General Information of the Cell Line
Cell Line ID
CL000009
Cell Line Name
LLC-PK1
Synonyms
LLC-PK(1)
LLC-PK-1
LLC PK-1
LLc-PK1
LLC PK1
LLCPK1
Lilly Laboratories Culture-Porcine Kidney 1
Category
Spontaneously immortalized cell line
Organism
Sus scrofa (Pig)
Cellosaurus ID
CVCL_0391
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT01546, ATP-dependent translocase ABCB1
Compound ID Compound Name Compound Formula
CP0667196
Ivermectin
   Show/Hide
C95H146O28
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0036222
(3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33-[(1R,2R,4E)-1-hydroxy-2-methylhex-4-en-1-yl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-bis(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecaazacyclotritriacontan-2,5,8,11,14,17,20,23,26,29,32-undecone
   Show/Hide
C62H111N11O12
 3
1
IC50 = 800 nM
   TI
   LI
   LO
   TS
2
Ki = 1300 nM
   TI
   LI
   LO
   TS
3
Ki = 4660 nM
   TI
   LI
   LO
   TS
CP0040184
1-[(4-fluorophenyl)methyl]-N-{1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}-1H-1,3-benzodiazol-2-amine
   Show/Hide
C28H31FN4O
 1
1
IC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0033565
(+/-)1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-ol
   Show/Hide
C32H41NO2
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0013607
2-methoxyacetic acid [(1S,2S)-2-[2-[3-(1H-benzimidazol-2-yl)propyl-methyl-amino]ethyl]-6-fluoro-1-isopropyl-tetralin-2-yl] ester;hydrate;hydrochloride
   Show/Hide
C29H38FN3O3
 1
1
IC50 = 1800 nM
   TI
   LI
   LO
   TS
CP0041632
ITRAZOLE
   Show/Hide
C35H38Cl2N8O4
 1
1
IC50 = 2100 nM
   TI
   LI
   LO
   TS
CP0055461
CHEBI:7550
   Show/Hide
C26H29N3O6
 3
1
IC50 = 2300 nM
   TI
   LI
   LO
   TS
2
IC50 = 4540 nM
   TI
   LI
   LO
   TS
3
IC50 = 17500 nM
   TI
   LI
   LO
   TS
CP0027419
1-(1-(4,4-bis(4-fluorophenyl)butyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
   Show/Hide
C28H29F2N3O
 1
1
IC50 = 2900 nM
   TI
   LI
   LO
   TS
CP0010655
(3S,4aS,8aS)-N-tert-butyl-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylphenyl)formamido]-4-(phenylsulfanyl)butyl]-decahydroisoquinoline-3-carboxamide
   Show/Hide
C32H45N3O4S
 1
1
IC50 = 3400 nM
   TI
   LI
   LO
   TS
CP0063077
1-[2-(2,4-dichlorobenzyl)oxy-2-(2,4-dichlorophenyl)ethyl]imidazole;nitric acid
   Show/Hide
C18H14Cl4N2O
 3
1
IC50 = 3500 nM
   TI
   LI
   LO
   TS
2
Ki = 26360 nM
   TI
   LI
   LO
   TS
3
Ki = 55500 nM
   TI
   LI
   LO
   TS
CP0035563
US20230414632, Compound I-g
   Show/Hide
C35H38N4O6
 2
1
IC50 = 4600 nM
   TI
   LI
   LO
   TS
2
IC50 = 4650 nM
   TI
   LI
   LO
   TS
CP0005212
US8987315, Ketoconazole
   Show/Hide
C26H28Cl2N4O4
 3
1
IC50 = 4800 nM
   TI
   LI
   LO
   TS
2
Ki = 5270 nM
   TI
   LI
   LO
   TS
3
Ki = 24900 nM
   TI
   LI
   LO
   TS
CP0088895
Benidipine
   Show/Hide
C28H31N3O6
 2
1
IC50 = 4960 nM
   TI
   LI
   LO
   TS
2
IC50 = 9500 nM
   TI
   LI
   LO
   TS
CP0034615
(6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2.2.2]oct-2-yl)-methanol
   Show/Hide
C20H24N2O2
 1
1
IC50 = 5600 nM
   TI
   LI
   LO
   TS
CP0036382
CAS_52-53-9
   Show/Hide
C27H38N2O4
 1
1
IC50 = 6300 nM
   TI
   LI
   LO
   TS
CP0030899
1-[(2-chlorophenyl)-diphenylmethyl]imidazole
   Show/Hide
C22H17ClN2
 3
1
IC50 = 6700 nM
   TI
   LI
   LO
   TS
2
Ki = 29920 nM
   TI
   LI
   LO
   TS
3
Ki = 44000 nM
   TI
   LI
   LO
   TS
CP0406367
Barnidipine
   Show/Hide
C27H29N3O6
 2
1
IC50 = 8600 nM
   TI
   LI
   LO
   TS
2
IC50 = 12600 nM
   TI
   LI
   LO
   TS
CP0036175
1,3-thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[(2S)-3-methyl-2-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})carbamoyl]amino}butanamido]-1,6-diphenylhexan-2-yl]carbamate
   Show/Hide
C37H48N6O5S2
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0048327
(2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarbamoyl)-decahydroisoquinolin-2-yl]-3-hydroxy-1-phenylbutan-2-yl]-2-(quinolin-2-ylformamido)butanediamide
   Show/Hide
C38H50N6O5
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0924097
Efonidipine
   Show/Hide
C34H38N3O7P
 3
1
IC50 = 13000 nM
   TI
   LI
   LO
   TS
2
IC50 = 17300 nM
   TI
   LI
   LO
   TS
3
IC50 = 20600 nM
   TI
   LI
   LO
   TS
CP0077818
CL-287389
   Show/Hide
C19H19N3O6
 1
1
IC50 = 18000 nM
   TI
   LI
   LO
   TS
CP0055077
Amlodipine
   Show/Hide
C20H25ClN2O5
 1
1
IC50 = 22000 nM
   TI
   LI
   LO
   TS
CP0072914
US20230414632, Compound I-e
   Show/Hide
C20H24N2O6
 1
1
IC50 = 44100 nM
   TI
   LI
   LO
   TS
CP0000305
(-)-(etorphine)
   Show/Hide
C17H19NO3
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0008077
(1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,13,15-trimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-3,6-dien-5-one
   Show/Hide
C22H29FO5
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0035927
(Cimetidine) N-Methyl-N''''-[2-(5-methyl-1H-imidazol-4-ylmethylsulfanyl)-ethyl]-guanidine,cyanide
   Show/Hide
C10H16N6S
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0036823
(-)-etoposide
   Show/Hide
C29H32O13
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0037274
(S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-oxobenzo[a]heptalen-7-yl)acetamide
   Show/Hide
C22H25NO6
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0038098
(1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-en-5-one
   Show/Hide
C21H30O5
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0038418
13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid
   Show/Hide
C30H39N5O7S2
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0054979
DIGOXIN
   Show/Hide
C41H64O14
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0055087
(3R,4S,5S,6R,7R,9R,11R,12R,13S,14R)-6-[(2S,3R,4S,6R)-4-(dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-14-ethyl-7,12,13-trihydroxy-4-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-3,5,7,9,11,13-hexamethyl-oxacyclotetradecane-2,10-dione
   Show/Hide
C37H67NO13
 2
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
2
Ki = 37790 nM
   TI
   LI
   LO
   TS
CP0075209
(2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLASTINE
   Show/Hide
C46H58N4O9
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0078108
12-chloro-9-(2-fluorophenyl)-3-methyl-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,8,11,13-hexaene
   Show/Hide
C18H13ClFN3
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0663086
Ranitidine
   Show/Hide
C13H22N4O3S
 1
1
IC50 > 50000 nM
   TI
   LI
   LO
   TS
CP0072374
BAY-E-5009
   Show/Hide
C18H20N2O6
 1
1
IC50 = 68200 nM
   TI
   LI
   LO
   TS
CP0077731
(+)-cis-Diltiazem
   Show/Hide
C22H26N2O4S
 1
1
IC50 = 77700 nM
   TI
   LI
   LO
   TS
CP0035720
(-)-reserpine
   Show/Hide
C33H40N2O9
 2
1
Ki = 970 nM
   TI
   LI
   LO
   TS
2
Ki = 12200 nM
   TI
   LI
   LO
   TS
CP0084033
BROMOCRIPTINE
   Show/Hide
C32H40BrN5O5
 2
1
Ki = 2810 nM
   TI
   LI
   LO
   TS
2
Ki = 3960 nM
   TI
   LI
   LO
   TS
CP0068493
(2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-diiodophenoxy}ethyl)diethylamine
   Show/Hide
C25H29I2NO3
 1
1
Ki = 5780 nM
   TI
   LI
   LO
   TS
CP0047240
(6aR,9R)-N-[(1S,2S,4R,7S)-2-hydroxy-7-(2-methylpropyl)-5,8-dioxo-4-propan-2-yl-3-oxa-6,9-diazatricyclo[7.3.0.02,6]dodecan-4-yl]-7-methyl-6,6a,8,9-tetrahydro-4H-indolo[4,3-fg]quinoline-9-carboxamide
   Show/Hide
C32H41N5O5
 2
1
Ki = 6430 nM
   TI
   LI
   LO
   TS
2
Ki = 12200 nM
   TI
   LI
   LO
   TS
CP0194869
ERGOCRISTINE
   Show/Hide
C35H39N5O5
 2
1
Ki = 13330 nM
   TI
   LI
   LO
   TS
2
Ki = 42800 nM
   TI
   LI
   LO
   TS
CP0045584
(5'alpha)-12'-hydroxy-2'-methyl-5'-(phenylmethyl)ergotoman-3',6',18-trione
   Show/Hide
C33H35N5O5
 2
1
Ki = 14250 nM
   TI
   LI
   LO
   TS
2
Ki = 98900 nM
   TI
   LI
   LO
   TS
CP0208538
(6aR,9R,10aR)-N-[(1S,2S,4R,7S)-7-benzyl-2-hydroxy-5,8-dioxo-4-propan-2-yl-3-oxa-6,9-diazatricyclo[7.3.0.02,6]dodecan-4-yl]-7-methyl-6,6a,8,9,10,10a-hexahydro-4H-indolo[4,3-fg]quinoline-9-carboxamide
   Show/Hide
C35H41N5O5
 1
1
Ki = 16000 nM
   TI
   LI
   LO
   TS
CP0870792
alpha-Dihydroergocriptine
   Show/Hide
C32H43N5O5
 1
1
Ki = 19820 nM
   TI
   LI
   LO
   TS
CP0076396
ERGOCORNINE
   Show/Hide
C31H39N5O5
 1
1
Ki = 24500 nM
   TI
   LI
   LO
   TS
CP0057947
TROLEANDOMYCIN
   Show/Hide
C41H67NO15
 1
1
Ki = 87640 nM
   TI
   LI
   LO
   TS
CP0047294
ERGONOVINE
   Show/Hide
C19H23N3O2
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
Cell Viability or Cytotoxicity Assay
Compound ID Compound Name Compound Formula
CP0041805
(E)-resveratrol
   Show/Hide
C14H12O3  1
1
IC50 = 52500 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
GeneBLAzer AR-UAS-bla Griptite 293 Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -