Brief Information of the Cell Line and Protein
Cell Line ID: CL000009 , LLC-PK1
Synonyms
LLC-PK(1)
LLC-PK-1
LLC PK-1
LLc-PK1
LLC PK1
LLCPK1
Lilly Laboratories Culture-Porcine Kidney 1
Category Spontaneously immortalized cell line
Organism
Sus scrofa (Pig)
Cellosaurus ID
CVCL_0391
Protein ID: PT06345 , Solute carrier family 15 member 2
Gene Name SLC15A2
Organism Rattus norvegicus, Rat
Protein Classification Transporter
Uniprot ID Q63424
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000009  Protein ID: PT06345
 
Compound ID Compound Name Compound Formula
CP0178740
BL-S578
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C16H17N3O5S
 1
1
Ki = 3000 nM
   TI
   LI
   LO
   TS
CP0133817
(S)-2-(2-Amino-acetylamino)-4-methyl-pentanoic acid
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C8H16N2O3
 1
1
Ki = 6000 nM
   TI
   LI
   LO
   TS
CP0228451
((S)-2-Amino-3-phenyl-propionylamino)-acetic acid
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C11H14N2O3
 1
1
Ki = 7000 nM
   TI
   LI
   LO
   TS
CP0233448
(S)-2-(2-Amino-acetylamino)-3-(1H-indol-3-yl)-propionic acid
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C13H15N3O3
 1
1
Ki = 7000 nM
   TI
   LI
   LO
   TS
CP0056548
(S)-2-(2-Amino-acetylamino)-3-phenyl-propionic acid
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C11H14N2O3
 1
1
Ki = 8000 nM
   TI
   LI
   LO
   TS
CP0354596
(2S)-2-[[(2S)-2-[(2-aminoacetyl)amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoic acid
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C17H25N3O5
 1
1
Ki = 8000 nM
   TI
   LI
   LO
   TS
CP0102052
(S)-2-(2-Amino-acetylamino)-3-(4-hydroxy-phenyl)-propionic acid
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C11H14N2O4
 1
1
Ki = 14000 nM
   TI
   LI
   LO
   TS
CP0288946
CHEBI:74394
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C8H16N2O3S
 1
1
Ki = 17000 nM
   TI
   LI
   LO
   TS
CP0037780
(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
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C16H24N2O4
 1
1
Ki = 18000 nM
   TI
   LI
   LO
   TS
CP0219242
((S)-2,6-Diamino-hexanoylamino)-acetic acid
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C8H17N3O3
 1
1
Ki = 21000 nM
   TI
   LI
   LO
   TS
CP0354595
CHEBI:73888
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C6H11N3O4
 1
1
Ki = 22000 nM
   TI
   LI
   LO
   TS
CP0049376
CICLACILLIN
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C15H23N3O4S
 1
1
Ki = 27000 nM
   TI
   LI
   LO
   TS
CP0233435
CHEBI:73905
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C13H17N3O4
 1
1
Ki = 29000 nM
   TI
   LI
   LO
   TS
CP0275781
(2S)-2-amino-N-(4-nitrophenyl)propanamide
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C9H11N3O3
 1
1
Ki = 29000 nM
   TI
   LI
   LO
   TS
CP0310662
(S)-2-(2-Amino-acetylamino)-3-(3H-imidazol-4-yl)-propionic acid
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C8H12N4O3
 1
1
Ki = 39000 nM
   TI
   LI
   LO
   TS
CP0213590
Substrate analogue, 16
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C4H8N2O3
 1
1
Ki = 42000 nM
   TI
   LI
   LO
   TS
CP0045560
(S)-3-Amino-N-carboxymethyl-succinamic acid
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C6H10N2O5
 1
1
Ki = 46000 nM
   TI
   LI
   LO
   TS
CP0271018
Anspor
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C16H19N3O4S
 1
1
Ki = 47000 nM
   TI
   LI
   LO
   TS
CP0099743
(6R,7R)-7-((R)-2-Amino-2-phenyl-acetylamino)-3-methyl-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid
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C16H17N3O4S
 1
1
Ki = 49000 nM
   TI
   LI
   LO
   TS
CP0219176
(S)-2-(2-Amino-acetylamino)-succinic acid
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C6H10N2O5
 1
1
Ki = 60000 nM
   TI
   LI
   LO
   TS
CP0119429
CHEBI:15727
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C9H14N4O3
 1
1
Ki = 66000 nM
   TI
   LI
   LO
   TS
CP0448888
(2S)-6-amino-2-[[(2S)-2,6-diaminohexanoyl]amino]hexanoic acid
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C12H26N4O3
 1
1
Ki = 96000 nM
   TI
   LI
   LO
   TS
CP0161781
2-(2-amino-N-methylacetamido)acetic acid
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C5H10N2O3
 1
1
Km = 110000 nM
   TI
   LI
   LO
   TS