[(3R)-7-fluoro-6-(2-methylpropyl)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]methanesulfonamide

6-[(3R)-7-fluoro-3-(methylsulfonylmethyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

2-[(3S)-7-chloro-6-(2-methylpropyl)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

2-[(3S)-7-fluoro-6-(2-methylpropyl)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

[(3R)-7-fluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]methanesulfonamide

2',15'-dimethyl-5,5'-dioxo-(9'R)-spiro[tetrahydrofuran-2,14'-tetracyclo[8.7.0.02,7.011,15]heptadec-6'-ene]-9-yl ethanethioate

US10017502, Example 5a

5-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1,3-dihydrobenzimidazol-2-one

US10017502, Example 8a

6-[(3S)-7-fluoro-3-(2-methylpropyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

6-[(3R)-3,7-dimethyl-3-(methylsulfonylmethyl)-2H-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

US10017502, Example 6b

2-[(3S)-6-cyclopropyl-7-fluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

N-methyl-2-[(3S)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-7-(trifluoromethyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

2-[(3S)-4-[2-(carbamoylamino)pyridine-4-carbonyl]-7-fluoro-6-(2-methylpropyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

N-methyl-2-[(3S)-7-methyl-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

2-[(2S)-6-chloro-1-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-3,4-dihydro-2H-quinoxalin-2-yl]acetamide

6-[(2R,5R)-2-methyl-5-phenylmorpholin-4-yl]-4H-pyrido[3,2-b][1,4]oxazin-3-one

2-[(3S)-7-fluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-6-propan-2-yloxy-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

[(3R)-4-(3,4-dihydro-2H-1,4-benzoxazine-6-carbonyl)-7-fluoro-2,3-dihydro-1,4-benzoxazin-3-yl]methanesulfonamide

6-[(3S)-6-(cyclohexylmethyl)-7-fluoro-3-(2-hydroxyethyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

[(3R)-7-fluoro-4-(1H-indole-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]methanesulfonamide

methyl 2-[(3S)-7-fluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetate

US10017502, Example 4b

6-[(3S)-7-fluoro-3-(2-hydroxyethyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

N-methyl-2-[(3S)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

2-{(3S or 3R)-7-Fluoro-4-[(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-yl}acetamide

2-[(3S)-5,7-difluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

methyl (1R,2S,9R,10R,11S,14R,15S,17R)-2,15-dimethyl-5,5'-dioxospiro[18-oxapentacyclo[8.8.0.01,17.02,7.011,15]octadec-6-ene-14,2'-oxolane]-9-carboxylate

6-[(2S)-6-fluoro-2-methyl-3,4-dihydro-2H-quinoline-1-carbonyl]-4H-1,4-benzoxazin-3-one

2-[(3S)-6-chloro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

6-[(3S)-7-fluoro-3-methyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

6-(2-methyl-3,4-dihydro-2H-quinoline-1-carbonyl)-4H-1,4-benzoxazin-3-one

6-(3,4-dihydro-2H-quinoline-1-carbonyl)-4H-1,4-benzoxazin-3-one

2-[(3S)-7-chloro-5-methyl-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

2-[(2R)-6-fluoro-1-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-3,4-dihydro-2H-quinolin-2-yl]-N-methylacetamide

7-[(3S)-7-fluoro-3-(2-methylpropyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-3,4-dihydro-1H-quinolin-2-one

6-(2,3-dihydro-1,4-benzoxazine-4-carbonyl)-4H-1,4-benzoxazin-3-one

2-[(3S)-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetonitrile

6-[(2-methyl-3,4-dihydro-2H-quinolin-1-yl)sulfonyl]-4H-1,4-benzoxazin-3-one

6-[2-(4-methylphenyl)piperidin-1-yl]sulfonyl-4H-1,4-benzoxazin-3-one

2-[(3S)-7-cyano-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide

US10017502, Example 4a

2-[(2S)-7-fluoro-1-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-3,5-dihydro-2H-4,1-benzoxazepin-2-yl]acetamide

N-ethyl-2-[7-fluoro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetamide

6-[(3S)-3-(2-aminoethyl)-7-fluoro-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

2-[(3S)-7-chloro-4-(3-oxo-4H-1,4-benzoxazine-6-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]acetic acid

6-[(3R)-7-fluoro-3-methyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

6-[(2R)-6-fluoro-2-methyl-3,4-dihydro-2H-quinoline-1-carbonyl]-4H-1,4-benzoxazin-3-one

6-[(3S)-3-methyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carbonyl]-4H-1,4-benzoxazin-3-one

6-[(2R)-5-chloro-2-(2-hydroxyethyl)-2,3-dihydroindole-1-carbonyl]-4H-1,4-benzoxazin-3-one

2-[(3S)-7-fluoro-4-(2-oxo-1,4-dihydro-3,1-benzoxazine-7-carbonyl)-2,3-dihydro-1,4-benzoxazin-3-yl]-N-methylacetamide