Protein Information

General Information of the Protein

Protein ID	PT00909
Protein Name	Peroxisome proliferator-activated receptor delta
Secondarily Protein Name	NUCI Nuclear hormone receptor 1 Nuclear receptor subfamily 1 group C member 2 Peroxisome proliferator-activated receptor beta
Gene Name	PPARD
Secondarily Gene Name	NR1C2 PPARB
Sequence	MEQPQEEAPEVREEEEKEEVAEAEGAPELNGGPQHALPSSSYTDLSRSSSPPSLLDQLQMGCDGASCGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCERSCKIQKKNRNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTANEGSQYNPQVADLKAFSKHIYNAYLKNFNMTKKKARSILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKEISVHVFYRCQCTTVETVRELTEFAKSIPSFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKDGLLVANGSGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGDRPGLMNVPRVEAIQDTILRALEFHLQANHPDAQYLFPKLLQKMADLRQLVTEHAQMMQRIKKTETETSLHPLLQEIYKDMY Show/Hide
Organism	Homo sapiens, Human
Protein Classification	Transcription factor > Nuclear receptor > Nuclear hormone receptor subfamily 1 > Nuclear hormone receptor subfamily 1 group C > Nuclear hormone receptor subfamily 1 group C member 2
Function	Ligand-activated transcription factor key mediator of energy metabolism in adipose tissues (PubMed:35675826). Receptor that binds peroxisome proliferators such as hypolipidemic drugs and fatty acids. Has a preference for poly-unsaturated fatty acids, such as gamma-linoleic acid and eicosapentanoic acid. Once activated by a ligand, the receptor binds to promoter elements of target genes. Regulates the peroxisomal beta-oxidation pathway of fatty acids. Functions as transcription activator for the acyl-CoA oxidase gene. Decreases expression of NPC1L1 once activated by a ligand. Show/Hide
Uniprot ID	Primary ID: Q03181 Secondarily ID: A8K6J6 B4E3V3 B6ZGS1 B7Z3W1 E9PE18 Q5D1P0 Q7Z5K0 Q9BUD4 Show/Hide
Ensembl ID	ENSG00000112033
HGNC ID	HGNC:9235
Subcellular Location	Nucleus

Map of Molecular Bioactivity Related to the Protein

Map of Molecular Bioactivity Related to the Protein Protein Cell Line Compound Bioactivity Value: <= 0.1 μM > 0.1 μM and <= 10 μM > 10 μM Imprecise Activity

Table of Molecular Bioactivities Related to the Protein

Cell Line ID: CL000044 , CV-1

Cell Line Info

Compound ID	Compound Name	Compound Formula
CP0451331 Compound Info	US10399958, Compound 2e Show/Hide	C25H25F3N2O4	1
1	EC50 = 0.3 nM Bioactivity Info	TI LI LO TS
CP0421004 Compound Info	(3R)-3-methyl-6-[2-[[5-methyl-2-[4-(trifluoromethoxy)phenyl]imidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C25H27F3N2O4	1
1	EC50 = 0.4 nM Bioactivity Info	TI LI LO TS
CP0457346 Compound Info	2-[2-methyl-4-[(1R)-2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C30H25F3O3S	1
1	EC50 = 0.7 nM Bioactivity Info	TI LI LO TS
CP0416556 Compound Info	(3R)-6-[2-[[2-[4-(furan-2-yl)phenyl]-5-(trifluoromethyl)imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C28H27F3N2O4	1
1	EC50 = 0.7 nM Bioactivity Info	TI LI LO TS
CP0444892 Compound Info	6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C27H28N2O4	1
1	EC50 = 0.7 nM Bioactivity Info	TI LI LO TS
CP0444891 Compound Info	(3R)-6-[2-[[2-(4-chloro-3-fluorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C24H26ClFN2O3	1
1	EC50 = 0.8 nM Bioactivity Info	TI LI LO TS
CP0054286 Compound Info	2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)acetic acid Show/Hide	C21H18F3NO3SSe	1
1	EC50 = 0.9 nM Bioactivity Info	TI LI LO TS
CP0075560 Compound Info	(R)-3-(4-(3-(1-(5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid Show/Hide	C30H30ClFN2O4	1
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
CP0051318 Compound Info	(R)-3-(4-(3-(2-benzoyl-4-ethylphenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C29H32O5	2
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
2	EC50 = 5 nM Bioactivity Info	TI LI LO TS
CP0039118 Compound Info	2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid Show/Hide	C21H18F3NO3S2	7
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
2	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
3	EC50 = 1.7 nM Bioactivity Info	TI LI LO TS
4	EC50 = 2 nM Bioactivity Info	TI LI LO TS
5	EC50 = 2.5 nM Bioactivity Info	TI LI LO TS
6	EC50 = 3.162 nM Bioactivity Info	TI LI LO TS
7	IC50 = 125.89 nM Bioactivity Info	TI LI LO TS
CP0057743 Compound Info	(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethyl-phenoxy)-butoxy]-phenyl}-propionic acid Show/Hide	C27H27F3O5	1
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
CP0498362 Compound Info	2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)acetic acid Show/Hide	C21H17F4NO3SSe	1
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
CP0385347 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]butylsulfanyl]phenoxy]acetic acid Show/Hide	C24H24F3NO3S2	1
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
CP0444893 Compound Info	(E)-6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H28N2O4	1
1	EC50 = 1 nM Bioactivity Info	TI LI LO TS
CP0432336 Compound Info	2-[4-[2-cyclopropyl-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C25H24F3NO3S2	1
1	EC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0454766 Compound Info	2-[2-methyl-4-[3-methyl-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]butyl]sulfanylphenoxy]acetic acid Show/Hide	C25H26F3NO3S2	1
1	EC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0447734 Compound Info	2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H22F7NO3S2	1
1	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0495382 Compound Info	2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C28H22ClF4NO3S2	1
1	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0568375 Compound Info	(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyl-1H-pyrazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H28N2O4	1
1	EC50 = 1.2 nM Bioactivity Info	TI LI LO TS
CP0527650 Compound Info	(E)-6-[2-[[5-[4-(furan-2-yl)phenyl]-3-methylimidazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H28N2O4	1
1	EC50 = 1.3 nM Bioactivity Info	TI LI LO TS
CP0517564 Compound Info	(3R)-6-[2-[[5-chloro-2-[4-(trifluoromethyl)phenyl]imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C24H24ClF3N2O3	1
1	EC50 = 1.5 nM Bioactivity Info	TI LI LO TS
CP0444762 Compound Info	(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyl-1,2-oxazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H27NO5	1
1	EC50 = 1.5 nM Bioactivity Info	TI LI LO TS
CP0134379 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-phenylethyl]sulfanylphenoxy]acetic acid Show/Hide	C28H24F3NO3S2	1
1	EC50 = 1.6 nM Bioactivity Info	TI LI LO TS
CP0381217 Compound Info	2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C23H21F4NO3SSe	1
1	EC50 = 1.8 nM Bioactivity Info	TI LI LO TS
CP0416092 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]propylsulfanyl]phenoxy]acetic acid Show/Hide	C23H22F3NO3S2	1
1	EC50 = 1.8 nM Bioactivity Info	TI LI LO TS
CP0171815 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]acetic acid Show/Hide	C27H30ClNO5S	1
1	EC50 = 1.995 nM Bioactivity Info	TI LI LO TS
CP0082065 Compound Info	(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acid Show/Hide	C27H27F3O6	1
1	EC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0540081 Compound Info	(3R)-6-[2-[[4-[3,5-difluoro-4-(furan-2-yl)phenyl]-2-methyl-1,3-thiazol-5-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C28H27F2NO4S	1
1	EC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0450700 Compound Info	2-[4-[2-(2,6-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C28H22F5NO3S2	1
1	EC50 = 2.1 nM Bioactivity Info	TI LI LO TS
CP0416093 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]pentylsulfanyl]phenoxy]acetic acid Show/Hide	C25H26F3NO3S2	1
1	EC50 = 2.3 nM Bioactivity Info	TI LI LO TS
CP0169972 Compound Info	2-[4-[butyl-[2-chloro-3-[4-(trifluoromethoxy)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO6S	1
1	EC50 = 2.512 nM Bioactivity Info	TI LI LO TS
CP0218060 Compound Info	2-[4-[butyl-[2-chloro-3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	EC50 = 2.512 nM Bioactivity Info	TI LI LO TS
CP0050852 Compound Info	2-[(1S)-5-{3-[2-propyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid Show/Hide	C30H35NO4S	1
1	EC50 = 2.6 nM Bioactivity Info	TI LI LO TS
CP0454802 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-3-phenylpropyl]sulfanylphenoxy]acetic acid Show/Hide	C29H26F3NO3S2	1
1	EC50 = 2.6 nM Bioactivity Info	TI LI LO TS
CP0365610 Compound Info	2-[2-methyl-4-[2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C30H25F3O3S	1
1	EC50 = 2.6 nM Bioactivity Info	TI LI LO TS
CP0416555 Compound Info	(3R)-3-methyl-6-[2-[[2-[4-(trifluoromethoxy)phenyl]-5-(trifluoromethyl)imidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C25H24F6N2O4	1
1	EC50 = 2.6 nM Bioactivity Info	TI LI LO TS
CP0717529 Compound Info	[(1S)-5-{3-[4-(6,7-dihydro-5H-pyrano[2,3-d]1,3thiazol-2-yl)-2-propylphenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid Show/Hide	C29H35NO5S	1
1	EC50 = 2.7 nM Bioactivity Info	TI LI LO TS
CP0421002 Compound Info	(3R)-6-[2-[[5-cyano-2-[4-(trifluoromethyl)phenyl]imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C25H24F3N3O3	1
1	EC50 = 2.7 nM Bioactivity Info	TI LI LO TS
CP0410207 Compound Info	2-[4-[2-(2,6-dichlorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C28H22Cl2F3NO3S2	1
1	EC50 = 2.8 nM Bioactivity Info	TI LI LO TS
CP0420999 Compound Info	(3R)-3-methyl-6-[2-[[5-(trifluoromethyl)-2-[4-(trifluoromethyl)phenyl]imidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C25H24F6N2O3	1
1	EC50 = 2.9 nM Bioactivity Info	TI LI LO TS
CP0466247 Compound Info	2-[2-methyl-4-[2-phenyl-1-[6-[4-(trifluoromethyl)phenyl]pyridin-3-yl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C29H24F3NO3S	1
1	EC50 = 3.2 nM Bioactivity Info	TI LI LO TS
CP0549476 Compound Info	(3R)-6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C28H30N2O4	1
1	EC50 = 3.7 nM Bioactivity Info	TI LI LO TS
CP0421000 Compound Info	6-[2-[[5-methyl-2-(2-methyl-1-benzofuran-5-yl)imidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C26H28N2O4	1
1	EC50 = 3.9 nM Bioactivity Info	TI LI LO TS
CP0035140 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-5-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	EC50 = 4 nM Bioactivity Info	TI LI LO TS
CP0075562 Compound Info	3-(4-(3-((5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C28H27ClN2O4	1
1	EC50 = 4 nM Bioactivity Info	TI LI LO TS
CP0409323 Compound Info	2-[2-methyl-4-(2-{4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}ethyl)phenoxy]acetic acid Show/Hide	C22H20F3NO3S	1
1	EC50 = 4 nM Bioactivity Info	TI LI LO TS
CP0396630 Compound Info	2-[4-[2-(2,6-difluorophenyl)-1-[4-(4-fluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H23F3O3S	1
1	EC50 = 4 nM Bioactivity Info	TI LI LO TS
CP0454767 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(4-phenylphenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C34H28F3NO3S2	1
1	EC50 = 4.4 nM Bioactivity Info	TI LI LO TS
CP0393242 Compound Info	2-methyl-2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)propanoic acid Show/Hide	C23H22F3NO3SSe	1
1	EC50 = 4.5 nM Bioactivity Info	TI LI LO TS
CP0396628 Compound Info	2-[2-methyl-4-[2-phenyl-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C29H23F3O3S	1
1	EC50 = 4.5 nM Bioactivity Info	TI LI LO TS
CP0451332 Compound Info	6-[2-[[2-[4-(furan-2-yl)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-2,2-dimethylhexanoic acid Show/Hide	C29H32N2O4	1
1	EC50 = 4.5 nM Bioactivity Info	TI LI LO TS
CP0548509 Compound Info	2-[4-[2-(2,4-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C28H22F5NO3S2	1
1	EC50 = 4.6 nM Bioactivity Info	TI LI LO TS
CP0421001 Compound Info	(3R)-6-[2-[[2-(4-cyanophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C25H27N3O3	1
1	EC50 = 4.6 nM Bioactivity Info	TI LI LO TS
CP0410206 Compound Info	2-[4-[2-(4-methoxyphenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H26F3NO4S2	1
1	EC50 = 4.8 nM Bioactivity Info	TI LI LO TS
CP0035354 Compound Info	(R)-3-(4-(3-(4-ethyl-2-(pyridin-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	EC50 = 5 nM Bioactivity Info	TI LI LO TS
CP0074936 Compound Info	(R)-3-{4-[3-(4-ethyl-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C28H32O5	1
1	EC50 = 5 nM Bioactivity Info	TI LI LO TS
CP0415613 Compound Info	2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C30H23ClF4O3S	1
1	EC50 = 5.3 nM Bioactivity Info	TI LI LO TS
CP0527652 Compound Info	(3R)-6-[2-[[2-(4-chlorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C24H27ClN2O3	1
1	EC50 = 5.5 nM Bioactivity Info	TI LI LO TS
CP0471906 Compound Info	2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C31H23F7O3S	1
1	EC50 = 5.8 nM Bioactivity Info	TI LI LO TS
CP0035136 Compound Info	3-(4-(3-((5-chloro-3-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H25ClN2O4	1
1	EC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0035360 Compound Info	3-{4-[(R)-3-(5-ethyl-biphenyl-2-yloxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C28H32O4	1
1	EC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0112273 Compound Info	3-(2-ethyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C27H28F3NO4	1
1	EC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0136164 Compound Info	3-(2-methyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C26H26F3NO4	1
1	EC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0221700 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-ethyl-phenyl}-propionic acid Show/Hide	C27H29ClO5	1
1	EC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0432345 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-4-phenylbutyl]sulfanylphenoxy]acetic acid Show/Hide	C30H28F3NO3S2	1
1	EC50 = 6.1 nM Bioactivity Info	TI LI LO TS
CP0539237 Compound Info	2-[2-methyl-4-[(1S)-2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C30H25F3O3S	1
1	EC50 = 6.1 nM Bioactivity Info	TI LI LO TS
CP0437343 Compound Info	2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)butanoic acid Show/Hide	C23H22F3NO3SSe	1
1	EC50 = 6.2 nM Bioactivity Info	TI LI LO TS
CP0415611 Compound Info	2-[4-[2-(2,6-difluorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H21F5O3S	1
1	EC50 = 6.3 nM Bioactivity Info	TI LI LO TS
CP0142828 Compound Info	2-[4-[butyl-[2-methyl-3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32F3NO5S	1
1	EC50 = 6.31 nM Bioactivity Info	TI LI LO TS
CP0410224 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C28H21F6NO3S2	1
1	EC50 = 6.7 nM Bioactivity Info	TI LI LO TS
CP0396626 Compound Info	2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H21ClF4O3S	1
1	EC50 = 6.9 nM Bioactivity Info	TI LI LO TS
CP0215238 Compound Info	(R)-3-(4-(3-(1-(5-chloro-3-methylbenzo[b]thiophene-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid Show/Hide	C29H27ClFNO4S	1
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0035358 Compound Info	3-(2-ethyl-4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C28H33NO4	1
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0221733 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C29H32O5	1
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0437345 Compound Info	2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)butanoic acid Show/Hide	C23H21F4NO3SSe	1
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0415614 Compound Info	2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-phenylethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H25FO3S	1
1	EC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0452176 Compound Info	(E)-6-[2-[[[3-chloro-4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C26H26ClNO5	1
1	EC50 = 7.4 nM Bioactivity Info	TI LI LO TS
CP0254225 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C26H27ClO5	1
1	EC50 = 8 nM Bioactivity Info	TI LI LO TS
CP0416592 Compound Info	(3R)-6-[2-[[2-(4-chlorophenyl)-5-(trifluoromethyl)imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C24H24ClF3N2O3	1
1	EC50 = 8 nM Bioactivity Info	TI LI LO TS
CP0410219 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(2,3,4,5,6-pentafluorophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C28H19F8NO3S2	1
1	EC50 = 8.1 nM Bioactivity Info	TI LI LO TS
CP0421003 Compound Info	(3R)-6-[2-[[2-(4-cyanophenyl)-5-(trifluoromethyl)imidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C25H24F3N3O3	1
1	EC50 = 8.2 nM Bioactivity Info	TI LI LO TS
CP0557787 Compound Info	(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methyltriazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C27H27N3O4	1
1	EC50 = 8.4 nM Bioactivity Info	TI LI LO TS
CP0437344 Compound Info	2-(4-((2-(3-fluoro-4-(trifluoromethyl)phenyl)-4-methylthiazol-5-yl)methylselanyl)-2-methylphenoxy)propanoic acid Show/Hide	C22H19F4NO3SSe	1
1	EC50 = 8.5 nM Bioactivity Info	TI LI LO TS
CP0264567 Compound Info	3-(4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	EC50 = 9 nM Bioactivity Info	TI LI LO TS
CP0396629 Compound Info	2-[4-[2-(2,6-difluorophenyl)-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C30H23F5O3S	1
1	EC50 = 9.1 nM Bioactivity Info	TI LI LO TS
CP0420883 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-[4-(trifluoromethyl)phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C29H23F6NO3S2	1
1	EC50 = 9.4 nM Bioactivity Info	TI LI LO TS
CP0415618 Compound Info	2-[4-[2-(2,6-dichlorophenyl)-1-[4-(3,4,5-trifluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H21Cl2F3O3S	1
1	EC50 = 9.5 nM Bioactivity Info	TI LI LO TS
CP0549453 Compound Info	(E)-6-[2-[[4-[4-(furan-2-yl)phenyl]-2-methyl-1,3-thiazol-5-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H27NO4S	1
1	EC50 = 9.5 nM Bioactivity Info	TI LI LO TS
CP0296472 Compound Info	2-[4-[butyl-[2-chloro-3-(4-chlorophenyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H29Cl2NO5S	1
1	EC50 = 10 nM Bioactivity Info	TI LI LO TS
CP0492681 Compound Info	2-[4-[2-[2-fluoro-6-(trifluoromethyl)phenyl]-1-(4-phenylphenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C30H24F4O3S	1
1	EC50 = 10 nM Bioactivity Info	TI LI LO TS
CP0381218 Compound Info	2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methylselanyl)phenoxy)propanoic acid Show/Hide	C22H20F3NO3SSe	1
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0459249 Compound Info	2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]-5-thiazolyl]ethyl]-5-methyl-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C27H27F3N2O4S	1
1	EC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0420998 Compound Info	(E)-4-methyl-6-[2-[[4-methyl-2-[4-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]phenoxy]hex-4-enoic acid Show/Hide	C25H25F3N2O3	1
1	EC50 = 11.2 nM Bioactivity Info	TI LI LO TS
CP0410222 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-6-phenylhexyl]sulfanylphenoxy]acetic acid Show/Hide	C32H32F3NO3S2	1
1	EC50 = 11.4 nM Bioactivity Info	TI LI LO TS
CP0396627 Compound Info	2-[2-methyl-4-[1-[4-[3-(trifluoromethyl)phenyl]phenyl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C30H22F6O3S	1
1	EC50 = 12 nM Bioactivity Info	TI LI LO TS
CP0206813 Compound Info	(2R)-2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 12.59 nM Bioactivity Info	TI LI LO TS
CP0527649 Compound Info	(3R)-6-[2-[[2-[4-(difluoromethoxy)phenyl]-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C25H28F2N2O4	1
1	EC50 = 13.5 nM Bioactivity Info	TI LI LO TS
CP0035355 Compound Info	3-(4-((R)-3-(4-ethyl-2-(pyridin-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	EC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0452177 Compound Info	(E)-6-[2-[[[3-fluoro-4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C26H26FNO5	1
1	EC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0281362 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2-cyclohexylphenoxy]propanoic acid Show/Hide	C32H38ClNO5S	1
1	EC50 = 15.85 nM Bioactivity Info	TI LI LO TS
CP0416105 Compound Info	2-[4-[2-(2,5-difluorophenyl)-1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C28H22F5NO3S2	1
1	EC50 = 16.7 nM Bioactivity Info	TI LI LO TS
CP0673789 Compound Info	2-(4-(2-chloro-4-((4-(trifluoromethyl)phenoxy)methyl)phenylthio)-5,6,7,8-tetrahydronaphthalen-1-yloxy)acetic acid Show/Hide	C26H22ClF3O4S	1
1	EC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0415617 Compound Info	2-[2-methyl-4-[2-phenyl-1-[4-[3-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]acetic acid Show/Hide	C30H25F3O3S	1
1	EC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0377839 Compound Info	2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid Show/Hide	C31H28F9NO4	1
1	EC50 = 19 nM Bioactivity Info	TI LI LO TS
CP0452175 Compound Info	(E)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]-4-methylphenoxy]-4-methylhex-4-enoic acid Show/Hide	C27H29NO5	1
1	EC50 = 19.8 nM Bioactivity Info	TI LI LO TS
CP0142785 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methoxyphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO6S	1
1	EC50 = 19.95 nM Bioactivity Info	TI LI LO TS
CP0461586 Compound Info	2-methyl-2-[4-(2-{4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}ethyl)phenoxy]propanoic acid Show/Hide	C23H22F3NO3S	1
1	EC50 = 20 nM Bioactivity Info	TI LI LO TS
CP0527651 Compound Info	(3R)-3-methyl-6-[2-[[5-methyl-2-(4-methylphenyl)imidazol-1-yl]methyl]phenoxy]hexanoic acid Show/Hide	C25H30N2O3	1
1	EC50 = 20 nM Bioactivity Info	TI LI LO TS
CP0502910 Compound Info	2-[3-[2-[4-Isopropyl-2-[4-(trifluoromethyl)phenyl]-5-thiazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C26H25F3N2O4S	1
1	EC50 = 21 nM Bioactivity Info	TI LI LO TS
CP0216421 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23F4NO5	1
1	EC50 = 22 nM Bioactivity Info	TI LI LO TS
CP0035191 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO4S	1
1	EC50 = 22 nM Bioactivity Info	TI LI LO TS
CP0051320 Compound Info	3-(4-((R)-3-(4-chloro-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H26ClNO4	1
1	EC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0035353 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO4S	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0166832 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-pentyloxy]-2-methyl-phenyl}-propionic acid Show/Hide	C30H34O5	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0376052 Compound Info	2-(3-(2-(2-(2,4-dichlorophenyl)-5-isopropyloxazol-4-yl)ethyl)-5-methylbenzo[d]isoxazol-6-yloxy)acetic acid Show/Hide	C24H22Cl2N2O5	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0404373 Compound Info	2-[4-[2-(2-chloro-6-fluorophenyl)-1-[4-(4-fluorophenyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H23ClF2O3S	1
1	EC50 = 25 nM Bioactivity Info	TI LI LO TS
CP0266172 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 25.12 nM Bioactivity Info	TI LI LO TS
CP0415619 Compound Info	2-[4-[2-(2-chloro-6-fluorophenyl)-1-(4-phenylphenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H24ClFO3S	1
1	EC50 = 26 nM Bioactivity Info	TI LI LO TS
CP0524605 Compound Info	(E)-4-methyl-6-[2-[[2-methyl-4-(2-methyl-1-benzofuran-5-yl)-1,3-thiazol-5-yl]methyl]phenoxy]hex-4-enoic acid Show/Hide	C27H27NO4S	1
1	EC50 = 29.7 nM Bioactivity Info	TI LI LO TS
CP0136124 Compound Info	2-(4-(3-((2-methoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H26F3NO6	1
1	EC50 = 30 nM Bioactivity Info	TI LI LO TS
CP0248504 Compound Info	2-[4-[butyl-[2-methyl-3-(4-methylphenyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H35NO5S	1
1	EC50 = 31.62 nM Bioactivity Info	TI LI LO TS
CP0035141 Compound Info	3-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenyl)propanoic acid Show/Hide	C26H24F3NO4	1
1	EC50 = 33 nM Bioactivity Info	TI LI LO TS
CP0057749 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-fluoro-phenyl}-propionic acid Show/Hide	C25H24ClFO5	1
1	EC50 = 34 nM Bioactivity Info	TI LI LO TS
CP0136122 Compound Info	2-(4-(3-((2-bromo-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23BrF3NO5	1
1	EC50 = 36 nM Bioactivity Info	TI LI LO TS
CP0062441 Compound Info	(E)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C26H27NO5	2
1	EC50 = 37 nM Bioactivity Info	TI LI LO TS
2	EC50 = 56 nM Bioactivity Info	TI LI LO TS
CP0216422 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C27H26F3NO5	1
1	EC50 = 38 nM Bioactivity Info	TI LI LO TS
CP0549063 Compound Info	2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-[2-fluoro-6-(trifluoromethyl)phenyl]ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C30H23F5O3S	1
1	EC50 = 38 nM Bioactivity Info	TI LI LO TS
CP0416104 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-5-phenylpentyl]sulfanylphenoxy]acetic acid Show/Hide	C31H30F3NO3S2	1
1	EC50 = 38.8 nM Bioactivity Info	TI LI LO TS
CP0549452 Compound Info	(3R)-6-[2-[[2-(4-fluorophenyl)-5-methylimidazol-1-yl]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C24H27FN2O3	1
1	EC50 = 39 nM Bioactivity Info	TI LI LO TS
CP0212514 Compound Info	2-[4-[butyl-[3-(4-methoxyphenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H35NO6S	1
1	EC50 = 39.81 nM Bioactivity Info	TI LI LO TS
CP0281363 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-4-fluorophenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H29ClFNO5S	1
1	EC50 = 39.81 nM Bioactivity Info	TI LI LO TS
CP0341774 Compound Info	2-[4-[butyl-[2-methyl-3-[4-(trifluoromethoxy)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32F3NO6S	1
1	EC50 = 39.81 nM Bioactivity Info	TI LI LO TS
CP0145989 Compound Info	2-[(1S)-5-{3-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)phenoxy]propoxy}-2,3-dihydro-1H-inden-1-yl]acetic acid Show/Hide	C27H29NO4S	1
1	EC50 = 40 nM Bioactivity Info	TI LI LO TS
CP0415530 Compound Info	(E)-6-[4-fluoro-2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C26H26FNO5	1
1	EC50 = 40 nM Bioactivity Info	TI LI LO TS
CP0035359 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiophen-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O4S	1
1	EC50 = 41 nM Bioactivity Info	TI LI LO TS
CP0051319 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiophen-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O4S	1
1	EC50 = 42 nM Bioactivity Info	TI LI LO TS
CP0280556 Compound Info	alkynyl ether, 20 Show/Hide	C30H27F3O5S	1
1	EC50 = 43 nM Bioactivity Info	TI LI LO TS
CP0136386 Compound Info	alkynyl ether, 21 Show/Hide	C31H29F3O5S	1
1	EC50 = 44 nM Bioactivity Info	TI LI LO TS
CP0082061 Compound Info	2-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-phenoxy}-2-methyl-propionic acid Show/Hide	C29H32O6	1
1	EC50 = 45 nM Bioactivity Info	TI LI LO TS
CP0221348 Compound Info	3-(4-(3-((5-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	EC50 = 47 nM Bioactivity Info	TI LI LO TS
CP0053319 Compound Info	2-(4-(3-(2-benzoyl-4-ethylphenoxy)propoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C28H30O6	1
1	EC50 = 47 nM Bioactivity Info	TI LI LO TS
CP0412452 Compound Info	US10188627, Comparator Cmpd. 1 Show/Hide	C25H27NO5	1
1	EC50 = 47 nM Bioactivity Info	TI LI LO TS
CP0296984 Compound Info	2-(4-(3-fluoro-5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H22F5NO5	1
1	EC50 = 48 nM Bioactivity Info	TI LI LO TS
CP0035146 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethoxy)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C27H26F3NO6	1
1	EC50 = 50 nM Bioactivity Info	TI LI LO TS
CP0274499 Compound Info	3-(4-((R)-3-(4-ethyl-2-(oxazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO5	1
1	EC50 = 50 nM Bioactivity Info	TI LI LO TS
CP0292417 Compound Info	alkynyl ether, 19 Show/Hide	C29H25F3O5S	1
1	EC50 = 52 nM Bioactivity Info	TI LI LO TS
CP0274904 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-hexyloxy]-2-methyl-phenyl}-propionic acid Show/Hide	C31H36O5	1
1	EC50 = 52 nM Bioactivity Info	TI LI LO TS
CP0322303 Compound Info	alkynyl ether, 10 Show/Hide	C27H23F3O5S	1
1	EC50 = 54 nM Bioactivity Info	TI LI LO TS
CP0455776 Compound Info	2-[2-methyl-4-[1-[6-[4-(trifluoromethyl)phenyl]pyridin-3-yl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C29H21F6NO3S	1
1	EC50 = 56 nM Bioactivity Info	TI LI LO TS
CP0410223 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-8-phenyloctyl]sulfanylphenoxy]acetic acid Show/Hide	C34H36F3NO3S2	1
1	EC50 = 57.2 nM Bioactivity Info	TI LI LO TS
CP0035149 Compound Info	2-(4-(3-((2-chloro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23ClF3NO5	1
1	EC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0261714 Compound Info	3-(4-(3-((5,6-dichloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H22Cl2N2O4	1
1	EC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0444890 Compound Info	(E)-6-[2-[[3-[4-(furan-2-yl)phenyl]-5-methylimidazol-4-yl]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C28H28N2O4	1
1	EC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0410205 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-(4-nitrophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C28H23F3N2O5S2	1
1	EC50 = 60 nM Bioactivity Info	TI LI LO TS
CP0341227 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dichlorophenoxy]propanoic acid Show/Hide	C26H26Cl3NO5S	1
1	EC50 = 63.1 nM Bioactivity Info	TI LI LO TS
CP0415615 Compound Info	2-[4-[1-[4-(4-fluorophenyl)phenyl]-2-(3,4,5-trifluorophenyl)ethyl]sulfanyl-2-methylphenoxy]acetic acid Show/Hide	C29H22F4O3S	1
1	EC50 = 65 nM Bioactivity Info	TI LI LO TS
CP0131907 Compound Info	3-{4-[3-(2-benzyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C29H34O4	1
1	EC50 = 70 nM Bioactivity Info	TI LI LO TS
CP0221734 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-trifluoromethyl-phenyl}-propionic acid Show/Hide	C26H24ClF3O5	1
1	EC50 = 73 nM Bioactivity Info	TI LI LO TS
CP0240934 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-propylsulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H30ClNO5S	1
1	EC50 = 79.43 nM Bioactivity Info	TI LI LO TS
CP0035138 Compound Info	3-(4-(3-((6-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	EC50 = 80 nM Bioactivity Info	TI LI LO TS
CP0261716 Compound Info	2-(4-(3-((2-ethyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C28H28F3NO5	1
1	EC50 = 81 nM Bioactivity Info	TI LI LO TS
CP0424426 Compound Info	(1S,2R)-2-[3-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]propyl]cyclopropane-1-carboxylic acid Show/Hide	C26H27NO5	2
1	EC50 = 82.5 nM Bioactivity Info	TI LI LO TS
2	EC50 = 330 nM Bioactivity Info	TI LI LO TS
CP0035142 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	EC50 = 86 nM Bioactivity Info	TI LI LO TS
CP0455775 Compound Info	2-[2-methyl-4-[1-(4-phenylphenyl)-2-(3,4,5-trifluorophenyl)ethyl]sulfanylphenoxy]acetic acid Show/Hide	C29H23F3O3S	1
1	EC50 = 86 nM Bioactivity Info	TI LI LO TS
CP0051472 Compound Info	3-(4-(3-((5-chloro-1-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H25ClN2O4	1
1	EC50 = 87 nM Bioactivity Info	TI LI LO TS
CP0374481 Compound Info	2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(3,4-dichloro-phenoxy)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid Show/Hide	C30H27Cl2F6NO5	1
1	EC50 = 93 nM Bioactivity Info	TI LI LO TS
CP0035196 Compound Info	3-(4-(3-((5-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23BrN2O4	1
1	EC50 = 93 nM Bioactivity Info	TI LI LO TS
CP0075559 Compound Info	2-methyl-2-(2-methyl-4-(3-((4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C26H24F3NO5	1
1	EC50 = 95 nM Bioactivity Info	TI LI LO TS
CP0035143 Compound Info	2-(4-(5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-2-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	EC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0204433 Compound Info	3-(4-(2-(5-(3-chlorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C22H23ClN2O5	1
1	EC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0171813 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-5-(trifluoromethyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	EC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0459248 Compound Info	2-[3-[2-[2-(2,4-Dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H24Cl2N2O5	1
1	EC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0075561 Compound Info	2-(4-(4-fluoro-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H22F5NO5	1
1	EC50 = 119 nM Bioactivity Info	TI LI LO TS
CP0142827 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-4-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 125.89 nM Bioactivity Info	TI LI LO TS
CP0169971 Compound Info	2-[4-[butyl-[3-(3,4-dichlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H31Cl2NO5S	1
1	EC50 = 125.89 nM Bioactivity Info	TI LI LO TS
CP0219135 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]butanoic acid Show/Hide	C29H34ClNO5S	1
1	EC50 = 125.89 nM Bioactivity Info	TI LI LO TS
CP0420884 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-11-phenylundecyl]sulfanylphenoxy]acetic acid Show/Hide	C37H42F3NO3S2	1
1	EC50 = 132 nM Bioactivity Info	TI LI LO TS
CP0248505 Compound Info	2-[2-methyl-4-[3-methylbutyl-[3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]phenoxy]acetic acid Show/Hide	C27H28F3NO5S	1
1	EC50 = 158.49 nM Bioactivity Info	TI LI LO TS
CP0468295 Compound Info	4-Isocyanato-benzoic acid 2-((2,4-bis-trifluoromethyl-benzyl)-{3-[3-(1-carboxy-1-methyl-ethoxy)-phenyl]-propyl}-amino)-ethyl ester Show/Hide	C32H30F6N2O6	1
1	EC50 = 160 nM Bioactivity Info	TI LI LO TS
CP0286632 Compound Info	3-(4-((5-(3,5-difluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C21H20F2N2O5	1
1	EC50 = 160 nM Bioactivity Info	TI LI LO TS
CP0086935 Compound Info	alkynyl ether, 23 Show/Hide	C30H27F3O6S	1
1	EC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0035108 Compound Info	2-(4-(3-((4-chloro-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H26ClNO5	1
1	EC50 = 254 nM Bioactivity Info	TI LI LO TS
CP0145397 Compound Info	3-(4-((R)-3-(4-ethyl-2-(oxazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO5	1
1	EC50 = 274 nM Bioactivity Info	TI LI LO TS
CP0210104 Compound Info	2-(4-(3-((2,4-dimethylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H29NO5	1
1	EC50 = 286 nM Bioactivity Info	TI LI LO TS
CP0169970 Compound Info	(2S)-2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 316.23 nM Bioactivity Info	TI LI LO TS
CP0206814 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-3-chloro-2-methoxyphenoxy]propanoic acid Show/Hide	C27H29Cl2NO6S	1
1	EC50 = 316.23 nM Bioactivity Info	TI LI LO TS
CP0341782 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-difluorophenoxy]propanoic acid Show/Hide	C26H26ClF2NO5S	1
1	EC50 = 316.23 nM Bioactivity Info	TI LI LO TS
CP0204434 Compound Info	3-(4-((5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C23H20F6N2O5	1
1	EC50 = 320 nM Bioactivity Info	TI LI LO TS
CP0274937 Compound Info	(S)-3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]2-methyl-phenyl}propionic acid Show/Hide	C29H32O5	1
1	EC50 = 339 nM Bioactivity Info	TI LI LO TS
CP0167310 Compound Info	alkynyl ether, 26 Show/Hide	C31H29F3O6S	1
1	EC50 = 340 nM Bioactivity Info	TI LI LO TS
CP0036483 Compound Info	alkynyl ether, 31 Show/Hide	C30H29ClO5S	1
1	EC50 = 350 nM Bioactivity Info	TI LI LO TS
CP0086940 Compound Info	alkynyl ether, 32 Show/Hide	C31H31ClO5S	1
1	EC50 = 370 nM Bioactivity Info	TI LI LO TS
CP0035145 Compound Info	2-(4-(3-((4-methoxy-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H29NO6	1
1	EC50 = 376 nM Bioactivity Info	TI LI LO TS
CP0219137 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-pentylsulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H34ClNO5S	1
1	EC50 = 398.11 nM Bioactivity Info	TI LI LO TS
CP0291942 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-3-chloro-2-fluorophenoxy]propanoic acid Show/Hide	C26H26Cl2FNO5S	1
1	EC50 = 398.11 nM Bioactivity Info	TI LI LO TS
CP0145396 Compound Info	3-(4-((R)-3-(4-ethyl-2-(furan-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O5	1
1	EC50 = 399 nM Bioactivity Info	TI LI LO TS
CP0035147 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-phenoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C32H28F3NO6	1
1	EC50 = 409 nM Bioactivity Info	TI LI LO TS
CP0412471 Compound Info	(3R)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C26H29NO5	1
1	EC50 = 417 nM Bioactivity Info	TI LI LO TS
CP0086938 Compound Info	alkynyl ether, 29 Show/Hide	C31H29F3O5S	1
1	EC50 = 420 nM Bioactivity Info	TI LI LO TS
CP0463084 Compound Info	2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-[2-(4-trifluoromethyl-phenyl)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid Show/Hide	C33H32F3N3O5	1
1	EC50 = 430 nM Bioactivity Info	TI LI LO TS
CP0036481 Compound Info	alkynyl ether, 27 Show/Hide	C32H31F3O6S	1
1	EC50 = 470 nM Bioactivity Info	TI LI LO TS
CP0495380 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-naphthalen-1-ylethyl]sulfanylphenoxy]acetic acid Show/Hide	C32H26F3NO3S2	1
1	EC50 = 490.1 nM Bioactivity Info	TI LI LO TS
CP0114160 Compound Info	3-(4-((5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C21H21ClN2O5	1
1	EC50 = 500 nM Bioactivity Info	TI LI LO TS
CP0233674 Compound Info	2-Isopropoxy-3-(4-{2-[5-(3-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-propionic acid Show/Hide	C23H23F3N2O5	1
1	EC50 = 500 nM Bioactivity Info	TI LI LO TS
CP0342886 Compound Info	2-Isopropoxy-3-{4-[5-(4-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid Show/Hide	C22H21F3N2O5	1
1	EC50 = 500 nM Bioactivity Info	TI LI LO TS
CP0142823 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2-fluoro-3-methoxyphenoxy]propanoic acid Show/Hide	C27H29ClFNO6S	1
1	EC50 = 501.19 nM Bioactivity Info	TI LI LO TS
CP0142825 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(cyclobutylmethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32ClNO5S	1
1	EC50 = 501.19 nM Bioactivity Info	TI LI LO TS
CP0206836 Compound Info	2-[4-[butyl-[3-(3-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 501.19 nM Bioactivity Info	TI LI LO TS
CP0310287 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(2-methoxyethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H30ClNO6S	1
1	EC50 = 501.19 nM Bioactivity Info	TI LI LO TS
CP0447760 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2,2-diphenylethyl]sulfanylphenoxy]acetic acid Show/Hide	C34H28F3NO3S2	1
1	EC50 = 523 nM Bioactivity Info	TI LI LO TS
CP0261715 Compound Info	3-(4-(3-((7-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23BrN2O4	1
1	EC50 = 527 nM Bioactivity Info	TI LI LO TS
CP0424429 Compound Info	6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C26H29NO5	1
1	EC50 = 566 nM Bioactivity Info	TI LI LO TS
CP0408488 Compound Info	6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy)-2-methylhexanoic acid Show/Hide	C26H29NO5	1
1	EC50 = 640 nM Bioactivity Info	TI LI LO TS
CP0847204 Compound Info	2-methyl-2-[4-{[(5-methyl-2-[4-trifluoromethylphenyl]-thiazol-4-ylcarbonyl)amino]methyl}phenoxy]propionic acid Show/Hide	C17H20N2O4S	1
1	EC50 = 660 nM Bioactivity Info	TI LI LO TS
CP0086937 Compound Info	alkynyl ether, 28 Show/Hide	C34H28F3NO5S	1
1	EC50 = 680 nM Bioactivity Info	TI LI LO TS
CP0459247 Compound Info	2-[3-[2-[2-(4-Butylphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C29H34N2O5	1
1	EC50 = 700 nM Bioactivity Info	TI LI LO TS
CP0404578 Compound Info	2-(4-{2-[1-Cycloheptyl-3-(2,4-difluoro-phenyl)-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid Show/Hide	C26H32F2N2O4	1
1	EC50 = 790 nM Bioactivity Info	TI LI LO TS
CP0114159 Compound Info	3-(4-((5-(4-bromophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C21H21BrN2O5	1
1	EC50 = 790 nM Bioactivity Info	TI LI LO TS
CP0206815 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(cyclopropylmethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H30ClNO5S	1
1	EC50 = 794.33 nM Bioactivity Info	TI LI LO TS
CP0295054 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 794.33 nM Bioactivity Info	TI LI LO TS
CP0445956 Compound Info	2-methyl-2-phenoxypropanoic acid, 25j Show/Hide	C23H21F3N2O4S	1
1	EC50 = 808 nM Bioactivity Info	TI LI LO TS
CP0201561 Compound Info	alkynyl ether, 36 Show/Hide	C29H34O5S	1
1	EC50 = 900 nM Bioactivity Info	TI LI LO TS
CP0505001 Compound Info	2-[3-[2-[2-(2-Hydroxyphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H26N2O6	1
1	EC50 = 900 nM Bioactivity Info	TI LI LO TS
CP0389163 Compound Info	6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhexanoic acid Show/Hide	C26H29NO5	2
1	EC50 = 990 nM Bioactivity Info	TI LI LO TS
2	EC50 = 998 nM Bioactivity Info	TI LI LO TS
CP0377750 Compound Info	2-(3-{3-[(3,4-Bis-trifluoromethyl-benzoyl)-(2-cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-amino]-propyl}-phenoxy)-2-methyl-propionic acid Show/Hide	C33H29F6N3O5	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0448498 Compound Info	2-[3-(3-{(2-Cyclopropyl-3-[1,2,4]oxadiazol-3-yl-phenyl)-[2-(3,4-dichloro-phenoxy)-acetyl]-amino}-propyl)-phenoxy]-2-methyl-propionic acid Show/Hide	C32H31Cl2N3O6	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0296470 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2-(trifluoromethoxy)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO6S	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0380840 Compound Info	2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(2-methoxy-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C30H42N2O4S	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0086939 Compound Info	alkynyl ether, 30 Show/Hide	C31H29F3O5S	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0194611 Compound Info	phenoxyacetic acid-ether, 12 Show/Hide	C26H22F3NO5S	1
1	EC50 = 1100 nM Bioactivity Info	TI LI LO TS
CP0086936 Compound Info	alkynyl ether, 25 Show/Hide	C31H29F3O6S	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0145069 Compound Info	alkynyl ether, 33 Show/Hide	C30H28F3NO5S	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0441380 Compound Info	2-[3-[2-[2-(4-tert-Butylphenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C29H34N2O5	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0142780 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2,4-difluorophenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H28ClF2NO5S	1
1	EC50 = 1258.93 nM Bioactivity Info	TI LI LO TS
CP0035109 Compound Info	3-(4-(3-((4-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	EC50 = 1300 nM Bioactivity Info	TI LI LO TS
CP0376050 Compound Info	2-[3-[2-[2-(2-Chlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H25ClN2O5	1
1	EC50 = 1300 nM Bioactivity Info	TI LI LO TS
CP0424428 Compound Info	2-[4-[[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]methyl]phenyl]acetic acid Show/Hide	C28H25NO5	1
1	EC50 = 1316 nM Bioactivity Info	TI LI LO TS
CP0170396 Compound Info	2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)amino}ethyl)phenyl]sulfanyl}-2-methylpropanoic acid Show/Hide	C26H34F2N2O3S	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0167306 Compound Info	alkynyl ether, 22 Show/Hide	C32H31F3O6S	1
1	EC50 = 1400 nM Bioactivity Info	TI LI LO TS
CP0208857 Compound Info	alkynyl ether, 37 Show/Hide	C28H32O5S	1
1	EC50 = 1500 nM Bioactivity Info	TI LI LO TS
CP0071095 Compound Info	2-Isopropoxy-3-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid Show/Hide	C22H24N2O5	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0231601 Compound Info	2-Isopropoxy-3-[4-(5-o-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid Show/Hide	C22H24N2O5	1
1	EC50 = 1600 nM Bioactivity Info	TI LI LO TS
CP0481942 Compound Info	(1R,2R)-2-[3-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]propyl]cyclopropane-1-carboxylic acid Show/Hide	C26H27NO5	1
1	EC50 = 1630 nM Bioactivity Info	TI LI LO TS
CP0276403 Compound Info	phenoxyacetic acid-ether, 11 Show/Hide	C27H27F3O6S	1
1	EC50 = 1700 nM Bioactivity Info	TI LI LO TS
CP0035144 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methylbenzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C26H27NO5	1
1	EC50 = 1878 nM Bioactivity Info	TI LI LO TS
CP0201564 Compound Info	phenoxyacetic acid-ether, 9 Show/Hide	C28H29F3O6S	1
1	EC50 = 1900 nM Bioactivity Info	TI LI LO TS
CP0266173 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(4,4,4-trifluorobutyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	EC50 = 1995.26 nM Bioactivity Info	TI LI LO TS
CP0281364 Compound Info	2-[4-[butyl-[3-(2-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	EC50 = 1995.26 nM Bioactivity Info	TI LI LO TS
CP0128464 Compound Info	alkynyl ether, 24 Show/Hide	C31H29F3O6S	1
1	EC50 = 2000 nM Bioactivity Info	TI LI LO TS
CP0482215 Compound Info	2-[3-[2-[2-(2-Chlorophenyl)-5-hexyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C28H31ClN2O5	1
1	EC50 = 2000 nM Bioactivity Info	TI LI LO TS
CP0039791 Compound Info	phenoxyacetic acid-ether, 13 Show/Hide	C29H26F3NO6S	1
1	EC50 = 2200 nM Bioactivity Info	TI LI LO TS
CP0231600 Compound Info	2-Isopropoxy-3-[4-(5-p-tolyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid Show/Hide	C22H24N2O5	1
1	EC50 = 2500 nM Bioactivity Info	TI LI LO TS
CP0233673 Compound Info	2-Isopropoxy-3-(4-{2-[5-(2-trifluoromethyl-phenyl)-[1,2,4]oxadiazol-3-yl]-ethoxy}-phenyl)-propionic acid Show/Hide	C23H23F3N2O5	1
1	EC50 = 2500 nM Bioactivity Info	TI LI LO TS
CP0268622 Compound Info	2-methyl-2-phenoxypropanoic acid, 25a Show/Hide	C23H21F3N2O4S	2
1	EC50 = 2600 nM Bioactivity Info	TI LI LO TS
2	EC50 = 2830 nM Bioactivity Info	TI LI LO TS
CP0075564 Compound Info	2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H23F6NO5	1
1	EC50 = 2870 nM Bioactivity Info	TI LI LO TS
CP0086886 Compound Info	phenoxyacetic acid-ether, 14 Show/Hide	C30H26F3NO5S	1
1	EC50 = 2900 nM Bioactivity Info	TI LI LO TS
CP0077439 Compound Info	(R)-2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acid Show/Hide	C28H27NO5	1
1	EC50 = 3014 nM Bioactivity Info	TI LI LO TS
CP0374670 Compound Info	2-(4-{2-[3-(4-Fluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-propionic acid Show/Hide	C26H35FN2O4	1
1	EC50 = 3100 nM Bioactivity Info	TI LI LO TS
CP0086881 Compound Info	alkynyl ether, 34 Show/Hide	C31H30F3NO4S	1
1	EC50 = 3100 nM Bioactivity Info	TI LI LO TS
CP0160737 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-4-fluoro-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H31ClFNO5S	1
1	EC50 = 3162.28 nM Bioactivity Info	TI LI LO TS
CP0043337 Compound Info	(2S)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-pyrrol-1-ylpropanoic acid Show/Hide	C25H24N2O4	1
1	EC50 = 3800 nM Bioactivity Info	TI LI LO TS
CP0406324 Compound Info	3-(4-(2-(5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)ethoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C22H23FN2O5	1
1	EC50 = 4000 nM Bioactivity Info	TI LI LO TS
CP0460135 Compound Info	2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2,4-dimethoxy-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C35H38N2O5S	1
1	EC50 = 4000 nM Bioactivity Info	TI LI LO TS
CP0445955 Compound Info	2-methyl-2-(4-{[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)amino]methyl}phenoxy)propanoic acid Show/Hide	C23H23F3N2O3S	1
1	EC50 = 4050 nM Bioactivity Info	TI LI LO TS
CP0146580 Compound Info	phenoxyacetic acid-ether, 15 Show/Hide	C30H26F3NO5S	1
1	EC50 = 4100 nM Bioactivity Info	TI LI LO TS
CP0409204 Compound Info	2-methyl-2-phenoxypropanoic acid, 25c Show/Hide	C23H21F3N2O5S	1
1	EC50 = 4600 nM Bioactivity Info	TI LI LO TS
CP0401328 Compound Info	3-(4-((5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C25H30N2O5	1
1	EC50 = 5000 nM Bioactivity Info	TI LI LO TS
CP0381165 Compound Info	2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-cyclohexyl-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C33H40N2O3S	1
1	EC50 = 5000 nM Bioactivity Info	TI LI LO TS
CP0409332 Compound Info	2-[4-({[2-(4-chlorophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C22H21ClN2O4S	1
1	EC50 = 5400 nM Bioactivity Info	TI LI LO TS
CP0376049 Compound Info	2-[3-[2-[2-(2-Chlorophenyl)-5-propyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H25ClN2O5	1
1	EC50 = 5400 nM Bioactivity Info	TI LI LO TS
CP0023801 Compound Info	2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)ethyl)phenylthio)-2-methylpropanoic acid Show/Hide	C29H46N2O3S	1
1	EC50 = 6200 nM Bioactivity Info	TI LI LO TS
CP0409333 Compound Info	2-methyl-2-phenoxypropanoic acid, 34 Show/Hide	C23H21F3N2O4S	1
1	EC50 = 6260 nM Bioactivity Info	TI LI LO TS
CP0482211 Compound Info	2-[3-[2-[5-Ethyl-2-phenyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C24H24N2O5	1
1	EC50 = 6700 nM Bioactivity Info	TI LI LO TS
CP0086887 Compound Info	phenoxyacetic acid-ether, 16 Show/Hide	C29H29F3O6S	1
1	EC50 = 7100 nM Bioactivity Info	TI LI LO TS
CP0085230 Compound Info	3-(4-((5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C21H21FN2O5	1
1	EC50 = 7900 nM Bioactivity Info	TI LI LO TS
CP0114157 Compound Info	2-Isopropoxy-3-{4-[5-(4-isopropyl-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid Show/Hide	C24H28N2O5	1
1	EC50 = 7900 nM Bioactivity Info	TI LI LO TS
CP0114158 Compound Info	2-Isopropoxy-3-{4-[5-(4-trifluoromethoxy-phenyl)-[1,2,4]oxadiazol-3-ylmethoxy]-phenyl}-propionic acid Show/Hide	C22H21F3N2O6	1
1	EC50 = 7900 nM Bioactivity Info	TI LI LO TS
CP0367813 Compound Info	3-(4-((5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl)methoxy)phenyl)-2-isopropoxypropanoic acid Show/Hide	C21H21FN2O5	1
1	EC50 = 7900 nM Bioactivity Info	TI LI LO TS
CP0409327 Compound Info	2-methyl-2-[4-({[4-(trifluoromethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]formamido}methyl)phenoxy]propanoic acid Show/Hide	C23H18F6N2O4S	1
1	EC50 = 8240 nM Bioactivity Info	TI LI LO TS
CP0441423 Compound Info	2-[3-[2-[2-Phenyl-5-propyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H26N2O5	1
1	EC50 = 9800 nM Bioactivity Info	TI LI LO TS
CP0071096 Compound Info	2-Isopropoxy-3-[4-(5-phenyl-[1,2,4]oxadiazol-3-ylmethoxy)-phenyl]-propionic acid Show/Hide	C21H22N2O5	1
1	EC50 = 10000 nM Bioactivity Info	TI LI LO TS
CP0406631 Compound Info	2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2,4,5-trimethyl-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C36H40N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0409243 Compound Info	2-(4-{2-[3-(3-Cyano-phenyl)-1-(4-cyclohexyl-butyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C30H39N3O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0460136 Compound Info	2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(4-methyl-3-nitro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C30H41N3O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0465322 Compound Info	2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(3,5-dichloro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C33H32Cl2N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0515829 Compound Info	2-(4-{2-[1-(4-Cyclohexyl-butyl)-3-(3,5-dichloro-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C29H38Cl2N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0518415 Compound Info	2-(4-{2-[1-(2-Biphenyl-4-yl-ethyl)-3-(2-methoxy-5-methyl-phenyl)-ureido]-ethyl}-phenylsulfanyl)-2-methyl-propionic acid Show/Hide	C35H38N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0086888 Compound Info	phenoxyacetic acid-ether, 18 Show/Hide	C30H32F3NO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0208859 Compound Info	alkynyl ether, 35 Show/Hide	C29H34O6S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0275263 Compound Info	phenoxyacetic acid-ether, 17 Show/Hide	C30H32F3NO6S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0372105 Compound Info	2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C26H30N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0409324 Compound Info	2-[4-({[2-(4-aminophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C22H23N3O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0409325 Compound Info	2-methyl-2-phenoxypropanoic acid, 25l Show/Hide	C23H24N2O7S2	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0409326 Compound Info	2-[4-({[2-(4-methoxyphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C23H24N2O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0409331 Compound Info	2-[4-({[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C22H21FN2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0442419 Compound Info	2-methyl-2-[4-({[4-methyl-2-(4-nitrophenyl)-1,3-thiazol-5-yl]formamido}methyl)phenoxy]propanoic acid Show/Hide	C22H21N3O6S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0442420 Compound Info	2-[4-({[2-(4-hydroxyphenyl)-4-methyl-1,3-thiazol-5-yl]formamido}methyl)phenoxy]-2-methylpropanoic acid Show/Hide	C22H22N2O5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0442421 Compound Info	2-methyl-2-phenoxypropanoic acid, 27 Show/Hide	C24H23F3N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0453688 Compound Info	2-methyl-2-phenoxypropanoic acid, 37 Show/Hide	C24H23F3N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0503895 Compound Info	2-methyl-2-[4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-}amido)phenoxy]propanoic acid Show/Hide	C22H19F3N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0938856 Compound Info	2-methyl-2-[4-{[(4-methyl-2-phenylthiazol-5-ylcarbonyl)amino]-methyl}phenoxy]propionic acid Show/Hide	C21H20N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0083167 Compound Info	4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidazol)-1'-yl)methyl)-(1,1'-biphenyl)-2-carboxylic acid Show/Hide	C33H30N4O2	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0320788 Compound Info	4'-((2-methyl-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C33H30N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0371730 Compound Info	4'-((2,3-dimethyl-5-(3-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C34H32N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0429811 Compound Info	4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C34H32N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0429825 Compound Info	4'-((5-(benzylcarbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C32H28N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0430855 Compound Info	4'-((2-methyl-6-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C33H30N2O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0447683 Compound Info	4'-((6-(1-phenylpropylcarbamoyl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C34H33N3O3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0452274 Compound Info	4'-((3-(methylthio)-5-(2-phenylbutanamido)-2-propyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C36H36N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0492739 Compound Info	4'-((2-methyl-3-(methylthio)-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid Show/Hide	C34H32N2O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0206812 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]hexanoic acid Show/Hide	C31H38ClNO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0240988 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2,4,6-trimethylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C30H36ClNO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0291982 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]pentanoic acid Show/Hide	C30H36ClNO5S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0296471 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethoxyphenoxy]propanoic acid Show/Hide	C28H32ClNO7S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0005387 Compound Info	Avandamet Show/Hide	C18H19N3O3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0375119 Compound Info	2-[3-[2-[2-(2,6-Dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C25H24Cl2N2O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0390776 Compound Info	2-[3-[2-[5-Isopropyl-2-[2-(trifluoromethyl)phenyl]-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C26H25F3N2O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0482214 Compound Info	2-[3-[2-[5-tert-Butyl-2-(2-chlorophenyl)-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C26H27ClN2O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0687662 Compound Info	5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(4-trifluoromethyl-benzyl)-benzamide Show/Hide	C20H17F3N2O4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0389162 Compound Info	6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy)-2,2-dimethylhexanoic acid Show/Hide	C27H31NO5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0408487 Compound Info	(E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy)-3-methylhex-2-enoic acid Show/Hide	C26H27NO5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0408489 Compound Info	(3S)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-3-methylhexanoic acid Show/Hide	C26H29NO5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0482177 Compound Info	(E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy)-2-methylhex-2-enoic acid Show/Hide	C26H27NO5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0008406 Compound Info	(3S)-3-[4-[[5-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]thiophen-2-yl]methoxy]phenyl]hex-4-ynoic acid Show/Hide	C28H29NO4S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0010598 Compound Info	(3S)-3-[4-[[5-(spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylmethyl)thiophen-2-yl]methoxy]phenyl]hex-4-ynoic acid Show/Hide	C31H33NO3S	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0013323 Compound Info	(3S)-3-[4-[[4-(spiro[indene-1,4'-piperidine]-1'-ylmethyl)phenyl]methoxy]phenyl]hex-4-ynoic acid Show/Hide	C33H33NO3	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0450935 Compound Info	2-[4-[3-[4-[(3-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C31H35N3O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0450936 Compound Info	2-[4-[3-[4-[(4-chlorophenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C30H32ClN3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0450937 Compound Info	2-[4-[3-[1-[(4-ethenylphenyl)methyl]-4-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C32H35N3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0450938 Compound Info	2-[4-[3-[4-[(4-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C31H35N3O5	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0538367 Compound Info	2-[4-[3-[1,4-bis[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C31H35N3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0538368 Compound Info	2-methyl-2-[4-[3-[1-[(4-methylphenyl)methyl]-5-oxo-4-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-triazol-3-yl]propyl]phenoxy]propanoic acid Show/Hide	C33H39N3O7	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0551890 Compound Info	2-[4-[3-[4-benzyl-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C30H33N3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0568641 Compound Info	2-[4-[3-[4-[(4-fluorophenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acid Show/Hide	C30H32FN3O4	1
1	EC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0390775 Compound Info	2-[3-[2-[5-Methyl-2-phenyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yloxy]-2-methylpropionic acid Show/Hide	C23H22N2O5	1
1	EC50 = 14900 nM Bioactivity Info	TI LI LO TS
CP0015504 Compound Info	2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-2-methylpropanoic acid Show/Hide	C19H20ClNO4	2
1	EC50 = 20000 nM Bioactivity Info	TI LI LO TS
2	EC50 = 30000 nM Bioactivity Info	TI LI LO TS
CP0409330 Compound Info	2-methyl-2-phenoxypropanoic acid, 25i Show/Hide	C23H21F3N2O4S	1
1	EC50 > 25000 nM Bioactivity Info	TI LI LO TS
CP0441016 Compound Info	2-methyl-2-[6-(5-methyl-2-phenyl-1,3-oxazol-4-yl)hexoxy]propanoic acid Show/Hide	C20H27NO4	1
1	EC50 = 30000 nM Bioactivity Info	TI LI LO TS
CP0042877 Compound Info	2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic acid Show/Hide	C17H15ClO4	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0372747 Compound Info	(2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-yl)butyl)-1,3-dioxane-2-carboxylic acid Show/Hide	C21H27NO5	1
1	EC50 > 100000 nM Bioactivity Info	TI LI LO TS
CP0378531 Compound Info	(S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-4-yl)(methyl)amino)propoxy)-2,3-dihydro-1H-inden-1-yl)acetic acid Show/Hide	C28H33N3O3	1
1	IC50 = 30 nM Bioactivity Info	TI LI LO TS
CP0427747 Compound Info	(S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimidin-4-yl)(methyl)amino)propoxy)-2,3-dihydro-1H-inden-1-yl)acetic acid Show/Hide	C29H35N3O3	1
1	IC50 = 49 nM Bioactivity Info	TI LI LO TS
CP0427720 Compound Info	2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyridin-2-yloxy)propoxy)-2,3-dihydro-1H-inden-1-yl)acetic acid Show/Hide	C25H26N2O5S	1
1	IC50 = 56 nM Bioactivity Info	TI LI LO TS
CP0074619 Compound Info	4-bromo-2-fluoro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11BrF4N2O3S	1
1	IC50 = 79.43 nM Bioactivity Info	TI LI LO TS
CP0043623 Compound Info	4-chloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H12ClF3N2O3S	1
1	IC50 = 125.89 nM Bioactivity Info	TI LI LO TS
CP0149424 Compound Info	4-(2-methylpropyl)-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C19H21F3N2O3S	1
1	IC50 = 199.53 nM Bioactivity Info	TI LI LO TS
CP0290360 Compound Info	2,4-dichloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11Cl2F3N2O3S	1
1	IC50 = 199.53 nM Bioactivity Info	TI LI LO TS
CP0128531 Compound Info	4-chloro-3-methyl-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C16H14ClF3N2O3S	1
1	IC50 = 251.19 nM Bioactivity Info	TI LI LO TS
CP0214965 Compound Info	4-phenyl-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C21H17F3N2O3S	1
1	IC50 = 251.19 nM Bioactivity Info	TI LI LO TS
CP0239873 Compound Info	3-bromo-4-chloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11BrClF3N2O3S	1
1	IC50 = 251.19 nM Bioactivity Info	TI LI LO TS
CP0177179 Compound Info	methyl 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]thiophene-2-carboxylate Show/Hide	C19H18N2O5S2	1
1	IC50 = 316.23 nM Bioactivity Info	TI LI LO TS

Cell Line ID: CL000011 , CHO

Cell Line Info

Cell Line ID: CL000026 , CHO-K1

Cell Line Info

Cell Line ID: CL000109 , COS-1

Cell Line Info

Cell Line ID: CL000053 , COS-7

Cell Line Info

Cell Line ID: CL000025 , HEK-293T

Cell Line Info

Cell Line ID: CL000006 , HEK293

Cell Line Info

Cell Line ID: CL000017 , HeLa

Cell Line Info

Cell Line ID: CL000063 , Hep-G2

Cell Line Info

Cell Line ID: CL000148 , Huh-7

Cell Line Info

Biochemical Assays

Compound ID	Compound Name	Compound Formula
CP0039118 Compound Info	2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid Show/Hide	C21H18F3NO3S2	14
1	EC50 = 0.5 nM
2	EC50 = 1 nM
3	EC50 = 1.4 nM
4	EC50 = 6 nM
5	EC50 = 24 nM
6	EC50 = 700 nM
7	IC50 = 1 nM
8	IC50 = 2.6 nM
9	IC50 = 5.012 nM
10	Ki = 0.048 nM
11	Ki = 0.82 nM
12	Ki = 1 nM
13	Ki = 6.08 nM
14	Ki = 80 nM
CP0060839 Compound Info	2-[4-[[2-[3-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl]methylsulfanyl]-2-methylphenoxy]acetic acid Show/Hide	C21H17F4NO3S2	8
1	EC50 = 1 nM
2	EC50 = 2 nM
3	EC50 = 2.9 nM
4	EC50 = 4 nM
5	EC50 = 13 nM
6	EC50 = 67.11 nM
7	IC50 = 1 nM
8	Kd = 0.4 nM
CP0564413 Compound Info	2-[4-[2-[2-(3-methylphenoxy)ethylamino]-2-oxoethoxy]phenyl]acetic acid Show/Hide	C19H21NO5	1
1	EC50 = 4 nM
CP0064381 Compound Info	2-(4-((5-(4-Biphenyl)-4-(pyridin-3-yl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C30H24N2O5	1
1	EC50 = 6 nM
CP0261946 Compound Info	2-[2,6-dimethyl-4-[[5-oxo-4-[4-(trifluoromethoxy)phenyl]-1,2,4-triazol-1-yl]methyl]phenoxy]-2-methylpropanoic acid Show/Hide	C22H22F3N3O5	1
1	EC50 = 8.4 nM
CP0039614 Compound Info	2-(4-((4-(4-Isopropoxyphenyl)-5-(4-biphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C34H31NO5S	1
1	EC50 = 10 nM
CP0043946 Compound Info	2-[2-methyl-4-[[4-(4-propan-2-yloxyphenyl)-5-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]methoxy]phenoxy]acetic acid Show/Hide	C29H26F3NO6S	1
1	EC50 = 10 nM
CP0043958 Compound Info	2-(4-((4-(6-Methoxypyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C26H21F3N2O7	1
1	EC50 = 10 nM
CP0221663 Compound Info	2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-propylphenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C27H27N3O6	1
1	EC50 = 10 nM
CP0076831 Compound Info	Elafibranor Show/Hide	C22H24O4S	3
1	EC50 = 10 nM
2	EC50 = 115 nM
3	EC50 = 842.9 nM
CP0096783 Compound Info	2-(3-chloro-4-(3-(3-ethyl-7-propylbenzo[d]isoxazol-6-yloxy)propylthio)phenyl)acetic acid Show/Hide	C23H26ClNO4S	2
1	EC50 = 11 nM
2	IC50 = 4 nM
CP0221664 Compound Info	2-(4-((4-(6-Isopropoxypyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C28H25F3N2O6S	1
1	EC50 = 12 nM
CP0244640 Compound Info	2-[4-[[4-(6-methoxypyridin-3-yl)-5-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]methoxy]-2-methylphenoxy]acetic acid Show/Hide	C26H21F3N2O6S	1
1	EC50 = 12 nM
CP0287050 Compound Info	2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C31H28F3NO7	1
1	EC50 = 12 nM
CP0043959 Compound Info	2-(4-((4-(4-Isopropoxyphenyl)-5-(4-propylphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C31H33NO5S	1
1	EC50 = 13 nM
CP0345351 Compound Info	2-(4-((4-(4-Isopropoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C29H26F3NO7	1
1	EC50 = 13 nM
CP0134379 Compound Info	2-[2-methyl-4-[1-[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-phenylethyl]sulfanylphenoxy]acetic acid Show/Hide	C28H24F3NO3S2	1
1	EC50 = 13 nM
CP0057167 Compound Info	2-[2-methyl-4-[[4-(6-propan-2-yloxypyridin-3-yl)-5-[4-(trifluoromethoxy)phenyl]-1,3-oxazol-2-yl]methoxy]phenoxy]acetic acid Show/Hide	C28H25F3N2O7	1
1	EC50 = 14 nM
CP0237930 Compound Info	2-(4-((4-(4-Morpholinophenyl)-5-(4-biphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C35H32N2O5S	1
1	EC50 = 14 nM
CP0244563 Compound Info	2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C27H24F3N3O6S	1
1	EC50 = 14 nM
CP0254301 Compound Info	2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C31H28F3NO6S	1
1	EC50 = 15 nM
CP0346384 Compound Info	(S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-2-methylphenoxy)acetic acid Show/Hide	C26H24Cl2N2O4	1
1	EC50 = 15 nM
CP0043947 Compound Info	2-(4-((4-(4-Isopropoxyphenyl)-5-(3-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C29H26F3NO6S	1
1	EC50 = 16 nM
CP0287052 Compound Info	2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-isopropoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid Show/Hide	C29H26F3NO5S	1
1	EC50 = 16 nM
CP0155637 Compound Info	(3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)oxy]butoxy}phenyl)acetic acid Show/Hide	C28H29NO5	2
1	EC50 = 20 nM
2	Ki = 0.3 nM
CP0428318 Compound Info	2-hydroxyethyl-[(E)-14-iodotetradec-13-en-3,5-diynoxy]phosphinic acid Show/Hide	C16H24IO4P	1
1	EC50 = 23.7 nM
CP0041706 Compound Info	2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy)phenoxy)acetic acid Show/Hide	C22H26O7	2
1	EC50 = 61 nM
2	Kd = 76.4 nM
CP0111046 Compound Info	2-[4-[[1-[(2,4-dichlorophenyl)carbamoyl]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-2-methylphenoxy]acetic acid Show/Hide	C26H24Cl2N2O4	1
1	EC50 = 70 nM
CP0562409 Compound Info	2-[4-[[4-(2-fluorophenyl)-5-oxo-1-[4-(trifluoromethyl)phenyl]-1,2,4-triazol-3-yl]methoxy]phenoxy]-2-methylpropanoic acid Show/Hide	C26H21F4N3O5	1
1	EC50 = 71.4 nM
CP0200400 Compound Info	2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C28H31FO6	1
1	EC50 = 106 nM
CP0185199 Compound Info	(S)-3-{4-[3,3-Bis-(4-bromo-phenyl)-allyloxy]-phenyl}-2-ethoxy-propionic acid Show/Hide	C26H24Br2O4	1
1	EC50 = 400 nM
CP0159874 Compound Info	2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C26H26ClFO6	1
1	EC50 = 545 nM
CP0034705 Compound Info	2-(3-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C25H24ClFO6	1
1	EC50 = 2230 nM
CP0261934 Compound Info	4-[1-(1,3-benzothiazol-6-ylsulfonyl)-5-chloroindol-2-yl]butanoic acid Show/Hide	C19H15ClN2O4S2	1
1	EC50 = 2962 nM
CP0177179 Compound Info	methyl 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]thiophene-2-carboxylate Show/Hide	C19H18N2O5S2	6
1	EC50 = 3400 nM
2	EC50 = 4000 nM
3	EC50 = 4340 nM
4	EC50 = 5400 nM
5	IC50 = 158.49 nM
6	Ki = 4.65 nM
CP0005387 Compound Info	Avandamet Show/Hide	C18H19N3O3S	5
1	EC50 = 3620 nM
2	IC50 > 5 nM
3	IC50 > 10000 nM
4	IC50 > 50000 nM
5	Ki > 33300 nM
CP0086778 Compound Info	3-[(3S)-3-[[4-methyl-2-(4-methylphenyl)-1,3-thiazole-5-carbonyl]amino]piperidin-1-yl]benzoic acid Show/Hide	C24H25N3O3S	1
1	EC50 = 11000 nM
CP0142812 Compound Info	3-[(3S)-3-[[2-(4-chlorophenyl)-4-methyl-1,3-thiazole-5-carbonyl]amino]piperidin-1-yl]benzoic acid Show/Hide	C23H22ClN3O3S	1
1	EC50 = 13000 nM
CP0427686 Compound Info	5-(4-Butoxy-3-{[2-fluoro-4-(trifluoromethyl)phenylamido]methyl}phenyl)-4,6-dimethylpyridine-3-carboxylic acid Show/Hide	C27H26F4N2O4	1
1	EC50 = 76000 nM
CP0043623 Compound Info	4-chloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H12ClF3N2O3S	7
1	IC50 = 1.21 nM
2	IC50 = 199.53 nM
3	IC50 = 233 nM
4	IC50 = 284 nM
5	IC50 = 648 nM
6	IC50 = 825 nM
7	IC50 = 1329 nM
CP0103788 Compound Info	2-(7-(2-(4-(trifluoromethyl)benzyloxy)-5-fluorobenzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H22F4O4S	1
1	IC50 = 1.7 nM
CP0186126 Compound Info	2-(4-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-5-methoxy-2-methylphenoxy)acetic acid Show/Hide	C25H23F3O5S	1
1	IC50 = 1.7 nM
CP0051320 Compound Info	3-(4-((R)-3-(4-chloro-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H26ClNO4	1
1	IC50 = 2 nM
CP0039115 Compound Info	2-(5-((4-methyl-2-(trifluoromethyl)thiazol-5-yl)methylthio)-1H-indol-1-yl)acetic acid Show/Hide	C16H13F3N2O2S2	1
1	IC50 = 2.8 nM
CP0035136 Compound Info	3-(4-(3-((5-chloro-3-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H25ClN2O4	1
1	IC50 = 3 nM
CP0035138 Compound Info	3-(4-(3-((6-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	IC50 = 3 nM
CP0035143 Compound Info	2-(4-(5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-2-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	IC50 = 3 nM
CP0035149 Compound Info	2-(4-(3-((2-chloro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23ClF3NO5	1
1	IC50 = 3 nM
CP0051472 Compound Info	3-(4-(3-((5-chloro-1-methyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H25ClN2O4	1
1	IC50 = 3 nM
CP0075561 Compound Info	2-(4-(4-fluoro-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H22F5NO5	1
1	IC50 = 3 nM
CP0075562 Compound Info	3-(4-(3-((5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C28H27ClN2O4	1
1	IC50 = 3 nM
CP0136122 Compound Info	2-(4-(3-((2-bromo-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23BrF3NO5	1
1	IC50 = 3 nM
CP0216422 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C27H26F3NO5	1
1	IC50 = 3 nM
CP0221348 Compound Info	3-(4-(3-((5-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	IC50 = 3 nM
CP0296984 Compound Info	2-(4-(3-fluoro-5-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H22F5NO5	1
1	IC50 = 3 nM
CP0035191 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO4S	1
1	IC50 = 3 nM
CP0035358 Compound Info	3-(2-ethyl-4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C28H33NO4	1
1	IC50 = 3 nM
CP0051318 Compound Info	(R)-3-(4-(3-(2-benzoyl-4-ethylphenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C29H32O5	1
1	IC50 = 3 nM
CP0112273 Compound Info	3-(2-ethyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C27H28F3NO4	1
1	IC50 = 3 nM
CP0264567 Compound Info	3-(4-((R)-3-(4-ethyl-2-(pyridin-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	IC50 = 3 nM
CP0173291 Compound Info	2-(6-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C22H16F3NO3S2	1
1	IC50 = 3.1 nM
CP0092761 Compound Info	2-(6-(4-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C25H19F3O4S	1
1	IC50 = 3.6 nM
CP0035196 Compound Info	3-(4-(3-((5-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23BrN2O4	1
1	IC50 = 4 nM
CP0136124 Compound Info	2-(4-(3-((2-methoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H26F3NO6	1
1	IC50 = 4 nM
CP0210104 Compound Info	2-(4-(3-((2,4-dimethylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H29NO5	1
1	IC50 = 4 nM
CP0216421 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H23F4NO5	1
1	IC50 = 4 nM
CP0261716 Compound Info	2-(4-(3-((2-ethyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C28H28F3NO5	1
1	IC50 = 4 nM
CP0136164 Compound Info	3-(2-methyl-4-((R)-3-(2-(pyridin-2-yl)-4-(trifluoromethyl)phenoxy)butoxy)phenyl)propanoic acid Show/Hide	C26H26F3NO4	1
1	IC50 = 4 nM
CP0057749 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-fluoro-phenyl}-propionic acid Show/Hide	C25H24ClFO5	1
1	IC50 = 4 nM
CP0074936 Compound Info	(R)-3-{4-[3-(4-ethyl-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C28H32O5	1
1	IC50 = 4 nM
CP0221700 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-ethyl-phenyl}-propionic acid Show/Hide	C27H29ClO5	1
1	IC50 = 4 nM
CP0254225 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C26H27ClO5	1
1	IC50 = 4 nM
CP0035140 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-5-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	IC50 = 5 nM
CP0035141 Compound Info	3-(2-methyl-4-(3-((2-methyl-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenyl)propanoic acid Show/Hide	C26H24F3NO4	1
1	IC50 = 5 nM
CP0075560 Compound Info	(R)-3-(4-(3-(1-(5-chloro-1,3-dimethyl-1H-indole-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid Show/Hide	C30H30ClFN2O4	1
1	IC50 = 5 nM
CP0215238 Compound Info	(R)-3-(4-(3-(1-(5-chloro-3-methylbenzo[b]thiophene-2-carboxamido)ethyl)-5-fluorophenoxy)-2-ethylphenyl)propanoic acid Show/Hide	C29H27ClFNO4S	1
1	IC50 = 5 nM
CP0261714 Compound Info	3-(4-(3-((5,6-dichloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H22Cl2N2O4	1
1	IC50 = 5 nM
CP0035354 Compound Info	(R)-3-(4-(3-(4-ethyl-2-(pyridin-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	IC50 = 5 nM
CP0035355 Compound Info	3-(4-((R)-3-(4-ethyl-2-(pyridin-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C27H31NO4	1
1	IC50 = 5 nM
CP0035360 Compound Info	3-{4-[(R)-3-(5-ethyl-biphenyl-2-yloxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C28H32O4	1
1	IC50 = 5 nM
CP0274499 Compound Info	3-(4-((R)-3-(4-ethyl-2-(oxazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO5	1
1	IC50 = 5 nM
CP0057743 Compound Info	(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethyl-phenoxy)-butoxy]-phenyl}-propionic acid Show/Hide	C27H27F3O5	1
1	IC50 = 5 nM
CP0082061 Compound Info	2-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-phenoxy}-2-methyl-propionic acid Show/Hide	C29H32O6	1
1	IC50 = 5 nM
CP0082065 Compound Info	(R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acid Show/Hide	C27H27F3O6	1
1	IC50 = 5 nM
CP0221734 Compound Info	(R)-3-{4-[3-(4-chloro-2-phenoxy-phenoxy)-butoxy]-2-trifluoromethyl-phenyl}-propionic acid Show/Hide	C26H24ClF3O5	1
1	IC50 = 5 nM
CP0035108 Compound Info	2-(4-(3-((4-chloro-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C26H26ClNO5	1
1	IC50 = 6 nM
CP0035142 Compound Info	2-(4-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methylphenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H25F4NO5	1
1	IC50 = 6 nM
CP0075559 Compound Info	2-methyl-2-(2-methyl-4-(3-((4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C26H24F3NO5	1
1	IC50 = 6 nM
CP0053319 Compound Info	2-(4-(3-(2-benzoyl-4-ethylphenoxy)propoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C28H30O6	1
1	IC50 = 6 nM
CP0166832 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-pentyloxy]-2-methyl-phenyl}-propionic acid Show/Hide	C30H34O5	1
1	IC50 = 6 nM
CP0218060 Compound Info	2-[4-[butyl-[2-chloro-3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	IC50 = 6.31 nM
CP0039117 Compound Info	2-(5-((4-methyl-2-(trifluoromethyl)thiazol-5-yl)methoxy)-1H-indol-1-yl)acetic acid Show/Hide	C16H13F3N2O3S	1
1	IC50 = 6.8 nM
CP0221733 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C29H32O5	1
1	IC50 = 7 nM
CP0039114 Compound Info	2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C20H14ClNO4S	1
1	IC50 = 7.7 nM
CP0296472 Compound Info	2-[4-[butyl-[2-chloro-3-(4-chlorophenyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H29Cl2NO5S	1
1	IC50 = 7.943 nM
CP0051319 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiophen-3-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O4S	1
1	IC50 = 8 nM
CP0131907 Compound Info	3-{4-[3-(2-benzyl-4-ethyl-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acid Show/Hide	C29H34O4	1
1	IC50 = 8 nM
CP0261715 Compound Info	3-(4-(3-((7-bromo-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23BrN2O4	1
1	IC50 = 9 nM
CP0035359 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiophen-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O4S	1
1	IC50 = 9 nM
CP0274904 Compound Info	3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-hexyloxy]-2-methyl-phenyl}-propionic acid Show/Hide	C31H36O5	1
1	IC50 = 9 nM
CP0162445 Compound Info	2-(7-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H23F3O4S	1
1	IC50 = 10 nM
CP0245147 Compound Info	2-(7-(2-(4-(trifluoromethyl)benzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H23F3O4S	1
1	IC50 = 10.4 nM
CP0083062 Compound Info	2-(6-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C21H14F3NO4S	1
1	IC50 = 11 nM
CP0035109 Compound Info	3-(4-(3-((4-chloro-1H-indole-2-carboxamido)methyl)phenoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H23ClN2O4	1
1	IC50 = 12 nM
CP0035145 Compound Info	2-(4-(3-((4-methoxy-2-methylbenzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H29NO6	1
1	IC50 = 12 nM
CP0035353 Compound Info	3-(4-((R)-3-(4-ethyl-2-(thiazol-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO4S	1
1	IC50 = 12 nM
CP0171815 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]acetic acid Show/Hide	C27H30ClNO5S	1
1	IC50 = 12.59 nM
CP0145397 Compound Info	3-(4-((R)-3-(4-ethyl-2-(oxazol-4-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C25H29NO5	1
1	IC50 = 13 nM
CP0083519 Compound Info	2-(5-(3-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)-1H-indol-1-yl)acetic acid Show/Hide	C25H20F3NO4	1
1	IC50 = 13 nM
CP0145396 Compound Info	3-(4-((R)-3-(4-ethyl-2-(furan-2-yl)phenoxy)butoxy)-2-methylphenyl)propanoic acid Show/Hide	C26H30O5	1
1	IC50 = 14 nM
CP0167041 Compound Info	2-(6-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methoxy)benzofuran-3-yl)acetic acid Show/Hide	C22H16F3NO4S	1
1	IC50 = 14 nM
CP0083099 Compound Info	2-(6-(3-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C25H19F3O4S	1
1	IC50 = 15 nM
CP0142828 Compound Info	2-[4-[butyl-[2-methyl-3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32F3NO5S	1
1	IC50 = 15.85 nM
CP0169972 Compound Info	2-[4-[butyl-[2-chloro-3-[4-(trifluoromethoxy)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO6S	1
1	IC50 = 15.85 nM
CP0281362 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2-cyclohexylphenoxy]propanoic acid Show/Hide	C32H38ClNO5S	1
1	IC50 = 15.85 nM
CP0156775 Compound Info	2-(4-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-2-methylphenoxy)acetic acid Show/Hide	C24H21F3O4S	1
1	IC50 = 19 nM
CP0161265 Compound Info	2-(4-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-5-chloro-2-methylphenoxy)acetic acid Show/Hide	C24H20ClF3O4S	1
1	IC50 = 20 nM
CP0199852 Compound Info	2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-methylbenzo[b]thiophen-3-yl)acetic acid Show/Hide	C21H16ClNO4S	1
1	IC50 = 23 nM
CP0176539 Compound Info	2-(6-(3-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzofuran-3-yl)acetic acid Show/Hide	C25H19F3O5	1
1	IC50 = 24.1 nM
CP0083528 Compound Info	2-(6-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methoxy)benzofuran-3-yl)acetic acid Show/Hide	C21H14F3NO5	1
1	IC50 = 25 nM
CP0142785 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methoxyphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO6S	1
1	IC50 = 25.12 nM
CP0206813 Compound Info	(2R)-2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 25.12 nM
CP0296303 Compound Info	2-(5-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methoxy)-1H-indol-1-yl)acetic acid Show/Hide	C21H15F3N2O4	1
1	IC50 = 31 nM
CP0035147 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-phenoxy-4-(trifluoromethyl)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C32H28F3NO6	1
1	IC50 = 32 nM
CP0083527 Compound Info	2-(4-methyl-6-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C22H16F3NO4S	1
1	IC50 = 37 nM
CP0173293 Compound Info	2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-5-methylbenzo[b]thiophen-3-yl)acetic acid Show/Hide	C21H16ClNO4S	1
1	IC50 = 37 nM
CP0075564 Compound Info	2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid Show/Hide	C27H23F6NO5	1
1	IC50 = 40 nM
CP0083525 Compound Info	2-(6-(2-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)-5-methylbenzo[b]thiophen-3-yl)acetic acid Show/Hide	C26H21F3O4S	1
1	IC50 = 43 nM
CP0074619 Compound Info	4-bromo-2-fluoro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11BrF4N2O3S	1
1	IC50 = 50.12 nM
CP0266172 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 50.12 nM
CP0035146 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methyl-4-(trifluoromethoxy)benzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C27H26F3NO6	1
1	IC50 = 54 nM
CP0173294 Compound Info	2-(4-chloro-6-((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C22H15ClF3NO3S2	1
1	IC50 = 58 nM
CP0171813 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-5-(trifluoromethyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	IC50 = 63.1 nM
CP0219135 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]butanoic acid Show/Hide	C29H34ClNO5S	1
1	IC50 = 63.1 nM
CP0035144 Compound Info	2-methyl-2-(2-methyl-4-(3-((2-methylbenzamido)methyl)phenoxy)phenoxy)propanoic acid Show/Hide	C26H27NO5	1
1	IC50 = 64 nM
CP0235279 Compound Info	2-(7-(4-(2,5-dichlorobenzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C25H22Cl2O4S	1
1	IC50 = 69 nM
CP0164151 Compound Info	2-(7-(4-(4-(trifluoromethoxy)benzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H23F3O5S	1
1	IC50 = 76 nM
CP0248504 Compound Info	2-[4-[butyl-[2-methyl-3-(4-methylphenyl)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H35NO5S	1
1	IC50 = 79.43 nM
CP0341227 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dichlorophenoxy]propanoic acid Show/Hide	C26H26Cl3NO5S	1
1	IC50 = 79.43 nM
CP0341774 Compound Info	2-[4-[butyl-[2-methyl-3-[4-(trifluoromethoxy)phenyl]phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32F3NO6S	1
1	IC50 = 79.43 nM
CP0083520 Compound Info	2-(6-(4-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzofuran-3-yl)acetic acid Show/Hide	C25H19F3O5	1
1	IC50 = 81 nM
CP0083521 Compound Info	2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)benzofuran-3-yl)acetic acid Show/Hide	C20H14ClNO5	1
1	IC50 = 81 nM
CP0292208 Compound Info	2-(7-(4-(4-chlorobenzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C25H23ClO4S	1
1	IC50 = 89 nM
CP0339540 Compound Info	2-(5-(4-(4-(trifluoromethyl)phenoxy)benzyloxy)-1H-indol-1-yl)acetic acid Show/Hide	C24H18F3NO4	1
1	IC50 = 91 nM
CP0172622 Compound Info	2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxazol-6-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C24H23F3N2O5	1
1	IC50 = 96 nM
CP0167039 Compound Info	2-(4-chloro-6-((5-(4-(trifluoromethyl)phenyl)isoxazol-3-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C21H13ClF3NO4S	1
1	IC50 = 97 nM
CP0212514 Compound Info	2-[4-[butyl-[3-(4-methoxyphenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H35NO6S	1
1	IC50 = 100 nM
CP0103781 Compound Info	2-(7-(4-(4-methoxybenzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H26O5S	1
1	IC50 = 120 nM
CP0038172 Compound Info	2-(7-(4-(benzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C25H24O4S	1
1	IC50 = 125 nM
CP0128531 Compound Info	4-chloro-3-methyl-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C16H14ClF3N2O3S	1
1	IC50 = 125.89 nM
CP0239873 Compound Info	3-bromo-4-chloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11BrClF3N2O3S	1
1	IC50 = 125.89 nM
CP0169971 Compound Info	2-[4-[butyl-[3-(3,4-dichlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H31Cl2NO5S	1
1	IC50 = 125.89 nM
CP0240934 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-propylsulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H30ClNO5S	1
1	IC50 = 125.89 nM
CP0161178 Compound Info	2-(8-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)chroman-5-yloxy)acetic acid Show/Hide	C26H23F3O5S	1
1	IC50 = 136 nM
CP0103789 Compound Info	2-(7-(4-(4-tert-butylbenzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C29H32O4S	1
1	IC50 = 148 nM
CP0290360 Compound Info	2,4-dichloro-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C15H11Cl2F3N2O3S	1
1	IC50 = 158.49 nM
CP0206812 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]hexanoic acid Show/Hide	C31H38ClNO5S	1
1	IC50 = 158.49 nM
CP0206814 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-3-chloro-2-methoxyphenoxy]propanoic acid Show/Hide	C27H29Cl2NO6S	1
1	IC50 = 158.49 nM
CP0291982 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]pentanoic acid Show/Hide	C30H36ClNO5S	1
1	IC50 = 158.49 nM
CP0274937 Compound Info	(S)-3-{4-[3-(2-benzoyl-4-ethyl-phenoxy)-butoxy]2-methyl-phenyl}propionic acid Show/Hide	C29H32O5	1
1	IC50 = 183 nM
CP0159997 Compound Info	2-(7-(4-(4-fluorobenzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C25H23FO4S	1
1	IC50 = 191 nM
CP0214965 Compound Info	4-phenyl-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C21H17F3N2O3S	1
1	IC50 = 199.53 nM
CP0281363 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-4-fluorophenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H29ClFNO5S	1
1	IC50 = 199.53 nM
CP0099056 Compound Info	(5-{3-[(6-BENZOYL-1-PROPYL-2-NAPHTHYL)OXY]PROPOXY}-1H-INDOL-1-YL)ACETIC ACID Show/Hide	C33H31NO5	1
1	IC50 = 223 nM
CP0039148 Compound Info	2-(6-(2-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C25H19F3O4S	1
1	IC50 = 244 nM
CP0291942 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-3-chloro-2-fluorophenoxy]propanoic acid Show/Hide	C26H26Cl2FNO5S	1
1	IC50 = 251.19 nM
CP0065352 Compound Info	4-methyl-2-[4-(trifluoromethyl)phenyl]-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]-1,3-thiazole-5-carboxamide Show/Hide	C20H15F6N3O3S2	5
1	IC50 = 284 nM
2	IC50 = 301 nM
3	IC50 = 423 nM
4	IC50 = 581 nM
5	IC50 = 949 nM
CP0210529 Compound Info	2-(7-(2-(4-(trifluoromethyl)benzyloxy)-6-fluorobenzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H22F4O4S	1
1	IC50 = 286 nM
CP0160000 Compound Info	2-(8-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-6-methylchroman-5-yloxy)acetic acid Show/Hide	C27H25F3O5S	1
1	IC50 = 313 nM
CP0149424 Compound Info	4-(2-methylpropyl)-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]benzamide Show/Hide	C19H21F3N2O3S	1
1	IC50 = 316.23 nM
CP0038170 Compound Info	2-(7-(4-(4-fluoro-2-(trifluoromethyl)benzyloxy)benzylthio)-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C26H22F4O4S	1
1	IC50 = 356 nM
CP0039157 Compound Info	2-(4-chloro-6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)benzo[b]thiophen-3-yl)acetic acid Show/Hide	C20H13Cl2NO4S	1
1	IC50 = 375 nM
CP0142827 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-4-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 398.11 nM
CP0142823 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2-fluoro-3-methoxyphenoxy]propanoic acid Show/Hide	C27H29ClFNO6S	1
1	IC50 = 501.19 nM
CP0310287 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(2-methoxyethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H30ClNO6S	1
1	IC50 = 501.19 nM
CP0103782 Compound Info	2-(7-(4-(4-(trifluoromethyl)benzyloxy)benzylthio)-5-methyl-2,3-dihydro-1H-inden-4-yloxy)acetic acid Show/Hide	C27H25F3O4S	1
1	IC50 = 586 nM
CP0169970 Compound Info	(2S)-2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 630.96 nM
CP0206836 Compound Info	2-[4-[butyl-[3-(3-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 630.96 nM
CP0341782 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-difluorophenoxy]propanoic acid Show/Hide	C26H26ClF2NO5S	1
1	IC50 = 630.96 nM
CP0159334 Compound Info	2-(5-(3-(4-(4-fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C29H28FNO5	1
1	IC50 = 649 nM
CP0083524 Compound Info	2-(6-(2-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)benzofuran-3-yl)acetic acid Show/Hide	C25H19F3O5	1
1	IC50 = 662 nM
CP0039116 Compound Info	2-(5-(2-((4-(trifluoromethyl)phenoxy)methyl)benzyloxy)-1H-indol-1-yl)acetic acid Show/Hide	C25H20F3NO4	1
1	IC50 = 734 nM
CP0206815 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(cyclopropylmethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H30ClNO5S	1
1	IC50 = 794.33 nM
CP0219137 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-pentylsulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H34ClNO5S	1
1	IC50 = 794.33 nM
CP0684997 Compound Info	5-(3-chloro-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H26ClNO5S	1
1	IC50 = 880 nM
CP0734398 Compound Info	5-(4-(3-(4-phenoxy-2-propylphenoxy)propoxy)-3-propylphenyl)thiazolidine-2,4-dione Show/Hide	C30H33NO5S	1
1	IC50 = 1000 nM
CP0142825 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(cyclobutylmethyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C29H32ClNO5S	1
1	IC50 = 1000 nM
CP0248505 Compound Info	2-[2-methyl-4-[3-methylbutyl-[3-[4-(trifluoromethyl)phenyl]phenyl]sulfamoyl]phenoxy]acetic acid Show/Hide	C27H28F3NO5S	1
1	IC50 = 1258.93 nM
CP0266173 Compound Info	2-[4-[[3-(4-chlorophenyl)-2-methylphenyl]-(4,4,4-trifluorobutyl)sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO5S	1
1	IC50 = 1258.93 nM
CP0281364 Compound Info	2-[4-[butyl-[3-(2-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 1584.89 nM
CP0295054 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H32ClNO5S	1
1	IC50 = 1584.89 nM
CP0783387 Compound Info	5-(3-fluoro-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H26FNO5S	1
1	IC50 = 2000 nM
CP0077688 Compound Info	2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propoxy)phenoxy)-2-methylpropanoic acid Show/Hide	C25H24ClFO6	1
1	IC50 = 2390 nM
CP0154580 Compound Info	2-(6-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C33H31NO5	1
1	IC50 = 2398 nM
CP0194328 Compound Info	2-(6-(3-(6-benzoylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C30H25NO5	1
1	IC50 = 2568 nM
CP0104519 Compound Info	2-(6-(3-(4-(4-fluorobenzoyl)phenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C26H22FNO5	1
1	IC50 = 3153 nM
CP0142780 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2,4-difluorophenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C27H28ClF2NO5S	1
1	IC50 = 3162.28 nM
CP0296470 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-2-(trifluoromethoxy)phenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H29ClF3NO6S	1
1	IC50 = 3162.28 nM
CP0194312 Compound Info	2-(4-(3-(4-(4-fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C29H28FNO5	1
1	IC50 = 3256 nM
CP0661032 Compound Info	5-(3-{3-[4-(4-Hydroxy-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C27H27NO6S	1
1	IC50 = 3800 nM
CP0186632 Compound Info	2-(5-(3-(6-benzoylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C30H25NO5	1
1	IC50 = 4430 nM
CP0160737 Compound Info	2-[4-[butyl-[5-(4-chlorophenyl)-4-fluoro-2-methylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C28H31ClFNO5S	1
1	IC50 = 5011.87 nM
CP0296471 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2-methylphenyl]sulfamoyl]-2,3-dimethoxyphenoxy]propanoic acid Show/Hide	C28H32ClNO7S	1
1	IC50 = 5011.87 nM
CP0099080 Compound Info	2-(4-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C33H31NO5	1
1	IC50 = 5377 nM
CP0680900 Compound Info	5-(3-methyl-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C28H29NO5S	1
1	IC50 = 6000 nM
CP0278453 Compound Info	2-(6-(3-(4-(4-fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C29H28FNO5	1
1	IC50 = 7616 nM
CP0240988 Compound Info	2-[4-[butyl-[3-(4-chlorophenyl)-2,4,6-trimethylphenyl]sulfamoyl]-2,3-dimethylphenoxy]propanoic acid Show/Hide	C30H36ClNO5S	1
1	IC50 = 10000 nM
CP0646515 Compound Info	5-(3-{3-[4-(4-Fluoro-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C27H26FNO5S	1
1	IC50 > 5000 nM
CP0651087 Compound Info	5-(3-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H27NO5S	2
1	IC50 > 10000 nM
2	IC50 > 50000 nM
CP0654439 Compound Info	5-(3-{3-[4-(4-Methoxy-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C28H29NO6S	1
1	IC50 > 10000 nM
CP0654730 Compound Info	5-(4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H27NO5S	1
1	IC50 > 10000 nM
CP0677669 Compound Info	5-(3-methoxy-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C28H29NO6S	1
1	IC50 > 10000 nM
CP0761598 Compound Info	5-(4-(4-(4-phenoxy-2-propylphenoxy)butoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C28H29NO5S	1
1	IC50 > 10000 nM
CP0099074 Compound Info	2-(4-(3-(4-(4-fluorobenzoyl)phenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C26H22FNO5	1
1	IC50 > 10000 nM
CP0099078 Compound Info	2-(4-(3-(6-benzoylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C30H25NO5	1
1	IC50 > 10000 nM
CP0159276 Compound Info	2-(5-(3-(4-(4-fluorobenzoyl)phenoxy)propoxy)-1H-indol-1-yl)acetic acid Show/Hide	C26H22FNO5	1
1	IC50 > 10000 nM
CP0654731 Compound Info	5-(3-{3-[4-(4-Chloro-3-methyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C28H28ClNO5S	1
1	IC50 > 50000 nM
CP0672145 Compound Info	5-(3-{3-[4-(4-Cyclopentyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C32H35NO5S	1
1	IC50 > 50000 nM
CP0672411 Compound Info	5-(3-{3-[4-(4-Fluoro-3-methyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C28H28FNO5S	1
1	IC50 > 50000 nM
CP0686397 Compound Info	5-(3-{3-[4-(4-Chloro-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C27H26ClNO5S	1
1	IC50 > 50000 nM
CP0708518 Compound Info	5-(3-(3-(4-(3,4-dichlorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H25Cl2NO5S	1
1	IC50 > 50000 nM
CP0727828 Compound Info	5-(3-{3-[4-(Biphenyl-4-yloxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C33H31NO5S	1
1	IC50 > 50000 nM
CP0782507 Compound Info	5-(3-{3-[4-(4-Isopropyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione Show/Hide	C30H33NO5S	1
1	IC50 > 50000 nM
CP0645378 Compound Info	5-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H26FNO5S	1
1	IC50 > 50000 nM
CP0658355 Compound Info	5-(4-(3-(4-(4-methoxyphenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C28H29NO6S	1
1	IC50 > 50000 nM
CP0672440 Compound Info	5-(4-(3-(4-(4-chlorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C27H26ClNO5S	1
1	IC50 > 50000 nM
CP0679717 Compound Info	5-(4-(3-(4-(biphenyl-4-yloxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C33H31NO5S	1
1	IC50 > 50000 nM
CP0705705 Compound Info	5-(4-(3-(4-(4-isobutylphenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C31H35NO5S	1
1	IC50 > 50000 nM
CP0716559 Compound Info	N-(4-(4-(3-(4-(2,4-dioxothiazolidin-5-yl)phenoxy)propoxy)-3-propylphenoxy)phenyl)-4-methylbenzenesulfonamide Show/Hide	C34H34N2O7S2	1
1	IC50 > 50000 nM
CP0761841 Compound Info	5-(4-(3-(4-(4-(methylsulfonyl)phenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione Show/Hide	C28H29NO7S2	1
1	IC50 > 50000 nM
CP0062441 Compound Info	(E)-6-[2-[[[4-(furan-2-yl)benzoyl]-methylamino]methyl]phenoxy]-4-methylhex-4-enoic acid Show/Hide	C26H27NO5	1
1	Kd = 57 nM
CP0128464 Compound Info	alkynyl ether, 24 Show/Hide	C31H29F3O6S	1
1	Ki = 0.6 nM
CP0086935 Compound Info	alkynyl ether, 23 Show/Hide	C30H27F3O6S	1
1	Ki = 2 nM
CP0130403 Compound Info	2-[3-chloro-4-[3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propylsulfanyl]phenyl]acetic acid Show/Hide	C27H26ClNO4S	1
1	Ki = 3.7 nM
CP0220490 Compound Info	2-[4-[3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propoxy]phenoxy]acetic acid Show/Hide	C27H27NO6	1
1	Ki = 3.7 nM
CP0036481 Compound Info	alkynyl ether, 27 Show/Hide	C32H31F3O6S	1
1	Ki = 4 nM
CP0322303 Compound Info	alkynyl ether, 10 Show/Hide	C27H23F3O5S	1
1	Ki = 4 nM
CP0078110 Compound Info	2-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenoxy}-propionic acid Show/Hide	C28H29NO6	1
1	Ki = 4.6 nM
CP0213824 Compound Info	2-(4-(3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy)propoxy)phenyl)acetic acid Show/Hide	C27H27NO5	1
1	Ki = 5 nM
CP0136386 Compound Info	alkynyl ether, 21 Show/Hide	C31H29F3O5S	1
1	Ki = 5 nM
CP0086936 Compound Info	alkynyl ether, 25 Show/Hide	C31H29F3O6S	1
1	Ki = 6 nM
CP0280556 Compound Info	alkynyl ether, 20 Show/Hide	C30H27F3O5S	1
1	Ki = 6 nM
CP0292417 Compound Info	alkynyl ether, 19 Show/Hide	C29H25F3O5S	1
1	Ki = 7 nM
CP0673789 Compound Info	2-(4-(2-chloro-4-((4-(trifluoromethyl)phenoxy)methyl)phenylthio)-5,6,7,8-tetrahydronaphthalen-1-yloxy)acetic acid Show/Hide	C26H22ClF3O4S	1
1	Ki = 7 nM
CP0201564 Compound Info	phenoxyacetic acid-ether, 9 Show/Hide	C28H29F3O6S	1
1	Ki = 8 nM
CP0167310 Compound Info	alkynyl ether, 26 Show/Hide	C31H29F3O6S	1
1	Ki = 9 nM
CP0145069 Compound Info	alkynyl ether, 33 Show/Hide	C30H28F3NO5S	1
1	Ki = 11 nM
CP0276403 Compound Info	phenoxyacetic acid-ether, 11 Show/Hide	C27H27F3O6S	1
1	Ki = 11 nM
CP0086937 Compound Info	alkynyl ether, 28 Show/Hide	C34H28F3NO5S	1
1	Ki = 16 nM
CP0194611 Compound Info	phenoxyacetic acid-ether, 12 Show/Hide	C26H22F3NO5S	1
1	Ki = 16 nM
CP0036288 Compound Info	(E)-3-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenyl}-acrylic acid Show/Hide	C28H27NO5	1
1	Ki = 18 nM
CP0167306 Compound Info	alkynyl ether, 22 Show/Hide	C32H31F3O6S	1
1	Ki = 22 nM
CP0208054 Compound Info	2-Methyl-2-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenoxy}-propionic acid Show/Hide	C30H33NO6	1
1	Ki = 23 nM
CP0086940 Compound Info	alkynyl ether, 32 Show/Hide	C31H31ClO5S	1
1	Ki = 28 nM
CP0039791 Compound Info	phenoxyacetic acid-ether, 13 Show/Hide	C29H26F3NO6S	1
1	Ki = 35 nM
CP0086938 Compound Info	alkynyl ether, 29 Show/Hide	C31H29F3O5S	1
1	Ki = 35 nM
CP0036483 Compound Info	alkynyl ether, 31 Show/Hide	C30H29ClO5S	1
1	Ki = 36 nM
CP0086886 Compound Info	phenoxyacetic acid-ether, 14 Show/Hide	C30H26F3NO5S	1
1	Ki = 36 nM
CP0324132 Compound Info	4-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenyl}-butyric acid Show/Hide	C29H31NO5	1
1	Ki = 38 nM
CP0146580 Compound Info	phenoxyacetic acid-ether, 15 Show/Hide	C30H26F3NO5S	1
1	Ki = 47 nM
CP0086887 Compound Info	phenoxyacetic acid-ether, 16 Show/Hide	C29H29F3O6S	1
1	Ki = 70 nM
CP0086939 Compound Info	alkynyl ether, 30 Show/Hide	C31H29F3O5S	1
1	Ki = 120 nM
CP0208857 Compound Info	alkynyl ether, 37 Show/Hide	C28H32O5S	1
1	Ki = 120 nM
CP0201561 Compound Info	alkynyl ether, 36 Show/Hide	C29H34O5S	1
1	Ki = 150 nM
CP0257979 Compound Info	2-Methyl-2-{3-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid Show/Hide	C30H33NO5	1
1	Ki = 165 nM
CP0100328 Compound Info	(E)-3-{4-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-acrylic acid Show/Hide	C29H29NO5	1
1	Ki = 265 nM
CP0275263 Compound Info	phenoxyacetic acid-ether, 17 Show/Hide	C30H32F3NO6S	1
1	Ki = 270 nM
CP0178891 Compound Info	2,2-Dimethyl-3-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid Show/Hide	C31H35NO5	1
1	Ki = 317 nM
CP0086881 Compound Info	alkynyl ether, 34 Show/Hide	C31H30F3NO4S	1
1	Ki = 660 nM
CP0208859 Compound Info	alkynyl ether, 35 Show/Hide	C29H34O6S	1
1	Ki = 1200 nM
CP0043337 Compound Info	(2S)-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-pyrrol-1-ylpropanoic acid Show/Hide	C25H24N2O4	1
1	Ki = 2500 nM
CP0086888 Compound Info	phenoxyacetic acid-ether, 18 Show/Hide	C30H32F3NO5S	1
1	Ki > 10000 nM

Clinical Information about the Protein

Target 1 ( Peroxisome proliferator-activated receptor delta (PPARD) )

Target Type	Clinical trial Target
Disease	3 Target-related Diseases				3
1	Obesity [ICD-11: 5B81]
2	Non-alcoholic steatohepatitis [ICD-11: DB92.1]
3	Type-1 diabetes [ICD-11: 5A10]
Clinical Trial Drug(s)	2 Clinical Trial Drugs				2
1	MBX-8025	Drug Info	Phase 2/3	Obesity
2	GFT-505	Drug Info	Phase 3	Non-alcoholic steatohepatitis
Discontinued Drug(s)	1 Discontinued Drug				1
1	GW-501516	Drug Info	Discontinued in Phase 4	Type-1 diabetes

Similar Protein(s) and Bioactivity Statistics

90% Identity

Protein ID	Protein Name	Protein Organism
PT03063	Peroxisome proliferator-activated receptor delta	Mus musculus, Mouse	Protein Info

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About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han