General Information of the Cell Line
Cell Line ID
CL000154
Cell Line Name
HEK293-EBNA1-6E
Synonyms
HEK 293EBNA1-6E
HEK293-6E
HEK2936E
293-6E
293FEt-clone 6E
Category
Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_HF20
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT03627, Catechol O-methyltransferase
Compound ID Compound Name Compound Formula
CP0080125
5-(4-methylphenyl)sulfonylquinolin-8-ol
   Show/Hide
C16H13NO3S
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0438323
7-fluoro-5-(4-methylphenyl)sulfonylquinolin-8-ol
   Show/Hide
C16H12FNO3S
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0534904
5-cyclopentylsulfonylquinolin-8-ol
   Show/Hide
C14H15NO3S
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0521500
5-[4-(trifluoromethyl)phenyl]sulfonylquinolin-8-ol
   Show/Hide
C16H10F3NO3S
 1
1
IC50 = 1258.93 nM
   TI
   LI
   LO
   TS
CP0159103
7-fluoro-5-pyrrolidin-1-ylsulfonylquinolin-8-ol
   Show/Hide
C13H13FN2O3S
 1
1
IC50 = 1584.89 nM
   TI
   LI
   LO
   TS
CP0404794
7-fluoro-5-(4-fluorophenyl)sulfonylquinolin-8-ol
   Show/Hide
C15H9F2NO3S
 1
1
IC50 = 1584.89 nM
   TI
   LI
   LO
   TS
CP0438319
5-ethylsulfonylquinolin-8-ol
   Show/Hide
C11H11NO3S
 1
1
IC50 = 1584.89 nM
   TI
   LI
   LO
   TS
CP0387334
5-(2-benzylpyrrolidin-1-yl)sulfonylquinolin-8-ol
   Show/Hide
C20H20N2O3S
 1
1
IC50 = 1995.26 nM
   TI
   LI
   LO
   TS
CP0476687
5-pyrrolidin-1-ylsulfonylquinolin-8-ol
   Show/Hide
C13H14N2O3S
 1
1
IC50 = 1995.26 nM
   TI
   LI
   LO
   TS
CP0427211
5-cyclopentylsulfonyl-7-fluoroquinolin-8-ol
   Show/Hide
C14H14FNO3S
 1
1
IC50 = 2511.89 nM
   TI
   LI
   LO
   TS
CP0484717
7-methyl-5-pyrrolidin-1-ylsulfonylquinolin-8-ol
   Show/Hide
C14H16N2O3S
 1
1
IC50 = 3162.28 nM
   TI
   LI
   LO
   TS
CP0519742
7-chloro-5-pyrrolidin-1-ylsulfonylquinolin-8-ol
   Show/Hide
C13H13ClN2O3S
 1
1
IC50 = 3162.28 nM
   TI
   LI
   LO
   TS
CP0438321
7-fluoro-5-[4-(trifluoromethyl)phenyl]sulfonylquinolin-8-ol
   Show/Hide
C16H9F4NO3S
 1
1
IC50 = 6309.57 nM
   TI
   LI
   LO
   TS
CP0483087
7-chloro-5-cyclopentylsulfonylquinolin-8-ol
   Show/Hide
C14H14ClNO3S
 1
1
IC50 = 7943.28 nM
   TI
   LI
   LO
   TS
CP0412358
7-chloro-5-(4-fluorophenyl)sulfonylquinolin-8-ol
   Show/Hide
C15H9ClFNO3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0438325
5-cyclopentylsulfonyl-7-(trifluoromethyl)quinolin-8-ol
   Show/Hide
C15H14F3NO3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0438326
7-chloro-5-(4-methylphenyl)sulfonylquinolin-8-ol
   Show/Hide
C16H12ClNO3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0476688
5-(4-methylphenyl)sulfonyl-7-(trifluoromethyl)quinolin-8-ol
   Show/Hide
C17H12F3NO3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0567266
7-bromo-5-(4-methylphenyl)sulfonylquinolin-8-ol
   Show/Hide
C16H12BrNO3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0355617
2-[(2,4-dichlorophenyl)methyl]-7-hydroxy-3,4-dihydro-1H-pyrido[1,2-a]pyrazin-8-one
   Show/Hide
C15H14Cl2N2O2
 1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
CP0437962
2-[(2,6-dimethylphenyl)methyl]-7-hydroxy-3,4-dihydro-1H-pyrido[1,2-a]pyrazin-8-one
   Show/Hide
C17H20N2O2
 1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
CP0437965
2-[(2-chlorophenyl)methyl]-7-hydroxy-3,4-dihydro-1H-pyrido[1,2-a]pyrazin-8-one
   Show/Hide
C15H15ClN2O2
 1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
CP0474014
2-[(2-chloro-6-fluorophenyl)methyl]-7-hydroxy-3,4-dihydro-1H-pyrido[1,2-a]pyrazin-8-one
   Show/Hide
C15H14ClFN2O2
 1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
CP0556289
2-benzyl-7-hydroxy-3,4-dihydro-1H-pyrido[1,2-a]pyrazin-8-one
   Show/Hide
C15H16N2O2
 1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -