General Information of the Cell Line
Cell Line ID
CL000541
Cell Line Name
HEK-2
Synonyms
Human Embryo Kidney-2
Category
Finite cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_WZ56
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT01584, Steroid 17-alpha-hydroxylase/17,20 lyase
Compound ID Compound Name Compound Formula
CP0443737
US8969586, 1
   Show/Hide
C19H14N2O
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0492512
US8916553, 198
   Show/Hide
C15H15F3N2O3S
 1
1
IC50 = 1.4 nM
   TI
   LI
   LO
   TS
CP0535595
US8916553, 225
   Show/Hide
C16H18N2O3S
 1
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
CP0536972
US8916553, 217
   Show/Hide
C14H16N2O3S
 1
1
IC50 = 2.5 nM
   TI
   LI
   LO
   TS
CP0492511
US8916553, 147
   Show/Hide
C23H20N2O4S
 1
1
IC50 = 2.7 nM
   TI
   LI
   LO
   TS
CP0536969
US8916553, 143
   Show/Hide
C22H18N2O3S
 1
1
IC50 = 2.9 nM
   TI
   LI
   LO
   TS
CP0535596
US8916553, 228
   Show/Hide
C17H13F3N2O3S
 1
1
IC50 = 3.2 nM
   TI
   LI
   LO
   TS
CP0468224
US8969586, 6
   Show/Hide
C19H13FN2O
 1
1
IC50 = 3.2 nM
   TI
   LI
   LO
   TS
CP0560555
US8916553, 173
   Show/Hide
C19H18ClN3O3S
 1
1
IC50 = 3.4 nM
   TI
   LI
   LO
   TS
CP0509202
US8969586, 86
   Show/Hide
C18H12FN3O
 1
1
IC50 = 3.9 nM
   TI
   LI
   LO
   TS
CP0573593
US8969586, 99
   Show/Hide
C20H14FN3S
 1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
CP0574878
US8969586, 103
   Show/Hide
C17H10ClFN4S
 1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
CP0506883
US8916553, 165
   Show/Hide
C18H17N3O3S
 1
1
IC50 = 5.4 nM
   TI
   LI
   LO
   TS
CP0459450
4-(4-methylpyridin-3-yl)-1-pyridin-2-ylbenzimidazole
   Show/Hide
C18H14N4
 1
1
IC50 = 5.8 nM
   TI
   LI
   LO
   TS
CP0575689
US8916553, 160
   Show/Hide
C21H17N3O3S
 1
1
IC50 = 6 nM
   TI
   LI
   LO
   TS
CP0556511
US8916553, 159
   Show/Hide
C19H18N2O3S
 1
1
IC50 = 6.2 nM
   TI
   LI
   LO
   TS
CP0520326
US8916553, 142
   Show/Hide
C17H16N2O3S
 1
1
IC50 = 6.6 nM
   TI
   LI
   LO
   TS
CP0550979
US8916553, 184
   Show/Hide
C17H17F3N2O3S
 1
1
IC50 = 7.7 nM
   TI
   LI
   LO
   TS
CP0533160
US8969586, 98
   Show/Hide
C18H12FN3S
 1
1
IC50 = 8 nM
   TI
   LI
   LO
   TS
CP0450087
US8916553, 156
   Show/Hide
C18H18N2O3S
 1
1
IC50 = 8.1 nM
   TI
   LI
   LO
   TS
CP0556918
US9145419, 35
   Show/Hide
C16H12N4S
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0575691
US8916553, 168
   Show/Hide
C19H19N3O3S
 1
1
IC50 = 9.6 nM
   TI
   LI
   LO
   TS
CP0484581
1-(6-fluoropyridin-2-yl)-4-(4-methylpyridin-3-yl)benzimidazole
   Show/Hide
C18H13FN4
 1
1
IC50 = 11 nM
   TI
   LI
   LO
   TS
CP0539544
US8916553, 144
   Show/Hide
C26H20N2O3S
 1
1
IC50 = 11 nM
   TI
   LI
   LO
   TS
CP0102366
4-(4-methylpyridin-3-yl)-1-(2,2,2-trifluoroethyl)benzimidazole
   Show/Hide
C15H12F3N3
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0518576
US9145419, 3
   Show/Hide
C20H16N4O
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0511961
US9266880, 7
   Show/Hide
C21H15N5O2S
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
CP0550981
US8916553, 240
   Show/Hide
C14H13F3N2O2S
 1
1
IC50 = 26 nM
   TI
   LI
   LO
   TS
CP0550977
US8916553, 154
   Show/Hide
C25H19N3O3S
 1
1
IC50 = 27 nM
   TI
   LI
   LO
   TS
CP0549963
US8916553, 23
   Show/Hide
C15H16F2N2O3S
 1
1
IC50 = 32 nM
   TI
   LI
   LO
   TS
CP0404501
4-(4-methylpyridin-3-yl)-1-pyrazin-2-ylbenzimidazole
   Show/Hide
C17H13N5
 1
1
IC50 = 37 nM
   TI
   LI
   LO
   TS
CP0536976
US8916553, 243
   Show/Hide
C16H15F3N2O2S
 1
1
IC50 = 39 nM
   TI
   LI
   LO
   TS
CP0489074
4-(4-methylpyridin-3-yl)-1-[6-(trifluoromethyl)pyridin-2-yl]benzimidazole
   Show/Hide
C19H13F3N4
 1
1
IC50 = 40 nM
   TI
   LI
   LO
   TS
CP0535597
US8916553, 234
   Show/Hide
C18H17FN2O3S
 1
1
IC50 = 40 nM
   TI
   LI
   LO
   TS
CP0553483
US9145419, 1
   Show/Hide
C18H14N4
 1
1
IC50 = 41 nM
   TI
   LI
   LO
   TS
CP0490137
US9266880, 3
   Show/Hide
C20H12FN5
 1
1
IC50 = 41 nM
   TI
   LI
   LO
   TS
CP0508996
US8916553, 24
   Show/Hide
C15H15F3N2O3S
 1
1
IC50 = 42 nM
   TI
   LI
   LO
   TS
CP0561900
US8969586, 52
   Show/Hide
C19H11ClN6O
 1
1
IC50 = 42 nM
   TI
   LI
   LO
   TS
CP0536975
US8916553, 241
   Show/Hide
C17H13F3N2O2S
 1
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0468225
US8969586, 30
   Show/Hide
C15H11ClN2O
 1
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0509001
US8916553, 218
   Show/Hide
C14H17N3O3S
 1
1
IC50 = 49 nM
   TI
   LI
   LO
   TS
CP0494899
US9266880, 4
   Show/Hide
C16H12FN5
 1
1
IC50 = 50 nM
   TI
   LI
   LO
   TS
CP0550980
US8916553, 239
   Show/Hide
C17H16FN3O3S
 1
1
IC50 = 51 nM
   TI
   LI
   LO
   TS
CP0546689
US8916553, 195
   Show/Hide
C13H13ClN2O2S
 1
1
IC50 = 52 nM
   TI
   LI
   LO
   TS
CP0450088
US8916553, 170
   Show/Hide
C19H19N3O4S
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0450091
US8916553, 233
   Show/Hide
C15H15F3N2O4S
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0509203
US8969586, 109
   Show/Hide
C23H14FNS
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0574708
US9145419, 7
   Show/Hide
C18H13FN4
 1
1
IC50 = 56 nM
   TI
   LI
   LO
   TS
CP0450092
US8916553, 245
   Show/Hide
C13H15N3O4S
 1
1
IC50 = 57 nM
   TI
   LI
   LO
   TS
CP0556512
US8916553, 175
   Show/Hide
C22H19N3O3S
 1
1
IC50 = 59 nM
   TI
   LI
   LO
   TS
CP0563049
US8916553, 232
   Show/Hide
C18H15F3N2O3S
 1
1
IC50 = 59 nM
   TI
   LI
   LO
   TS
CP0450800
US8969586, 26
   Show/Hide
C17H10F3N5O2
 1
1
IC50 = 65 nM
   TI
   LI
   LO
   TS
CP0574811
US8969586, 94
   Show/Hide
C16H11N3S2
 1
1
IC50 = 76 nM
   TI
   LI
   LO
   TS
CP0565789
US9266880, 8
   Show/Hide
C19H11F2N5
 1
1
IC50 = 76 nM
   TI
   LI
   LO
   TS
CP0492543
US8969586, 129
   Show/Hide
C21H18N2O3
 1
1
IC50 = 79 nM
   TI
   LI
   LO
   TS
CP0406850
US9145419, 11
   Show/Hide
C18H13ClN4
 1
1
IC50 = 97 nM
   TI
   LI
   LO
   TS
CP0546688
US8916553, 164
   Show/Hide
C16H21N3O3S
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0560556
US8916553, 221
   Show/Hide
C18H23N3O3S
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0450089
US8916553, 220
   Show/Hide
C15H19N3O3S
 1
1
IC50 = 103 nM
   TI
   LI
   LO
   TS
CP0506881
US8916553, 12
   Show/Hide
C19H18N2O2S
 1
1
IC50 = 104 nM
   TI
   LI
   LO
   TS
CP0575690
US8916553, 161
   Show/Hide
C13H15N3O3S
 1
1
IC50 = 112 nM
   TI
   LI
   LO
   TS
CP0508999
US8916553, 172
   Show/Hide
C18H16ClN3O3S
 1
1
IC50 = 117 nM
   TI
   LI
   LO
   TS
CP0415281
US8916553, 158
   Show/Hide
C21H20N4O3S
 1
1
IC50 = 118 nM
   TI
   LI
   LO
   TS
CP0509000
US8916553, 176
   Show/Hide
C21H18N4O3S
 1
1
IC50 = 118 nM
   TI
   LI
   LO
   TS
CP0508998
US8916553, 169
   Show/Hide
C20H21N3O3S
 1
1
IC50 = 119 nM
   TI
   LI
   LO
   TS
CP0509002
US8916553, 250
   Show/Hide
C15H15N3O3S
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0491467
US9145419, 9
   Show/Hide
C19H16N4
 1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
CP0511960
US9266880, 1
   Show/Hide
C21H13FN4
 1
1
IC50 = 128 nM
   TI
   LI
   LO
   TS
CP0494898
US9145419, 37
   Show/Hide
C19H13F3N4
 1
1
IC50 = 129 nM
   TI
   LI
   LO
   TS
CP0550978
US8916553, 166
   Show/Hide
C17H16N4O3S
 1
1
IC50 = 131 nM
   TI
   LI
   LO
   TS
CP0508997
US8916553, 163
   Show/Hide
C15H19N3O3S
 1
1
IC50 = 134 nM
   TI
   LI
   LO
   TS
CP0557414
4-(4-ethoxypyrimidin-5-yl)-1-(2,2,2-trifluoroethyl)benzimidazole
   Show/Hide
C15H13F3N4O
 1
1
IC50 = 135 nM
   TI
   LI
   LO
   TS
CP0539545
US8916553, 167
   Show/Hide
C14H14F3N3O3S
 1
1
IC50 = 158 nM
   TI
   LI
   LO
   TS
CP0520327
US8916553, 162
   Show/Hide
C15H17N3O3S
 1
1
IC50 = 169 nM
   TI
   LI
   LO
   TS
CP0536973
US8916553, 236
   Show/Hide
C14H14ClFN2O3S
 1
1
IC50 = 174 nM
   TI
   LI
   LO
   TS
CP0442048
US8969586, 14
   Show/Hide
C20H12FN3O
 1
1
IC50 = 192 nM
   TI
   LI
   LO
   TS
CP0576875
US9266880, 5
   Show/Hide
C20H14N6O2S
 1
1
IC50 = 206 nM
   TI
   LI
   LO
   TS
CP0567695
US9133160, 6
   Show/Hide
C17H13N5
 1
1
IC50 = 250 nM
   TI
   LI
   LO
   TS
CP0554830
US8969586, 128
   Show/Hide
C20H15ClN2O2
 1
1
IC50 = 251 nM
   TI
   LI
   LO
   TS
CP0566358
US9266880, 6
   Show/Hide
C16H14N6O2S
 1
1
IC50 = 271 nM
   TI
   LI
   LO
   TS
CP0500222
US9145419, 38
   Show/Hide
C20H18N4
 1
1
IC50 = 279 nM
   TI
   LI
   LO
   TS
CP0489075
2-[4-(4-methylpyridin-3-yl)benzimidazol-1-yl]acetonitrile
   Show/Hide
C15H12N4
 1
1
IC50 = 330 nM
   TI
   LI
   LO
   TS
CP0450799
US8969586, 4
   Show/Hide
C18H13N3O
 1
1
IC50 = 357 nM
   TI
   LI
   LO
   TS
CP0512108
4-(4-chloropyridin-3-yl)-1-(2,2,2-trifluoroethyl)benzimidazole
   Show/Hide
C14H9ClF3N3
 1
1
IC50 = 361 nM
   TI
   LI
   LO
   TS
CP0435588
1-cyclopropyl-4-(4-methylpyridin-3-yl)benzimidazole
   Show/Hide
C16H15N3
 1
1
IC50 = 396 nM
   TI
   LI
   LO
   TS
CP0441622
4-(4-methylpyridin-3-yl)-1-pyridin-4-ylbenzimidazole
   Show/Hide
C18H14N4
 1
1
IC50 = 405 nM
   TI
   LI
   LO
   TS
CP0539227
US8969586, 57
   Show/Hide
C19H11ClN6O
 1
1
IC50 = 524 nM
   TI
   LI
   LO
   TS
CP0550065
US8969586, 68
   Show/Hide
C16H16N2O3
 1
1
IC50 = 524 nM
   TI
   LI
   LO
   TS
CP0553890
US9145419, 26
   Show/Hide
C17H11FN4
 1
1
IC50 = 524 nM
   TI
   LI
   LO
   TS
CP0492542
US8969586, 124
   Show/Hide
C24H18N2O2
 1
1
IC50 = 611 nM
   TI
   LI
   LO
   TS
CP0575908
US9266880, 2
   Show/Hide
C15H10FN5
 1
1
IC50 = 640 nM
   TI
   LI
   LO
   TS
CP0534412
4-(4-methylpyridin-3-yl)-1-pyrimidin-4-ylbenzimidazole
   Show/Hide
C17H13N5
 1
1
IC50 = 656 nM
   TI
   LI
   LO
   TS
CP0406851
US9145419, 34
   Show/Hide
C18H12Cl2N4
 1
1
IC50 = 664 nM
   TI
   LI
   LO
   TS
CP0453356
5-[1-(2,2,2-trifluoroethyl)benzimidazol-4-yl]pyrimidin-4-amine
   Show/Hide
C13H10F3N5
 1
1
IC50 = 674 nM
   TI
   LI
   LO
   TS
CP0549879
1-(3,5-difluoropyridin-2-yl)-4-(4-methylpyridin-3-yl)benzimidazole
   Show/Hide
C18H12F2N4
 1
1
IC50 = 758 nM
   TI
   LI
   LO
   TS
CP0471287
5-[1-(2,4-difluorophenyl)benzimidazol-4-yl]pyrimidin-4-amine
   Show/Hide
C17H11F2N5
 1
1
IC50 = 797 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -