General Information of the Cell Line
Cell Line ID
CL000883
Cell Line Name
HTLA
Category
Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT00834, Cannabinoid receptor 2
Compound ID Compound Name Compound Formula
CP0382825
N-(3-pentyl-1,3-benzothiazol-2-ylidene)naphthalene-1-carboxamide
   Show/Hide
C23H22N2OS
 2
1
EC50 = 12.88 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382775
N-(3-pentyl-1,3-benzothiazol-2-ylidene)adamantane-1-carboxamide
   Show/Hide
C23H30N2OS
 2
1
EC50 = 26.3 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0152977
5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid ((1S,2S,4R)-1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
   Show/Hide
C29H34ClN3O
 2
1
EC50 = 41 nM
   TI
   LI
   LO
   TS
2
EC50 = 1360 nM
   TI
   LI
   LO
   TS
CP0462464
N-(3-pentyl-1,3-benzothiazol-2-ylidene)-3-(trifluoromethyl)benzamide
   Show/Hide
C20H19F3N2OS
 2
1
EC50 = 128.82 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382751
2,4-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-5-carboxamide
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C16H18N2OS
 2
1
EC50 = 436.5 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382776
N-(3-pentyl-1,3-benzothiazol-2-ylidene)-4-(trifluoromethyl)benzamide
   Show/Hide
C20H19F3N2OS
 2
1
EC50 = 2511.8 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382783
N-[(2-chlorophenyl)methyl]-1,3-benzothiazole-2-carboxamide
   Show/Hide
C15H11ClN2OS
 2
1
EC50 = 3311 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382826
N-(1-adamantyl)-2-tert-butyl-4-methyl-1,3-thiazole-5-carboxamide
   Show/Hide
C19H28N2OS
 2
1
EC50 = 3981 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382752
N-(1,3-benzothiazol-2-yl)adamantane-1-carboxamide
   Show/Hide
C18H20N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382754
N-hexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C17H22N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382755
N-cyclopentyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C16H18N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382759
N-(1,3-benzothiazol-2-yl)-4-(trifluoromethyl)benzamide
   Show/Hide
C15H9F3N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382778
N-naphthalen-1-yl-1,3-benzothiazole-2-carboxamide
   Show/Hide
C18H12N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382785
(4-methyl-2-phenyl-1,3-thiazol-5-yl)-morpholin-4-ylmethanone
   Show/Hide
C15H16N2O2S
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382820
N-(cyclohexylmethyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C18H22N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382821
N-(1-adamantyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
   Show/Hide
C16H22N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382822
N-butyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C15H18N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382823
N-[(4-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C18H15FN2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382824
N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-benzothiazole-2-carboxamide
   Show/Hide
C18H16N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382827
N-benzyl-2,4-dimethyl-1,3-thiazole-5-carboxamide
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C13H14N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382828
N-(cyclohexylmethyl)-1,3-benzothiazole-2-carboxamide
   Show/Hide
C15H18N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427555
N-[(2-chlorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C18H15ClN2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427556
N-naphthalen-2-yl-1,3-benzothiazole-2-carboxamide
   Show/Hide
C18H12N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0431627
N-(1,3-benzothiazol-2-yl)-3-(trifluoromethyl)benzamide
   Show/Hide
C15H9F3N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0431630
N-(1,3-benzothiazol-2-yl)naphthalene-1-carboxamide
   Show/Hide
C18H12N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382756
N-benzyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C18H16N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382757
N-[(2-fluorophenyl)methyl]-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C18H15FN2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382758
N-benzyl-1,3-benzothiazole-2-carboxamide
   Show/Hide
C15H12N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0382781
N-cyclopropyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C14H14N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0402060
N-(1-adamantyl)-1,3-benzothiazole-2-carboxamide
   Show/Hide
C18H20N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427553
N-cyclohexyl-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C17H20N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427554
N-(1-adamantyl)-4-methyl-2-phenyl-1,3-thiazole-5-carboxamide
   Show/Hide
C21H24N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0427561
4-methyl-2-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-5-carboxamide
   Show/Hide
C21H20N2OS
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -