2-[4-(2-phenylphenyl)piperazin-1-yl]ethyl]-1H-indole
Show/Hide
|
C26H26FN3
|
1
|
| 1 |
Ki = 0.26 nM
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CP0112368
|
3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
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C22H26ClN3O
|
2
|
| 1 |
Ki = 0.38 nM
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| 2 |
Ki = 7 nM
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CP0436292
|
3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H30ClN3O
|
1
|
| 1 |
Ki = 0.38 nM
|
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CP0353494
|
2,8-Dimethyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C22H26N2
|
1
|
| 1 |
Ki = 0.389 nM
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CP0437044
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H30ClN3O
|
2
|
| 1 |
Ki = 0.4 nM
|
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| 2 |
Ki = 0.41 nM
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CP0451972
|
3-ethyl-3-[4-[4-(4-fluorophenyl)piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C24H30FN3O
|
1
|
| 1 |
Ki = 0.43 nM
|
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CP0436293
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
|
C22H26ClN3O
|
1
|
| 1 |
Ki = 0.49 nM
|
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CP0446202
|
5-fluoro-3-[3-[4-[3-fluoro-2-(3-fluorophenyl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C27H26F3N3
|
1
|
| 1 |
Ki = 0.55 nM
|
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CP0394524
|
3-[4-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H29ClFN3O
|
1
|
| 1 |
Ki = 0.6 nM
|
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CP0074213
|
2-(6-Phenylpyridin-2-ylthio)-N,N-dimethylethan-amine
Show/Hide
|
C15H18N2S
|
1
|
| 1 |
Ki = 0.6 nM
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CP0451971
|
3-[4-[4-(3,4-dichlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H29Cl2N3O
|
2
|
| 1 |
Ki = 0.6 nM
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| 2 |
Ki = 0.63 nM
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CP0498670
|
N-(diaminomethylidene)-9-ethyl-9-methoxyfluorene-2-carboxamide;hydrochloride
Show/Hide
|
C18H20ClN3O2
|
1
|
| 1 |
Ki = 0.6 nM
|
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CP0373135
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3-[4-[4-(3-chloro-4-methylphenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C25H32ClN3O
|
1
|
| 1 |
Ki = 0.66 nM
|
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CP0399742
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
Show/Hide
|
C24H29ClFN3O
|
1
|
| 1 |
Ki = 0.67 nM
|
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CP0418395
|
2-(6-cyclohexylpyridin-2-ylthio)-N,N-dimethylethanamine
Show/Hide
|
C15H24N2S
|
1
|
| 1 |
Ki = 0.7 nM
|
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CP0414362
|
N-(diaminomethylidene)-9-methoxy-9-(methoxymethyl)fluorene-2-carboxamide;hydrochloride
Show/Hide
|
C18H20ClN3O3
|
1
|
| 1 |
Ki = 0.76 nM
|
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CP0109472
|
3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
Show/Hide
|
C24H29ClFN3O
|
1
|
| 1 |
Ki = 0.79 nM
|
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CP0455706
|
5-fluoro-3-[2-[4-[2-(3-fluorophenyl)phenyl]piperazin-1-yl]ethyl]-1H-indole
Show/Hide
|
C26H25F2N3
|
1
|
| 1 |
Ki = 0.79 nM
|
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CP0420806
|
(5Z)-3-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-5-[(3,4-dimethoxyphenyl)methylidene]imidazolidine-2,4-dione
Show/Hide
|
C26H30Cl2N4O4
|
1
|
| 1 |
Ki = 0.8 nM
|
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CP0434333
|
5-fluoro-3-[3-[4-[4-fluoro-2-(1H-pyrazol-4-yl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C24H25F2N5
|
1
|
| 1 |
Ki = 0.9 nM
|
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CP0468921
|
3-[4-[2-(5-fluoro-1H-indol-3-yl)ethyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C21H21FN4S
|
1
|
| 1 |
Ki = 0.99 nM
|
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CP0039958
|
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C23H27FN4O2
|
1
|
| 1 |
Ki = 1 nM
|
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|
CP0420807
|
(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]imidazolidine-2,4-dione
Show/Hide
|
C31H40N4O5
|
1
|
| 1 |
Ki = 1 nM
|
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|
CP0528467
|
3-[4-[4-(4-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C25H29ClN2O
|
1
|
| 1 |
Ki = 1.02 nM
|
|
|
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CP0373134
|
5-chloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H29Cl2N3O
|
2
|
| 1 |
Ki = 1.1 nM
|
|
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| 2 |
Ki = 3.72 nM
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CP0450959
|
5-fluoro-3-[3-[4-[2-(3-fluorophenyl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C27H27F2N3
|
1
|
| 1 |
Ki = 1.1 nM
|
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|
|
CP0467698
|
5-fluoro-3-[3-[4-(2-phenylphenyl)piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C27H28FN3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
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CP0437191
|
3-ethyl-3-[4-[4-(4-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C25H29FN2O
|
2
|
| 1 |
Ki = 1.19 nM
|
|
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| 2 |
Ki = 1.2 nM
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CP0414363
|
N-(diaminomethylidene)-9-ethyl-9-hydroxyfluorene-2-carboxamide;hydrochloride
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0407910
|
3-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C25H32ClN3O
|
1
|
| 1 |
Ki = 1.24 nM
|
|
|
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CP0418396
|
(2-tert-Butylsulfanyl-ethyl)-dimethyl-amine
Show/Hide
|
C8H19NS
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
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CP0866566
|
N-(Diaminomethylene)-2',3',5',6'-tetrahydrospiro[fluorene-9,4'-pyran]-2-carboxamide hydrochloride
Show/Hide
|
C19H20ClN3O2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0539786
|
N-(diaminomethylidene)-9-methoxy-9-methylfluorene-2-carboxamide;hydrochloride
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0437194
|
3-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C25H32ClN3O
|
1
|
| 1 |
Ki = 1.45 nM
|
|
|
|
CP0437192
|
3-ethyl-5-fluoro-3-[4-[4-(4-fluorophenyl)piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C24H29F2N3O
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0037955
|
METHIOTHEPIN
Show/Hide
|
C20H24N2S2
|
2
|
| 1 |
Ki = 1.7 nM
|
|
|
| 2 |
Ki = 2.2 nM
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CP0408009
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-(2-methylpropyl)-1H-indol-2-one
Show/Hide
|
C26H34ClN3O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0921389
|
N-(Diaminomethylene)spiro[cyclopentane-1,9'-fluorene]-2'-carboxamide hydrochloride
Show/Hide
|
C19H20ClN3O
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
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CP0307921
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H26FN3O3S2
|
1
|
| 1 |
Ki = 1.9 nM
|
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|
|
CP0373136
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-5-fluoro-1,3-dihydroindol-2-one
Show/Hide
|
C22H25ClFN3O
|
1
|
| 1 |
Ki = 1.96 nM
|
|
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CP0485520
|
5-fluoro-3-[3-[4-(4-fluoro-2-thiophen-3-ylphenyl)piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C25H25F2N3S
|
1
|
| 1 |
Ki = 2 nM
|
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|
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CP0435715
|
3-ethyl-3-[4-(4-phenylpiperazin-1-yl)butyl]-1H-indol-2-one
Show/Hide
|
C24H31N3O
|
1
|
| 1 |
Ki = 2.07 nM
|
|
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|
CP0474956
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-5-fluoro-1H-indol-2-one
Show/Hide
|
C24H29ClFN3O
|
2
|
| 1 |
Ki = 2.1 nM
|
|
|
| 2 |
Ki = 2.11 nM
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CP0367059
|
2a-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3,4,5-tetrahydrobenzo[cd]indol-2-one
Show/Hide
|
C26H33N3O2
|
1
|
| 1 |
Ki = 2.138 nM
|
|
|
|
CP0402331
|
3-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]-1,2-benzothiazole
Show/Hide
|
C22H23FN4S
|
1
|
| 1 |
Ki = 2.2 nM
|
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CP0920595
|
N-(Diaminomethylene)-5-ethyl-9-hydroxy-9-methyl-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
|
C18H20ClN3O2
|
1
|
| 1 |
Ki = 2.3 nM
|
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CP0446201
|
5-fluoro-3-[2-[4-[2-(2-fluorophenyl)phenyl]piperazin-1-yl]ethyl]-1H-indole
Show/Hide
|
C26H25F2N3
|
1
|
| 1 |
Ki = 2.3 nM
|
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CP0386218
|
3-ethyl-3-[4-[4-(3-methoxyphenyl)piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C25H33N3O2
|
1
|
| 1 |
Ki = 2.55 nM
|
|
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CP0394365
|
5-fluoro-3-[3-[4-[5-fluoro-2-(3-fluorophenyl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C27H26F3N3
|
1
|
| 1 |
Ki = 2.6 nM
|
|
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CP0436490
|
3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-5-fluoro-1H-indol-2-one
Show/Hide
|
C24H29ClFN3O
|
1
|
| 1 |
Ki = 2.81 nM
|
|
|
|
CP0394364
|
5-fluoro-3-[3-[4-(4-fluoro-2-phenylphenyl)piperazin-1-yl]propyl]-1H-indole
Show/Hide
|
C27H27F2N3
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0455696
|
2a-[4-(4-phenylpiperazin-1-yl)butyl]-1,3,4,5,8a,9-hexahydrobenzo[cd]indol-2-one
Show/Hide
|
C25H33N3O
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0500623
|
5-fluoro-3-[4-[4-(4-fluorophenyl)piperazin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
|
C22H25F2N3O
|
1
|
| 1 |
Ki = 3.4 nM
|
|
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CP0208718
|
N-methyl-2-[2-[4-(2-oxo-1,3,4,5-tetrahydrobenzo[cd]indol-2a-yl)butyl]-3,4-dihydro-1H-pyrido[3,4-b]indol-9-yl]acetamide
Show/Hide
|
C29H34N4O2
|
1
|
| 1 |
Ki = 3.548 nM
|
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|
|
CP0472795
|
3-ethyl-3-[4-(4-pyridin-2-ylpiperazin-1-yl)butyl]-1H-indol-2-one
Show/Hide
|
C23H30N4O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0920594
|
N-(Diaminomethylene)-9-hydroxy-5,9-dimethyl-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
|
C17H18ClN3O2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0366518
|
2-(6-Bromopyridin-2-ylthio)-N,N-dimethylethanamine
Show/Hide
|
C9H13BrN2S
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0425896
|
N-(diaminomethylidene)-5-ethyl-9-hydroxy-9H-fluorene-2-carboxamide
Show/Hide
|
C17H17N3O2
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0851268
|
N-(Diaminomethylene)-9-methyl-9H-fluorene-2-carboxamide hydrochloride
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0535226
|
3-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C21H26N2OS
|
1
|
| 1 |
Ki = 4.31 nM
|
|
|
|
CP0528469
|
7-chloro-3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-5-fluoro-1H-indol-2-one
Show/Hide
|
C24H28Cl2FN3O
|
1
|
| 1 |
Ki = 4.75 nM
|
|
|
|
CP0921388
|
N-(Diaminomethylene)spiro[cyclopropane-1,9'-fluorene]-2'-carboxamide hydrochloride
Show/Hide
|
C17H16ClN3O
|
1
|
| 1 |
Ki = 4.9 nM
|
|
|
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CP0512806
|
3-[4-[4-(4-fluorophenyl)piperazin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
|
C22H26FN3O
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0056386
|
5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6-chloroindolin-2-one
Show/Hide
|
C21H21ClN4OS
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0512805
|
3-ethyl-3-[4-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C25H30F3N3O
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0437042
|
3-[4-[4-(2-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H30ClN3O
|
2
|
| 1 |
Ki = 5.11 nM
|
|
|
| 2 |
Ki = 53 nM
|
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CP0407906
|
3-ethyl-3-[4-[4-(4-fluorophenyl)piperidin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C25H31FN2O
|
2
|
| 1 |
Ki = 5.3 nM
|
|
|
| 2 |
Ki = 6.9 nM
|
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|
CP0422072
|
3-ethyl-3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
|
C25H33N3O2
|
2
|
| 1 |
Ki = 5.38 nM
|
|
|
| 2 |
Ki = 5.4 nM
|
|
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|
CP0373133
|
7-chloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-5-fluoro-1H-indol-2-one
Show/Hide
|
C24H28Cl2FN3O
|
1
|
| 1 |
Ki = 5.97 nM
|
|
|
|
CP0467800
|
2-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline
Show/Hide
|
C22H33NO2S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0427792
|
(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]imidazolidine-2,4-dione
Show/Hide
|
C30H38N4O5
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0373137
|
1-benzyl-3-ethyl-3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]indol-2-one
Show/Hide
|
C32H39N3O2
|
1
|
| 1 |
Ki = 6.57 nM
|
|
|
|
CP0417895
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-6-fluoro-1,3-dihydroindol-2-one
Show/Hide
|
C22H25ClFN3O
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0437041
|
5-chloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
Show/Hide
|
C24H28Cl2FN3O
|
2
|
| 1 |
Ki = 6.99 nM
|
|
|
| 2 |
Ki = 10 nM
|
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|
|
CP0475223
|
1-[4-(benzenesulfonyl)-4-methylpentyl]-3-phenylpiperidine
Show/Hide
|
C23H31NO2S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0502111
|
1-[6-(2-Dimethylamino-ethylsulfanyl)-pyridin-2-yl]-cyclohexanol
Show/Hide
|
C15H24N2OS
|
1
|
| 1 |
Ki = 7.2 nM
|
|
|
|
CP0041133
|
6-chloro-2a-[4-[4-(4-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-1,3,4,5-tetrahydrobenzo[cd]indol-2-one
Show/Hide
|
C26H28Cl2N2O
|
1
|
| 1 |
Ki = 7.244 nM
|
|
|
|
CP0412527
|
3-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
Ki = 7.65 nM
|
|
|
|
CP0407867
|
(R)-8-(4-(3-(5-fluoro-1H-indol-3-yl)propyl)piperazin-1-yl)-2-methyl-2H-benzo[b][1,4]oxazin-3(4H)-one
Show/Hide
|
C24H27FN4O2
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0017601
|
2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-3,4-dihydro-1H-pyrido[4,3-b]indole
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C21H25N3
|
1
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| 1 |
Ki = 7.943 nM
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CP0475222
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2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4-tetrahydroisoquinoline
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C22H27NO2S
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1
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| 1 |
Ki = 8 nM
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CP0475224
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(4aS,8aR)-2-[4-(benzenesulfonyl)-4-methylpentyl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline
Show/Hide
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C21H33NO2S
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1
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| 1 |
Ki = 8 nM
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CP0382391
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N-(3-hydroxyphenyl)-N-methyl-6-(4-naphthalen-1-ylpiperazin-1-yl)hexanamide;hydrochloride
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C27H33N3O2
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1
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| 1 |
Ki = 8.1 nM
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CP0407905
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5-chloro-3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
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C24H29Cl2N3O
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1
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| 1 |
Ki = 8.27 nM
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CP0475221
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-3-phenylpyrrolidine
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C23H29NO2S
|
1
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| 1 |
Ki = 9 nM
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CP0464236
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5-chloro-3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
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C24H28Cl2FN3O
|
1
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| 1 |
Ki = 9.07 nM
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CP0528468
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5,7-dichloro-3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
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C24H28Cl3N3O
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1
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| 1 |
Ki = 9.46 nM
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CP0485745
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5,7-dichloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
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C24H28Cl3N3O
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2
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| 1 |
Ki = 9.5 nM
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| 2 |
Ki = 10.13 nM
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CP0091593
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2a-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)butyl]-1-methyl-4,5-dihydro-3H-benzo[cd]indol-2-one
Show/Hide
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C23H28N2OS
|
1
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| 1 |
Ki = 9.772 nM
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CP0472796
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3-[4-(4-pyridin-2-ylpiperazin-1-yl)butyl]-1,3-dihydroindol-2-one
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C21H26N4O
|
1
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| 1 |
Ki = 10.9 nM
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CP0472798
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3-ethyl-3-[4-[4-(3-fluorophenyl)piperazin-1-yl]butyl]-1H-indol-2-one
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C24H30FN3O
|
1
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| 1 |
Ki = 11 nM
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CP0412084
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5-fluoro-3-[3-[4-[4-fluoro-2-(furan-3-yl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
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C25H25F2N3O
|
1
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| 1 |
Ki = 11 nM
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CP0542141
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5-fluoro-3-[3-[4-(4-fluoro-2-thiophen-2-ylphenyl)piperazin-1-yl]propyl]-1H-indole
Show/Hide
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C25H25F2N3S
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1
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| 1 |
Ki = 11 nM
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CP0494256
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3-[4-[4-[3-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
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C24H25F3N2O
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1
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| 1 |
Ki = 11.1 nM
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CP0411071
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3-[2-(4-naphthalen-1-ylpiperazin-1-yl)ethyl]-1H-indol-5-ol
Show/Hide
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C24H25N3O
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1
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| 1 |
Ki = 11.6 nM
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CP0424601
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N,N-dimethyl-2-[(4-phenyl-1,3-thiazol-2-yl)sulfanyl]ethanamine
Show/Hide
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C13H16N2S2
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1
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| 1 |
Ki = 12 nM
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CP0477204
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5-fluoro-3-[3-[4-[4-fluoro-2-(3-fluorophenyl)phenyl]piperazin-1-yl]propyl]-1H-indole
Show/Hide
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C27H26F3N3
|
1
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| 1 |
Ki = 12 nM
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CP0210428
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N-(diaminomethylidene)-9H-fluorene-2-carboxamide
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C15H13N3O
|
1
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| 1 |
Ki = 12.4 nM
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CP0475220
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1-[4-[1-(benzenesulfonyl)cyclobutyl]butyl]-3-phenylpyrrolidine
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C24H31NO2S
|
1
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| 1 |
Ki = 13 nM
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CP0474955
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3-[4-[4-(3-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-6-fluoro-1,3-dihydroindol-2-one
Show/Hide
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C23H24ClFN2O
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1
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| 1 |
Ki = 13 nM
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CP0851267
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5-Methyl-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
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C16H16ClN3O2
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1
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| 1 |
Ki = 14 nM
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CP0475225
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5-[1-[4-(benzenesulfonyl)-4-methylpentyl]piperidin-3-yl]-1,3-oxazole
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C20H28N2O3S
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1
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| 1 |
Ki = 15 nM
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CP0867161
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1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride
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C22H31ClN2O2
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1
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| 1 |
Ki = 15 nM
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CP0494258
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3-[4-(4-phenylpiperazin-1-yl)butyl]-1,3-dihydroindol-2-one
Show/Hide
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C22H27N3O
|
1
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| 1 |
Ki = 16 nM
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CP0427793
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(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]imidazolidine-2,4-dione
Show/Hide
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C27H34N4O5
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1
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| 1 |
Ki = 16 nM
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CP0494257
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6-fluoro-3-[4-(4-pyridin-2-ylpiperazin-1-yl)butyl]-1,3-dihydroindol-2-one
Show/Hide
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C21H25FN4O
|
1
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| 1 |
Ki = 16.8 nM
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CP0718312
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N-(9-Hydroxy-9H-fluorene-2-carbonyl)guanidinemonohydrochloride
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C15H14ClN3O2
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1
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| 1 |
Ki = 17.6 nM
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CP0506963
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N-(diaminomethylidene)-9-hydroxy-9H-fluorene-2-carboxamide
Show/Hide
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C15H13N3O2
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1
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| 1 |
Ki = 18 nM
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CP0025667
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2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
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C18H19ClN4
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1
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| 1 |
Ki = 19.95 nM
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CP0247158
|
3-[methyl-[3-(4-phenylpiperazin-1-yl)propyl]amino]phenol
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C20H27N3O
|
1
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| 1 |
Ki = 20 nM
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CP0407903
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3-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-3-ethyl-1H-indol-2-one
Show/Hide
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C23H28ClN3O
|
1
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| 1 |
Ki = 21 nM
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CP0514330
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-4-phenylpiperazine
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C23H30N2O2S
|
1
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| 1 |
Ki = 22 nM
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CP0424605
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2-[(4-tert-butyl-1,3-thiazol-2-yl)sulfanyl]-N,N-dimethylethanamine
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C11H20N2S2
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1
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| 1 |
Ki = 22 nM
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CP0424508
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(5Z)-3-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propyl]-5-[(3,4-dimethoxyphenyl)methylidene]imidazolidine-2,4-dione
Show/Hide
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C25H28Cl2N4O4
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1
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| 1 |
Ki = 22 nM
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CP0376451
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ethyl (3R)-1-[4-(benzenesulfonyl)-4-methylpentyl]piperidine-3-carboxylate
Show/Hide
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C20H31NO4S
|
1
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| 1 |
Ki = 24 nM
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CP0860616
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3-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
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C20H22ClN3O2S
|
1
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| 1 |
Ki = 24 nM
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CP0472799
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3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-6-fluoro-1,3-dihydroindol-2-one
Show/Hide
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C22H25ClFN3O
|
1
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| 1 |
Ki = 25 nM
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CP0065912
|
CAS_15574-96-6
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C19H21NS
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1
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| 1 |
Ki = 25 nM
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CP0427995
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Amisulpride
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C17H27N3O4S
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1
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| 1 |
Ki = 25.12 nM
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CP0464237
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3-ethyl-3-[4-[4-(4-methoxyphenyl)piperazin-1-yl]butyl]-1H-indol-2-one
Show/Hide
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C25H33N3O2
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1
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| 1 |
Ki = 25.4 nM
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CP0505629
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-4-phenylpiperidine
Show/Hide
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C24H31NO2S
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1
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| 1 |
Ki = 26 nM
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CP0394360
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1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine
Show/Hide
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C18H22N2S
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1
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| 1 |
Ki = 26 nM
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CP0497712
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N,N-dimethyl-2-[(4-pyridin-4-yl-1,3-thiazol-2-yl)sulfanyl]ethanamine
Show/Hide
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C12H15N3S2
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1
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| 1 |
Ki = 27 nM
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CP0379189
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2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine
Show/Hide
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C16H16N2O2S
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1
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| 1 |
Ki = 29 nM
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CP0907774
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5-Fluoro-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
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C15H13ClFN3O2
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1
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| 1 |
Ki = 29 nM
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CP0033479
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(chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine
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C17H19ClN2S
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1
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| 1 |
Ki = 31.62 nM
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CP0946032
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8-Chloro-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
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C15H13Cl2N3O2
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1
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| 1 |
Ki = 33 nM
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CP0373138
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3-ethyl-1-methyl-3-[4-(4-phenylpiperazin-1-yl)butyl]indol-2-one
Show/Hide
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C25H33N3O
|
1
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| 1 |
Ki = 33.38 nM
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CP0512705
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3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-5-fluoro-1,3-dihydroindol-2-one
Show/Hide
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C22H25ClFN3O
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1
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| 1 |
Ki = 40 nM
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CP0532181
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5-fluoro-3-[4-[4-[3-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
|
C24H24F4N2O
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1
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| 1 |
Ki = 40 nM
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CP0907775
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5-Chloro-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
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C15H13Cl2N3O2
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1
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| 1 |
Ki = 41 nM
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CP0957283
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N-(Diaminomethylene)-9-hydroxy-5-(hydroxymethyl)-9H-fluorene-2-carboxamide hydrochloride
Show/Hide
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C16H16ClN3O3
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1
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| 1 |
Ki = 41 nM
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CP0848922
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N-(Diaminomethylene)-9H-carbazole-2-carboxamidemonohydrochloride
Show/Hide
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C14H13ClN4O
|
1
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| 1 |
Ki = 42 nM
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CP0424512
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(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]imidazolidine-2,4-dione
Show/Hide
|
C26H32N4O5
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1
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| 1 |
Ki = 42 nM
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CP0865101
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9-Amino-N-(diaminomethylene)-9H-fluorene-2-carboxamide dihydrochloride
Show/Hide
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C15H15ClN4O
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1
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| 1 |
Ki = 43 nM
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CP0162073
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5-fluoro-3-[4-(4-phenylpiperazin-1-yl)butyl]-1,3-dihydroindol-2-one
Show/Hide
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C22H26FN3O
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2
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| 1 |
Ki = 44 nM
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| 2 |
Ki = 47 nM
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CP0907776
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N-(Diaminomethylene)-9-hydroxy-5-(methoxymethyl)-9H-fluorene-2-carboxamide hydrochloride
Show/Hide
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C17H18ClN3O3
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1
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| 1 |
Ki = 50 nM
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CP0532180
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3-[4-[4-(3-chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-ethyl-5-fluoro-1H-indol-2-one
Show/Hide
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C25H28ClFN2O
|
1
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| 1 |
Ki = 52 nM
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CP0553842
|
1-[2-[1-(benzenesulfonyl)cyclobutyl]ethyl]-3-phenylpyrrolidine
Show/Hide
|
C22H27NO2S
|
1
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| 1 |
Ki = 53 nM
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CP0386567
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1-[4-(benzenesulfonyl)-4-methylpentyl]-3-(trifluoromethyl)piperidine
Show/Hide
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C18H26F3NO2S
|
1
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| 1 |
Ki = 54 nM
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CP0922197
|
N-(9-Fluoro-9H-fluorene-2-carbonyl)guanidine hydrochloride
Show/Hide
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C15H13ClFN3O
|
1
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| 1 |
Ki = 57 nM
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CP0040250
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2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol
Show/Hide
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C21H25N3O2S
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1
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| 1 |
Ki = 63.1 nM
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CP0042927
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7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one
Show/Hide
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C23H27Cl2N3O2
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1
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| 1 |
Ki = 63.1 nM
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CP0291324
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1-(2,3-dihydro-1,4-benzodioxin-5-yl)-4-[[5-(4-fluorophenyl)pyridin-3-yl]methyl]piperazine
Show/Hide
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C24H24FN3O2
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1
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| 1 |
Ki = 63.1 nM
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CP0123937
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3-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-indol-5-ol
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 63.1 nM
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CP0864251
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1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride
Show/Hide
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C24H36Cl2N2O3
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1
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| 1 |
Ki = 70 nM
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CP0512794
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5,7-dichloro-3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
Show/Hide
|
C24H27Cl3FN3O
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1
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| 1 |
Ki = 72 nM
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CP0873359
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2-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
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1
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| 1 |
Ki = 74 nM
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CP0420924
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(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-[3-(4-pyrimidin-2-ylpiperazin-1-yl)propyl]imidazolidine-2,4-dione
Show/Hide
|
C23H28N6O4
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1
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| 1 |
Ki = 74 nM
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CP0045063
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2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
Show/Hide
|
C17H20N4S
|
1
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| 1 |
Ki = 79.43 nM
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CP0376362
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2-(1,3-benzothiazol-2-ylsulfanyl)-N,N-dimethylethanamine
Show/Hide
|
C11H14N2S2
|
1
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| 1 |
Ki = 84 nM
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CP0920597
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8-Methyl-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
|
C16H16ClN3O2
|
1
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| 1 |
Ki = 87 nM
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CP0873149
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1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride
Show/Hide
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C24H36Cl2N2O3
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1
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| 1 |
Ki = 89 nM
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CP0873148
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1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride
Show/Hide
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C20H27Cl3N2O
|
1
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| 1 |
Ki = 90 nM
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CP0382081
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2-[4-(benzenesulfonyl)butyl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinoline
Show/Hide
|
C19H29NO2S
|
1
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| 1 |
Ki = 96 nM
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CP0532182
|
5,7-dichloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3-ethyl-6-fluoro-1H-indol-2-one
Show/Hide
|
C24H27Cl3FN3O
|
1
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| 1 |
Ki = 96 nM
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CP0418433
|
N,N-dimethyl-2-(2-phenylpyridin-4-yl)sulfanylethanamine
Show/Hide
|
C15H18N2S
|
1
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| 1 |
Ki = 100 nM
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CP0466838
|
2-(4-(4-(5-fluoro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)butyl)isoindoline-1,3-dione
Show/Hide
|
C25H24FN3O2
|
1
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| 1 |
Ki = 100 nM
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CP0512807
|
5,7-dichloro-3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1,3-dihydroindol-2-one
Show/Hide
|
C22H24Cl3N3O
|
1
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| 1 |
Ki = 107 nM
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CP0438711
|
(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]imidazolidine-2,4-dione
Show/Hide
|
C30H36Cl2N4O4
|
1
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| 1 |
Ki = 125 nM
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CP0530973
|
3-[4-[4-(2,4-dichlorophenyl)piperazin-1-yl]butyl]-3-ethyl-1H-indol-2-one
Show/Hide
|
C24H29Cl2N3O
|
1
|
| 1 |
Ki = 139 nM
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CP0848923
|
N-(Diaminomethylene)-10H-phenoxazine-2-carboxamide monohydrochloride
Show/Hide
|
C14H13ClN4O2
|
1
|
| 1 |
Ki = 144 nM
|
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CP0920596
|
6-Chloro-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
Show/Hide
|
C15H13Cl2N3O2
|
1
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| 1 |
Ki = 160 nM
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CP0429362
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N,N-dimethyl-2-[(5-methyl-4-phenyl-1,3-thiazol-2-yl)sulfanyl]ethanamine
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C14H18N2S2
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1
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| 1 |
Ki = 170 nM
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CP0922196
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9-(Acetylamino)-N-(diaminomethylene)-9H-fluorene-2-carboxamide monohydrochloride
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C17H17ClN4O2
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1
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| 1 |
Ki = 180 nM
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CP0379280
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2-[3-[4-[1-(benzenesulfonyl)indol-4-yl]piperazin-1-yl]propoxy]benzamide
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C28H30N4O4S
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1
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| 1 |
Ki = 180 nM
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CP0918281
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N-(Diaminomethylene)-9-oxo-9H-fluorene-2-carboxamide
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C15H11N3O2
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1
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| 1 |
Ki = 185 nM
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CP0874364
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N-(9H-Fluorene-1-carbonyl)guanidinemonohydrochloride
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C15H14ClN3O
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1
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| 1 |
Ki = 239 nM
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CP0424507
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(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[4-(4-pyrimidin-2-ylpiperazin-1-yl)butyl]imidazolidine-2,4-dione
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C28H36N6O4
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1
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| 1 |
Ki = 298 nM
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CP0008601
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4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
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C21H23ClFNO2
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1
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| 1 |
Ki = 316.23 nM
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CP0777252
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2-Iodo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
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C20H22IN3O2S
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1
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| 1 |
Ki = 329 nM
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CP0420922
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(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propyl]imidazolidine-2,4-dione
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C29H34Cl2N4O4
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1
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| 1 |
Ki = 380 nM
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CP0853339
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1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride
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C24H36Cl2N2O2
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1
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| 1 |
Ki = 388 nM
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CP0376430
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ethyl (3S)-1-[4-(benzenesulfonyl)-4-methylpentyl]piperidine-3-carboxylate
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C20H31NO4S
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1
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| 1 |
Ki = 455 nM
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CP0330654
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2-[1-(benzenesulfonyl)indol-4-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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1
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| 1 |
Ki = 460 nM
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CP0318039
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3-(2-Dimethylamino-ethyl)-1H-indole-2-carboxylic acid ethyl ester
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C15H20N2O2
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1
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| 1 |
Ki = 510 nM
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CP0527087
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-4-methylpiperidine
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C19H29NO2S
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1
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| 1 |
Ki = 550 nM
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CP0144949
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2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulfonyl)-1H-indol-3-yl]ethan-1-amine
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C15H13ClN4O2S2
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1
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| 1 |
Ki = 679 nM
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CP0420923
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(5Z)-5-[(3,4-dimethoxyphenyl)methylidene]-3-[4-(4-pyrimidin-2-ylpiperazin-1-yl)butyl]imidazolidine-2,4-dione
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C24H30N6O4
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1
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| 1 |
Ki = 933 nM
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CP0902025
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1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride
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C25H38Cl2N2O2
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1
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| 1 |
Ki = 1050 nM
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CP0439649
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N,N-dimethyl-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethanamine
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C12H16N4S
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1
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| 1 |
Ki = 1200 nM
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CP0418991
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[1-(benzenesulfonyl)-4-[2-(dimethylamino)ethyl]indol-2-yl]-phenylmethanone
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C25H24N2O3S
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1
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| 1 |
Ki = 1300 nM
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CP0376998
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4-[3-(1,2,3,6-Tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
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C19H19N3O2S
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1
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| 1 |
Ki = 1555 nM
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CP0409092
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[3-[2-(dimethylamino)ethyl]-5-hydroxyindol-1-yl]-phenylmethanone
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C19H20N2O2
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1
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| 1 |
Ki = 1600 nM
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CP0045069
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2-[1-(benzenesulfonyl)-5-methoxyindol-3-yl]-N,N-dimethylethanamine
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C19H22N2O3S
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1
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| 1 |
Ki = 1900 nM
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CP0497215
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]piperidine
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C18H27NO2S
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1
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| 1 |
Ki = 2700 nM
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CP0853338
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1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride
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C23H34Cl2N2O2
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1
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| 1 |
Ki = 3027 nM
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CP0874185
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2-(4-{2-[2-(2,3,5-Trimethylphenoxy)ethoxy]ethyl}piperazin-1-yl)ethanol dihydrochloride
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C19H34Cl2N2O3
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1
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| 1 |
Ki = 3142 nM
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CP0864252
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1-Benzyl-4-{2-[2-(mesityloxy)ethoxy]ethyl}piperazine dihydrochloride
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C24H36Cl2N2O2
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1
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| 1 |
Ki = 3160 nM
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CP0405226
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N,N-dimethyl-2-[(5-phenyl-1,3-thiazol-2-yl)sulfanyl]ethanamine
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C13H16N2S2
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1
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| 1 |
Ki = 3200 nM
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CP0255950
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2-[1-(benzenesulfonyl)indol-3-yl]-N,N-dimethylethanamine
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C18H20N2O2S
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1
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| 1 |
Ki = 3700 nM
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CP0024732
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5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1-yl}-benzofuran-2-carboxylic acid amide
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C26H27N5O2
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1
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| 1 |
Ki = 3900 nM
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CP0527086
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1-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]-4-methylpiperazine
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C18H28N2O2S
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1
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| 1 |
Ki = 5800 nM
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CP0505978
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N,N-dimethyl-2-(1,3-thiazol-2-ylsulfanyl)ethanamine
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C7H12N2S2
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1
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| 1 |
Ki = 6800 nM
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CP0850547
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N-(Diaminomethylene)dibenzo[b,d]furan-3-carboxamidemonohydrochloride
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C14H12ClN3O2
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1
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| 1 |
Ki > 100 nM
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CP0895764
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(2E)-N-(Diaminomethylene)-3-(9-hydroxy-9H-fluoren-2-yl)acrylamide monohydrochloride
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C17H16ClN3O2
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1
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| 1 |
Ki > 100 nM
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CP0415200
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9-butyl-N-(diaminomethylidene)-9-hydroxyfluorene-2-carboxamide;hydrochloride
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C19H22ClN3O2
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1
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| 1 |
Ki > 100 nM
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CP0848920
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N-(9-Hydroxy-9H-fluorene-3-carbonyl)guanidinemonohydrochloride
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C15H14ClN3O2
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1
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| 1 |
Ki > 1000 nM
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CP0882311
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N-(9H-Fluorene-4-carbonyl)guanidinemonohydrochloride
Show/Hide
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C15H14ClN3O
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1
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| 1 |
Ki > 1000 nM
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CP0905129
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N-(Diaminomethylene)-10H-phenoxazine-3-carboxamide monohydrochloride
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C14H13ClN4O2
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1
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| 1 |
Ki > 1000 nM
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CP0865100
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7-Chloro-N-(diaminomethylene)-9-hydroxy-9Hfluorene-2-carboxamide hydrochloride
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C15H13Cl2N3O2
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1
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| 1 |
Ki > 1000 nM
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CP0458060
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(5Z)-5-[(3-cyclopentyloxy-4-methoxyphenyl)methylidene]-3-[3-(4-pyrimidin-2-ylpiperazin-1-yl)propyl]imidazolidine-2,4-dione
Show/Hide
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C27H34N6O4
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1
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| 1 |
Ki > 1000 nM
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CP0393293
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4-(6-Chloro-3-piperidin-4-yl-indole-1-sulfonyl)-phenylamine
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C19H20ClN3O2S
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1
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| 1 |
Ki > 2000 nM
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CP0469570
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N,N-dimethyl-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethanamine
Show/Hide
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C12H15N3OS
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1
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| 1 |
Ki > 4000 nM
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CP0377633
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4-[5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-indole-1-sulfonyl]-phenylamine
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C20H21N3O3S
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1
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| 1 |
Ki > 5000 nM
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CP0186950
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(4S,5S)-4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tetrahydro-benzo[cd]indol-5-ol
Show/Hide
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C20H22N2O3S
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1
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| 1 |
Ki > 5800 nM
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CP0436926
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3-[1-(benzenesulfonyl)cyclobutyl]-N,N-dimethylpropan-1-amine
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C15H23NO2S
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1
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| 1 |
Ki > 7000 nM
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CP0514331
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4-[3-[1-(benzenesulfonyl)cyclobutyl]propyl]morpholine
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C17H25NO3S
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1
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| 1 |
Ki > 7000 nM
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CP0370584
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4-(2-bromo-6-piperazin-1-ylpyridin-4-yl)sulfonylaniline
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C15H17BrN4O2S
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1
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| 1 |
Ki < 10000 nM
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CP0415376
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4-(4-aminophenyl)sulfonyl-6-bromo-N-methylpyridin-2-amine
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C12H12BrN3O2S
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1
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| 1 |
Ki < 10000 nM
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CP0874735
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4-Amino-N-(2,6-bis-methylamino-pyrimidin-4-yl)-benzenesulfonamide dihydrobromide
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C12H18Br2N6O2S
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1
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| 1 |
Ki < 10000 nM
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CP0370117
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4-(2-Bromo-6-pyrrolidin-1-yl-pyridine-4-sulfonyl)-phenylamine
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C15H16BrN3O2S
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1
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| 1 |
Ki < 100000 nM
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