| Compound ID |
Compound Name |
Compound Formula |
|
CP0416475
|
N-(2-hydroxyethyl)-3-methyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C23H20F3N3O2S
|
1
|
| 1 |
EC50 = 5.2 nM
|
|
|
|
CP0476663
|
N-(2-methoxyethyl)-3-methyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C24H22F3N3O2S
|
1
|
| 1 |
EC50 = 9.6 nM
|
|
|
|
CP0539172
|
4-[2-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C20H16F4N2OS
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0466025
|
N-(2-hydroxyethyl)-3,5-dimethyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C24H22F3N3O2S
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0511769
|
N-(2-methoxyethyl)-3,5-dimethyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C25H24F3N3O2S
|
1
|
| 1 |
EC50 = 17 nM
|
|
|
|
CP0416474
|
N-(2-hydroxyethyl)-5-(hydroxymethyl)-3-methyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C24H22F3N3O3S
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0419766
|
4-[5-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]-2-methylpyrazol-3-yl]-2-methylbenzamide
Show/Hide
|
C20H17F4N3O
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0419767
|
4-[2-[(3-chloro-5-fluorophenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C19H16ClFN2OS
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0398813
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-4-yl]benzamide
Show/Hide
|
C25H20F3NO3
|
1
|
| 1 |
EC50 = 28.18 nM
|
|
|
|
CP0334329
|
3-[2-[(3-chloro-5-fluorophenyl)methyl]-1-benzothiophen-7-yl]-N-(2-methoxyethyl)benzamide
Show/Hide
|
C25H21ClFNO2S
|
1
|
| 1 |
EC50 = 29.51 nM
|
|
|
|
CP0523051
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-7-yl]benzamide
Show/Hide
|
C25H20F3NO3
|
1
|
| 1 |
EC50 = 34.67 nM
|
|
|
|
CP0532168
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]benzamide
Show/Hide
|
C25H20F3NO2S
|
1
|
| 1 |
EC50 = 37.15 nM
|
|
|
|
CP0555255
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-4-yl]benzamide
Show/Hide
|
C25H20F3NO2S
|
1
|
| 1 |
EC50 = 38.02 nM
|
|
|
|
CP0555256
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]indazol-4-yl]benzamide
Show/Hide
|
C24H20F3N3O2
|
1
|
| 1 |
EC50 = 38.9 nM
|
|
|
|
CP0475963
|
N-(2-methoxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]benzamide
Show/Hide
|
C26H22F3NO2S
|
1
|
| 1 |
EC50 = 42.66 nM
|
|
|
|
CP0466024
|
N-(2-hydroxyethyl)-2-methyl-5-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-3-carboxamide
Show/Hide
|
C23H20F3N3O2S
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0398817
|
N-(2-amino-2-oxoethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]benzamide
Show/Hide
|
C25H19F3N2O2S
|
1
|
| 1 |
EC50 = 54.95 nM
|
|
|
|
CP0407281
|
4-[4-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]-2-methylimidazol-1-yl]-2-methylbenzamide
Show/Hide
|
C20H17F4N3O
|
1
|
| 1 |
EC50 = 59 nM
|
|
|
|
CP0547139
|
N-(2-methoxyethyl)-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C23H20F3N3O2S
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0578013
|
N-(2-methoxyethyl)-5-methyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C24H22F3N3O2S
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0398815
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]indazol-7-yl]benzamide
Show/Hide
|
C24H20F3N3O2
|
1
|
| 1 |
EC50 = 64.57 nM
|
|
|
|
CP0414086
|
2-methyl-4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C20H17F3N2OS
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
|
CP0033447
|
4-[3-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]-5-methyl-1,2,4-triazol-1-yl]-2-methylbenzamide
Show/Hide
|
C19H16F4N4O
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0398814
|
N-(2-hydroxyethyl)-3-[3-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-7-yl]benzamide
Show/Hide
|
C26H22F3NO3
|
1
|
| 1 |
EC50 = 81.28 nM
|
|
|
|
CP0510805
|
2-ethyl-4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C21H19F3N2OS
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0448356
|
N-(2-amino-2-oxoethyl)-3-[4-fluoro-2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]benzamide
Show/Hide
|
C25H18F4N2O2S
|
1
|
| 1 |
EC50 = 83.18 nM
|
|
|
|
CP0519760
|
N-(2-hydroxyethyl)-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C22H18F3N3O2S
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0547944
|
4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]-2-(trifluoromethyl)benzamide
Show/Hide
|
C20H14F6N2OS
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0543059
|
4-[2-[(3-chlorophenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C19H17ClN2OS
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0519759
|
N-(2-hydroxyethyl)-3-(hydroxymethyl)-5-methyl-1-[2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzothiophen-7-yl]pyrazole-4-carboxamide
Show/Hide
|
C24H22F3N3O3S
|
1
|
| 1 |
EC50 = 146 nM
|
|
|
|
CP0402870
|
4-[2-[(3-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C20H20N2O2S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0407282
|
2-methoxy-4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C20H17F3N2O2S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0523053
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-2,3-dihydro-1-benzofuran-7-yl]benzamide
Show/Hide
|
C25H22F3NO3
|
1
|
| 1 |
EC50 = 208.93 nM
|
|
|
|
CP0432823
|
4-[2-[(4-chlorophenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C19H17ClN2OS
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0447332
|
4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C19H15F3N2OS
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0539173
|
4-[2-[(3-fluorophenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C19H17FN2OS
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0419769
|
4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]-2-propan-2-ylbenzamide
Show/Hide
|
C22H21F3N2OS
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0543061
|
2-fluoro-4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C19H14F4N2OS
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0565934
|
6-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]pyridine-3-carboxamide
Show/Hide
|
C18H14F3N3OS
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0523052
|
N-(2-hydroxyethyl)-3-[2-[[3-(trifluoromethyl)phenyl]methyl]-2,3-dihydro-1-benzofuran-4-yl]benzamide
Show/Hide
|
C25H22F3NO3
|
1
|
| 1 |
EC50 = 645.65 nM
|
|
|
|
CP0558689
|
4-[2-[[3-(dimethylamino)phenyl]methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C21H23N3OS
|
1
|
| 1 |
EC50 = 690 nM
|
|
|
|
CP0432830
|
3-methyl-4-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]benzamide
Show/Hide
|
C20H17F3N2OS
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0419768
|
4-[2-[(2-chlorophenyl)methyl]-4-methyl-1,3-thiazol-5-yl]-2-methylbenzamide
Show/Hide
|
C19H17ClN2OS
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0489437
|
N-(2-hydroxyethyl)-3-[3-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1-benzofuran-4-yl]benzamide
Show/Hide
|
C26H22F3NO3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0865725
|
N-(3,4-dimethoxyphenethyl)-4-(4-methoxyphenyl)pyrimidin-2-amine
Show/Hide
|
C21H23N3O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0030334
|
5-[4-methyl-2-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-5-yl]pyridine-2-carboxamide
Show/Hide
|
C18H14F3N3OS
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
