Brief Information of the Compound and Protein
| Compound Name |
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
5-hydroxytryptamine receptor 7
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Protein Classification |
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
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| Uniprot ID | Gene Name | HTR7 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Biochemical Assays
| 1 | Ki = 9 nM | ||
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| 2 | Ki = 12.59 nM | ||
| 3 | Ki = 39.81 nM | ||
| 4 | Ki = 40 nM | ||
| 5 | Ki = 45.5 nM | ||
| 6 | Ki = 48 nM | ||
| 7 | Ki = 100 nM | ||