Cell Line ID	CL000044
Cell Line Name	CV-1
Synonyms	Cv-1 CV 1 CV-1.K CV1
Category	Finite cell line
Organism	Chlorocebus aethiops (Green monkey)
Cellosaurus ID	CVCL_0229
Tissue Information	Kidney
Disease	None

Map of Molecular Bioactivity Related to the Cell Line Cell Line Protein Compound Bioactivity Value: <= 0.1 μM > 0.1 μM and <= 10 μM > 10 μM Imprecise Activity

Compound ID	Compound Name	Compound Formula
CP0489029  Compound Info	4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)-3-methyl-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H11F6NO	1
1	EC50 = 0.03162 nM  Bioactivity Info	TI    LI    LO    TS
CP0416203  Compound Info	1-[(2S)-3-(4-cyano-2-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H16FN3O3	2
1	EC50 = 0.039 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.14 nM  Bioactivity Info	TI    LI    LO    TS
CP0416204  Compound Info	1-[(2S)-3-(2-bromo-4-cyanophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H16BrN3O3	2
1	EC50 = 0.06 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.41 nM  Bioactivity Info	TI    LI    LO    TS
CP0415630  Compound Info	1-[(2S)-3-(2-cyano-4-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H16FN3O3	2
1	EC50 = 0.074 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.74 nM  Bioactivity Info	TI    LI    LO    TS
CP0415628  Compound Info	1-[(2S)-3-(4-bromo-2-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H16BrFN2O3	2
1	EC50 = 0.11 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.93 nM  Bioactivity Info	TI    LI    LO    TS
CP0392181  Compound Info	5-(2,6-difluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H8F2N2O	2
1	EC50 = 0.14 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.71 nM  Bioactivity Info	TI    LI    LO    TS
CP0399810  Compound Info	1-[(2S)-3-(2-cyanophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H17N3O3	2
1	EC50 = 0.15 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.77 nM  Bioactivity Info	TI    LI    LO    TS
CP0429385  Compound Info	4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H9F6NO	1
1	EC50 = 0.1585 nM  Bioactivity Info	TI    LI    LO    TS
CP0482531  Compound Info	5-(2,6-dichloro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H8Cl2N2O	2
1	EC50 = 0.17 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0429399  Compound Info	2,3-dichloro-4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)benzonitrile    Show/Hide	C12H8Cl2F3NO	1
1	EC50 = 0.1995 nM  Bioactivity Info	TI    LI    LO    TS
CP0447519  Compound Info	2-chloro-4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)-3-methylbenzonitrile    Show/Hide	C13H11ClF3NO	1
1	EC50 = 0.1995 nM  Bioactivity Info	TI    LI    LO    TS
CP0570939  Compound Info	4-(1-cyclobutyl-2,2,2-trifluoro-1-hydroxyethyl)-3-methyl-2-(trifluoromethyl)benzonitrile    Show/Hide	C15H13F6NO	1
1	EC50 = 0.1995 nM  Bioactivity Info	TI    LI    LO    TS
CP0170782  Compound Info	6-[bis(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H9F9N2O	3
1	EC50 = 0.2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 1.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0416200  Compound Info	1-[(2S)-3-(2,4-dichlorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H16Cl2N2O3	2
1	EC50 = 0.25 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0510613  Compound Info	3-methyl-4-[2,2,2-trifluoro-1-(furan-2-yl)-1-hydroxyethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C15H9F6NO2	1
1	EC50 = 0.2512 nM  Bioactivity Info	TI    LI    LO    TS
CP0570940  Compound Info	3-methyl-4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H13F6NO	1
1	EC50 = 0.2512 nM  Bioactivity Info	TI    LI    LO    TS
CP0434291  Compound Info	1-[(2S)-3-(4-chloro-2-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H16ClFN2O3	2
1	EC50 = 0.28 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 0.85 nM  Bioactivity Info	TI    LI    LO    TS
CP0394102  Compound Info	(1R,2S,10S,11S,14S,15S,17S)-1-fluoro-14,17-dihydroxy-2,14,15-trimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-en-5-one    Show/Hide	C20H29FO3	2
1	EC50 = 0.3 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0395575  Compound Info	1-[(2S)-3-(4-bromophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17BrN2O3	2
1	EC50 = 0.34 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 7.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0078041  Compound Info	5-(2-fluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9FN2O	2
1	EC50 = 0.34 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1205.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0558047  Compound Info	2-chloro-4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)benzonitrile    Show/Hide	C12H9ClF3NO	1
1	EC50 = 0.3981 nM  Bioactivity Info	TI    LI    LO    TS
CP0203867  Compound Info	6-[ethyl(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H12F6N2O	2
1	EC50 = 0.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0382042  Compound Info	1-[(2S)-3-(2-bromo-4-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H16BrFN2O3	2
1	EC50 = 0.4 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 39.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0558043  Compound Info	3-methyl-4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-oxazol-4-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H8F6N2O2	1
1	EC50 = 0.5012 nM  Bioactivity Info	TI    LI    LO    TS
CP0434507  Compound Info	1-[(2S)-3-(2-chloro-4-methoxyphenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H19ClN2O4	2
1	EC50 = 0.61 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 54.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0558045  Compound Info	2,3-dichloro-4-(1-cyclobutyl-2,2,2-trifluoro-1-hydroxyethyl)benzonitrile    Show/Hide	C13H10Cl2F3NO	1
1	EC50 = 0.631 nM  Bioactivity Info	TI    LI    LO    TS
CP0456182  Compound Info	2,3-dichloro-4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)benzonitrile    Show/Hide	C12H10Cl2F3NO	1
1	EC50 = 0.7943 nM  Bioactivity Info	TI    LI    LO    TS
CP0570934  Compound Info	2-chloro-3-methyl-4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)benzonitrile    Show/Hide	C13H13ClF3NO	1
1	EC50 = 0.7943 nM  Bioactivity Info	TI    LI    LO    TS
CP0374902  Compound Info	7-Ethyl-6-methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0429807  Compound Info	(6S,7S)-6-ethyl-7-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0417190  Compound Info	(R)-3-ethyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C16H14F6N2O2	2
1	EC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0417188  Compound Info	(2R)-2-methyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H12F6N2O2	3
1	EC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 70 nM  Bioactivity Info	TI    LI    LO    TS
3	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0373227  Compound Info	tert-butyl 4-methyl-2,5-dioxo-1H-chromeno[3,4-f]quinoline-10-carboxylate    Show/Hide	C22H19NO5	2
1	EC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0411231  Compound Info	1-[(2S)-3-(4-fluoro-2-methylphenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H19FN2O3	2
1	EC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 72.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0036705  Compound Info	(1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-en-5-one    Show/Hide	C19H28O2	1
1	EC50 = 1.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0558044  Compound Info	4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-oxazol-4-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H6F6N2O2	1
1	EC50 = 1.259 nM  Bioactivity Info	TI    LI    LO    TS
CP0567860  Compound Info	4-[2,2,2-trifluoro-1-(furan-2-yl)-1-hydroxyethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H7F6NO2	1
1	EC50 = 1.259 nM  Bioactivity Info	TI    LI    LO    TS
CP0441554  Compound Info	2-(difluoromethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H10F8N2O2	1
1	EC50 = 1.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0159674  Compound Info	1-(cyclopropylmethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H15F3N2O2	2
1	EC50 = 1.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0359750  Compound Info	6-(dipropylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C16H19F3N2O	2
1	EC50 = 1.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0447522  Compound Info	4-(1-cyclopropyl-2,2,2-trifluoro-1-hydroxyethyl)-2,3-dimethylbenzonitrile    Show/Hide	C14H14F3NO	1
1	EC50 = 1.585 nM  Bioactivity Info	TI    LI    LO    TS
CP0447526  Compound Info	4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-3-methyl-2-(trifluoromethyl)benzonitrile    Show/Hide	C12H6F9NO	1
1	EC50 = 1.585 nM  Bioactivity Info	TI    LI    LO    TS
CP0549434  Compound Info	4-(1-cyclobutyl-2,2,2-trifluoro-1-hydroxyethyl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H11F6NO	1
1	EC50 = 1.585 nM  Bioactivity Info	TI    LI    LO    TS
CP0561936  Compound Info	2-chloro-4-(1-cyclobutyl-2,2,2-trifluoro-1-hydroxyethyl)benzonitrile    Show/Hide	C13H11ClF3NO	1
1	EC50 = 1.585 nM  Bioactivity Info	TI    LI    LO    TS
CP0482570  Compound Info	1-[(2S)-2-hydroxy-2-methyl-3-[2-(trifluoromethyl)phenoxy]propanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H17F3N2O3	2
1	EC50 = 1.7 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 372 nM  Bioactivity Info	TI    LI    LO    TS
CP0392184  Compound Info	5-(2-chloro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9ClN2O	2
1	EC50 = 1.7 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1556 nM  Bioactivity Info	TI    LI    LO    TS
CP0411228  Compound Info	1-[(2S)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H17N3O3	2
1	EC50 = 1.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 71.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0416202  Compound Info	1-[(2S)-2-hydroxy-2-methyl-3-[4-(trifluoromethyl)phenoxy]propanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H17F3N2O3	2
1	EC50 = 1.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0390933  Compound Info	6-[bis(cyclopropylmethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C18H19F3N2O	2
1	EC50 = 1.9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0432984  Compound Info	1-(cyclopropylmethyl)-2-methyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C17H17F3N2O2	1
1	EC50 = 1.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0451594  Compound Info	4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-thiazol-4-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H6F6N2OS	1
1	EC50 = 1.995 nM  Bioactivity Info	TI    LI    LO    TS
CP0475457  Compound Info	4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-thiazol-2-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H6F6N2OS	1
1	EC50 = 1.995 nM  Bioactivity Info	TI    LI    LO    TS
CP0561872  Compound Info	2-chloro-3-methyl-4-(1,1,1-trifluoro-2-hydroxybutan-2-yl)benzonitrile    Show/Hide	C12H11ClF3NO	1
1	EC50 = 1.995 nM  Bioactivity Info	TI    LI    LO    TS
CP0049794  Compound Info	(4aS,12bS)-11-(trifluoromethyl)-2,3,4,4a,5,6,8,12b-octahydro-1H-pyrido[3,2-b]phenanthridin-9-one    Show/Hide	C17H17F3N2O	2
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0375501  Compound Info	5-Ethyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C15H14F3NO2	2
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0375820  Compound Info	4,5-Bis-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C14H9F6NO2	2
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0404519  Compound Info	5-Methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C14H12F3NO2	2
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0394257  Compound Info	(2R)-1-(2,2,2-trifluoroethyl)-2,9-bis(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H9F9N2O2	1
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0412815  Compound Info	(2R)-2-(methoxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C16H14F6N2O3	1
1	EC50 = 2 nM  Bioactivity Info	TI    LI    LO    TS
CP0203868  Compound Info	6-(diethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H15F3N2O	2
1	EC50 = 2.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0390934  Compound Info	6-[ethyl(propan-2-yl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H17F3N2O	2
1	EC50 = 2.2 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0202560  Compound Info	1-(cyclopropylmethyl)-2-ethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C18H19F3N2O2	1
1	EC50 = 2.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0433610  Compound Info	1-propyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H15F3N2O2	2
1	EC50 = 2.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0060255  Compound Info	1-[(2S)-3-(4-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17FN2O3	2
1	EC50 = 2.5 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0447517  Compound Info	4-[1-(5-chlorofuran-2-yl)-2,2,2-trifluoro-1-hydroxyethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H6ClF6NO2	1
1	EC50 = 2.512 nM  Bioactivity Info	TI    LI    LO    TS
CP0456183  Compound Info	2,3-dichloro-4-(1,1,1-trifluoro-2-hydroxybutan-2-yl)benzonitrile    Show/Hide	C11H8Cl2F3NO	1
1	EC50 = 2.512 nM  Bioactivity Info	TI    LI    LO    TS
CP0253730  Compound Info	2-methyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H12F6N2O2	1
1	EC50 = 2.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0432982  Compound Info	(2R)-2-ethyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H14F6N2O2	1
1	EC50 = 2.7 nM  Bioactivity Info	TI    LI    LO    TS
CP0390988  Compound Info	6-[(cyclopropylmethyl)(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C16H14F6N2O	2
1	EC50 = 2.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0451593  Compound Info	4-[1-(5-chlorofuran-2-yl)-2,2,2-trifluoro-1-hydroxyethyl]-3-methyl-2-(trifluoromethyl)benzonitrile    Show/Hide	C15H8ClF6NO2	1
1	EC50 = 2.884 nM  Bioactivity Info	TI    LI    LO    TS
CP0411210  Compound Info	1-[(2S)-3-(2-fluoro-4-methoxyphenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H19FN2O4	2
1	EC50 = 2.9 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0189598  Compound Info	(4aR,12bS)-11-(trifluoromethyl)-2,3,4,4a,5,6,8,12b-octahydro-1H-pyrido[3,2-b]phenanthridin-9-one    Show/Hide	C17H17F3N2O	2
1	EC50 = 3 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0192403  Compound Info	6-Isopropyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 3 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0105842  Compound Info	(7S,8R)-7,8-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 = 3 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0419488  Compound Info	2,3-dichloro-4-(1,1,1-trifluoro-2-hydroxy-4,4-dimethylpentan-2-yl)benzonitrile    Show/Hide	C14H14Cl2F3NO	1
1	EC50 = 3.162 nM  Bioactivity Info	TI    LI    LO    TS
CP0419489  Compound Info	2,3-dichloro-4-(1,1,1-trifluoro-2-hydroxy-4-methylpentan-2-yl)benzonitrile    Show/Hide	C13H12Cl2F3NO	1
1	EC50 = 3.162 nM  Bioactivity Info	TI    LI    LO    TS
CP0570936  Compound Info	2-chloro-4-(1-cyclopentyl-2,2,2-trifluoro-1-hydroxyethyl)benzonitrile    Show/Hide	C14H13ClF3NO	1
1	EC50 = 3.162 nM  Bioactivity Info	TI    LI    LO    TS
CP0431961  Compound Info	1-(2-methylpropyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H17F3N2O2	1
1	EC50 = 3.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0485798  Compound Info	2-(ethoxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C17H16F6N2O3	1
1	EC50 = 3.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0435178  Compound Info	1-[(2S)-3-(4-chlorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17ClN2O3	2
1	EC50 = 3.4 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 172.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0436363  Compound Info	4-(cyclopropylmethyl)-3-phenyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C22H19F3N2O2	2
1	EC50 = 3.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0320793  Compound Info	1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C14H10F6N2O2	2
1	EC50 = 3.5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0434484  Compound Info	(2S)-2-methyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H12F6N2O2	1
1	EC50 = 3.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0412810  Compound Info	(2R)-2-(fluoromethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H11F7N2O2	1
1	EC50 = 3.8 nM  Bioactivity Info	TI    LI    LO    TS
CP0483870  Compound Info	1,2-diethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H17F3N2O2	1
1	EC50 = 3.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0429405  Compound Info	2-chloro-3-methyl-4-(1,1,1-trifluoro-2-hydroxy-4,4-dimethylpentan-2-yl)benzonitrile    Show/Hide	C15H17ClF3NO	1
1	EC50 = 3.981 nM  Bioactivity Info	TI    LI    LO    TS
CP0447525  Compound Info	4-(1,1,1-trifluoro-2-hydroxybutan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C12H9F6NO	1
1	EC50 = 3.981 nM  Bioactivity Info	TI    LI    LO    TS
CP0489030  Compound Info	3-methyl-4-(1,1,1-trifluoro-2-hydroxypropan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C12H9F6NO	1
1	EC50 = 3.981 nM  Bioactivity Info	TI    LI    LO    TS
CP0549431  Compound Info	2-chloro-4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)benzonitrile    Show/Hide	C12H11ClF3NO	1
1	EC50 = 3.981 nM  Bioactivity Info	TI    LI    LO    TS
CP0049184  Compound Info	6-ethyl-4-(trifluoromethyl)-1H,2H,6H,7H,8H,9H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	4
1	EC50 = 4 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 4.1 nM  Bioactivity Info	TI    LI    LO    TS
3	IC50 = 4580 nM  Bioactivity Info	TI    LI    LO    TS
4	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0433824  Compound Info	2-(propoxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C18H18F6N2O3	1
1	EC50 = 4.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0407007  Compound Info	(2R,3R)-2,3-Dimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C14H13F3N2O	1
1	EC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0460983  Compound Info	(5bR,9aR)-4-Trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C16H15F3N2O	1
1	EC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0372391  Compound Info	5-Propyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0404427  Compound Info	(6R,7R)-6,7-diethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C17H18F3NO2	2
1	EC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0461022  Compound Info	(6S,7S)-6,7-diethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C17H18F3NO2	2
1	EC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1400 nM  Bioactivity Info	TI    LI    LO    TS
CP0044960  Compound Info	(1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-5-one    Show/Hide	C19H30O2	5
1	EC50 = 5.1 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 5.7 nM  Bioactivity Info	TI    LI    LO    TS
3	EC50 = 6 nM  Bioactivity Info	TI    LI    LO    TS
4	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
5	Ki = 0.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0441553  Compound Info	(2R)-2-phenyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C20H14F6N2O2	1
1	EC50 = 5.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0475157  Compound Info	5-(2-cyano-6-fluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H8FN3O	2
1	EC50 = 5.3 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 28.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0394489  Compound Info	(R)-3-methyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C15H12F6N2O2	2
1	EC50 = 5.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0475456  Compound Info	4-[1-(5-chlorothiophen-2-yl)-2,2,2-trifluoro-1-hydroxyethyl]-3-methyl-2-(trifluoromethyl)benzonitrile    Show/Hide	C15H8ClF6NOS	1
1	EC50 = 5.623 nM  Bioactivity Info	TI    LI    LO    TS
CP0456181  Compound Info	3-methyl-4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-thiazol-4-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H8F6N2OS	1
1	EC50 = 5.888 nM  Bioactivity Info	TI    LI    LO    TS
CP0437277  Compound Info	(2R)-2-(propan-2-yl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C17H16F6N2O2	1
1	EC50 = 5.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0865304  Compound Info	(+/-)-1-(2,2,2-trifluoroethyl)-2,9-bis(trifluoromethyl)-2,3-dihydro-1H-[1,4]oxazino[3,2-g]quinolin-7(6H)-one    Show/Hide	C15H9F9N2O2	1
1	EC50 = 5.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0082236  Compound Info	2-ethyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H14F6N2O2	1
1	EC50 = 6 nM  Bioactivity Info	TI    LI    LO    TS
CP0041416  Compound Info	(6alpha)-17-(Acetyloxy)-6-methylpreg-4-ene-3,20-dione    Show/Hide	C24H34O4	2
1	EC50 = 6.1 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 6.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0395573  Compound Info	1-[(2S)-3-(2-chlorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17ClN2O3	2
1	EC50 = 6.1 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 4818.2 nM  Bioactivity Info	TI    LI    LO    TS
CP0155404  Compound Info	1-ethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C14H13F3N2O2	2
1	EC50 = 6.4 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0412808  Compound Info	(2S)-2-(hydroxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H12F6N2O3	2
1	EC50 = 6.6 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 165 nM  Bioactivity Info	TI    LI    LO    TS
CP0492849  Compound Info	methyl 4-[(2S)-3-(4-cyano-2,3-dihydroindol-1-yl)-2-hydroxy-2-methyl-3-oxopropoxy]benzoate    Show/Hide	C21H20N2O5	2
1	EC50 = 6.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0208631  Compound Info	(7R)-6-ethyl-7-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 7 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 2710 nM  Bioactivity Info	TI    LI    LO    TS
CP0212830  Compound Info	(6R,7S)-6-ethyl-7-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 7 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0398020  Compound Info	8-ethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C15H14F3NO2	2
1	EC50 = 7 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0415647  Compound Info	(6R,7S)-6-ethyl-7-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 7 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0382041  Compound Info	1-[(2S)-2-hydroxy-2-methyl-3-[4-(1,3-oxazol-4-yl)phenoxy]propanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C22H19N3O4	2
1	EC50 = 7.2 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0434506  Compound Info	1-[(2S)-3-(4-cyano-2-methoxyphenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C21H19N3O4	2
1	EC50 = 7.6 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 2118.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0394101  Compound Info	1-tert-butyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H17F3N2O2	2
1	EC50 = 7.8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0429386  Compound Info	4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H11F6NO	1
1	EC50 = 7.943 nM  Bioactivity Info	TI    LI    LO    TS
CP0397374  Compound Info	8-ethyl-6-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 8 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0415629  Compound Info	1-[(2S)-2-hydroxy-3-(4-methoxyphenoxy)-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H20N2O4	2
1	EC50 = 8.6 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 624.3 nM  Bioactivity Info	TI    LI    LO    TS
CP0208771  Compound Info	(11S,15R)-7-(trifluoromethyl)-4,17-diazatetracyclo[8.7.0.03,8.011,15]heptadeca-1(10),2,6,8-tetraen-5-one    Show/Hide	C16H15F3N2O	2
1	EC50 = 9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0375509  Compound Info	7,7-Dimethyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C15H14F3NO2	2
1	EC50 = 9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0278665  Compound Info	(7S,8R)-7-Ethyl-8-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 9 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0377494  Compound Info	(5bR,9aR)-1-Methyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C17H17F3N2O	1
1	EC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0183809  Compound Info	(7R)-6,7-dimethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0217196  Compound Info	(7R,8R)-7-Ethyl-8-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0432985  Compound Info	1-ethyl-2-methyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H15F3N2O2	1
1	EC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0035186  Compound Info	(10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]-14-hydroxy-15-methyl-14-(prop-1-yn-1-yl)tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-5-one    Show/Hide	C29H35NO2	3
1	EC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 1 nM  Bioactivity Info	TI    LI    LO    TS
3	IC50 = 5 nM  Bioactivity Info	TI    LI    LO    TS
CP0447516  Compound Info	3-methyl-4-[2,2,2-trifluoro-1-hydroxy-1-(1,3-thiazol-2-yl)ethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H8F6N2OS	1
1	EC50 = 10.47 nM  Bioactivity Info	TI    LI    LO    TS
CP0373218  Compound Info	10-methoxy-4-methyl-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C18H13NO4	2
1	EC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0386694  Compound Info	(2R)-2-(hydroxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H12F6N2O3	2
1	EC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 60 nM  Bioactivity Info	TI    LI    LO    TS
CP0373226  Compound Info	10-(hydroxymethyl)-4-methyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H15NO3	2
1	EC50 = 12 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0429400  Compound Info	4-(1,1,1-trifluoro-2-hydroxybut-3-en-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C12H7F6NO	1
1	EC50 = 12.59 nM  Bioactivity Info	TI    LI    LO    TS
CP0570937  Compound Info	2,3-dimethyl-4-(1,1,1-trifluoro-2-hydroxy-3-methylbutan-2-yl)benzonitrile    Show/Hide	C14H16F3NO	1
1	EC50 = 12.59 nM  Bioactivity Info	TI    LI    LO    TS
CP0213338  Compound Info	(7R)-7-methyl-4-(trifluoromethyl)-6-(3,3,3-trifluoropropyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H16F6N2O	2
1	EC50 = 13 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 61 nM  Bioactivity Info	TI    LI    LO    TS
CP0398685  Compound Info	5-Pentafluoroethyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C15H9F8NO2	2
1	EC50 = 13 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0358612  Compound Info	4-(trifluoromethyl)-1,2,7,8,9,10,10a,11-octahydro-12-oxa-1,6000100-diazatetraphen-2-one    Show/Hide	C16H15F3N2O2	1
1	EC50 = 14 nM  Bioactivity Info	TI    LI    LO    TS
CP0382551  Compound Info	1-[(2S)-3-(2-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17FN2O3	2
1	EC50 = 14.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0377287  Compound Info	(2R,3R)-2,3,8-Trimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 9182 nM  Bioactivity Info	TI    LI    LO    TS
CP0049409  Compound Info	6-Methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C14H13F3N2O	2
1	EC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 259 nM  Bioactivity Info	TI    LI    LO    TS
CP0434033  Compound Info	3-ethyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H14F6N2O2	2
1	EC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0475159  Compound Info	5-[4-hydroxy-2-(trifluoromethyl)phenyl]-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H9F3N2O	2
1	EC50 = 15.2 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0451595  Compound Info	2-chloro-4-(4-cyclopropyl-1,1,1-trifluoro-2-hydroxybut-3-yn-2-yl)-3-methylbenzonitrile    Show/Hide	C15H11ClF3NO	1
1	EC50 = 15.85 nM  Bioactivity Info	TI    LI    LO    TS
CP0451596  Compound Info	4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C11H4F9NO	1
1	EC50 = 15.85 nM  Bioactivity Info	TI    LI    LO    TS
CP0456184  Compound Info	3-methyl-4-(4,4,4-trifluoro-3-hydroxy-2-methylbutan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H13F6NO	1
1	EC50 = 15.85 nM  Bioactivity Info	TI    LI    LO    TS
CP0449306  Compound Info	(6S,8R)-6-ethyl-8-methyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0309686  Compound Info	(7S,8R)-8-Ethyl-7-propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	2
1	EC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0373230  Compound Info	10-hydroxy-4-(trifluoromethyl)-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C17H10F3NO3	2
1	EC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0383826  Compound Info	1-[(2S)-3-(4-chloro-2-methoxyphenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C20H19ClN2O4	2
1	EC50 = 17.1 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0468784  Compound Info	5-(7-hydroxy-2,3-dihydro-1H-inden-4-yl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C15H14N2O	2
1	EC50 = 17.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0421959  Compound Info	(S)-4-(cyclopropylmethyl)-3-phenyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C22H19F3N2O2	2
1	EC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0444567  Compound Info	1-methyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C13H11F3N2O2	2
1	EC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0433628  Compound Info	9-ethoxy-10-methoxy-4-methyl-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C20H17NO5	2
1	EC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0228036  Compound Info	6-Propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0461021  Compound Info	4-Trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C13H10F3NO2	2
1	EC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0432004  Compound Info	(2R)-2-(3-methylphenyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C21H16F6N2O2	1
1	EC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0419286  Compound Info	2-chloro-4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-3-methylbenzonitrile    Show/Hide	C11H6ClF6NO	1
1	EC50 = 19.95 nM  Bioactivity Info	TI    LI    LO    TS
CP0549432  Compound Info	2,3-dimethyl-4-(1,1,1-trifluoro-2-hydroxy-4,4-dimethylpentan-2-yl)benzonitrile    Show/Hide	C16H20F3NO	1
1	EC50 = 19.95 nM  Bioactivity Info	TI    LI    LO    TS
CP0567859  Compound Info	4-[1-(5-chlorothiophen-2-yl)-2,2,2-trifluoro-1-hydroxyethyl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H6ClF6NOS	1
1	EC50 = 19.95 nM  Bioactivity Info	TI    LI    LO    TS
CP0373320  Compound Info	(R)-2,8-Dimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C14H13F3N2O	1
1	EC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0461096  Compound Info	(7R,8R)-7,8-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0424753  Compound Info	(R)-3-isopropyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C17H16F6N2O2	2
1	EC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0373224  Compound Info	10-methoxy-4-(trifluoromethyl)-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H12F3NO3	2
1	EC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0364001  Compound Info	(R)-8-Methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C14H13F3N2O	2
1	EC50 = 21 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0399724  Compound Info	9-hydroxy-10-methoxy-4-methyl-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C18H13NO5	2
1	EC50 = 21 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0309668  Compound Info	(7S)-6,7-dimethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0373217  Compound Info	10-methoxy-4-methyl-9-propan-2-yloxy-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C21H19NO5	2
1	EC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0412809  Compound Info	(2R)-2-(2-methylsulfanylethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C17H16F6N2O2S	1
1	EC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0458065  Compound Info	(2R)-1,2-bis(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C16H11F9N2O2	1
1	EC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0463444  Compound Info	(5bR,9aR)-5b-Methyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C17H17F3N2O	1
1	EC50 = 25 nM  Bioactivity Info	TI    LI    LO    TS
CP0214521  Compound Info	6-Isobutyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 = 25 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0460898  Compound Info	6,8-diethyl-4-(trifluoromethyl)-6,7,8,9-tetrahydropyrano[3,2-g]quinolin-2-one    Show/Hide	C17H18F3NO2	2
1	EC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0483839  Compound Info	(15R)-7-(trifluoromethyl)-17-oxa-4,11-diazatetracyclo[8.7.0.0^{3,8}.0^{11,15}]heptadeca-1,3(8),6,9-tetraen-5-one    Show/Hide	C15H13F3N2O2	1
1	EC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
CP0437275  Compound Info	(2R)-2-(2-methylpropyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C18H18F6N2O2	1
1	EC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0412811  Compound Info	2-(methylsulfanylmethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C16H14F6N2O2S	2
1	EC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 25 nM  Bioactivity Info	TI    LI    LO    TS
CP0482533  Compound Info	5-(2-cyano-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H9N3O	2
1	EC50 = 29.7 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0394105  Compound Info	(2S)-2-ethyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H14F6N2O2	1
1	EC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0394253  Compound Info	2-[7-oxo-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-2-yl]acetonitrile    Show/Hide	C16H11F6N3O2	1
1	EC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0378461  Compound Info	1,3-diethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C16H17F3N2O2	2
1	EC50 = 31 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0549433  Compound Info	4-(1,1,1-trifluoro-2-hydroxy-3-methylbut-3-en-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C13H9F6NO	1
1	EC50 = 31.62 nM  Bioactivity Info	TI    LI    LO    TS
CP0318127  Compound Info	(6S,8R)-6,8-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0389662  Compound Info	(5bR,9aR)-1,5b-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C18H19F3N2O	1
1	EC50 = 33 nM  Bioactivity Info	TI    LI    LO    TS
CP0183422  Compound Info	(7R,8R)-7,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 34 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 74 nM  Bioactivity Info	TI    LI    LO    TS
CP0468788  Compound Info	5-(4-hydroxy-2,3-dimethylphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C14H14N2O	2
1	EC50 = 34.6 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0464182  Compound Info	(R)-4-allyl-3-isopropyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C18H19F3N2O2	2
1	EC50 = 35 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0412813  Compound Info	(2S)-2-(fluoromethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H11F7N2O2	2
1	EC50 = 35 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 199 nM  Bioactivity Info	TI    LI    LO    TS
CP0394310  Compound Info	(2R)-2-(4-methylphenyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C21H16F6N2O2	1
1	EC50 = 36 nM  Bioactivity Info	TI    LI    LO    TS
CP0392188  Compound Info	5-(4-hydroxy-3-methylphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H12N2O	2
1	EC50 = 37.3 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1542.6 nM  Bioactivity Info	TI    LI    LO    TS
CP0416201  Compound Info	1-[(2S)-3-(3-fluorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17FN2O3	2
1	EC50 = 37.4 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1530.4 nM  Bioactivity Info	TI    LI    LO    TS
CP0447523  Compound Info	4-[(E)-1,1,1-trifluoro-2-hydroxy-3-methylpent-3-en-2-yl]-2-(trifluoromethyl)benzonitrile    Show/Hide	C14H11F6NO	1
1	EC50 = 39.81 nM  Bioactivity Info	TI    LI    LO    TS
CP0491543  Compound Info	3,3-Dimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C14H13F3N2O	2
1	EC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0394222  Compound Info	(2S)-1-(2,2,2-trifluoroethyl)-2,9-bis(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C15H9F9N2O2	2
1	EC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 34 nM  Bioactivity Info	TI    LI    LO    TS
CP0449133  Compound Info	(R)-3-benzyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C21H16F6N2O2	2
1	EC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0394285  Compound Info	trifluoromethyl 10-methoxy-4-methyl-2,5-dioxo-1H-chromeno[3,4-f]quinoline-9-carboxylate    Show/Hide	C20H12F3NO6	2
1	EC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0433974  Compound Info	1,3-dimethyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C14H13F3N2O2	1
1	EC50 = 47 nM  Bioactivity Info	TI    LI    LO    TS
CP0373229  Compound Info	10-methoxy-4-methyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H15NO3	2
1	EC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0461126  Compound Info	(R)-4-allyl-3-ethyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C17H17F3N2O2	2
1	EC50 = 51 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0378430  Compound Info	3-ethyl-1-methyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H15F3N2O2	2
1	EC50 = 52 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 67 nM  Bioactivity Info	TI    LI    LO    TS
CP0213792  Compound Info	(6R,7R)-7-methyl-6-(2-methylpropyl)-4-(trifluoromethyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	2
1	EC50 = 56 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 29 nM  Bioactivity Info	TI    LI    LO    TS
CP0412071  Compound Info	(6S,8R)-6,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 59 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0432040  Compound Info	4-(trifluoromethyl)-1,6-dihydroisochromeno[3,4-f]quinolin-2-one    Show/Hide	C17H10F3NO2	2
1	EC50 = 60 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0429114  Compound Info	(S)-3-Methyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C13H11F3N2O	1
1	EC50 = 62 nM  Bioactivity Info	TI    LI    LO    TS
CP0570935  Compound Info	2,3-dichloro-4-(1,1,1-trifluoro-2-hydroxypropan-2-yl)benzonitrile    Show/Hide	C10H6Cl2F3NO	1
1	EC50 = 63.1 nM  Bioactivity Info	TI    LI    LO    TS
CP0377288  Compound Info	(5bR,7S,9aR)-7-Methyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C17H17F3N2O	1
1	EC50 = 64 nM  Bioactivity Info	TI    LI    LO    TS
CP0442162  Compound Info	6-alkyl, 7-amino-2-quinolinone, 11d (+/-)    Show/Hide	C14H15F3N2O	3
1	EC50 = 65 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 14 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 13 nM  Bioactivity Info	TI    LI    LO    TS
CP0360625  Compound Info	(6S,8R)-6-Ethyl-8-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 66 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0407407  Compound Info	6,6-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 68 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 16 nM  Bioactivity Info	TI    LI    LO    TS
CP0379126  Compound Info	7-[bis(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-2H-chromen-2-one    Show/Hide	C14H8F9NO2	2
1	EC50 = 73 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 63 nM  Bioactivity Info	TI    LI    LO    TS
CP0412814  Compound Info	(2S)-2-(methoxymethyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C16H14F6N2O3	2
1	EC50 = 77 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 17 nM  Bioactivity Info	TI    LI    LO    TS
CP0429403  Compound Info	2-chloro-3-methyl-4-(1,1,1-trifluoro-2-hydroxy-5,5-dimethylhex-3-yn-2-yl)benzonitrile    Show/Hide	C16H15ClF3NO	1
1	EC50 = 79.43 nM  Bioactivity Info	TI    LI    LO    TS
CP0475458  Compound Info	2-chloro-3-methyl-4-(1,1,1-trifluoro-2-hydroxy-3,3-dimethylbutan-2-yl)benzonitrile    Show/Hide	C14H15ClF3NO	1
1	EC50 = 79.43 nM  Bioactivity Info	TI    LI    LO    TS
CP0310025  Compound Info	(6R,7S)-7-methyl-4-(trifluoromethyl)-6-(3,3,3-trifluoropropyl)-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H16F6N2O	2
1	EC50 = 82 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 63 nM  Bioactivity Info	TI    LI    LO    TS
CP0433372  Compound Info	6-alkyl, 7-amino-2-quinolinone, 11c    Show/Hide	C13H13F3N2O	3
1	EC50 = 83 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 9 nM  Bioactivity Info	TI    LI    LO    TS
CP0394282  Compound Info	10-methoxy-4-(trifluoromethyl)-1H-isochromeno[3,4-f]quinoline-2,6-dione    Show/Hide	C18H10F3NO4	2
1	EC50 = 90 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0482530  Compound Info	5-(4-hydroxy-2-methylphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H12N2O	2
1	EC50 = 94.8 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 1550.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0373219  Compound Info	10-hydroxy-4-(trifluoromethyl)-1H-isochromeno[3,4-f]quinoline-2,6-dione    Show/Hide	C17H8F3NO4	2
1	EC50 = 97 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0424756  Compound Info	(R)-3-isobutyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C18H18F6N2O2	1
1	EC50 = 98 nM  Bioactivity Info	TI    LI    LO    TS
CP0406506  Compound Info	(R)-2,3,3-Trimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C15H15F3N2O	2
1	EC50 = 99 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 48 nM  Bioactivity Info	TI    LI    LO    TS
CP0374883  Compound Info	6-(propan-2-ylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H13F3N2O	2
1	EC50 = 106 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 16.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0428659  Compound Info	6-[(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H8F6N2O	3
1	EC50 = 108 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 18 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 16 nM  Bioactivity Info	TI    LI    LO    TS
CP0288503  Compound Info	(6S,8R)-8-Ethyl-6-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 119 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 137 nM  Bioactivity Info	TI    LI    LO    TS
CP0458132  Compound Info	2-methyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C13H11F3N2O2	1
1	EC50 = 133 nM  Bioactivity Info	TI    LI    LO    TS
CP0223867  Compound Info	4-Ethyl-8-oxo-6-trifluoromethyl-3,4,8,9-tetrahydro-2H-pyrido[3,2-g]quinoline-1-carbaldehyde    Show/Hide	C16H15F3N2O2	2
1	EC50 = 137 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0146696  Compound Info	Bicalutamide    Show/Hide	C18H14F4N2O4S	7
1	EC50 = 157 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
3	IC50 = 157 nM  Bioactivity Info	TI    LI    LO    TS
4	IC50 = 162 nM  Bioactivity Info	TI    LI    LO    TS
5	IC50 = 300 nM  Bioactivity Info	TI    LI    LO    TS
6	IC50 = 338 nM  Bioactivity Info	TI    LI    LO    TS
7	Ki = 151 nM  Bioactivity Info	TI    LI    LO    TS
CP0342695  Compound Info	6-Ethyl-9-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 158 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0447520  Compound Info	2-chloro-4-(1,1,1-trifluoro-2-hydroxy-3,3-dimethylbutan-2-yl)benzonitrile    Show/Hide	C13H13ClF3NO	1
1	EC50 = 158.49 nM  Bioactivity Info	TI    LI    LO    TS
CP0393742  Compound Info	(R)-2-Methyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C13H11F3N2O	2
1	EC50 = 168 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 7 nM  Bioactivity Info	TI    LI    LO    TS
CP0373222  Compound Info	5,10-dimethoxy-4-methyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C19H17NO4	2
1	EC50 = 184 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0421963  Compound Info	4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C14H10F6N2O2	1
1	EC50 = 190 nM  Bioactivity Info	TI    LI    LO    TS
CP0373228  Compound Info	5-hydroxy-10-methoxy-4-methyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H15NO4	2
1	EC50 = 208 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0375502  Compound Info	5-Ethyl-8-methyl-4-trifluoromethyl-5,6,7,8-tetrahydro-1-oxa-8-aza-anthracen-2-one    Show/Hide	C16H16F3NO2	2
1	EC50 = 209 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10 nM  Bioactivity Info	TI    LI    LO    TS
CP0436364  Compound Info	(R)-3-ethyl-4-isobutyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C18H21F3N2O2	2
1	EC50 = 227 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0391193  Compound Info	(R)-4-allyl-3-methyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C16H15F3N2O2	1
1	EC50 = 228 nM  Bioactivity Info	TI    LI    LO    TS
CP0431638  Compound Info	5-(2,5-difluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H8F2N2O	2
1	EC50 = 229.1 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0482532  Compound Info	5-(4-hydroxy-2-nitrophenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9N3O3	2
1	EC50 = 233 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0394256  Compound Info	9-fluoro-4-methyl-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C17H10FNO3	2
1	EC50 = 240 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0428667  Compound Info	6-[(2,2,3,3,3-pentafluoropropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H8F8N2O	3
1	EC50 = 246 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 17 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 78 nM  Bioactivity Info	TI    LI    LO    TS
CP0456705  Compound Info	(R)-4-ethyl-3-isopropyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C17H19F3N2O2	2
1	EC50 = 272 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0395572  Compound Info	1-[(2S)-3-(3-chlorophenoxy)-2-hydroxy-2-methylpropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H17ClN2O3	2
1	EC50 = 275 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0436360  Compound Info	(R)-3-isopropyl-4-methyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C16H17F3N2O2	1
1	EC50 = 276 nM  Bioactivity Info	TI    LI    LO    TS
CP0394477  Compound Info	(R)-3-ethyl-4-(2-hydroxy-2-methylpropyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C18H21F3N2O3	2
1	EC50 = 300 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0373223  Compound Info	9-hydroxy-10-methoxy-4-methyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H15NO4	2
1	EC50 = 306 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0223868  Compound Info	4-Trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C13H11F3N2O	2
1	EC50 = 317 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 12 nM  Bioactivity Info	TI    LI    LO    TS
CP0402619  Compound Info	(5bR,9aR)-1-Methyl-10-propyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C20H23F3N2O	2
1	EC50 = 324 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0407178  Compound Info	(R)-2,3,3,8-Tetramethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 380 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
CP0392183  Compound Info	5-(3-ethyl-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C14H14N2O	2
1	EC50 = 391 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0424754  Compound Info	(R)-3-ethyl-4-propyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C17H19F3N2O2	2
1	EC50 = 394 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0379130  Compound Info	6-[(2-methylpropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H15F3N2O	3
1	EC50 = 404 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 59 nM  Bioactivity Info	TI    LI    LO    TS
CP0384335  Compound Info	(R)-3-methyl-4-propyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C16H17F3N2O2	1
1	EC50 = 406 nM  Bioactivity Info	TI    LI    LO    TS
CP0424755  Compound Info	(R)-3,4-diethyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C16H17F3N2O2	2
1	EC50 = 410 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0391189  Compound Info	(R)-4-ethyl-3-methyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C15H15F3N2O2	1
1	EC50 = 420 nM  Bioactivity Info	TI    LI    LO    TS
CP0463355  Compound Info	5-(4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H10N2O	2
1	EC50 = 573.2 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 = 2014.9 nM  Bioactivity Info	TI    LI    LO    TS
CP0428660  Compound Info	6-alkyl, 7-amino-2-quinolinone, 11b    Show/Hide	C12H11F3N2O	3
1	EC50 = 593 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0395571  Compound Info	1-[(2S)-2-hydroxy-2-methyl-3-phenoxypropanoyl]-2,3-dihydroindole-4-carbonitrile    Show/Hide	C19H18N2O3	2
1	EC50 = 689 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0427877  Compound Info	7-[(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H8F6N2O	3
1	EC50 = 905 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 21 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0513304  Compound Info	5-(3-chloro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9ClN2O	2
1	EC50 = 909.5 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0463354  Compound Info	5-(2,3-difluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H8F2N2O	2
1	EC50 = 980 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0431632  Compound Info	1-ethyl-5-(2-fluoro-4-hydroxyphenyl)pyrrole-2-carbonitrile    Show/Hide	C13H11FN2O	2
1	EC50 = 1136.4 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0390992  Compound Info	6-(dibutylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C18H23F3N2O	2
1	EC50 = 1283 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 29.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0379122  Compound Info	7-amino-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C10H7F3N2O	3
1	EC50 = 1300 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 407 nM  Bioactivity Info	TI    LI    LO    TS
CP0482529  Compound Info	5-(4-hydroxyphenyl)-1-methyl-3-(trifluoromethyl)pyrrole-2-carbonitrile    Show/Hide	C13H9F3N2O	2
1	EC50 = 1341.7 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0463358  Compound Info	methyl 2-(5-cyano-1-methylpyrrol-2-yl)-5-hydroxybenzoate    Show/Hide	C14H12N2O3	2
1	EC50 = 1450.3 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0468785  Compound Info	5-(3-fluoro-4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9FN2O	2
1	EC50 = 1517.7 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0510662  Compound Info	4-bromo-5-(4-hydroxyphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C12H9BrN2O	2
1	EC50 = 1644.6 nM  Bioactivity Info	TI    LI    LO    TS
2	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0151164  Compound Info	(7S,8R)-8-Ethyl-7-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 1668 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0374643  Compound Info	5-Trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C12H9F3N2O	2
1	EC50 = 1897 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0390987  Compound Info	6-(propylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H13F3N2O	2
1	EC50 = 2022 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 27.5 nM  Bioactivity Info	TI    LI    LO    TS
CP0134234  Compound Info	(7R,8R)-8-Ethyl-7-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 = 2468 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0475459  Compound Info	2,3-dimethyl-4-(1,1,1-trifluoro-2-hydroxypropan-2-yl)benzonitrile    Show/Hide	C12H12F3NO	1
1	EC50 = 2511.89 nM  Bioactivity Info	TI    LI    LO    TS
CP0061327  Compound Info	6-Ethyl-1-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 20 nM  Bioactivity Info	TI    LI    LO    TS
CP0107976  Compound Info	6-Ethyl-1,9-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 216 nM  Bioactivity Info	TI    LI    LO    TS
CP0189599  Compound Info	6-(3,5-Bis-trifluoromethyl-phenyl)-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C21H13F9N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 251 nM  Bioactivity Info	TI    LI    LO    TS
CP0208826  Compound Info	6,6-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 73 nM  Bioactivity Info	TI    LI    LO    TS
CP0390990  Compound Info	6-(dimethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H11F3N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 34 nM  Bioactivity Info	TI    LI    LO    TS
CP0428662  Compound Info	6-amino-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C10H7F3N2O	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
CP0399739  Compound Info	(R)-3-ethyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C14H13F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 84 nM  Bioactivity Info	TI    LI    LO    TS
CP0399740  Compound Info	(R)-3,4-dimethyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C14H13F3N2O2	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0417185  Compound Info	(R)-3-methyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C13H11F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 72 nM  Bioactivity Info	TI    LI    LO    TS
CP0417187  Compound Info	(R)-3-phenyl-4-(2,2,2-trifluoroethyl)-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C20H14F6N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 65 nM  Bioactivity Info	TI    LI    LO    TS
CP0421842  Compound Info	(R)-3-ethyl-4-methyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C15H15F3N2O2	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0436362  Compound Info	10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C12H9F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 1500 nM  Bioactivity Info	TI    LI    LO    TS
CP0449115  Compound Info	(R)-3-phenyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C18H13F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 1480 nM  Bioactivity Info	TI    LI    LO    TS
CP0461130  Compound Info	(R)-3-propyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C15H15F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 113 nM  Bioactivity Info	TI    LI    LO    TS
CP0464181  Compound Info	(R)-4-(cyclopropylmethyl)-3-phenyl-10-(trifluoromethyl)-3,4-dihydro-2H-[1,4]oxazino[2,3-f]quinolin-8(7H)-one    Show/Hide	C22H19F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 45 nM  Bioactivity Info	TI    LI    LO    TS
CP0394087  Compound Info	7H-[1,4]Oxazino[3,2-g]quinolin-7-one based compound, 11a    Show/Hide	C12H9F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 296 nM  Bioactivity Info	TI    LI    LO    TS
CP0431962  Compound Info	1-benzyl-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C19H15F3N2O2	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 224 nM  Bioactivity Info	TI    LI    LO    TS
CP0373221  Compound Info	10-methoxy-4-methyl-5-prop-2-enyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C21H19NO3	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 144 nM  Bioactivity Info	TI    LI    LO    TS
CP0373249  Compound Info	10-methoxy-4,5-dimethyl-1,5-dihydrochromeno[3,4-f]quinolin-2-one    Show/Hide	C19H17NO3	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 62 nM  Bioactivity Info	TI    LI    LO    TS
CP0432039  Compound Info	10-methoxy-4-(trifluoromethyl)-1,6-dihydroisochromeno[3,4-f]quinolin-2-one    Show/Hide	C18H12F3NO3	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 78 nM  Bioactivity Info	TI    LI    LO    TS
CP0432041  Compound Info	9-methoxy-4-methyl-1H-chromeno[3,4-f]quinoline-2,5-dione    Show/Hide	C18H13NO4	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 48 nM  Bioactivity Info	TI    LI    LO    TS
CP0284048  Compound Info	4-chloro-13-(2-chlorophenyl)-6-methyl-11-oxo-8-thia-3,10-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5-tetraene-5-carbonitrile    Show/Hide	C18H11Cl2N3OS	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0090808  Compound Info	3-(3-fluorophenyl)-1-(4-methylphenyl)-3-(4-nitroanilino)propan-1-one    Show/Hide	C22H19FN2O3	2
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 140 nM  Bioactivity Info	TI    LI    LO    TS
CP0570938  Compound Info	4-(1,1,1-trifluoro-2,3-dihydroxypropan-2-yl)-2-(trifluoromethyl)benzonitrile    Show/Hide	C11H7F6NO2	1
1	EC50 = 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0392182  Compound Info	1-(cyanomethyl)-5-(2-fluoro-4-hydroxyphenyl)pyrrole-2-carbonitrile    Show/Hide	C13H8FN3O	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0392186  Compound Info	5-(4-hydroxy-2-methylsulfonylphenyl)-1-methylpyrrole-2-carbonitrile    Show/Hide	C13H12N2O3S	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0392187  Compound Info	2-[2-cyano-5-(2-fluoro-4-hydroxyphenyl)pyrrol-1-yl]acetic acid    Show/Hide	C13H9FN2O3	1
1	EC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0107746  Compound Info	(R)-8-Ethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0122738  Compound Info	(R)-8-Ethyl-7,7-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
CP0168794  Compound Info	(R)-8-Propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
CP0187275  Compound Info	8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0217015  Compound Info	(S)-8-Isopropyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 25 nM  Bioactivity Info	TI    LI    LO    TS
CP0291483  Compound Info	(R)-7,7,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 24 nM  Bioactivity Info	TI    LI    LO    TS
CP0360576  Compound Info	(R)-7,7,8-Triethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C19H23F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 48 nM  Bioactivity Info	TI    LI    LO    TS
CP0361134  Compound Info	2-hydroxy-N-[2-hydroxy-4-nitro-3-(trifluoromethyl)phenyl]-2-methylpropanamide    Show/Hide	C11H11F3N2O5	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
CP0394271  Compound Info	(7S,8R)-7,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	EC50 < 10000 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 33 nM  Bioactivity Info	TI    LI    LO    TS
CP0460051  Compound Info	8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinoline-2-carbonitrile    Show/Hide	C16H14F3N3	1
1	IC50 = 9 nM  Bioactivity Info	TI    LI    LO    TS
CP0428661  Compound Info	8-ethyl-4-(trifluoromethyl)-1H,2H,6H,7H,8H,9H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H15F3N2O	2
1	IC50 = 14 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 11 nM  Bioactivity Info	TI    LI    LO    TS
CP0040191  Compound Info	2-Hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-phenyl)-propionamide    Show/Hide	C11H11F3N2O4	2
1	IC50 = 15 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
CP0215260  Compound Info	1,8,8,9-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 19 nM  Bioactivity Info	TI    LI    LO    TS
CP0316819  Compound Info	6,8,8,10-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
CP0419190  Compound Info	8-Fluoro-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C15H14F4N2	1
1	IC50 = 22 nM  Bioactivity Info	TI    LI    LO    TS
CP0041854  Compound Info	6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclopropa[1,2]pregna-4,6-dien-17-yl acetate    Show/Hide	C24H29ClO4	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0276572  Compound Info	8-Ethyl-8-methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0328159  Compound Info	6,8,8,10-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H17F3N2O	1
1	IC50 = 23 nM  Bioactivity Info	TI    LI    LO    TS
CP0041439  Compound Info	8-Ethyl-1,8,9-trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	1
1	IC50 = 24 nM  Bioactivity Info	TI    LI    LO    TS
CP0449258  Compound Info	(5bR,9aS)-9,9-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
CP0041137  Compound Info	6,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	1
1	IC50 = 26 nM  Bioactivity Info	TI    LI    LO    TS
CP0378067  Compound Info	(5bR,9aS)-1,9,9,10-Tetramethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C20H23F3N2O	1
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0102250  Compound Info	8,8-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0332143  Compound Info	6-Ethyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0352184  Compound Info	3a,10-Dimethyl-7-trifluoromethyl-1,2,3a,4,5,10-hexahydro-3H-10,11b-diaza-cyclopenta[a]anthracen-9-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
CP0163588  Compound Info	8,8-dimethyl-4-(trifluoromethyl)-1H,2H,8H,9H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C15H13F3N2O	3
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
2	IC50 = 58 nM  Bioactivity Info	TI    LI    LO    TS
3	Ki = 73 nM  Bioactivity Info	TI    LI    LO    TS
CP0427879  Compound Info	6-[(2,2-dimethylpropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H17F3N2O	2
1	IC50 = 27 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 56 nM  Bioactivity Info	TI    LI    LO    TS
CP0106239  Compound Info	6,8,8-Trimethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H15F3N2O	1
1	IC50 = 28 nM  Bioactivity Info	TI    LI    LO    TS
CP0220774  Compound Info	7,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	1
1	IC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0377716  Compound Info	8-Chloro-2,2,4-trimethyl-6-trifluoromethyl-1,2-dihydro-pyrido[3,2-g]quinoline    Show/Hide	C16H14ClF3N2	1
1	IC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0453376  Compound Info	8-Chloro-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C15H14ClF3N2	1
1	IC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0433371  Compound Info	7-(methylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C11H9F3N2O	2
1	IC50 = 30 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 83 nM  Bioactivity Info	TI    LI    LO    TS
CP0237260  Compound Info	1,6,8,8,10-Pentamethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	1
1	IC50 = 31 nM  Bioactivity Info	TI    LI    LO    TS
CP0442685  Compound Info	8-Fluoro-2,2,4-trimethyl-6-trifluoromethyl-1,2-dihydro-pyrido[3,2-g]quinoline    Show/Hide	C16H14F4N2	1
1	IC50 = 31 nM  Bioactivity Info	TI    LI    LO    TS
CP0379125  Compound Info	7-(propylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H13F3N2O	2
1	IC50 = 32 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 37 nM  Bioactivity Info	TI    LI    LO    TS
CP0295804  Compound Info	1,6,8,8-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H17F3N2O	1
1	IC50 = 34 nM  Bioactivity Info	TI    LI    LO    TS
CP0041438  Compound Info	6'-trifluoromethylspiro[cyclohexane-1,2'-(1',2',3',4',8',9'-hexahydropyrido[3,2-g]quinoline)]-8'-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 35 nM  Bioactivity Info	TI    LI    LO    TS
CP0405760  Compound Info	7-(ethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H11F3N2O	2
1	IC50 = 35 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 29 nM  Bioactivity Info	TI    LI    LO    TS
CP0374711  Compound Info	(5bR,9aR)-1,10-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 36 nM  Bioactivity Info	TI    LI    LO    TS
CP0130624  Compound Info	4,6,8,8-Tetramethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H18N2O	1
1	IC50 = 36 nM  Bioactivity Info	TI    LI    LO    TS
CP0246106  Compound Info	1,8,8-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C16H17F3N2O	1
1	IC50 = 36 nM  Bioactivity Info	TI    LI    LO    TS
CP0038813  Compound Info	(1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-en-5-one    Show/Hide	C21H30O2	1
1	IC50 = 37 nM  Bioactivity Info	TI    LI    LO    TS
CP0216906  Compound Info	8-Methyl-8-propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
CP0442163  Compound Info	6-(cyclopentylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H15F3N2O	2
1	IC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 74 nM  Bioactivity Info	TI    LI    LO    TS
CP0442166  Compound Info	7-[ethyl(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H12F6N2O	2
1	IC50 = 42 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0428663  Compound Info	7-(cyclobutylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H13F3N2O	2
1	IC50 = 43 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 161 nM  Bioactivity Info	TI    LI    LO    TS
CP0435851  Compound Info	(2S)-2-(4-methylphenyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C21H16F6N2O2	1
1	IC50 = 44 nM  Bioactivity Info	TI    LI    LO    TS
CP0464622  Compound Info	8,8,9-Trimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinoline-2-carbonitrile    Show/Hide	C17H16F3N3	1
1	IC50 = 45 nM  Bioactivity Info	TI    LI    LO    TS
CP0101361  Compound Info	1,6,8,8,9-Pentamethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 46 nM  Bioactivity Info	TI    LI    LO    TS
CP0292537  Compound Info	7-Ethyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 46 nM  Bioactivity Info	TI    LI    LO    TS
CP0377889  Compound Info	(5bR,7S,9aR)-1,7-Dimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 48 nM  Bioactivity Info	TI    LI    LO    TS
CP0036037  Compound Info	8-Ethyl-1,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 48 nM  Bioactivity Info	TI    LI    LO    TS
CP0379127  Compound Info	7-[(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-2H-chromen-2-one    Show/Hide	C12H7F6NO2	1
1	IC50 = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0375432  Compound Info	(5bR,9aR)-5b,9,9-Trimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C19H21F3N2O	1
1	IC50 = 51 nM  Bioactivity Info	TI    LI    LO    TS
CP0433826  Compound Info	(2R)-2-benzyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C21H16F6N2O2	1
1	IC50 = 51 nM  Bioactivity Info	TI    LI    LO    TS
CP0454739  Compound Info	(5bR,9aR)-1,5b,10-Trimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C19H21F3N2O	1
1	IC50 = 53 nM  Bioactivity Info	TI    LI    LO    TS
CP0378063  Compound Info	(5bR,7S,9aR)-1,7,10-Trimethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C19H21F3N2O	1
1	IC50 = 54 nM  Bioactivity Info	TI    LI    LO    TS
CP0374712  Compound Info	(R)-1,2,3,3,8-Pentamethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 56 nM  Bioactivity Info	TI    LI    LO    TS
CP0440277  Compound Info	8-Methyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C13H11F3N2O	1
1	IC50 = 56 nM  Bioactivity Info	TI    LI    LO    TS
CP0379129  Compound Info	7-(propan-2-ylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H13F3N2O	2
1	IC50 = 56 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 79 nM  Bioactivity Info	TI    LI    LO    TS
CP0368335  Compound Info	6,7,7,8,8-Pentamethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	1
1	IC50 = 57 nM  Bioactivity Info	TI    LI    LO    TS
CP0444507  Compound Info	7-[(2,2,3,3,3-pentafluoropropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C13H8F8N2O	2
1	IC50 = 58 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 36 nM  Bioactivity Info	TI    LI    LO    TS
CP0408426  Compound Info	8-Methanesulfinyl-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H17F3N2OS	1
1	IC50 = 63 nM  Bioactivity Info	TI    LI    LO    TS
CP0427881  Compound Info	7-(butylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H15F3N2O	2
1	IC50 = 67 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 50 nM  Bioactivity Info	TI    LI    LO    TS
CP0088296  Compound Info	6,7,8,8-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H17F3N2O	1
1	IC50 = 68 nM  Bioactivity Info	TI    LI    LO    TS
CP0379059  Compound Info	8-Bromo-1,2,2-trimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H16BrF3N2	1
1	IC50 = 72 nM  Bioactivity Info	TI    LI    LO    TS
CP0406515  Compound Info	8-Bromo-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C15H14BrF3N2	1
1	IC50 = 72 nM  Bioactivity Info	TI    LI    LO    TS
CP0198388  Compound Info	1,6,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 73 nM  Bioactivity Info	TI    LI    LO    TS
CP0433370  Compound Info	7-[(2-methylpropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H15F3N2O	2
1	IC50 = 74 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 65 nM  Bioactivity Info	TI    LI    LO    TS
CP0442165  Compound Info	6-alkyl, 7-amino-2-quinolinone, 11a    Show/Hide	C11H9F3N2O	2
1	IC50 = 76 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 30 nM  Bioactivity Info	TI    LI    LO    TS
CP0272980  Compound Info	7,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 83 nM  Bioactivity Info	TI    LI    LO    TS
CP0442168  Compound Info	7-[(2,2-dimethylpropyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H17F3N2O	2
1	IC50 = 98 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 134 nM  Bioactivity Info	TI    LI    LO    TS
CP0379123  Compound Info	6-(ethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H11F3N2O	1
1	IC50 = 111 nM  Bioactivity Info	TI    LI    LO    TS
CP0428664  Compound Info	7-[(2-methylbut-3-en-2-yl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H15F3N2O	2
1	IC50 = 122 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 118 nM  Bioactivity Info	TI    LI    LO    TS
CP0428666  Compound Info	7-(cyclopentylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H15F3N2O	2
1	IC50 = 149 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 1000 nM  Bioactivity Info	TI    LI    LO    TS
CP0267990  Compound Info	6,8,8,9-Tetramethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H17F3N2O	1
1	IC50 = 156 nM  Bioactivity Info	TI    LI    LO    TS
CP0141600  Compound Info	6-Isopropyl-8,8-dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H21F3N2O	1
1	IC50 = 159 nM  Bioactivity Info	TI    LI    LO    TS
CP0161755  Compound Info	(6R,7S)-6,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 164 nM  Bioactivity Info	TI    LI    LO    TS
CP0393389  Compound Info	8-Fluoro-1,2,2-trimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H16F4N2	1
1	IC50 = 172 nM  Bioactivity Info	TI    LI    LO    TS
CP0380168  Compound Info	1,8-Dimethyl-5-trifluoromethyl-1,2,3,8-tetrahydro-pyrrolo[3,2-g]quinolin-7-one    Show/Hide	C14H13F3N2O	1
1	IC50 = 197 nM  Bioactivity Info	TI    LI    LO    TS
CP0379128  Compound Info	7-[(2-methylbutan-2-yl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H17F3N2O	2
1	IC50 = 209 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 110 nM  Bioactivity Info	TI    LI    LO    TS
CP0457283  Compound Info	2,2-Dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C15H15F3N2	1
1	IC50 = 212 nM  Bioactivity Info	TI    LI    LO    TS
CP0379131  Compound Info	6-alkyl, 7-alkylamino-2-quinolinone, 11h    Show/Hide	C14H12F6N2O	2
1	IC50 = 216 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 157 nM  Bioactivity Info	TI    LI    LO    TS
CP0407064  Compound Info	(5bR,9aR)-1-Ethyl-4-trifluoromethyl-1,5b,6,7,8,9,9a,10-octahydro-pyrido[2,3-b]carbazol-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 230 nM  Bioactivity Info	TI    LI    LO    TS
CP0453816  Compound Info	2,2,4,10-Tetramethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C17H19F3N2	1
1	IC50 = 244 nM  Bioactivity Info	TI    LI    LO    TS
CP0454002  Compound Info	8-Chloro-1,2,2-trimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H16ClF3N2	1
1	IC50 = 251 nM  Bioactivity Info	TI    LI    LO    TS
CP0063640  Compound Info	5-(3-Chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H22ClNO	1
1	IC50 = 253 nM  Bioactivity Info	TI    LI    LO    TS
CP0428669  Compound Info	7-(benzylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C17H13F3N2O	2
1	IC50 = 294 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 163 nM  Bioactivity Info	TI    LI    LO    TS
CP0428668  Compound Info	6-alkyl, 7-alkylamino-2-quinolinone, 11f    Show/Hide	C15H17F3N2O	2
1	IC50 = 301 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 650 nM  Bioactivity Info	TI    LI    LO    TS
CP0163667  Compound Info	2,2,4-Trimethyl-5-(3-trifluoromethyl-phenyl)-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22F3NO	1
1	IC50 = 315 nM  Bioactivity Info	TI    LI    LO    TS
CP0087434  Compound Info	3a-Methyl-7-trifluoromethyl-1,2,3a,4,5,10-hexahydro-3H-10,11b-diaza-cyclopenta[a]anthracen-9-one    Show/Hide	C17H17F3N2O	1
1	IC50 = 325 nM  Bioactivity Info	TI    LI    LO    TS
CP0494337  Compound Info	8-(Butane-1-sulfinyl)-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C19H23F3N2OS	1
1	IC50 = 335 nM  Bioactivity Info	TI    LI    LO    TS
CP0437428  Compound Info	8-Chloro-1,2,2,4-tetramethyl-6-trifluoromethyl-1,2-dihydro-pyrido[3,2-g]quinoline    Show/Hide	C17H16ClF3N2	1
1	IC50 = 336 nM  Bioactivity Info	TI    LI    LO    TS
CP0471355  Compound Info	(2S)-2-phenyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C20H14F6N2O2	1
1	IC50 = 340 nM  Bioactivity Info	TI    LI    LO    TS
CP0205607  Compound Info	5-(3-Bromo-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H22BrNO	1
1	IC50 = 401 nM  Bioactivity Info	TI    LI    LO    TS
CP0392963  Compound Info	2,2-Dimethyl-6,8-bis-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H14F6N2	1
1	IC50 = 467 nM  Bioactivity Info	TI    LI    LO    TS
CP0379056  Compound Info	8-Methanesulfonyl-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H17F3N2O2S	1
1	IC50 = 479 nM  Bioactivity Info	TI    LI    LO    TS
CP0235429  Compound Info	5-(4-Bromo-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H22BrNO	1
1	IC50 = 481 nM  Bioactivity Info	TI    LI    LO    TS
CP0473748  Compound Info	17-[(6S)-6-Methyl-5,6-dihydropyridin-2(1H)-one-6-yl]-androst-4-ene-3-one    Show/Hide	C25H35NO2	1
1	IC50 = 500 nM  Bioactivity Info	TI    LI    LO    TS
CP0380719  Compound Info	N-[2,2-dimethyl-6-(trifluoromethyl)-3,4-dihydro-1H-pyrido[3,2-g]quinolin-8-yl]methanesulfonamide    Show/Hide	C16H18F3N3O2S	1
1	IC50 = 503 nM  Bioactivity Info	TI    LI    LO    TS
CP0442164  Compound Info	6-alkyl, 7-alkylamino-2-quinolinone, 11g    Show/Hide	C13H13F3N2O	2
1	IC50 = 504 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 869 nM  Bioactivity Info	TI    LI    LO    TS
CP0427880  Compound Info	7-(cyclohexylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C16H17F3N2O	2
1	IC50 = 507 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 1000 nM  Bioactivity Info	TI    LI    LO    TS
CP0379132  Compound Info	7-[propyl(2,2,2-trifluoroethyl)amino]-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C15H14F6N2O	2
1	IC50 = 549 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 241 nM  Bioactivity Info	TI    LI    LO    TS
CP0412812  Compound Info	(2S)-2-(3-methylphenyl)-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-3,6-dihydro-2H-pyrido[3,2-g][1,4]benzoxazin-7-one    Show/Hide	C21H16F6N2O2	1
1	IC50 = 574 nM  Bioactivity Info	TI    LI    LO    TS
CP0428665  Compound Info	7-(diethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C14H15F3N2O	2
1	IC50 = 591 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 463 nM  Bioactivity Info	TI    LI    LO    TS
CP0379024  Compound Info	N-[2,2-dimethyl-6-(trifluoromethyl)-3,4-dihydro-1H-pyrido[3,2-g]quinolin-8-yl]-N-methylsulfonylmethanesulfonamide    Show/Hide	C17H20F3N3O4S2	1
1	IC50 = 636 nM  Bioactivity Info	TI    LI    LO    TS
CP0193631  Compound Info	2,2,4-Trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H23NO	1
1	IC50 = 650 nM  Bioactivity Info	TI    LI    LO    TS
CP0442169  Compound Info	6-alkyl, 7-alkylamino-2-quinolinone, 11e    Show/Hide	C14H15F3N2O	2
1	IC50 = 674 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 641 nM  Bioactivity Info	TI    LI    LO    TS
CP0377719  Compound Info	8-Chloro-2,2,4,10-tetramethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C17H18ClF3N2	1
1	IC50 = 675 nM  Bioactivity Info	TI    LI    LO    TS
CP0043208  Compound Info	1-Ethyl-6,8,8-trimethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 692 nM  Bioactivity Info	TI    LI    LO    TS
CP0437332  Compound Info	1,2,2-Trimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H17F3N2	1
1	IC50 = 725 nM  Bioactivity Info	TI    LI    LO    TS
CP0050558  Compound Info	2,2,4-Trimethyl-5-phenyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H23NO	1
1	IC50 = 745 nM  Bioactivity Info	TI    LI    LO    TS
CP0414948  Compound Info	2,2-Dimethyl-8-methylsulfanyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C16H17F3N2S	1
1	IC50 = 751 nM  Bioactivity Info	TI    LI    LO    TS
CP0414926  Compound Info	8-Bromo-2,2,4,10-tetramethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C17H18BrF3N2	1
1	IC50 = 785 nM  Bioactivity Info	TI    LI    LO    TS
CP0301665  Compound Info	5-[1-(3-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22FNO	1
1	IC50 = 795 nM  Bioactivity Info	TI    LI    LO    TS
CP0537884  Compound Info	2,2-Dimethyl-8-(2,2,2-trifluoro-ethylsulfanyl)-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C17H16F6N2S	1
1	IC50 = 889 nM  Bioactivity Info	TI    LI    LO    TS
CP0146748  Compound Info	5-[1-(3,4-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H21F2NO	1
1	IC50 = 916 nM  Bioactivity Info	TI    LI    LO    TS
CP0200882  Compound Info	5-(3,4-Dichloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H21Cl2NO	1
1	IC50 = 946 nM  Bioactivity Info	TI    LI    LO    TS
CP0104425  Compound Info	2,2,4-Trimethyl-5-[1-o-tolyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C27H25NO	1
1	IC50 = 1062 nM  Bioactivity Info	TI    LI    LO    TS
CP0250549  Compound Info	5-(3,5-Dichloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H21Cl2NO	1
1	IC50 = 1089 nM  Bioactivity Info	TI    LI    LO    TS
CP0405090  Compound Info	8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinolin-2-ylamine    Show/Hide	C15H16F3N3	1
1	IC50 = 1159 nM  Bioactivity Info	TI    LI    LO    TS
CP0379124  Compound Info	7-(dimethylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one    Show/Hide	C12H11F3N2O	2
1	IC50 = 1160 nM  Bioactivity Info	TI    LI    LO    TS
2	Ki = 761 nM  Bioactivity Info	TI    LI    LO    TS
CP0057358  Compound Info	5-(3-Fluoro-4-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H24FNO	1
1	IC50 = 1220 nM  Bioactivity Info	TI    LI    LO    TS
CP0051650  Compound Info	5-(3-Bromo-5-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H24BrNO	1
1	IC50 = 1236 nM  Bioactivity Info	TI    LI    LO    TS
CP0184222  Compound Info	2,2,4-Trimethyl-5-p-tolyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H25NO	1
1	IC50 = 1239 nM  Bioactivity Info	TI    LI    LO    TS
CP0134558  Compound Info	5-(4-Chloro-3-methyl-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H24ClNO	1
1	IC50 = 1426 nM  Bioactivity Info	TI    LI    LO    TS
CP0447848  Compound Info	8-Fluoro-2,2,4,10-tetramethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C17H18F4N2	1
1	IC50 = 1448 nM  Bioactivity Info	TI    LI    LO    TS
CP0185464  Compound Info	5-(4-Chloro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H22ClNO	1
1	IC50 = 1550 nM  Bioactivity Info	TI    LI    LO    TS
CP0134269  Compound Info	5-[1-(2,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H21F2NO	1
1	IC50 = 1600 nM  Bioactivity Info	TI    LI    LO    TS
CP0454276  Compound Info	8-Butylsulfanyl-2,2-dimethyl-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrido[3,2-g]quinoline    Show/Hide	C19H23F3N2S	1
1	IC50 = 1866 nM  Bioactivity Info	TI    LI    LO    TS
CP0411966  Compound Info	17-[(6R)-6-Methyl-5,6-dihydropyridin-2(1H)-one-6-yl]-androst-4-ene-3-one    Show/Hide	C25H35NO2	1
1	IC50 = 2000 nM  Bioactivity Info	TI    LI    LO    TS
CP0411967  Compound Info	17-[(6R)-6-Methyl-5,6-dihydropyridin-2(1H)-one-6-yl]-androst-5-ene-3beta-ol    Show/Hide	C25H37NO2	1
1	IC50 = 2000 nM  Bioactivity Info	TI    LI    LO    TS
CP0051168  Compound Info	5-(4-Chloro-3-fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C25H21ClFNO	1
1	IC50 = 2205 nM  Bioactivity Info	TI    LI    LO    TS
CP0259897  Compound Info	1,6,8,8,10-Pentamethyl-4-trifluoromethyl-8,9-dihydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C18H19F3N2O	1
1	IC50 = 2413 nM  Bioactivity Info	TI    LI    LO    TS
CP0428431  Compound Info	17-[(6S)-6-Methyl-5,6-dihydropyridin-2(1H)-one-6-yl]-androst-5-ene-3beta-ol    Show/Hide	C25H37NO2	1
1	IC50 = 3000 nM  Bioactivity Info	TI    LI    LO    TS
CP0538402  Compound Info	(8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinolin-2-yl)-(4-methoxy-benzyl)-amine    Show/Hide	C23H24F3N3O	1
1	IC50 = 3217 nM  Bioactivity Info	TI    LI    LO    TS
CP0208002  Compound Info	(6S,7S)-6,7,8,8-Tetramethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2-g]quinolin-2-one    Show/Hide	C17H19F3N2O	1
1	IC50 = 7042 nM  Bioactivity Info	TI    LI    LO    TS
CP0408608  Compound Info	(8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinolin-2-yl)-dimethyl-amine    Show/Hide	C17H20F3N3	1
1	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0409720  Compound Info	(8,8-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-pyrido[3,2-g]quinolin-2-yl)-methyl-amine    Show/Hide	C16H18F3N3	1
1	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0309228  Compound Info	3-methyl-1-(2,2,2-trifluoroethyl)-9-(trifluoromethyl)-1H,2H,3H,6H,7H-quinolino[7,6-b][1,4]oxazin-7-one    Show/Hide	C15H12F6N2O2	1
1	IC50 > 10000 nM  Bioactivity Info	TI    LI    LO    TS
CP0060594  Compound Info	WAY-362450    Show/Hide	C25H24F2N2O3	1
1	IC50 = 10000 nM  Bioactivity Info	TI    LI    LO    TS

Compound ID	Compound Name	Compound Formula
CP0134269  Compound Info	5-[1-(2,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H21F2NO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0146748  Compound Info	5-[1-(3,4-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H21F2NO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0193631  Compound Info	2,2,4-Trimethyl-5-[1-phenyl-meth-(Z)-ylidene]-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H23NO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0256867  Compound Info	12-Episcalarin    Show/Hide	C27H40O5	1
1	IC50 = 75100 nM	TI    LI    LO    TS
CP0268369  Compound Info	5-[1-(2-Chloro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22ClNO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0289306  Compound Info	(R)-sargachromenol    Show/Hide	C27H36O4	1
1	IC50 = 45000 nM	TI    LI    LO    TS
CP0301665  Compound Info	5-[1-(3-Fluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22FNO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0303823  Compound Info	5-[1-(2,6-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H21F2NO	1
1	IC50 = 220 nM	TI    LI    LO    TS
CP0334888  Compound Info	5-[1-(2-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22BrNO	1
1	IC50 > 10000 nM	TI    LI    LO    TS
CP0345741  Compound Info	12-O-deacetyl-12-epi-scalarin    Show/Hide	C25H38O4	1
1	IC50 = 77200 nM	TI    LI    LO    TS
CP0392067  Compound Info	(1R,5bR,11aS,13R,13aS,13bS)-1-hydroxy-5b,8,8,11a,13a-pentamethyl-1,3,5,5a,5b,6,7,7a,8,9,10,11,11a,11b,12,13,13a,13b-octadecahydrochryseno[2,1-c]furan-13-yl acetate    Show/Hide	C27H42O4	1
1	IC50 = 98500 nM	TI    LI    LO    TS
CP0408425  Compound Info	(1R,5bR,11aS,13R,13aS,13bS)-1-methoxy-5b,8,8,11a,13a-pentamethyl-1,3,5,5a,5b,6,7,7a,8,9,10,11,11a,11b,12,13,13a,13b-octadecahydrochryseno[2,1-c]furan-13-ol    Show/Hide	C26H42O3	1
1	IC50 = 86900 nM	TI    LI    LO    TS
CP0439641  Compound Info	(1R,5bS,11aS,13R,13aS,13bS)-5b-(hydroxymethyl)-8,8,11a,13a-tetramethyl-1,3,5,5a,5b,6,7,7a,8,9,10,11,11a,11b,12,13,13a,13b-octadecahydrochryseno[2,1-c]furan-1,13-diol    Show/Hide	C25H40O4	1
1	IC50 > 100000 nM	TI    LI    LO    TS
CP0496783  Compound Info	((1R,5bS,11aS,13R,13aS,13bS)-1,13-dihydroxy-8,8,11a,13a-tetramethyl-1,3,5,5a,5b,6,7,7a,8,9,10,11,11a,11b,12,13,13a,13b-octadecahydrochryseno[2,1-c]furan-5b-yl)methyl acetate    Show/Hide	C27H42O5	1
1	IC50 = 29200 nM	TI    LI    LO    TS
CP0531862  Compound Info	5-[1-(4-Bromo-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene    Show/Hide	C26H22BrNO	1
1	IC50 > 10000 nM	TI    LI    LO    TS