General Information of the Cell Line
Cell Line ID
CL000079
Cell Line Name
Expi293F
Category
Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_D615
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT00862, Adenosine receptor A2a
Compound ID Compound Name Compound Formula
CP0053494
4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-7-yl]amino}ethyl)phenol
   Show/Hide
C16H15N7O2
 2
1
Kd = 0.286 nM
   TI
   LI
   LO
   TS
2
Ki = 0.395 nM
   TI
   LI
   LO
   TS
CP0056600
2-(Phenylamino)ado (CV-1808)
   Show/Hide
C16H18N6O4
 2
1
Kd = 9.1 nM
   TI
   LI
   LO
   TS
2
Ki = 76 nM
   TI
   LI
   LO
   TS
CP0001102
(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol
   Show/Hide
C10H13N5O4
 2
1
Kd = 17.3 nM
   TI
   LI
   LO
   TS
2
Ki = 150 nM
   TI
   LI
   LO
   TS
CP0015475
3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophenyl)-2,5-dihydro-1H-pyrrole-2,5-dione
   Show/Hide
C16H10Cl2N2O3
 1
1
Kd = 110 nM
   TI
   LI
   LO
   TS
CP0016654
N-[5-bromo-6-(furan-2-yl)-1H-pyrazolo[3,4-b]pyridin-3-yl]cyclopropanecarboxamide
   Show/Hide
C14H11BrN4O2
 1
1
Kd = 560 nM
   TI
   LI
   LO
   TS
CP0546728
3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-amine
   Show/Hide
C11H9N5
 1
1
Kd = 1110 nM
   TI
   LI
   LO
   TS
CP0568020
BENZOGUANAMINE
   Show/Hide
C9H9N5
 1
1
Kd = 1500 nM
   TI
   LI
   LO
   TS
CP0042654
1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
   Show/Hide
C7H8N4O2
 1
1
Kd = 3630 nM
   TI
   LI
   LO
   TS
CP0043620
1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
   Show/Hide
C8H10N4O2
 1
1
Kd = 5510 nM
   TI
   LI
   LO
   TS
CP0019682
2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]pyridine
   Show/Hide
C18H12FN3
 1
1
Kd = 8900 nM
   TI
   LI
   LO
   TS
CP0543485
pteridine-2,4-diamine
   Show/Hide
C6H6N6
 1
1
Kd = 9600 nM
   TI
   LI
   LO
   TS
CP0547170
N-(3-chlorophenyl)-4-methylsulfonylbenzamide
   Show/Hide
C14H12ClNO3S
 1
1
Kd = 13500 nM
   TI
   LI
   LO
   TS
CP0546737
5-(4-chlorophenyl)-1,2,4-thiadiazol-3-amine
   Show/Hide
C8H6ClN3S
 1
1
Kd = 21800 nM
   TI
   LI
   LO
   TS
CP0546740
3-methyl-1H-quinazoline-2,4-dione
   Show/Hide
C9H8N2O2
 1
1
Kd = 28800 nM
   TI
   LI
   LO
   TS
CP0551935
5-phenyl-1,3-oxazole-4-carboxamide
   Show/Hide
C10H8N2O2
 1
1
Kd = 31800 nM
   TI
   LI
   LO
   TS
CP0562631
N-quinolin-2-ylfuran-2-carboxamide
   Show/Hide
C14H10N2O2
 1
1
Kd = 40000 nM
   TI
   LI
   LO
   TS
CP0568019
3-phenyl-N-propan-2-yl-1H-pyrazole-5-carboxamide
   Show/Hide
C13H15N3O
 1
1
Kd = 49000 nM
   TI
   LI
   LO
   TS
CP0546739
5-(4-bromophenyl)-1,2,4-triazin-3-amine
   Show/Hide
C9H7BrN4
 1
1
Kd = 50000 nM
   TI
   LI
   LO
   TS
CP0546741
1-phenyl-3-pyridin-2-ylurea
   Show/Hide
C12H11N3O
 1
1
Kd = 50900 nM
   TI
   LI
   LO
   TS
CP0036281
ALLOPURINOL
   Show/Hide
C5H4N4O
 1
1
Kd = 77000 nM
   TI
   LI
   LO
   TS
CP0562630
N-benzyl-2,1,3-benzoxadiazole-5-carboxamide
   Show/Hide
C14H11N3O2
 1
1
Kd = 100000 nM
   TI
   LI
   LO
   TS
CP0547178
3-phenyl-1,2,4-thiadiazol-5-amine
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C8H7N3S
 1
1
Kd = 130000 nM
   TI
   LI
   LO
   TS
CP0492321
2-(benzylamino)pyrido[1,2-a]pyrimidin-4-one
   Show/Hide
C15H13N3O
 1
1
Kd = 131000 nM
   TI
   LI
   LO
   TS
CP0543588
US8993552, 1F4 Compound 44
   Show/Hide
C10H10N4O
 1
1
Kd = 410000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -