Brief Information of the Cell Line and Protein
Cell Line ID: CL000079 , Expi293F
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_D615
Protein ID: PT01278 , Adenosine receptor A2b
Gene Name ADORA2B
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P29275
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000079  Protein ID: PT01278
 
Compound ID Compound Name Compound Formula
CP0019682
2-(4-fluorophenyl)-3-(4-pyridinyl)pyrazolo-[1,5-a]pyridine
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C18H12FN3
 1
1
Kd = 280 nM
   TI
   LI
   LO
   TS
CP0106488
2-Amino-4-(4-hydroxy-phenyl)-6-(1H-imidazol-2-ylmethylsulfanyl)-pyridine-3,5-dicarbonitrile
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C17H12N6OS
 2
1
Kd = 3070 nM
   TI
   LI
   LO
   TS
2
Ki = 1 nM
   TI
   LI
   LO
   TS
CP0547170
N-(3-chlorophenyl)-4-methylsulfonylbenzamide
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C14H12ClNO3S
 1
1
Kd = 19300 nM
   TI
   LI
   LO
   TS
CP0562630
N-benzyl-2,1,3-benzoxadiazole-5-carboxamide
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C14H11N3O2
 1
1
Kd = 22000 nM
   TI
   LI
   LO
   TS
CP0546741
1-phenyl-3-pyridin-2-ylurea
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C12H11N3O
 1
1
Kd = 43300 nM
   TI
   LI
   LO
   TS
CP0546737
5-(4-chlorophenyl)-1,2,4-thiadiazol-3-amine
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C8H6ClN3S
 1
1
Kd = 45000 nM
   TI
   LI
   LO
   TS
CP0547178
3-phenyl-1,2,4-thiadiazol-5-amine
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C8H7N3S
 1
1
Kd = 60700 nM
   TI
   LI
   LO
   TS
CP0545286
N-(furan-2-ylmethyl)-1-propan-2-ylpyrazolo[3,4-b]pyridine-5-carboxamide
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C15H16N4O2
 1
1
Kd = 80000 nM
   TI
   LI
   LO
   TS
CP0568020
BENZOGUANAMINE
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C9H9N5
 1
1
Kd = 107000 nM
   TI
   LI
   LO
   TS
CP0546728
3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-amine
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C11H9N5
 1
1
Kd = 120000 nM
   TI
   LI
   LO
   TS
CP0562631
N-quinolin-2-ylfuran-2-carboxamide
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C14H10N2O2
 1
1
Kd = 123000 nM
   TI
   LI
   LO
   TS
CP0543588
US8993552, 1F4 Compound 44
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C10H10N4O
 1
1
Kd = 140100 nM
   TI
   LI
   LO
   TS
CP0492321
2-(benzylamino)pyrido[1,2-a]pyrimidin-4-one
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C15H13N3O
 1
1
Kd = 199000 nM
   TI
   LI
   LO
   TS