General Information of the Cell Line
Cell Line ID
CL000930
Cell Line Name
GeneBLAzer AR-UAS-bla Griptite 293
Synonyms
GeneBLAzer AR-UAS-bla Griptite
AR-UAS-bla GripTite 293
AR-UAS-bla Griptite
Category
Transformed cell line
Organism
Homo sapiens (Human)
Tissue Information
Kidney
Disease None
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT01486, Androgen receptor
Compound ID Compound Name Compound Formula
CP0217093
Enobosarm
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C19H14F3N3O3
 1
1
IC50 = 36.4 nM
   TI
   LI
   LO
   TS
CP0390712
3-(4-cyano-3-fluorophenoxy)-2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]propanamide
   Show/Hide
C18H13F4N3O5
 1
1
IC50 = 49.2 nM
   TI
   LI
   LO
   TS
CP0482952
[(2S,3S,5R,11R,12S,15R,16S)-15-acetyl-9-chloro-2,16-dimethyl-6-oxo-15-pentacyclo[9.7.0.02,8.03,5.012,16]octadeca-7,9-dienyl] acetate
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C24H29ClO4
 1
1
IC50 = 58.6 nM
   TI
   LI
   LO
   TS
CP0531002
3-[4-cyano-2-(trifluoromethyl)phenoxy]-2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]propanamide
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C19H13F6N3O5
 1
1
IC50 = 72.2 nM
   TI
   LI
   LO
   TS
CP0488255
5,5-dimethyl-1-[4-nitro-3-(trifluoromethyl)phenyl]-3-[4-(trifluoromethyl)phenyl]imidazolidine-2,4-dione
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C19H13F6N3O4
 1
1
IC50 = 80.3 nM
   TI
   LI
   LO
   TS
CP0410891
5,5-dimethyl-1-[4-nitro-2-(trifluoromethyl)phenyl]-3-[3-(trifluoromethyl)phenyl]imidazolidine-2,4-dione
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C19H13F6N3O4
 1
1
IC50 = 111 nM
   TI
   LI
   LO
   TS
CP0410878
5,5-dimethyl-1,3-bis[3-(trifluoromethyl)phenyl]imidazolidine-2,4-dione
   Show/Hide
C19H14F6N2O2
 1
1
IC50 = 123 nM
   TI
   LI
   LO
   TS
CP0482916
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[2-(trifluoromethyl)phenoxy]propanamide
   Show/Hide
C18H14F6N2O5
 1
1
IC50 = 183 nM
   TI
   LI
   LO
   TS
CP0390714
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[2-(trifluoromethoxy)phenoxy]propanamide
   Show/Hide
C18H14F6N2O6
 1
1
IC50 = 198 nM
   TI
   LI
   LO
   TS
CP0410877
3,3,3-trifluoro-2-hydroxy-N-[4-nitro-3-(trifluoromethyl)phenyl]-2-[[2-(trifluoromethyl)phenyl]sulfanylmethyl]propanamide
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C18H11F9N2O4S
 1
1
IC50 = 245 nM
   TI
   LI
   LO
   TS
CP0482951
5,5-dimethyl-1-[4-nitro-2-(trifluoromethyl)phenyl]-3-[4-(trifluoromethyl)phenyl]imidazolidine-2,4-dione
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C19H13F6N3O4
 1
1
IC50 = 265 nM
   TI
   LI
   LO
   TS
CP0543069
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[2-(trifluoromethyl)phenyl]sulfanylpropanamide
   Show/Hide
C18H14F6N2O4S
 1
1
IC50 = 280 nM
   TI
   LI
   LO
   TS
CP0446951
2-hydroxy-2-methyl-N-[4-nitro-2-(trifluoromethyl)phenyl]-3-[2-(trifluoromethyl)phenyl]sulfanylpropanamide
   Show/Hide
C18H14F6N2O4S
 1
1
IC50 = 332 nM
   TI
   LI
   LO
   TS
CP0095953
ENZALUTAMIDE
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C21H16F4N4O2S
 1
1
IC50 = 361 nM
   TI
   LI
   LO
   TS
CP0390711
4-[5,5-dimethyl-2,4-dioxo-3-[4-(trifluoromethyl)phenyl]imidazolidin-1-yl]-3-(trifluoromethyl)benzonitrile
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C20H13F6N3O2
 1
1
IC50 = 402 nM
   TI
   LI
   LO
   TS
CP0482950
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[3-(trifluoromethoxy)phenoxy]propanamide
   Show/Hide
C18H14F6N2O6
 1
1
IC50 = 407 nM
   TI
   LI
   LO
   TS
CP0410879
N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methyl-3-[2-(trifluoromethyl)phenyl]sulfanylpropanamide
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C19H14F6N2O2S
 1
1
IC50 = 425 nM
   TI
   LI
   LO
   TS
CP0037412
(2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorobenzene)sulfonyl]-2-hydroxy-2-methylpropanamide
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C18H14F4N2O4S
 1
1
IC50 = 490 nM
   TI
   LI
   LO
   TS
CP0410880
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[4-(trifluoromethoxy)phenoxy]propanamide
   Show/Hide
C18H14F6N2O6
 1
1
IC50 = 625 nM
   TI
   LI
   LO
   TS
CP0536551
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[3-(trifluoromethyl)phenyl]sulfanylpropanamide
   Show/Hide
C18H14F6N2O4S
 1
1
IC50 = 625 nM
   TI
   LI
   LO
   TS
CP0543070
3-[4-cyano-2-(trifluoromethyl)phenoxy]-N-[4-cyano-2-(trifluoromethyl)phenyl]-2-hydroxy-2-methylpropanamide
   Show/Hide
C20H13F6N3O3
 1
1
IC50 = 736 nM
   TI
   LI
   LO
   TS
CP0410881
(2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methyl-3-[4-(trifluoromethyl)phenyl]sulfonylpropanamide
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C19H14F6N2O4S
 1
1
IC50 = 775 nM
   TI
   LI
   LO
   TS
CP0390713
(2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methyl-3-[4-(trifluoromethoxy)phenyl]sulfonylpropanamide
   Show/Hide
C19H14F6N2O5S
 1
1
IC50 = 777 nM
   TI
   LI
   LO
   TS
CP0410892
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[2-(trifluoromethyl)phenyl]sulfonylpropanamide
   Show/Hide
C18H14F6N2O6S
 1
1
IC50 = 811 nM
   TI
   LI
   LO
   TS
CP0482949
2-hydroxy-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]-3-[3-(trifluoromethyl)phenyl]sulfonylpropanamide
   Show/Hide
C18H14F6N2O6S
 1
1
IC50 = 1070 nM
   TI
   LI
   LO
   TS
CP0390715
(2R)-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-hydroxy-2-methyl-3-[4-(trifluoromethyl)phenyl]sulfanylpropanamide
   Show/Hide
C19H14F6N2O2S
 1
1
IC50 = 2170 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Kidney)
Cell Line Name Organism Disease
G-402 Homo sapiens (Human) Kidney neoplasm
A-498 Homo sapiens (Human) Renal cell carcinoma
786-O Homo sapiens (Human) Renal cell carcinoma
SN12C Homo sapiens (Human) Renal cell carcinoma
G-401 Homo sapiens (Human) Rhabdoid tumor of the kidney
AU-BEK Bos taurus (Bovine) -
MDCK Canis lupus familiaris (Dog) -
MDCK-II Canis lupus familiaris (Dog) -
MDCK-I Canis lupus familiaris (Dog) -
MDCK-MDR1 Canis lupus familiaris (Dog) -
MDCKII-LE Canis lupus familiaris (Dog) -
DK Canis lupus familiaris (Dog) -
MDCK2/BCRP Canis lupus familiaris (Dog) -
MDCK-Net6 Canis lupus familiaris (Dog) -
MDCK-UT-A1-AQP1-YFP Canis lupus familiaris (Dog) -
CV-1 Chlorocebus aethiops (Green monkey) -
COS-7 Chlorocebus aethiops (Green monkey) -
COS-1 Chlorocebus aethiops (Green monkey) -
COS-M6 Chlorocebus aethiops (Green monkey) -
COS Chlorocebus aethiops (Green monkey) -
OAT1-COS7 Chlorocebus aethiops (Green monkey) -
BS-C-1 Chlorocebus pygerythrus (Vervet monkey) -
Vero Chlorocebus sabaeus (Green monkey) -
OK Didelphis virginiana (North American opossum) -
HEK293 Homo sapiens (Human) -
HEK-293T Homo sapiens (Human) -
tsA201 Homo sapiens (Human) -
HEK293-A Homo sapiens (Human) -
T-REx-293 Homo sapiens (Human) -
HEK293-EBNA Homo sapiens (Human) -
Expi293F Homo sapiens (Human) -
Flp-In-293 Homo sapiens (Human) -
HEK293S Homo sapiens (Human) -
HEK293-F Homo sapiens (Human) -
HEK293-EBNA1-6E Homo sapiens (Human) -
AD-293 Homo sapiens (Human) -
HEK293-H Homo sapiens (Human) -
HEK-Blue hNOD2 Homo sapiens (Human) -
HEK293T/17 Homo sapiens (Human) -
293T/ACE2 [Japan 2021] Homo sapiens (Human) -
GripTite 293 MSR Homo sapiens (Human) -
HL-2 Homo sapiens (Human) -
HEK-Blue hTLR8 Homo sapiens (Human) -
PathHunter HEK 293 EDG1 Total GPCR Internalization Homo sapiens (Human) -
Flp-In-T-REx-293 Homo sapiens (Human) -
HEKR2 Homo sapiens (Human) -
HEK-Blue IL-6 Homo sapiens (Human) -
HK-2 [Human kidney] Homo sapiens (Human) -
HEK293-FT Homo sapiens (Human) -
HEK-2 Homo sapiens (Human) -
HEK-Blue hTLR2 Homo sapiens (Human) -
HEK-Blue hTLR4 Homo sapiens (Human) -
HEK-Blue CD40L Homo sapiens (Human) -
Expi293F GnTI- Homo sapiens (Human) -
HEK-Blue hNOD1 Homo sapiens (Human) -
pEAK Rapid Homo sapiens (Human) -
HEK-Blue hTLR9 Homo sapiens (Human) -
HEK-Blue hTLR7 Homo sapiens (Human) -
293Ta Homo sapiens (Human) -
293-Dual hSTING-R232 Homo sapiens (Human) -
HEK293-CNG Homo sapiens (Human) -
FreeStyle 293-F Homo sapiens (Human) -
PrecisION hnAChR alpha7/ric3-HEK Homo sapiens (Human) -
GeneBLAzer ERbeta-UAS-bla GripTite 293 Homo sapiens (Human) -
HEK385-7 Homo sapiens (Human) -
HEK2935 Homo sapiens (Human) -
ACTOne CXCR4 Homo sapiens (Human) -
HEK298 Homo sapiens (Human) -
HEK273 Homo sapiens (Human) -
293/GFP Homo sapiens (Human) -
HEK293 AequoScreen Homo sapiens (Human) -
HEK-Blue Null1-v Homo sapiens (Human) -
HEK-GIRK-M4 Homo sapiens (Human) -
HTLA Homo sapiens (Human) -
HEK293/Galpha15 Homo sapiens (Human) -
HEK293-SF-hH4R-His6-CRE-Luc Homo sapiens (Human) -
HEK293-SF-mH4R-His6-CRE-Luc Homo sapiens (Human) -
293AD Homo sapiens (Human) -
HEK293T/Galpha16-gustducin 44 Homo sapiens (Human) -
CellSensor SBE-bla HEK 293T Homo sapiens (Human) -
NRK1-HEK293T Homo sapiens (Human) -
HEK293T-SF-His6-CRE-Luc Homo sapiens (Human) -
HEK293T-beta-arr2-rH4R Homo sapiens (Human) -
HEK293T-beta-arr2-mH4R Homo sapiens (Human) -
HEK293T-beta-arr2-hH4R Homo sapiens (Human) -
HEK293T-SP-FLAG-hH3R-CRE-CBR Homo sapiens (Human) -
293/AP1-luc Homo sapiens (Human) -
293GT Homo sapiens (Human) -
UAS-MR-bla HEK293 Homo sapiens (Human) -
HEK293-DR-GFP Homo sapiens (Human) -
PSC-HEK293 Homo sapiens (Human) -
HEK-293-A2B Homo sapiens (Human) -
HEK293-SF-rH4R-His6-CRE-Luc Homo sapiens (Human) -
Hana3A Homo sapiens (Human) -
HEK293S GnTI- Homo sapiens (Human) -
GeneBLAzer UAS-bla GripTite 293 Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293H Homo sapiens (Human) -
GeneBLAzer UAS-bla HEK 293T Homo sapiens (Human) -
HEKMSR2 Homo sapiens (Human) -
HEK-hNET Homo sapiens (Human) -
HEK-hDAT Homo sapiens (Human) -
HEK-hSERT Homo sapiens (Human) -
EE-HEK293 Homo sapiens (Human) -
HEK-A2A Homo sapiens (Human) -
HEK293EM Homo sapiens (Human) -
293-NB2 Homo sapiens (Human) -
HEK-SEAP Homo sapiens (Human) -
HEK293/Gal4 Homo sapiens (Human) -
Octn2-HEK Homo sapiens (Human) -
Octn1-HEK Homo sapiens (Human) -
Octn3-HEK Homo sapiens (Human) -
HEK293superTOP Homo sapiens (Human) -
HEK293T-ARRB1 Homo sapiens (Human) -
HEK293T-ARRB2 Homo sapiens (Human) -
HEK293T-qs5-HA Homo sapiens (Human) -
EDG3-Ga15-bla HEK293T Homo sapiens (Human) -
LLC-MK2 Macaca mulatta (Rhesus macaque) -
BHK-21 Mesocricetus auratus (Golden hamster) -
BHK-21 clone 13 Mesocricetus auratus (Golden hamster) -
BHK570 Mesocricetus auratus (Golden hamster) -
TK-TS 13 Mesocricetus auratus (Golden hamster) -
BHK/AC9 Mesocricetus auratus (Golden hamster) -
mIMCD-3 Mus musculus (Mouse) -
RK3E Rattus norvegicus (Rat) -
KNRK Rattus norvegicus (Rat) -
NRK-52E Rattus norvegicus (Rat) -
SKPT-0193 Cl.2 Rattus norvegicus (Rat) -
RKE Rattus norvegicus (Rat) -
LLC-PK1 Sus scrofa (Pig) -
LLC-GA5-CoL150 Sus scrofa (Pig) -
PK-15 Sus scrofa (Pig) -
HKRK-B28 Sus scrofa (Pig) -
PK15NTD Sus scrofa (Pig) -