General Information of the Cell Line
Cell Line ID
CL000750
Cell Line Name
PrecisION hnAChR alpha7/ric3-HEK
Synonyms
PrecisION hnAChR alpha7/ric3
Category
Transformed cell line
Organism
Homo sapiens (Human)
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT01846, Neuronal acetylcholine receptor subunit alpha-7
Compound ID Compound Name Compound Formula
CP0000479
(1S,5R)-7-pyridin-3-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H16N2
 1
1
Ki = 1.2 nM
   TI
   LI
   LO
   TS
CP0001444
(1R,5S)-7-pyridin-3-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H16N2
 1
1
Ki = 1.3 nM
   TI
   LI
   LO
   TS
CP0000799
3-pyridin-3-yl-3,7-diazabicyclo[3.3.1]nonane
   Show/Hide
C12H17N3
 1
1
Ki = 1.6 nM
   TI
   LI
   LO
   TS
CP0001445
(1S,5R)-7-(5-fluoropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15FN2
 1
1
Ki = 1.6 nM
   TI
   LI
   LO
   TS
CP0000786
(1R,5S)-7-(5-fluoropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15FN2
 1
1
Ki = 3.3 nM
   TI
   LI
   LO
   TS
CP0637839
7-(5-Fluoropyridin-3-yl)-3-azabicyclo[3.3.1]non-7-ene
   Show/Hide
C13H15FN2
 1
1
Ki = 3.6 nM
   TI
   LI
   LO
   TS
CP0633537
rac-7-(Pyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H16N2
 1
1
Ki = 4 nM
   TI
   LI
   LO
   TS
CP0000946
7-(5-methoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H18N2O
 1
1
Ki = 4.6 nM
   TI
   LI
   LO
   TS
CP0008520
7-[5-(4-fluorophenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H19FN2O
 1
1
Ki = 7.2 nM
   TI
   LI
   LO
   TS
CP0000952
7-[5-(3-methoxyphenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C20H22N2O2
 1
1
Ki = 13 nM
   TI
   LI
   LO
   TS
CP0005737
7-[5-(3-chlorophenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H19ClN2O
 1
1
Ki = 13 nM
   TI
   LI
   LO
   TS
CP0003288
7-(5-chloropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15ClN2
 1
1
Ki = 15 nM
   TI
   LI
   LO
   TS
CP0000950
3-methyl-7-(5-phenoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C20H22N2O
 1
1
Ki = 17 nM
   TI
   LI
   LO
   TS
CP0000935
7-pyrimidin-5-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C12H15N3
 1
1
Ki = 19 nM
   TI
   LI
   LO
   TS
CP0000937
7-(6-fluoropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15FN2
 1
1
Ki = 20 nM
   TI
   LI
   LO
   TS
CP0000942
7-(5-phenoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H20N2O
 1
1
Ki = 22 nM
   TI
   LI
   LO
   TS
CP0001667
7-[5-(4-methoxyphenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C20H22N2O2
 1
1
Ki = 23 nM
   TI
   LI
   LO
   TS
CP0009417
7-[5-(4-chlorophenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H19ClN2O
 1
1
Ki = 23 nM
   TI
   LI
   LO
   TS
CP0009416
7-[5-(2-methoxyphenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C20H22N2O2
 1
1
Ki = 30 nM
   TI
   LI
   LO
   TS
CP0001447
7-(4-chloropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15ClN2
 1
1
Ki = 33 nM
   TI
   LI
   LO
   TS
CP0000951
7-(6-chloropyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H15ClN2
 1
1
Ki = 39 nM
   TI
   LI
   LO
   TS
CP0011949
7-[5-(2-chlorophenoxy)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H19ClN2O
 1
1
Ki = 39 nM
   TI
   LI
   LO
   TS
CP0000787
7-(5-phenylmethoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C20H22N2O
 1
1
Ki = 43.9 nM
   TI
   LI
   LO
   TS
CP0000884
(1R,5S)-3-methyl-7-pyridin-3-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H18N2
 1
1
Ki = 70 nM
   TI
   LI
   LO
   TS
CP0000945
5-[(1R,5S)-3-azabicyclo[3.3.1]non-6-en-7-yl]pyridine-3-carbonitrile
   Show/Hide
C14H15N3
 1
1
Ki = 73 nM
   TI
   LI
   LO
   TS
CP0000944
(1S,5R)-3-methyl-7-pyridin-3-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H18N2
 1
1
Ki = 74 nM
   TI
   LI
   LO
   TS
CP0000478
7-(6-chloropyridazin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C12H14ClN3
 1
1
Ki = 77 nM
   TI
   LI
   LO
   TS
CP0000949
5-[(1S,5R)-3-azabicyclo[3.3.1]non-6-en-7-yl]pyridine-3-carbonitrile
   Show/Hide
C14H15N3
 1
1
Ki = 79 nM
   TI
   LI
   LO
   TS
CP0006458
7-(6-methylpyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H18N2
 1
1
Ki = 80 nM
   TI
   LI
   LO
   TS
CP0000882
7-(5-propan-2-yloxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C16H22N2O
 1
1
Ki = 105 nM
   TI
   LI
   LO
   TS
CP0000481
7-(6-chloro-5-methoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17ClN2O
 1
1
Ki = 111.4 nM
   TI
   LI
   LO
   TS
CP0636918
7-(5-Cyanopyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H15N3
 1
1
Ki = 160 nM
   TI
   LI
   LO
   TS
CP0000953
7-pyrazin-2-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C12H15N3
 1
1
Ki = 281 nM
   TI
   LI
   LO
   TS
CP0000947
3-(3-azabicyclo[3.3.1]non-6-en-7-yl)pyridine-4-carbonitrile
   Show/Hide
C14H15N3
 1
1
Ki = 330 nM
   TI
   LI
   LO
   TS
CP0000948
7-(6-phenylpyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H20N2
 1
1
Ki = 590 nM
   TI
   LI
   LO
   TS
CP0000943
7-(5-methoxypyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C15H20N2O
 1
1
Ki = 605 nM
   TI
   LI
   LO
   TS
CP0001666
7-[5-(trifluoromethyl)pyridin-3-yl]-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H15F3N2
 1
1
Ki = 641 nM
   TI
   LI
   LO
   TS
CP0009376
7-(5-fluoropyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17FN2
 1
1
Ki = 1007 nM
   TI
   LI
   LO
   TS
CP0001448
7-(6-fluoropyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17FN2
 1
1
Ki = 1305 nM
   TI
   LI
   LO
   TS
CP0001669
7-(4-chloropyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17ClN2
 1
1
Ki = 1421 nM
   TI
   LI
   LO
   TS
CP0000954
7-(6-methoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H18N2O
 1
1
Ki = 1849 nM
   TI
   LI
   LO
   TS
CP0000941
7-(5-phenylpyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C19H20N2
 1
1
Ki = 3220 nM
   TI
   LI
   LO
   TS
CP0008063
3-methyl-7-(5-phenylmethoxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C21H24N2O
 1
1
Ki = 4545 nM
   TI
   LI
   LO
   TS
CP0001670
3-(3-methyl-3-azabicyclo[3.3.1]non-6-en-7-yl)pyridine-4-carbonitrile
   Show/Hide
C15H17N3
 1
1
Ki = 4847 nM
   TI
   LI
   LO
   TS
CP0010089
7-(6-chloropyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17ClN2
 1
1
Ki = 6530 nM
   TI
   LI
   LO
   TS
CP0002106
7-(6-chloro-5-methoxypyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C15H19ClN2O
 1
1
Ki = 7565 nM
   TI
   LI
   LO
   TS
CP0004237
(E)-N-methyl-4-pyridin-3-ylbut-3-en-1-amine
   Show/Hide
C10H14N2
 1
1
Ki = 8000 nM
   TI
   LI
   LO
   TS
CP0004193
7-(5-chloropyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C14H17ClN2
 1
1
Ki = 8006 nM
   TI
   LI
   LO
   TS
CP0000480
7-(6-methoxypyridin-3-yl)-3-methyl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C15H20N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0000788
3-methyl-7-(5-propan-2-yloxypyridin-3-yl)-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C17H24N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0001446
6-(3-azabicyclo[3.3.1]non-6-en-7-yl)quinoxaline
   Show/Hide
C16H17N3
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0001668
7-pyridin-4-yl-3-azabicyclo[3.3.1]non-6-ene
   Show/Hide
C13H16N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0009375
5-(3-methyl-3-azabicyclo[3.3.1]non-6-en-7-yl)pyridine-3-carbonitrile
   Show/Hide
C15H17N3
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -