General Information of the Cell Line
Cell Line ID
CL000780
Cell Line Name
RKE
Category
Spontaneously immortalized cell line
Organism
Rattus norvegicus (Rat)
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT06150, Vasoactive intestinal polypeptide receptor 1
Compound ID Compound Name Compound Formula
CP0391381
[4-tert-butyl-2-(3,4-dimethylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C22H30O
 1
1
IC50 = 81 nM
   TI
   LI
   LO
   TS
CP0399087
[4-tert-butyl-2-(3-chlorophenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C20H25ClO
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0500255
(4-tert-butyl-2-naphthalen-2-yl-6-propan-2-ylphenyl)methanol
   Show/Hide
C24H28O
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0418759
[4-tert-butyl-2-(3-methylsulfanylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28OS
 1
1
IC50 = 170 nM
   TI
   LI
   LO
   TS
CP0418939
(4-tert-butyl-2-naphthalen-1-yl-6-propan-2-ylphenyl)methanol
   Show/Hide
C24H28O
 1
1
IC50 = 180 nM
   TI
   LI
   LO
   TS
CP0500254
[4-tert-butyl-2-(3-methoxyphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O2
 1
1
IC50 = 200 nM
   TI
   LI
   LO
   TS
CP0497377
[4-tert-butyl-2-(3-phenylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C26H30O
 1
1
IC50 = 210 nM
   TI
   LI
   LO
   TS
CP0456252
[4-tert-butyl-2-(3-methylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O
 1
1
IC50 = 240 nM
   TI
   LI
   LO
   TS
CP0391991
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-phenylpropanamide
   Show/Hide
C18H18N2OS
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0497376
[4-tert-butyl-2-(4-chlorophenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C20H25ClO
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0400835
[4-tert-butyl-2-(4-methylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O
 1
1
IC50 = 300 nM
   TI
   LI
   LO
   TS
CP0499549
[4-tert-butyl-2-[3-(dimethylamino)phenyl]-6-propan-2-ylphenyl]methanol
   Show/Hide
C22H31NO
 1
1
IC50 = 310 nM
   TI
   LI
   LO
   TS
CP0493871
(4-tert-butyl-2-phenyl-6-propan-2-ylphenyl)methanol
   Show/Hide
C20H26O
 1
1
IC50 = 390 nM
   TI
   LI
   LO
   TS
CP0456771
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(4-methoxyphenyl)propanamide
   Show/Hide
C19H20N2O2S
 1
1
IC50 = 410 nM
   TI
   LI
   LO
   TS
CP0177086
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)cyclohexanecarboxamide
   Show/Hide
C16H20N2OS
 1
1
IC50 = 470 nM
   TI
   LI
   LO
   TS
CP0416881
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)cyclopentanecarboxamide
   Show/Hide
C15H18N2OS
 1
1
IC50 = 470 nM
   TI
   LI
   LO
   TS
CP0392137
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(4-methylphenyl)propanamide
   Show/Hide
C19H20N2OS
 1
1
IC50 = 480 nM
   TI
   LI
   LO
   TS
CP0399088
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(3-methoxyphenyl)propanamide
   Show/Hide
C19H20N2O2S
 1
1
IC50 = 610 nM
   TI
   LI
   LO
   TS
CP0418862
[4-tert-butyl-2-(4-phenylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C26H30O
 1
1
IC50 = 680 nM
   TI
   LI
   LO
   TS
CP0462762
[4-tert-butyl-2-(4-fluorophenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C20H25FO
 1
1
IC50 = 740 nM
   TI
   LI
   LO
   TS
CP0495490
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(3-methylphenyl)propanamide
   Show/Hide
C19H20N2OS
 1
1
IC50 = 750 nM
   TI
   LI
   LO
   TS
CP0463019
[4-tert-butyl-2-(2-methoxyphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O2
 1
1
IC50 = 820 nM
   TI
   LI
   LO
   TS
CP0391993
3-(4-chlorophenyl)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)propanamide
   Show/Hide
C18H17ClN2OS
 1
1
IC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0403719
[4-tert-butyl-2-(4-methoxyphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O2
 1
1
IC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0166953
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-phenylacetamide
   Show/Hide
C17H16N2OS
 1
1
IC50 = 1600 nM
   TI
   LI
   LO
   TS
CP0391990
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)cyclobutanecarboxamide
   Show/Hide
C14H16N2OS
 1
1
IC50 = 1800 nM
   TI
   LI
   LO
   TS
CP0392412
2-(1-benzothiophen-2-yl)-N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)acetamide
   Show/Hide
C19H16N2OS2
 1
1
IC50 = 1900 nM
   TI
   LI
   LO
   TS
CP0392428
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-methylbutanamide
   Show/Hide
C14H18N2OS
 1
1
IC50 = 1900 nM
   TI
   LI
   LO
   TS
CP0391382
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)cyclopropanecarboxamide
   Show/Hide
C13H14N2OS
 1
1
IC50 = 2700 nM
   TI
   LI
   LO
   TS
CP0438144
[4-tert-butyl-2-(2-phenylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C26H30O
 1
1
IC50 = 3200 nM
   TI
   LI
   LO
   TS
CP0346544
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-methylpropanamide
   Show/Hide
C13H16N2OS
 1
1
IC50 = 3400 nM
   TI
   LI
   LO
   TS
CP0462996
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-(2,3-dihydro-1-benzofuran-2-yl)acetamide
   Show/Hide
C19H18N2O2S
 1
1
IC50 = 3800 nM
   TI
   LI
   LO
   TS
CP0458447
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-phenoxyacetamide
   Show/Hide
C17H16N2O2S
 1
1
IC50 = 9100 nM
   TI
   LI
   LO
   TS
CP0391992
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(2-methylphenyl)propanamide
   Show/Hide
C19H20N2OS
 1
1
IC50 = 11000 nM
   TI
   LI
   LO
   TS
CP0418863
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)propanamide
   Show/Hide
C12H14N2OS
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0461693
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-1,2,3,4-tetrahydronaphthalene-2-carboxamide
   Show/Hide
C20H20N2OS
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0218894
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)acetamide
   Show/Hide
C11H12N2OS
 1
1
IC50 = 13000 nM
   TI
   LI
   LO
   TS
CP0043252
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)benzamide
   Show/Hide
C16H14N2OS
 1
1
IC50 = 15000 nM
   TI
   LI
   LO
   TS
CP0462763
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2,3-dihydro-1H-indene-2-carboxamide
   Show/Hide
C19H18N2OS
 1
1
IC50 = 17000 nM
   TI
   LI
   LO
   TS
CP0376905
[4-tert-butyl-2-(2-methylphenyl)-6-propan-2-ylphenyl]methanol
   Show/Hide
C21H28O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0456253
[4-tert-butyl-2-propan-2-yl-6-[3-(trifluoromethyl)phenyl]phenyl]methanol
   Show/Hide
C21H25F3O
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0463018
3-[5-tert-butyl-2-(hydroxymethyl)-3-propan-2-ylphenyl]benzonitrile
   Show/Hide
C21H25NO
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0495491
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-(1H-indol-2-yl)acetamide
   Show/Hide
C19H17N3OS
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -