Compound ID |
Compound Name |
Compound Formula |
CP0955447
|
(1r,4r)-4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexanol
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|
C18H20N4O
|
1
|
1 |
Kd = 5.46 nM
|
|
|
CP0546739
|
5-(4-bromophenyl)-1,2,4-triazin-3-amine
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|
C9H7BrN4
|
1
|
1 |
Kd = 1100 nM
|
|
|
CP0084760
|
2-methoxy-4-[(E)-[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinylidene]methyl]phenol
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|
C19H16N6O2
|
1
|
1 |
Kd = 1210 nM
|
|
|
CP0016654
|
N-[5-bromo-6-(furan-2-yl)-1H-pyrazolo[3,4-b]pyridin-3-yl]cyclopropanecarboxamide
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|
C14H11BrN4O2
|
1
|
1 |
Kd = 2120 nM
|
|
|
CP0015475
|
3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophenyl)-2,5-dihydro-1H-pyrrole-2,5-dione
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|
C16H10Cl2N2O3
|
1
|
1 |
Kd = 2210 nM
|
|
|
CP0568020
|
BENZOGUANAMINE
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|
C9H9N5
|
1
|
1 |
Kd = 2210 nM
|
|
|
CP0019682
|
2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]pyridine
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|
C18H12FN3
|
1
|
1 |
Kd = 6050 nM
|
|
|
CP0547170
|
N-(3-chlorophenyl)-4-methylsulfonylbenzamide
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|
C14H12ClNO3S
|
1
|
1 |
Kd = 7600 nM
|
|
|
CP0546737
|
5-(4-chlorophenyl)-1,2,4-thiadiazol-3-amine
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|
C8H6ClN3S
|
1
|
1 |
Kd = 20700 nM
|
|
|
CP0546728
|
3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-amine
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|
C11H9N5
|
1
|
1 |
Kd = 22900 nM
|
|
|
CP0545286
|
N-(furan-2-ylmethyl)-1-propan-2-ylpyrazolo[3,4-b]pyridine-5-carboxamide
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|
C15H16N4O2
|
1
|
1 |
Kd = 27000 nM
|
|
|
CP0546740
|
3-methyl-1H-quinazoline-2,4-dione
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|
C9H8N2O2
|
1
|
1 |
Kd = 34300 nM
|
|
|
CP0546741
|
1-phenyl-3-pyridin-2-ylurea
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|
C12H11N3O
|
1
|
1 |
Kd = 41000 nM
|
|
|
CP0547178
|
3-phenyl-1,2,4-thiadiazol-5-amine
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|
C8H7N3S
|
1
|
1 |
Kd = 51700 nM
|
|
|
CP0562631
|
N-quinolin-2-ylfuran-2-carboxamide
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|
C14H10N2O2
|
1
|
1 |
Kd = 59000 nM
|
|
|
CP0568019
|
3-phenyl-N-propan-2-yl-1H-pyrazole-5-carboxamide
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|
C13H15N3O
|
1
|
1 |
Kd = 70000 nM
|
|
|
CP0543588
|
US8993552, 1F4 Compound 44
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|
C10H10N4O
|
1
|
1 |
Kd = 78000 nM
|
|
|
CP0562630
|
N-benzyl-2,1,3-benzoxadiazole-5-carboxamide
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|
C14H11N3O2
|
1
|
1 |
Kd = 92000 nM
|
|
|
CP0492321
|
2-(benzylamino)pyrido[1,2-a]pyrimidin-4-one
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|
C15H13N3O
|
1
|
1 |
Kd = 154000 nM
|
|
|